NCT01081834

Brief Summary

The purpose of this study is to evaluate the efficacy, safety, and tolerability of 2 different doses of canagliflozin administered as monotherapy compared with placebo in patients with type 2 diabetes mellitus (T2DM) inadequately controlled with diet and exercise.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
678

participants targeted

Target at P50-P75 for phase_3 diabetes-mellitus-type-2

Timeline
Completed

Started Mar 2010

Typical duration for phase_3 diabetes-mellitus-type-2

Geographic Reach
17 countries

74 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 1, 2010

Completed
3 days until next milestone

First Submitted

Initial submission to the registry

March 4, 2010

Completed
1 day until next milestone

First Posted

Study publicly available on registry

March 5, 2010

Completed
1.4 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2011

Completed
7 months until next milestone

Study Completion

Last participant's last visit for all outcomes

March 1, 2012

Completed
1.3 years until next milestone

Results Posted

Study results publicly available

June 3, 2013

Completed
Last Updated

February 23, 2017

Status Verified

June 1, 2013

Enrollment Period

1.4 years

First QC Date

March 4, 2010

Results QC Date

April 15, 2013

Last Update Submit

February 15, 2017

Conditions

Keywords

Diabetes Mellitus, Type 2CanagliflozinPlaceboHemoglobin A1cType 2 diabetes mellitus

Outcome Measures

Primary Outcomes (2)

  • Change in HbA1c From Baseline to Week 26 (Main Study)

    The table below shows the least-squares (LS) mean change in HbA1c from Baseline to Week 26 for each treatment group. The statistical analyses show the treatment differences (ie, each canagliflozin group minus placebo) in the LS mean change.

    Day 1 (Baseline) and Week 26

  • Change in HbA1c From Baseline to Week 26 (High Glycemic Substudy)

    The table below shows the least-squares (LS) mean change in HbA1c from Baseline to Week 26 for each treatment group in patients randomized to the High Glycemic Substudy.

    Day 1 (Baseline) and Week 26

Secondary Outcomes (14)

  • Percentage of Patients With HbA1c <7% at Week 26 (Main Study)

    Week 26

  • Change in Fasting Plasma Glucose (FPG) From Baseline to Week 26 (Main Study)

    Day 1 (Baseline) and Week 26

  • Change in 2-hour Post-prandial Glucose From Baseline to Week 26 (Main Study)

    Day 1 (Baseline) and Week 26

  • Percent Change in Body Weight From Baseline to Week 26 (Main Study)

    Day 1 (Baseline) and Week 26

  • Change in Systolic Blood Pressure (SBP) From Baseline to Week 26 (Main Study)

    Day 1 (Baseline) and Week 26

  • +9 more secondary outcomes

Study Arms (3)

Canagliflozin 100 mg

EXPERIMENTAL

Each patient will receive 100 mg of canagliflozin once daily for 52 weeks (Main Study) or 26 weeks only (High Glycemic Substudy).

Drug: Canagliflozin

Canagliflozin 300 mg

EXPERIMENTAL

Each patient will receive 300 mg of canagliflozin once daily for 52 weeks (Main Study) or 26 weeks only (High Glycemic Substudy).

Drug: Canagliflozin

Placebo/Sitagliptin

EXPERIMENTAL

In the Main Study, each patient will receive matching placebo once daily for 26 weeks and will then switch from placebo to 100 mg of sitagliptin once daily until Week 52.

Drug: PlaceboDrug: Sitagliptin

Interventions

One 100 mg or 300 mg over-encapsulated tablet orally (by mouth) once daily for 52 weeks (Main Study) or 26 weeks (High Glycemic Substudy)

Canagliflozin 100 mgCanagliflozin 300 mg

One matching placebo capsule orally once daily for 26 weeks (Main Study)

Placebo/Sitagliptin

One 100 mg over-encapsulated tablet orally once daily beginning at Week 26 until Week 52 (Main Study)

Placebo/Sitagliptin

Eligibility Criteria

Age18 Years - 80 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • All patients must have a diagnosis of T2DM
  • Patients in the main study must have a Hemoglobin A1c (HbA1c) between \>=7% and \<=10% and a fasting plasma glucose (FPG) \<270 mg/dL (15 mmol/L)
  • Patients in the High Glycemic Cohort Substudy must have an HbA1c between \>10% and \<=12% and a FPG \<=350 mg/dL (19.44 mmol/L)

You may not qualify if:

  • History of diabetic ketoacidosis, type 1 diabetes mellitus (T1DM), pancreas or beta cell transplantation, diabetes secondary to pancreatitis or pancreatectomy, or a severe hypoglycemic episode within 6 months before screening

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (78)

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Phoenix, Arizona, United States

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Concord, California, United States

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Greenbrae, California, United States

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Los Angeles, California, United States

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Spring Valley, California, United States

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Colorado Springs, Colorado, United States

