NCT05563272

Brief Summary

A prospective, open-label, phase 2 study to explore CAIX expression through 89Zirconium-labelled girentuximab deferoxamine (89Zr-girentuximab) PET/CT imaging in patients with solid tumors.

Trial Health

57
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
11

participants targeted

Target at below P25 for phase_2

Timeline
Completed

Started Jun 2023

Geographic Reach
1 country

10 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 23, 2022

Completed
10 days until next milestone

First Posted

Study publicly available on registry

October 3, 2022

Completed
8 months until next milestone

Study Start

First participant enrolled

June 6, 2023

Completed
1.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 9, 2025

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 9, 2025

Completed
Last Updated

July 10, 2025

Status Verified

July 1, 2025

Enrollment Period

1.9 years

First QC Date

September 23, 2022

Last Update Submit

July 7, 2025

Conditions

Outcome Measures

Primary Outcomes (2)

  • Qualitative assessment of 89Zr-girentuximab uptake within individual tumor deposits

    This outcome will be evaluated on all patients by using a PET/CT machine to qualitatively assess (yes / no) the uptake of the 89Zr-girentuximab uptake within individual tumor deposits.

    Single diagnostic administration, followed by a diagnostic scan on Day 5 ± 2 days. This assessment will be conducted throughout the patient dosing and imaging period, an average of 18 months

  • Quantitative assessment of 89Zr-girentuximab uptake within individual tumor deposits

    This outcome will be evaluated on all patients by using a PET/CT machine to quantitatively assess the uptake of the 89Zr-girentuximab uptake within individual tumor deposits.

    Single diagnostic administration, followed by a diagnostic scan on Day 5 ± 2 days. This assessment will be conducted throughout the patient dosing and imaging period, an average of 18 months

Secondary Outcomes (5)

  • To evaluate safety parameter of Heart rate in patients administered with 89Zr-girentuximab

    Patients will be evaluated for the period up to imaging following administration of 89Zr-girentuximab, at most 7 days.

  • To evaluate safety parameter of blood pressure in patients administered with 89Zr-girentuximab.

    Patients will be evaluated for the period up to imaging following administration of 89Zr-girentuximab, up to 7 days.

  • To evaluate safety parameter related to Liver function in patients administered 89Zr-girentuximab

    Patients will be evaluated for the period up to imaging following administration of 89Zr-girentuximab, up to 7 days.

  • To evaluate safety parameter related to Renal function in patients administered 89Zr-girentuximab

    Patients will be evaluated for the period up to imaging following administration of 89Zr-girentuximab, up to 7 days.

  • To evaluate safety parameter related to Full Blood Count in patients administered 89Zr-girentuximab

    Patients will be evaluated for the period up to imaging following administration of 89Zr-girentuximab, up to 7 days.

Study Arms (1)

89Zr-TLX250

EXPERIMENTAL
Diagnostic Test: 89Zr-girentuximab for PET/CT imaging of CAIX positive tumors

Interventions

On Day 0, participants will receive a single administration of 89Zr-girentuximab (37 Megabecquerel (MBq) \[1mCi\] ± 10%, containing a mass dose of 10 mg of girentuximab).

89Zr-TLX250

Eligibility Criteria

Age18 Years - 95 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • All participants must meet the following criteria:
  • Written and voluntarily given Informed Consent.
  • Male or female ≥18 years of age at time of consent.
  • Have the capacity to understand the study and be willing and able to comply with all protocol requirements.
  • Participants must have proven tumors of the following types, but not limited to:
  • Cervical cancer;
  • Colorectal cancer;
  • Esophageal SCC and esophageal/esophagogastric junction adenocarcinoma;
  • Gastric adenocarcinoma;
  • GBM;
  • Head and neck SCC and nasopharyngeal carcinoma;
  • cholangiocarcinoma and hepatocellular carcinoma;
  • non-small cell lung cancer;
  • small cell lung cancer;
  • epithelial ovarian carcinoma;
  • +11 more criteria

You may not qualify if:

