NCT01137812

Brief Summary

The purpose of this study is to evaluate the efficacy and safety of canagliflozin compared with sitagliptin in patients with type 2 diabetes mellitus who are receiving treatment with metformin and sulphonylurea and have inadequate glycemic (blood sugar) control.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
756

participants targeted

Target at P75+ for phase_3 diabetes-mellitus-type-2

Timeline
Completed

Started Jul 2010

Typical duration for phase_3 diabetes-mellitus-type-2

Geographic Reach
17 countries

184 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 3, 2010

Completed
1 day until next milestone

First Posted

Study publicly available on registry

June 4, 2010

Completed
27 days until next milestone

Study Start

First participant enrolled

July 1, 2010

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 1, 2012

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

March 1, 2012

Completed
1.2 years until next milestone

Results Posted

Study results publicly available

May 17, 2013

Completed
Last Updated

January 15, 2015

Status Verified

January 1, 2015

Enrollment Period

1.7 years

First QC Date

June 3, 2010

Results QC Date

April 2, 2013

Last Update Submit

January 5, 2015

Conditions

Keywords

CanagliflozinSitagliptin (Januvia)MetforminSulphonylureaHemoglobin A1cType 2 diabetes mellitus

Outcome Measures

Primary Outcomes (1)

  • Change in HbA1c From Baseline to Week 52

    The table below shows the least-squares (LS) mean change in HbA1c from Baseline to Week 52 for each treatment group. The statistical analysis shows the treatment difference (ie, between canagliflozin and sitagliptin) in the LS mean change.

    Day 1 (Baseline) and Week 52

Secondary Outcomes (6)

  • Percentage of Patients With HbA1c <7% at Week 52

    Week 52

  • Change in Fasting Plasma Glucose (FPG) From Baseline to Week 52

    Day 1 (Baseline) and Week 52

  • Percent Change in Body Weight From Baseline to Week 52

    Day 1 (Baseline) and Week 52

  • Change in Systolic Blood Pressure (SBP) From Baseline to Week 52

    Day 1 (Baseline) and Week 52

  • Percent Change in Triglycerides From Baseline to Week 52

    Day 1 (Baseline) and Week 52

  • +1 more secondary outcomes

Study Arms (2)

Canagliflozin 300 mg

EXPERIMENTAL

Each patient will receive 300 mg of canagliflozin once daily for 52 weeks with protocol-specified doses of metformin and sulphonylurea

Drug: Canagliflozin 300 mgDrug: MetforminDrug: Sulphonylurea

Sitagliptin 100 mg

ACTIVE COMPARATOR

Each patient will receive 100 mg of sitagliptin once daily for 52 weeks with protocol-specified doses of metformin and sulphonylurea

Drug: Sitagliptin 100 mgDrug: MetforminDrug: Sulphonylurea

Interventions

One 100 mg capsule once daily for 52 weeks with protocol-specified doses of metformin and sulphonylurea

Sitagliptin 100 mg

One 300 mg capsule once daily for 52 weeks with protocol-specified doses of metformin and sulphonylurea

Canagliflozin 300 mg

Patients will continue to take background therapy with Metformin for T2DM at maximally or near-maximally effective protocol-specified doses for the duration of the study.

Canagliflozin 300 mgSitagliptin 100 mg

Patients will continue to take background therapy with Sulphonylurea for T2DM at maximally or near-maximally effective protocol-specified doses for the duration of the study.

Canagliflozin 300 mgSitagliptin 100 mg

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • All patients must have a diagnosis of T2DM and be currently treated with metformin and sulphonylurea
  • Patients in the study must have a HbA1c between \>=7 and \<=10.5% and a fasting plasma glucose (FPG) \<300 mg/dL (16.7 mmol/L)

You may not qualify if:

  • History of diabetic ketoacidosis, type 1 diabetes mellitus (T1DM), pancreas or beta cell transplantation, or diabetes secondary to pancreatitis or pancreatectomy
  • or a severe hypoglycemic episode within 6 months before screening

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (184)

Unknown Facility

Mobile, Alabama, United States

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Goodyear, Arizona, United States

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Mesa, Arizona, United States

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Escondido, California, United States

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Fresno, California, United States

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Greenbrae, California, United States

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La Mesa, California, United States

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Laguna Hills, California, United States

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Lancaster, California, United States

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Long Beach, California, United States

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Los Angeles, California, United States

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Norwalk, California, United States

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Pismo Beach, California, United States

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Roseville, California, United States

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Spring Valley, California, United States

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Walnut Creek, California, United States

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Watsonville, California, United States

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Denver, Colorado, United States

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Northglenn, Colorado, United States

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Milford, Connecticut, United States

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Bradenton, Florida, United States

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Cape Coral, Florida, United States

