NCT03317392

Brief Summary

This phase I/II trial studies the best dose and side effects of olaparib and how well it works with radium Ra 223 dichloride in treating patients with castration-resistant prostate cancer that has spread to the bone and other places in the body (metastatic). PARPs are proteins that help repair DNA mutations. PARP inhibitors, such as olaparib, can keep PARP from working, so tumor cells can't repair themselves, and they may stop growing. Radioactive drugs, such as radium Ra 223 dichloride, may carry radiation directly to tumor cells and not harm normal cells. Giving olaparib and radium Ra 223 dichloride may help treat patients with castration-resistant prostate cancer.

Trial Health

75
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
132

participants targeted

Target at P75+ for phase_1

Timeline
10mo left

Started Feb 2019

Longer than P75 for phase_1

Geographic Reach
1 country

22 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress90%
Feb 2019Feb 2027

First Submitted

Initial submission to the registry

October 20, 2017

Completed
3 days until next milestone

First Posted

Study publicly available on registry

October 23, 2017

Completed
1.3 years until next milestone

Study Start

First participant enrolled

February 4, 2019

Completed
6.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 31, 2025

Completed
1.1 years until next milestone

Results Posted

Study results publicly available

May 5, 2026

Completed
10 months until next milestone

Study Completion

Last participant's last visit for all outcomes

February 16, 2027

Expected
Last Updated

May 5, 2026

Status Verified

April 1, 2026

Enrollment Period

6.2 years

First QC Date

October 20, 2017

Results QC Date

March 24, 2026

Last Update Submit

April 15, 2026

Conditions

Outcome Measures

Primary Outcomes (2)

  • Phase I: Maximum Tolerated Dose

    Determine the maximum tolerated dose (MTD) of olaparib in combination with radium Ra 223 dichloride (radium-223). (Phase I)

    56 days

  • Phase II: Radiographic Progression-free Survival (rPFS)

    Radiographic progression is defined by Prostate Cancer Working Group 3 criteria for bone metastases and RECIST version 1.1 for non-bone metastases. Median rPFS will be estimated using the Kaplan-Meier method by treatment arm. A stratified Cox proportional hazards regression model will estimate the rPFS treatment hazard ratio with 80% 2-sided confidence intervals (CIs). Progression is defined using Response Evaluation Criteria In Solid Tumors Criteria (RECIST v1.0), as a 20% increase in the sum of the longest diameter of target lesions, or a measurable increase in a non-target lesion, or the appearance of new lesions",

    From randomization to date of radiographic progression or death due to any cause, whichever occurs first, or censored at the date of last disease assessment. Up to approximately 2 years

Secondary Outcomes (5)

  • Phase II: rPFS in Patients Without Prior Docetaxel

    Up to approximately 2 years after randomization

  • Phase II: rPFS in Patients With Prior Docetaxel

    Up to approximately 2 years after randomization

  • Phase II: rPFS in Patients With ≤ 20 Bone Lesions

    Up to approximately 2 years after randomization

  • Phase II: rPFS in Patients With > 20 Bone Lesions

    Up to approximately 2 years after randomization

  • Phase II: Overall Survival (OS)

    From randomization to the date of death due to any cause, or censored at the date of last follow-up, assessed up to 3.5 years

Other Outcomes (6)

  • Phase II: rPFS in Patients Without Homologous Recombination Deficiency

    Up to approximately 2 years after randomization

  • Phase II: rPFS in Patients With Homologous Recombination Deficiency

    Up to approximately 2 years after randomization

  • Phase II: Prostate Specific Antigen (PSA) Response

    Up to approximately 2 years after randomization

  • +3 more other outcomes

Study Arms (4)

Phase II Arm I (radium Ra 223 dichloride, olaparib)

EXPERIMENTAL

Patients receive radium Ra 223 dichloride IV over 1 minute on day 1. Treatment repeats every 28 days for up to 6 cycles in the absence of disease progression or unacceptable toxicity. Patients also receive olaparib PO BID on days 1-28. Cycles repeat every 28 days in the absence of disease progression or unacceptable toxicity. Patients also undergo CT or MRI as well as blood sample collection and a tissue biopsy during screening and on study.