  • Participants will be excluded from participation in the study if one or more of the following criteria are met:
  • Have been administered any radionuclide within 10 half-lives (of the radionuclide) prior to the intended administration of 89Zr-girentuximab (i.e., within 10 half-lives of Day 0);
  • Have been exposed to any CAIX targeting compound (diagnostic/therapeutic) in the prior 3 months;
  • Have any serious non-malignant disease (e.g., psychiatric, infectious, autoimmune or metabolic) that may interfere with the objectives of the study or with the safety or compliance of the participant, as judged by the Investigator;
  • Have any clinically significant abnormalities detected during screening laboratory tests or physical exam that, in the opinion of the Investigator, would adversely affect the participant's ability to participate in the study;
  • Have a mental impairment that may compromise the ability to give Informed Consent and comply with the requirements of the study;
  • Have been exposed to any antineoplastic treatment from Day 0 (89Zr-girentuximab dosing) to completion of 89Zr-girentuximab PET/CT imaging (Day 5 ± 2 days);
  • Be a female who is pregnant or breastfeeding;
  • Have a known allergy, hypersensitivity, or intolerance to girentuximab, desferrioxamine (DFO), or any of the components of the investigational agent;
  • Have renal insufficiency with a glomerular filtration rate (GFR) ≤45 milliliters/min/1.73m2
  • Be a vulnerable participant (e.g., being in detention).

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (10)

University of California, Los Angeles(UCLA)

Los Angeles, California, 90095, United States

Location

Biogenix Molecular, LLC

Miami, Florida, 33165, United States

Location

Massachusetts General Hospital

Boston, Massachusetts, 02114, United States

Location

Munson Medical Center

Traverse City, Michigan, 49684, United States

Location

University Hospitals Cleveland Medical Center (UHCMC)

Cleveland, Ohio, 44106, United States

Location

Kettering Health Research Institute

Kettering, Ohio, 45429, United States

Location

University of Pittsburgh Medical Center

Pittsburgh, Pennsylvania, 15219, United States

Location

Austin Radiological Association (ARA)

Austin, Texas, 78705, United States

Location

Carilion Clinic

Roanoke, Virginia, 24018, United States

Location

Inland Imaging

Spokane, Washington, 99208, United States

Location

MeSH Terms

Conditions

Uterine Cervical NeoplasmsColorectal NeoplasmsEsophageal NeoplasmsStomach NeoplasmsGlioblastomaCholangiocarcinomaCarcinoma, HepatocellularSquamous Cell Carcinoma of Head and NeckNasopharyngeal CarcinomaCarcinoma, Non-Small-Cell LungSmall Cell Lung CarcinomaCarcinoma, Ovarian EpithelialSarcomaMesothelioma, MalignantUrinary Bladder Neoplasms

Condition Hierarchy (Ancestors)

Uterine NeoplasmsGenital Neoplasms, FemaleUrogenital NeoplasmsNeoplasms by SiteNeoplasmsUterine Cervical DiseasesUterine DiseasesGenital Diseases, FemaleFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesGenital DiseasesIntestinal NeoplasmsGastrointestinal NeoplasmsDigestive System NeoplasmsDigestive System DiseasesGastrointestinal DiseasesColonic DiseasesIntestinal DiseasesRectal DiseasesHead and Neck NeoplasmsEsophageal DiseasesStomach DiseasesAstrocytomaGliomaNeoplasms, NeuroepithelialNeuroectodermal TumorsNeoplasms, Germ Cell and EmbryonalNeoplasms by Histologic TypeNeoplasms, Glandular and EpithelialNeoplasms, Nerve TissueAdenocarcinomaCarcinomaLiver NeoplasmsLiver DiseasesCarcinoma, Squamous CellNasopharyngeal NeoplasmsPharyngeal NeoplasmsOtorhinolaryngologic NeoplasmsNasopharyngeal DiseasesPharyngeal DiseasesStomatognathic DiseasesOtorhinolaryngologic DiseasesCarcinoma, BronchogenicBronchial NeoplasmsLung NeoplasmsRespiratory Tract NeoplasmsThoracic NeoplasmsLung DiseasesRespiratory Tract DiseasesOvarian NeoplasmsEndocrine Gland NeoplasmsOvarian DiseasesAdnexal DiseasesEndocrine System DiseasesGonadal DisordersNeoplasms, Connective and Soft TissueMesotheliomaAdenomaNeoplasms, MesothelialPleural NeoplasmsUrologic NeoplasmsUrinary Bladder DiseasesUrologic DiseasesMale Urogenital Diseases

Study Design

Study Type
interventional
Phase
phase 2
Allocation
NA
Masking
NONE
Purpose
DIAGNOSTIC
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 23, 2022

First Posted

October 3, 2022

Study Start

June 6, 2023

Primary Completion

May 9, 2025

Study Completion

May 9, 2025

Last Updated

July 10, 2025

Record last verified: 2025-07

Locations