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Clearwater, Florida, United States

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Delray Beach, Florida, United States

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Miami, Florida, United States

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Pembroke Pines, Florida, United States

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Tampa, Florida, United States

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Atlanta, Georgia, United States

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Lewiston, Idaho, United States

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Chicago, Illinois, United States

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O'Fallon, Illinois, United States

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Springfield, Illinois, United States

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Topeka, Kansas, United States

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Bowling Green, Kentucky, United States

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Lexington, Kentucky, United States

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Madisonville, Kentucky, United States

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Baton Rouge, Louisiana, United States

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Mandeville, Louisiana, United States

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Metairie, Louisiana, United States

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Sunset, Louisiana, United States

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Brockton, Massachusetts, United States

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Saint Clair Shores, Michigan, United States

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Southfield, Michigan, United States

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Dakota Dunes, Nebraska, United States

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Toms River, New Jersey, United States

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Albuquerque, New Mexico, United States

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West Seneca, New York, United States

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Calabash, North Carolina, United States

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Greensboro, North Carolina, United States

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Moerhead City, North Carolina, United States

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Morganton, North Carolina, United States

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Cincinnati, Ohio, United States

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Gallipolis, Ohio, United States

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Marion, Ohio, United States

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Mason, Ohio, United States

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Toledo, Ohio, United States

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Zanesville, Ohio, United States

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Beaver, Pennsylvania, United States

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Bensalem, Pennsylvania, United States

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Norristown, Pennsylvania, United States

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Perryopolis, Pennsylvania, United States

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Philadelphia, Pennsylvania, United States

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Pittsburgh, Pennsylvania, United States

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Pottstown, Pennsylvania, United States

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Greenville, South Carolina, United States

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Spartanburg, South Carolina, United States

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Johnson City, Tennessee, United States

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Dallas, Texas, United States

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Fort Worth, Texas, United States

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Houston, Texas, United States

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Killeen, Texas, United States

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Richardson, Texas, United States

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San Antonio, Texas, United States

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Schertz, Texas, United States

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Sugar Land, Texas, United States

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Burke, Virginia, United States

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Danville, Virginia, United States

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Falls Church, Virginia, United States

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Hampton, Virginia, United States

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Henrico, Virginia, United States

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Manassas, Virginia, United States

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Norfolk, Virginia, United States

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Richmond, Virginia, United States

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Selah, Washington, United States

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Tacoma, Washington, United States

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Salzburg, Austria

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Vienna, Austria

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Hedersem (Aalst), Belgium

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Tremelo, Belgium

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Belém, Brazil

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Brasília, Brazil

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Fortaleza, Brazil

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Goiânia, Brazil

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Marília, Brazil

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Passo Fundo, Brazil

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Porto Alegre, Brazil

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Rio de Janeiro, Brazil

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São Paulo, Brazil

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Calgary, Alberta, Canada

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Red Deer, Alberta, Canada

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Vancouver, British Columbia, Canada

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Halifax, Nova Scotia, Canada

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Brampton, Ontario, Canada

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Oshawa, Ontario, Canada

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Toronto, Ontario, Canada

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Charlottetown, Prince Edward Island, Canada

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Sherbrooke, Quebec, Canada

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Ville, Laint-Laurent, Quebec, Canada

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Pointe-Claire, Canada

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Toronto, Canada

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Aalborg, Denmark

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Ballerup Municipality, Denmark

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Gentofte Municipality, Denmark

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Vejle, Denmark

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Vipperoed, Denmark

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Bondy, France

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Dijon, France

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Marseille, France

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Nantes, France

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Narbonne, France

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Paris, France

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Pessac, France

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Saint-Etienne, France

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Berlin, Germany

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Dresden, Germany

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Eisenach, Germany

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Großheirath, Germany

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Meißen, Germany

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Bangalore, India

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Coimbatore, India

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Hyderabad, India

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Jaipur, India

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Nagpur, India

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Nashik, India

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Pune, India

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Beersheba, Israel

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Jerusalem, Israel

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Kfar Saba, Israel

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Nazareth, Israel

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Rishon LeZiyyon, Israel

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Tel Aviv, Israel

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Ipoh, Malaysia

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Johor Bahru, Malaysia

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Kelantan, Malaysia

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Kuala Selangor, Malaysia

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Breda, Netherlands

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Eindhoven, Netherlands

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Groningen, Netherlands

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Leiderdorp, Netherlands

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Rotterdam, Netherlands

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Velp Gld, Netherlands

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Zoetermeer, Netherlands

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Christchurch, New Zealand

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Dunedin, New Zealand

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Rotorua, New Zealand

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Tauranga, New Zealand

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Wellington, New Zealand

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Bialystok, Poland

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Chrzanów, Poland

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Gdansk, Poland

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Kamieniec Ząbkowicki, Poland