Procedure: Biopsy ProcedureProcedure: Biospecimen CollectionProcedure: Computed TomographyOther: Laboratory Biomarker AnalysisProcedure: Magnetic Resonance ImagingDrug: OlaparibOther: Quality-of-Life AssessmentRadiation: Radium Ra 223 Dichloride

Phase II Arm II (radium Ra 223 dichloride)

EXPERIMENTAL

Patients receive radium Ra 223 dichloride as in Arm I. Patients with radiographic progression may crossover to Arm I. If patients have already completed all 6 infusions of radium, they will receive monotherapy with olaparib. If they have not yet completed all 6 radium-223 infusion, they will continue radium-223 infusion until completion and receive concurrent treatment with olaparib. Patients also undergo CT or MRI as well as blood sample collection and a tissue biopsy during screening and on study.

Procedure: Biopsy ProcedureProcedure: Biospecimen CollectionProcedure: Computed TomographyOther: Laboratory Biomarker AnalysisProcedure: Magnetic Resonance ImagingOther: Quality-of-Life AssessmentRadiation: Radium Ra 223 Dichloride

Phase I Radium223+Olaparib dose level 1

EXPERIMENTAL

Dose level I: Radium223 plus olaparib 200 mg orally twice daily

Procedure: Biopsy ProcedureProcedure: Biospecimen CollectionProcedure: Computed TomographyOther: Laboratory Biomarker AnalysisProcedure: Magnetic Resonance ImagingDrug: OlaparibOther: Quality-of-Life AssessmentRadiation: Radium Ra 223 Dichloride

Phase I Radium223+Olaparib dose level 2

EXPERIMENTAL

Dose level II: Radium223 plus olaparib 300 mg orally twice daily

Procedure: Biopsy ProcedureProcedure: Biospecimen CollectionProcedure: Computed TomographyOther: Laboratory Biomarker AnalysisProcedure: Magnetic Resonance ImagingDrug: OlaparibOther: Quality-of-Life AssessmentRadiation: Radium Ra 223 Dichloride

Interventions

Given IV

Also known as: Alpharadin, BAY 88-8223, BAY88-8223, Radium 223 Dichloride, RADIUM RA-223 DICHLORIDE, Radium-223 Chloride, Radium-223 Dichloride, Xofigo
Phase I Radium223+Olaparib dose level 1Phase I Radium223+Olaparib dose level 2Phase II Arm I (radium Ra 223 dichloride, olaparib)Phase II Arm II (radium Ra 223 dichloride)

Undergo tissue biopsy

Also known as: Biopsy, BIOPSY_TYPE, Bx
Phase I Radium223+Olaparib dose level 1Phase I Radium223+Olaparib dose level 2Phase II Arm I (radium Ra 223 dichloride, olaparib)Phase II Arm II (radium Ra 223 dichloride)

Undergo blood sample collection

Also known as: Biological Sample Collection, Biospecimen Collected, Specimen Collection
Phase I Radium223+Olaparib dose level 1Phase I Radium223+Olaparib dose level 2Phase II Arm I (radium Ra 223 dichloride, olaparib)Phase II Arm II (radium Ra 223 dichloride)

Undergo CT

Also known as: CAT, CAT Scan, Computed Axial Tomography, Computerized Axial Tomography, Computerized axial tomography (procedure), Computerized Tomography, Computerized Tomography (CT) scan, CT, CT Scan, Diagnostic CAT Scan, Diagnostic CAT Scan Service Type, tomography
Phase I Radium223+Olaparib dose level 1Phase I Radium223+Olaparib dose level 2Phase II Arm I (radium Ra 223 dichloride, olaparib)Phase II Arm II (radium Ra 223 dichloride)

Correlative studies

Phase I Radium223+Olaparib dose level 1Phase I Radium223+Olaparib dose level 2Phase II Arm I (radium Ra 223 dichloride, olaparib)Phase II Arm II (radium Ra 223 dichloride)

