NCT06131840

Brief Summary

This clinical trial is studying advanced solid tumors. Solid tumors are cancers that start in a part of your body like your lungs or liver instead of your blood. Once tumors have grown bigger in one place but haven't spread, they're called locally advanced. If your cancer has spread to other parts of your body, it's called metastatic. When a cancer has gotten so big it can't easily be removed or has spread to other parts of the body, it is called unresectable. These types of cancer are harder to treat. Participants in this study must have cancer that has come back or did not get better with treatment. Participants must have a solid tumor cancer that can't be treated with standard of care drugs. This clinical trial uses an experimental drug called PF-08046050. PF-08046050 is a type of antibody-drug conjugate or ADC. ADCs are designed to stick to cancer cells and kill them. They may also stick to some normal cells. This study will test the safety of PF-08046050 in participants with solid tumors that are hard to treat or have spread throughout the body. This study has 5 different study parts. Part A and Part B of the study will find out how much PF-08046050 should be given to participants. Part C will use the information from Parts A and B to see if PF-08046050 is safe and if it works to treat certain solid tumor cancers. Part D and E of the study, together with information from Parts A and B, will find out how much PF-08046050 should be given in combination with other anti-cancer agents. Part E will use the information from Parts A, B, and D to see if PF-08046050 is safe in combination with other anti-cancer agents and if it works to treat a certain solid tumor.

Trial Health

83
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
914

participants targeted

Target at P75+ for phase_1

Timeline
53mo left

Started Nov 2023

Longer than P75 for phase_1

Geographic Reach
8 countries

44 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress36%
Nov 2023Sep 2030

First Submitted

Initial submission to the registry

November 9, 2023

Completed
5 days until next milestone

First Posted

Study publicly available on registry

November 14, 2023

Completed
6 days until next milestone

Study Start

First participant enrolled

November 20, 2023

Completed
5.8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

September 12, 2029

Expected
1 year until next milestone

Study Completion

Last participant's last visit for all outcomes

September 12, 2030

Last Updated

April 20, 2026

Status Verified

April 1, 2026

Enrollment Period

5.8 years

First QC Date

November 9, 2023

Last Update Submit

April 17, 2026

Conditions

Keywords

CRCNSCLCPDACGCGEJSCLCSeattle Genetics

Outcome Measures

Primary Outcomes (5)

  • Number of participants with adverse events (AEs)

    An AE is any untoward medical occurrence in a clinical study participant, temporally associated with the use of study intervention, whether or not considered related to the study intervention

    Through 30-37 days after the last study treatment, up to approximately 2 years

  • Number of participants with laboratory abnormalities

    Through 30-37 days after the last study treatment, up to approximately 2 years

  • Number of dose modifications due to AEs

    Through end of treatment up to approximately 2 years

  • Number of participants with dose-limiting toxicities (DLTs)

    Up to 28 days

  • Number of participants with DLTs by dose level

    Up to 28 days

Secondary Outcomes (10)

  • Pharmacokinetic (PK) parameter - Area under the concentration-time curve (AUC)

    Through 30-37 days after the last study treatment, up to approximately 2 years

  • PK parameter - Maximum concentration (Cmax)

    Through 30-37 days after the last study treatment, up to approximately 2 years

  • PK parameter - Time to maximum concentration (Tmax)

    Through 30-37 days after the last study treatment, up to approximately 2 years

  • PK parameter - Trough concentration (Ctrough)

    Through 30-37 days after the last study treatment, up to approximately 2 years

  • Number of participants with antidrug antibodies (ADAs)

    Through 30-37 days after the last study treatment, up to approximately 2 years

  • +5 more secondary outcomes

Study Arms (6)

PF-08046050

EXPERIMENTAL

PF-08046050 monotherapy

Drug: PF-08046050

PF-08046050 +bevacizumab

EXPERIMENTAL

PF-08046050 combination with bevacizumab

Drug: PF-08046050Drug: bevacizumab

PF-08046050 + bevacizumab + 5FU/LV

EXPERIMENTAL

PF-08046050 combination with bevacizumab + 5FU/LV

Drug: PF-08046050Drug: bevacizumabDrug: 5-Fluorouracil (5-FU)Drug: Leucovorin (LV)

PF-08046050 + 5FU/LV + oxaliplatin + bevacizumab

EXPERIMENTAL

PF-08046050 combination with 5FU/LV + oxaliplatin + bevacizumab

Drug: PF-08046050Drug: bevacizumabDrug: 5-Fluorouracil (5-FU)Drug: OxaliplatinDrug: Leucovorin (LV)