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Denver, Colorado, United States

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Northglenn, Colorado, United States

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Springfield, Illinois, United States

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Evansville, Indiana, United States

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Baton Rouge, Louisiana, United States

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Metairie, Louisiana, United States

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Meridian, New Jersey, United States

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Albuquerque, New Mexico, United States

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New York, New York, United States

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West Seneca, New York, United States

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Mooresville, North Carolina, United States

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Perryopolis, Pennsylvania, United States

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Pittsburgh, Pennsylvania, United States

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Taylors, South Carolina, United States

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Dallas, Texas, United States

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Houston, Texas, United States

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San Antonio, Texas, United States

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Norfolk, Virginia, United States

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Horn, Austria

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Salzburg, Austria

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Vienna, Austria

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Barranquilla, Colombia

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Bogotá, Colombia

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Pärnu, Estonia

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Tartu, Estonia

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Viljandi, Estonia

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Guatemala City, Guatemala

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Reykjavik, Iceland

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Bangalore, India

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Hyderabad, India

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Nagpur, India

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Kaunas, Lithuania

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Klaipėda, Lithuania

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Šiauliai, Lithuania

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Vilnius, Lithuania

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Vilnius Lt, Lithuania

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Kelantan, Malaysia

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Kuala Lumpur, Malaysia

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Aguascalientes, Mexico

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Guadalajara, Mexico

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Mexico City, Mexico

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Monterrey, Mexico

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Zapopan, Mexico

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Makati, Philippines

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Manila, Philippines

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Marikina City, Philippines

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Pasay, Philippines

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Katowice, Poland

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Torun, Poland

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Warsaw, Poland

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Fajardo, Puerto Rico

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Ponce, Puerto Rico

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San Juan, Puerto Rico

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Baia Mare, Romania

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Brasov, Romania

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Bucharest, Romania

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Târgu Mureş, Romania

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Halfway, South Africa

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Pretoria, South Africa

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Busan, South Korea

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Goyang-si, South Korea

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Jeonju, South Korea

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Seoul, South Korea

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Wŏnju, South Korea

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Alcalá de Henares, Spain

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Elche, Spain

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Girona, Spain

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Pozuelo de Alarcón, Spain

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Gothenburg, Sweden

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Lund, Sweden

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Malmo, Sweden

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Skene, Sweden

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Related Publications (17)

  • Davies MJ, Merton K, Vijapurkar U, Yee J, Qiu R. Efficacy and safety of canagliflozin in patients with type 2 diabetes based on history of cardiovascular disease or cardiovascular risk factors: a post hoc analysis of pooled data. Cardiovasc Diabetol. 2017 Mar 21;16(1):40. doi: 10.1186/s12933-017-0517-7.

  • Pfeifer M, Townsend RR, Davies MJ, Vijapurkar U, Ren J. Effects of canagliflozin, a sodium glucose co-transporter 2 inhibitor, on blood pressure and markers of arterial stiffness in patients with type 2 diabetes mellitus: a post hoc analysis. Cardiovasc Diabetol. 2017 Feb 27;16(1):29. doi: 10.1186/s12933-017-0511-0.

  • Gilbert RE, Mende C, Vijapurkar U, Sha S, Davies MJ, Desai M. Effects of Canagliflozin on Serum Magnesium in Patients With Type 2 Diabetes Mellitus: A Post Hoc Analysis of Randomized Controlled Trials. Diabetes Ther. 2017 Apr;8(2):451-458. doi: 10.1007/s13300-017-0232-0. Epub 2017 Feb 14.

  • Qiu R, Balis D, Xie J, Davies MJ, Desai M, Meininger G. Longer-term safety and tolerability of canagliflozin in patients with type 2 diabetes: a pooled analysis. Curr Med Res Opin. 2017 Mar;33(3):553-562. doi: 10.1080/03007995.2016.1271780. Epub 2017 Jan 4.

  • John M, Cerdas S, Violante R, Deerochanawong C, Hassanein M, Slee A, Canovatchel W, Hamilton G. Efficacy and safety of canagliflozin in patients with type 2 diabetes mellitus living in hot climates. Int J Clin Pract. 2016 Sep;70(9):775-85. doi: 10.1111/ijcp.12868.

  • Watts NB, Bilezikian JP, Usiskin K, Edwards R, Desai M, Law G, Meininger G. Effects of Canagliflozin on Fracture Risk in Patients With Type 2 Diabetes Mellitus. J Clin Endocrinol Metab. 2016 Jan;101(1):157-66. doi: 10.1210/jc.2015-3167. Epub 2015 Nov 18.

  • Lavalle-Gonzalez FJ, Eliaschewitz FG, Cerdas S, Chacon Mdel P, Tong C, Alba M. Efficacy and safety of canagliflozin in patients with type 2 diabetes mellitus from Latin America. Curr Med Res Opin. 2016;32(3):427-39. doi: 10.1185/03007995.2015.1121865. Epub 2016 Jan 14.