Undergo MRI

Also known as: Magnetic Resonance, Magnetic Resonance Imaging (MRI), Magnetic resonance imaging (procedure), Magnetic Resonance Imaging Scan, Medical Imaging, Magnetic Resonance / Nuclear Magnetic Resonance, MR, MR Imaging, MRI, MRI Scan, MRIs, NMR Imaging, NMRI, Nuclear Magnetic Resonance Imaging, sMRI, Structural MRI
Phase I Radium223+Olaparib dose level 1Phase I Radium223+Olaparib dose level 2Phase II Arm I (radium Ra 223 dichloride, olaparib)Phase II Arm II (radium Ra 223 dichloride)

Given PO

Also known as: AZD 2281, AZD-2281, AZD2281, KU 0059436, KU-0059436, KU0059436, Lynparza, Olanib, Olaparix, PARP Inhibitor AZD2281
Phase I Radium223+Olaparib dose level 1Phase I Radium223+Olaparib dose level 2Phase II Arm I (radium Ra 223 dichloride, olaparib)

Ancillary studies

Also known as: Quality of Life Assessment
Phase I Radium223+Olaparib dose level 1Phase I Radium223+Olaparib dose level 2Phase II Arm I (radium Ra 223 dichloride, olaparib)Phase II Arm II (radium Ra 223 dichloride)

Eligibility Criteria

Age18 Years+
Sexmale
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participants must be male aged \>= 18 years of age
  • Participants must have histologically or cytologically confirmed adenocarcinoma of the prostate
  • Participants must have castrate levels of serum testosterone \< 50 ng/dL
  • Participants without orchiectomy must be maintained on luteinizing hormone releasing hormone (LHRH) agonist/antagonist; participants receiving prior docetaxel abiraterone, or next generation AR antagonist (enzalutamide, apalutamide, or darolutamide) for hormone sensitive disease are permitted
  • Participants must have progressive disease as defined by any of the following:
  • Castrate resistant disease as defined by PCWG-3 criteria; participants must have a rise in PSA on two successive determination at least one week apart and PSA levels \>= 2 ng/mL (only the screening PS needs to be \>= 2 ng/mL) and serum testosterone \< 50 ng/dL
  • Soft tissue progression as defined by RECIST version 1.1
  • Bone disease progression as defined by PCWG-3 criteria including the development of two or more new lesions on bone scan
  • Participants must have \>= 2 bone metastases by radiographic imaging and at least 1 lesion which has not been treated with prior radiation therapy
  • Participants must have tumor accessible for biopsy and be agreeable to baseline tumor biopsy; a metastatic focus is preferred but if not available and prostate is still intact prostate biopsy can be performed
  • Availability at the study site of formalin-fixed, paraffin-embedded (FFPE) archival tumor specimens, when available
  • Eastern Cooperative Oncology Group (ECOG) performance status =\< 1 (Karnofsky \>= 80%)
  • White blood cell count (WBC) \>= 3,000/mcL (within 28 days prior to administration of study treatment)
  • Absolute neutrophil count (ANC) \>= 1,500/mcL (within 28 days prior to administration of study treatment)
  • Platelets \>= 100,000/mcL (within 28 days prior to administration of study treatment)
  • +14 more criteria

You may not qualify if:

  • Pathology consistent with small cell carcinoma of the prostate
  • Presence of visceral metastases (liver, lung, brain, etc.) or malignant lymphadenopathy exceeding 4 centimeters (cm) in short diameter
  • Prior treatment with radium-223
  • Prior treatment with olaparib or other PARPi
  • Treatment with abiraterone, apalutamide, or darolutamide within 2 weeks of treatment initiation; treatment with cytotoxic chemotherapy within 3 weeks of treatment initiation; treatment with investigational prostate cancer directed therapy within 4 weeks of treatment initiation; treatment with enzalutamide within 4 weeks of treatment initiation
  • Prior hemibody external radiotherapy
  • Palliative radiation therapy to the bone or other sites within 2 weeks of treatment initiation
  • Participants who are receiving any other investigational agents
  • Imminent or established spinal cord compression based on clinical and/or imaging findings
  • Uncontrolled intercurrent illness including, but not limited to, ongoing or active infection requiring need for intravenous anti-microbials, symptomatic congestive heart failure, unstable angina pectoris, cardiac arrhythmia, or psychiatric illness/social situations that would limit compliance with study requirements
  • Clinically significant medical condition defined as:
  • Cerebral infarction within 6 months of study treatment
  • Transient ischemic attack within 3 months of study treatment
  • Myocardial infarction within 6 months of study treatment
  • Uncontrolled angina within 3 months of study treatment
  • +20 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (22)