PF-08046050 + 5FU/LV + oxaliplatin

EXPERIMENTAL

PF-08046050 combination with 5FU/LV + oxaliplatin

Drug: PF-08046050Drug: 5-Fluorouracil (5-FU)Drug: OxaliplatinDrug: Leucovorin (LV)

PF-08046050 + 5FU/LV

EXPERIMENTAL

PF-08046050 combination with 5FU/LV

Drug: PF-08046050Drug: 5-Fluorouracil (5-FU)Drug: Leucovorin (LV)

Interventions

Given into the vein (IV; intravenous)

PF-08046050 + 5FU/LV + oxaliplatinPF-08046050 + 5FU/LV + oxaliplatin + bevacizumab

Given into the vein (IV; intravenous)

PF-08046050 + 5FU/LVPF-08046050 + 5FU/LV + oxaliplatinPF-08046050 + 5FU/LV + oxaliplatin + bevacizumabPF-08046050 + bevacizumab + 5FU/LV

Given into the vein (IV; intravenous)

Also known as: SAR445953; SGN-CEACAM5C
PF-08046050PF-08046050 + 5FU/LVPF-08046050 + 5FU/LV + oxaliplatinPF-08046050 + 5FU/LV + oxaliplatin + bevacizumabPF-08046050 + bevacizumab + 5FU/LVPF-08046050 +bevacizumab

Given into the vein (IV; intravenous)

PF-08046050 + 5FU/LV + oxaliplatin + bevacizumabPF-08046050 + bevacizumab + 5FU/LVPF-08046050 +bevacizumab

Given into the vein (IV; intravenous)

PF-08046050 + 5FU/LVPF-08046050 + 5FU/LV + oxaliplatinPF-08046050 + 5FU/LV + oxaliplatin + bevacizumabPF-08046050 + bevacizumab + 5FU/LV

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Tumor type:
  • Participants in Part A (dose escalation) and Part B (dose optimization) must have histologically- or cytologically-confirmed metastatic or unresectable solid tumor malignancy. Must have relapsed, refractory, or progressive disease, and should have no appropriate standard therapy available.
  • Participants in Part A must have one of the following tumor types: colorectal cancer (CRC); gastric carcinoma (GC) or gastroesophageal junction adenocarcinoma (GEJ); non-small cell lung cancer (NSCLC); or pancreatic ductal adenocarcinoma (PDAC).
  • The tumor types to be enrolled in Part B will be identified by the sponsor from among those specified in Part A.
  • Participants in Part C (dose expansion) must have one of the following histologically- or cytologically-confirmed metastatic or unresectable solid tumor malignancies.
  • CRC (adenocarcinoma of the colon or rectum) and must have received no more than 2 prior chemotherapy regimens for the treatment of advanced colorectal cancer and evidence of either progressive disease or intolerance to their last regimen.
  • PDAC with one or more metastatic lesions measurable by computed tomography/magnetic resonance imaging according to RECIST v1.1 criteria; and must have received no more than 1 prior chemotherapy regimen for the treatment of advanced PDAC and evidence of either progressive disease or intolerance to that regimen.
  • GC or GEJ and must have received prior platinum and fluoropyrimidine-based chemotherapy.
  • NSCLC and must have received platinum-based therapy. If eligible and consistent with local standard of care must have received a PD-1/PD-L1 inhibitor. In addition, participants with tumor genomic mutations/alterations for which approved targeted therapies are available per local standard of care, must have received such therapies.
  • Small cell lung cancer (SCLC) and must have received platinum-based therapy for extensive-stage disease and no more than 3 prior lines of therapy. If eligible and consistent with local standard of care must have received a PD 1/PD-L1 inhibitor.
  • CRC participants in Part D and Part E (bevacizumab combination therapy) must have histologically confirmed unresectable or metastatic adenocarcinoma of the colon or rectum. Received a maximum of 2 prior chemotherapy regimens for the treatment of advanced colorectal cancer and had demonstrated progressive disease or intolerance to their last regimen.
  • CRC participants in Part D and Part E (5FU/LV + bevacizumab and 5FU/LV + oxaliplatin + bevacizumab combination therapy) must have histologically confirmed unresectable or metastatic adenocarcinoma of the colon or rectum. Must not have received a prior TOPO1 inhibitor (such as irinotecan or nanoliposomal irinotecan) in any setting. 1L cohorts: No prior chemotherapy for advanced disease. 2L cohorts (applicable to 5FU/LV + bevacizumab combination only): 1 prior chemotherapy regimen for the treatment of advanced disease, which must have included a fluoropyrimidine and oxaliplatin.
  • \> 2L PDAC participants in Part E (5FU/LV combination therapy) must have histologically or cytologically confirmed metastatic pancreatic ductal adenocarcinoma. One or more metastatic lesions measurable by computed tomography/magnetic resonance imaging according to Response Evaluation Criteria in Solid Tumors (RECIST) version 1.1 criteria.
  • \> 1L PDAC participants in Part E (5FU/LV + oxaliplatin combination therapy) must have histologically or cytologically confirmed metastatic pancreatic ductal adenocarcinoma that has not been previously treated in the metastatic setting. One or more metastatic lesions measurable by computed tomography/magnetic resonance imaging according to Response Evaluation Criteria in Solid Tumors (RECIST) version 1.1 criteria. No prior chemotherapy for PDAC with the following exception: Patients who received adjuvant/neoadjuvant chemotherapy and who had recurrence more than 12 months after completion of adjuvant/neoadjuvant chemotherapy are eligible.
  • Participants enrolled in the following study parts should have a tumor site that is accessible for biopsy(ies) and agree to biopsy(ies) and/or submission of archival tissue:
  • +4 more criteria