  • Blonde L, Woo V, Mathieu C, Yee J, Vijapurkar U, Canovatchel W, Meininger G. Achievement of treatment goals with canagliflozin in patients with type 2 diabetes mellitus: a pooled analysis of randomized controlled trials. Curr Med Res Opin. 2015 Nov;31(11):1993-2000. doi: 10.1185/03007995.2015.1082991. Epub 2015 Sep 28.

  • Gavin JR 3rd, Davies MJ, Davies M, Vijapurkar U, Alba M, Meininger G. The efficacy and safety of canagliflozin across racial groups in patients with type 2 diabetes mellitus. Curr Med Res Opin. 2015;31(9):1693-702. doi: 10.1185/03007995.2015.1067192. Epub 2015 Sep 4.

  • Cefalu WT, Stenlof K, Leiter LA, Wilding JP, Blonde L, Polidori D, Xie J, Sullivan D, Usiskin K, Canovatchel W, Meininger G. Effects of canagliflozin on body weight and relationship to HbA1c and blood pressure changes in patients with type 2 diabetes. Diabetologia. 2015 Jun;58(6):1183-7. doi: 10.1007/s00125-015-3547-2. Epub 2015 Mar 27.

  • Weir MR, Januszewicz A, Gilbert RE, Vijapurkar U, Kline I, Fung A, Meininger G. Effect of canagliflozin on blood pressure and adverse events related to osmotic diuresis and reduced intravascular volume in patients with type 2 diabetes mellitus. J Clin Hypertens (Greenwich). 2014 Dec;16(12):875-82. doi: 10.1111/jch.12425. Epub 2014 Oct 20.

  • Usiskin K, Kline I, Fung A, Mayer C, Meininger G. Safety and tolerability of canagliflozin in patients with type 2 diabetes mellitus: pooled analysis of phase 3 study results. Postgrad Med. 2014 May;126(3):16-34. doi: 10.3810/pgm.2014.05.2753.

  • Weir MR, Kline I, Xie J, Edwards R, Usiskin K. Effect of canagliflozin on serum electrolytes in patients with type 2 diabetes in relation to estimated glomerular filtration rate (eGFR). Curr Med Res Opin. 2014 Sep;30(9):1759-68. doi: 10.1185/03007995.2014.919907. Epub 2014 May 22.

  • Sinclair A, Bode B, Harris S, Vijapurkar U, Mayer C, Fung A, Shaw W, Usiskin K, Desai M, Meininger G. Efficacy and safety of canagliflozin compared with placebo in older patients with type 2 diabetes mellitus: a pooled analysis of clinical studies. BMC Endocr Disord. 2014 Apr 18;14:37. doi: 10.1186/1472-6823-14-37.

  • Polidori D, Mari A, Ferrannini E. Canagliflozin, a sodium glucose co-transporter 2 inhibitor, improves model-based indices of beta cell function in patients with type 2 diabetes. Diabetologia. 2014 May;57(5):891-901. doi: 10.1007/s00125-014-3196-x. Epub 2014 Mar 1.

  • Nyirjesy P, Sobel JD, Fung A, Mayer C, Capuano G, Ways K, Usiskin K. Genital mycotic infections with canagliflozin, a sodium glucose co-transporter 2 inhibitor, in patients with type 2 diabetes mellitus: a pooled analysis of clinical studies. Curr Med Res Opin. 2014 Jun;30(6):1109-19. doi: 10.1185/03007995.2014.890925. Epub 2014 Feb 21.

  • Stenlof K, Cefalu WT, Kim KA, Jodar E, Alba M, Edwards R, Tong C, Canovatchel W, Meininger G. Long-term efficacy and safety of canagliflozin monotherapy in patients with type 2 diabetes inadequately controlled with diet and exercise: findings from the 52-week CANTATA-M study. Curr Med Res Opin. 2014 Feb;30(2):163-75. doi: 10.1185/03007995.2013.850066. Epub 2013 Oct 28.

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

CanagliflozinSitagliptin Phosphate

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

ThiophenesSulfur CompoundsOrganic ChemicalsHeterocyclic Compounds, 1-RingHeterocyclic CompoundsGlucosidesGlycosidesCarbohydratesTriazolesAzolesPyrazines

Results Point of Contact

Title
Vice President, Franchise Medical Leader, Cardiovascular & Metabolism Franchise
Organization
Janssen Research & Development, LLC

Study Officials

  • Janssen Research & Development, LLC Clinical Trial

    Janssen Research & Development, LLC

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 4, 2010

First Posted

March 5, 2010

Study Start

March 1, 2010

Primary Completion

August 1, 2011

Study Completion

March 1, 2012

Last Updated

February 23, 2017

Results First Posted

June 3, 2013

Record last verified: 2013-06

Locations