UC San Diego Moores Cancer Center

La Jolla, California, 92093, United States

Location

University of California Davis Comprehensive Cancer Center

Sacramento, California, 95817, United States

Location

Smilow Cancer Center/Yale-New Haven Hospital

New Haven, Connecticut, 06510, United States

Location

Yale University

New Haven, Connecticut, 06520, United States

Location

University of Kansas Clinical Research Center

Fairway, Kansas, 66205, United States

Location

University of Kansas Cancer Center

Kansas City, Kansas, 66160, United States

Location

University of Kansas Cancer Center-Overland Park

Overland Park, Kansas, 66210, United States

Location

University of Kansas Hospital-Westwood Cancer Center

Westwood, Kansas, 66205, United States

Location

University of Maryland/Greenebaum Cancer Center

Baltimore, Maryland, 21201, United States

Location

Wayne State University/Karmanos Cancer Institute

Detroit, Michigan, 48201, United States

Location

Siteman Cancer Center at Saint Peters Hospital

City of Saint Peters, Missouri, 63376, United States

Location

Siteman Cancer Center at West County Hospital

Creve Coeur, Missouri, 63141, United States

Location

University of Kansas Cancer Center - North

Kansas City, Missouri, 64154, United States

Location

University of Kansas Cancer Center - Lee's Summit

Lee's Summit, Missouri, 64064, United States

Location

University of Kansas Cancer Center at North Kansas City Hospital

North Kansas City, Missouri, 64116, United States

Location

Washington University School of Medicine

St Louis, Missouri, 63110, United States

Location

Siteman Cancer Center-South County

St Louis, Missouri, 63129, United States

Location

Rutgers Cancer Institute of New Jersey

New Brunswick, New Jersey, 08903, United States

Location

Duke University Medical Center

Durham, North Carolina, 27710, United States

Location

Ohio State University Comprehensive Cancer Center

Columbus, Ohio, 43210, United States

Location

University of Pittsburgh Cancer Institute (UPCI)

Pittsburgh, Pennsylvania, 15232, United States

Location

University of Wisconsin Carbone Cancer Center - University Hospital

Madison, Wisconsin, 53792, United States

Location

MeSH Terms

Conditions

Prostatic Neoplasms

Interventions

BiopsySpecimen HandlingMagnetic Resonance Spectroscopyolaparibradium Ra 223 dichloride

Condition Hierarchy (Ancestors)

Genital Neoplasms, MaleUrogenital NeoplasmsNeoplasms by SiteNeoplasmsGenital Diseases, MaleGenital DiseasesUrogenital DiseasesProstatic DiseasesMale Urogenital Diseases

Intervention Hierarchy (Ancestors)

CytodiagnosisCytological TechniquesClinical Laboratory TechniquesDiagnostic Techniques and ProceduresDiagnosisDiagnostic Techniques, SurgicalSurgical Procedures, OperativeInvestigative TechniquesSpectrum AnalysisChemistry Techniques, Analytical

Results Point of Contact

Title
Rana Mckay
Organization
University of California, San Diego

Study Officials

  • Rana R McKay

    Yale University Cancer Center LAO

    PRINCIPAL INVESTIGATOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
LTE60
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
NIH
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 20, 2017

First Posted

October 23, 2017

Study Start

February 4, 2019

Primary Completion

March 31, 2025

Study Completion (Estimated)

February 16, 2027

Last Updated

May 5, 2026

Results First Posted

May 5, 2026

Record last verified: 2026-04

Data Sharing

IPD Sharing
Will share

NCI is committed to sharing data in accordance with NIH policy. For more details on how clinical trial data is shared, access the link to the NIH data sharing policy page.

More information

Locations