You may not qualify if:

  • Previous exposure to CEACAM5-targeted therapy.
  • Prior treatment with a TOPO1-targeting ADC (CPT payload), such as Enhertu (trastuzumab deruxtecan) or Trodelvy (sacituzumab govitecan).
  • History of another malignancy within 3 years before the first dose of study intervention, or any evidence of residual disease from a previously diagnosed malignancy.
  • Active cerebral/meningeal disease related to the underlying malignancy. Participants with a history of cerebral/meningeal disease related to the underlying malignancy are allowed if prior central nervous system disease has been treated and the participant is clinically stable (defined as not having received steroid treatment for symptoms related to cerebral/meningeal disease for at least 2 weeks prior to enrollment and with no ongoing related AEs).
  • \> Criteria related to bevacizumab administration (participants in Parts D and E)
  • History of allergic reactions or hypersensitivity to bevacizumab or any of its excipients.
  • History of hypersensitivity to Chinese Hamster Ovary cell products or other recombinant human or humanized antibodies.
  • Serious non-healing wound, non-healing ulcer, or non-healing bone fracture.
  • Deep venous thromboembolic event within 4 weeks prior to enrollment
  • Known coagulopathy that increases risk of bleeding, bleeding diatheses.
  • History of any life-threatening VEGF-related adverse event

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (44)

Mayo Clinic Hospital

Phoenix, Arizona, 85054, United States

RECRUITING

Mayo Clinic

Scottsdale, Arizona, 85259, United States

RECRUITING

City of Hope (City of Hope National Medical Center, City of Hope Medical Center)

Duarte, California, 91010, United States

RECRUITING

IP Address: City of Hope Investigational Drug Services(IDS)

Duarte, California, 91010, United States

RECRUITING

University of Colorado Hospital - Anschutz Cancer Pavilion (ACP)