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Krakow, Poland

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Lublin, Poland

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Sobótka, Poland

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Sopot, Poland

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Torun, Poland

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Wroclaw, Poland

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Zabrze, Poland

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Singapore, Singapore

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Busan, South Korea

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Daegu, South Korea

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Jeonju, South Korea

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Seongnam, South Korea

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Seoul, South Korea

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Dnipro, Ukraine

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Ivano-Frankivsk, Ukraine

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Kharkiv, Ukraine

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Kiev, Ukraine

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Odesa, Ukraine

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Poltava, Ukraine

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Sumy, Ukraine

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Ternopil, Ukraine

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Vinnitsa, Ukraine

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Zaporizhzhya, Ukraine

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Related Publications (8)

  • Cai J, Delahanty LM, Akapame S, Slee A, Traina S. Impact of Canagliflozin Treatment on Health-Related Quality of Life among People with Type 2 Diabetes Mellitus: A Pooled Analysis of Patient-Reported Outcomes from Randomized Controlled Trials. Patient. 2018 Jun;11(3):341-352. doi: 10.1007/s40271-017-0290-4.

  • Qiu R, Balis D, Xie J, Davies MJ, Desai M, Meininger G. Longer-term safety and tolerability of canagliflozin in patients with type 2 diabetes: a pooled analysis. Curr Med Res Opin. 2017 Mar;33(3):553-562. doi: 10.1080/03007995.2016.1271780. Epub 2017 Jan 4.

  • Schernthaner G, Lavalle-Gonzalez FJ, Davidson JA, Jodon H, Vijapurkar U, Qiu R, Canovatchel W. Canagliflozin provides greater attainment of both HbA1c and body weight reduction versus sitagliptin in patients with type 2 diabetes. Postgrad Med. 2016 Nov;128(8):725-730. doi: 10.1080/00325481.2016.1210988. Epub 2016 Jul 26.

  • Watts NB, Bilezikian JP, Usiskin K, Edwards R, Desai M, Law G, Meininger G. Effects of Canagliflozin on Fracture Risk in Patients With Type 2 Diabetes Mellitus. J Clin Endocrinol Metab. 2016 Jan;101(1):157-66. doi: 10.1210/jc.2015-3167. Epub 2015 Nov 18.

  • Lavalle-Gonzalez FJ, Eliaschewitz FG, Cerdas S, Chacon Mdel P, Tong C, Alba M. Efficacy and safety of canagliflozin in patients with type 2 diabetes mellitus from Latin America. Curr Med Res Opin. 2016;32(3):427-39. doi: 10.1185/03007995.2015.1121865. Epub 2016 Jan 14.

  • Bailey RA, Vijapurkar U, Meininger G, Rupnow MF, Blonde L. Diabetes-Related Composite Quality End Point Attainment: Canagliflozin Versus Sitagliptin Based on a Pooled Analysis of 2 Clinical Trials. Clin Ther. 2015 May 1;37(5):1045-54. doi: 10.1016/j.clinthera.2015.02.020. Epub 2015 Mar 18.

  • Polidori D, Mari A, Ferrannini E. Canagliflozin, a sodium glucose co-transporter 2 inhibitor, improves model-based indices of beta cell function in patients with type 2 diabetes. Diabetologia. 2014 May;57(5):891-901. doi: 10.1007/s00125-014-3196-x. Epub 2014 Mar 1.

  • Schernthaner G, Gross JL, Rosenstock J, Guarisco M, Fu M, Yee J, Kawaguchi M, Canovatchel W, Meininger G. Canagliflozin compared with sitagliptin for patients with type 2 diabetes who do not have adequate glycemic control with metformin plus sulfonylurea: a 52-week randomized trial. Diabetes Care. 2013 Sep;36(9):2508-15. doi: 10.2337/dc12-2491. Epub 2013 Apr 5.

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

Sitagliptin PhosphateCanagliflozinMetforminSulfonylurea Compounds

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

TriazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPyrazinesThiophenesSulfur CompoundsOrganic ChemicalsGlucosidesGlycosidesCarbohydratesBiguanidesGuanidinesAmidinesUreaAmidesSulfones

Results Point of Contact

Title
Vice President, Franchise Medical Leader, Cardiovascular & Metabolism Franchise
Organization
Janssen Research & Development, LLC

Study Officials

  • Janssen Research & Development, LLC C. Clinical Trial

    Janssen Research & Development, LLC

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 3, 2010

First Posted

June 4, 2010

Study Start

July 1, 2010

Primary Completion

March 1, 2012

Study Completion

March 1, 2012

Last Updated

January 15, 2015

Results First Posted

May 17, 2013

Record last verified: 2015-01

Locations