Aurora, Colorado, 80045, United States

RECRUITING

University of Colorado Hospital

Aurora, Colorado, 80045, United States

RECRUITING

Florida Cancer Specialists

Orlando, Florida, 32827, United States

RECRUITING

Sarah Cannon Research Institute at Florida Cancer Specialists

Orlando, Florida, 32827, United States

RECRUITING

Sidney Kimmel Comprehensive Cancer at Johns Hopkins

Baltimore, Maryland, 21287, United States

RECRUITING

The Johns Hopkins University

Baltimore, Maryland, 21287, United States

RECRUITING

Beth Israel Deaconess Medical Center

Boston, Massachusetts, 02115, United States

RECRUITING

Beth Israel Deaconess Medical Center

Boston, Massachusetts, 02215, United States

RECRUITING

START Midwest

Grand Rapids, Michigan, 49546, United States

RECRUITING

Mayo Clinic Cancer Center

Rochester, Minnesota, 55905, United States

RECRUITING

Mayo Clinic

Rochester, Minnesota, 55905, United States

RECRUITING

Sarah Cannon Research Institute - Pharmacy

Nashville, Tennessee, 37203, United States

RECRUITING

SCRI Oncology Partners

Nashville, Tennessee, 37203, United States

RECRUITING

The University of Texas MD Anderson Cancer Center

Houston, Texas, 77030, United States

RECRUITING

South Texas Accelerated Research Therapeutics, LLC

San Antonio, Texas, 78229, United States

RECRUITING

START Mountain Region

Salt Lake City, Utah, 84119, United States

RECRUITING

South Texas Accelerated Research Therapeutics Mountain Region

West Valley City, Utah, 84119, United States

RECRUITING

The Ottawa Hospital

Ottawa, Ontario, K1H 8L6, Canada

RECRUITING

University Health Network

Toronto, Ontario, M5G 2C4, Canada

RECRUITING

University Health Network, Princess Margaret Cancer Centre

Toronto, Ontario, M5G 2M9, Canada

RECRUITING

McGill University Health Centre

Montreal, Quebec, H4A 3J1, Canada

RECRUITING

The Sixth Affiliated Hospital of Sun Yat-sen University

Guangzhou, Guangdong, 510655, China

NOT YET RECRUITING

Institut Gustave Roussy

Villejuif, Paris, 94805, France

RECRUITING

Gustave Roussy

Villejuif, 94800, France

RECRUITING

Netherlands Cancer Institute

Amsterdam, 1066CX, Netherlands

RECRUITING

Institut Catala d'Oncologia - Hospital Duran i Reynals (ICO L'Hospitalet)

L'Hospitalet de Llobregat, Catalunya [cataluña], 08908, Spain

RECRUITING

Ascires Cetir

Barcelona, 08029, Spain

RECRUITING

Ascires CETIR

Esplugues de Llobregat, 08950, Spain

RECRUITING

Servicio de Farmacia ICO - Planta 0

L'Hospitalet de Llobregat, 08908, Spain

RECRUITING

Hospital Universitario HM Sanchinarro-CIOCC-START Madrid

Madrid, 28050, Spain

RECRUITING

Karolinska University Hospital

Solna, 171 64, Sweden

RECRUITING

ApoEx NKS

Stockholm, 17176, Sweden

RECRUITING

Diagnostic Centre

London, Others, WlG 7AF, United Kingdom

RECRUITING

The Harley Street Clinic (THSC)

London, Other, W1G 8BJ, United Kingdom

RECRUITING

Edinburgh Cancer Centre, Western General Hospital

Edinburgh, Scotland, EH4 2XU, United Kingdom

RECRUITING

Lothian Health Board

Edinburgh, EH3 9DN, United Kingdom

RECRUITING

Western General Hospital

Edinburgh, EH4 2XU, United Kingdom

RECRUITING

Sarah Cannon Research Institute UK

London, W1G 6AD, United Kingdom

RECRUITING

The Harley Street Clinic

London, W1G 7LJ, United Kingdom

RECRUITING

Radiology

London, W1G 8PP, United Kingdom

RECRUITING

Related Links

MeSH Terms

Conditions

Colorectal NeoplasmsCarcinoma, Non-Small-Cell LungStomach NeoplasmsSmall Cell Lung Carcinoma

Interventions

BevacizumabFluorouracilOxaliplatinLeucovorin

Condition Hierarchy (Ancestors)

Intestinal NeoplasmsGastrointestinal NeoplasmsDigestive System NeoplasmsNeoplasms by SiteNeoplasmsDigestive System DiseasesGastrointestinal DiseasesColonic DiseasesIntestinal DiseasesRectal DiseasesCarcinoma, BronchogenicBronchial NeoplasmsLung NeoplasmsRespiratory Tract NeoplasmsThoracic NeoplasmsLung DiseasesRespiratory Tract DiseasesStomach Diseases

Intervention Hierarchy (Ancestors)

Antibodies, Monoclonal, HumanizedAntibodies, MonoclonalAntibodiesImmunoglobulinsImmunoproteinsBlood ProteinsProteinsAmino Acids, Peptides, and ProteinsSerum GlobulinsGlobulinsUracilPyrimidinonesPyrimidinesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsCoordination ComplexesOrganic ChemicalsFormyltetrahydrofolatesTetrahydrofolatesFolic AcidPterinsPteridinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingCoenzymesEnzymes and Coenzymes

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Central Study Contacts

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

November 9, 2023

First Posted

November 14, 2023

Study Start

November 20, 2023

Primary Completion (Estimated)

September 12, 2029

Study Completion (Estimated)

September 12, 2030

Last Updated

April 20, 2026

Record last verified: 2026-04

Data Sharing

IPD Sharing
Will not share

Pfizer will provide access to individual de-identified participant data and related study documents (e.g. protocol, Statistical Analysis Plan (SAP), Clinical Study Report (CSR)) upon request from qualified researchers, and subject to certain criteria, conditions, and exceptions. Further details on Pfizer's data sharing criteria and process for requesting access can be found at: https://www.pfizer.com/science/clinical\_trials/trial\_data\_and\_results/data\_requests.

Locations