NCT04933617

Brief Summary

Background: Burkitt Lymphoma (BL) and diffuse large B-cell lymphoma (DLBCL) are aggressive B cell lymphomas. Frontline treatment does not always work. Researchers want to see if a combination of drugs can help. Objective: To learn if it is safe to give people with certain cancers copanlisib together with rituximab and combination chemotherapy dose-adjusted etoposide, prednisone, vincristine, cyclophosphamide, doxorubicin, and rituximab (DA-EPOCH-R). Eligibility: People ages 18 and older with relapsed and/or refractory highly aggressive B-cell lymphomas such as BL and certain types of diffuse large B-cell lymphoma (DLBCL). Design: Participants will be screened with: Medical history Physical exam Bone marrow aspiration and biopsy. A needle will be put into their hipbone. Marrow will be removed. Imaging scans of the chest, abdomen, pelvis, and/or brain Tumor biopsy (if needed) Blood and urine tests Heart function tests Treatment will be given in 21-day cycles for up to 6 cycles. Participants will get copanlisib by intravenous (IV) infusion. They will also get a group of medicines called DA-EPOCH-R, as follows. They will get rituximab by IV infusion. Doxorubicin, etoposide, and vincristine will be mixed together in an IV bag and given by continuous IV infusion over 4 days. They will get cyclophosphamide by IV infusion. They will take prednisone by mouth. Participants will have frequent study visits. At these visits, they will repeat some screening tests. They may give tissue, saliva, and cheek swab samples. They will have at least one spinal tap. For this, a needle will be inserted into the spinal canal. Fluid will be removed. Participants will have a visit 30 days after treatment ends. They will have follow-up visits for at least 5 years.

Trial Health

57
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
8

participants targeted

Target at below P25 for phase_1

Timeline
Completed

Started Mar 2022

Geographic Reach
1 country

1 active site

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 18, 2021

Completed
4 days until next milestone

First Posted

Study publicly available on registry

June 22, 2021

Completed
9 months until next milestone

Study Start

First participant enrolled

March 24, 2022

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

November 30, 2023

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

November 30, 2023

Completed
7 months until next milestone

Results Posted

Study results publicly available

July 9, 2024

Completed
Last Updated

July 9, 2024

Status Verified

June 1, 2024

Enrollment Period

1.7 years

First QC Date

June 18, 2021

Results QC Date

May 16, 2024

Last Update Submit

June 13, 2024

Conditions

Keywords

AliqopaBAY 80-6946Monoclonal AntibodyPI3K Target

Outcome Measures

Primary Outcomes (1)

  • Maximum Tolerated Dose (MTD) and Recommended Phase II Dose (RP2D)

    MTD and RP2D is defined as the dose level at which no more than 1 of up to 6 participants experience dose limiting toxicity (DLT) during the DLT period, and the dose below that at which at least 2 (of ≤6) participants have DLT as a result of treatment. A DLT is any treatment-emergent, clinically relevant, and related severe (grade ≥ 3) toxicity that is possibly, probably, or definitely related to copanlisib.

    21 days

Secondary Outcomes (6)

  • Overall Response Rate (ORR)

    Response was assessed after cycles 1, 3 and 6 (each cycle is 21 days), approximately 63 days.

  • Progression-free Survival (PFS)

    Time from enrollment to progression or death, approximately 9 months.

  • Complete Response Rate

    Response was assessed after cycles 1, 3 and 6 (each cycle is 21 days). Approximately 63 days.

  • Overall Survival (OS)

    Time from enrollment to death, approximately 1 year

  • Event-free Survival (EFS)

    Time from enrollment to next line of anti-lymphoma therapy, progressive disease, or death. Approximately 6 months.

  • +1 more secondary outcomes

Other Outcomes (2)

  • Number of Participants With Serious and/or Non-serious Adverse Events Assessed by the Common Terminology Criteria for Adverse Events (CTCAE v5.0)

    Date treatment consent signed to date off study, an average of 245.5 days

  • Number of Participants With Dose Limiting-toxicity (DLT)

    21 days

Study Arms (2)

Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)

EXPERIMENTAL

Copanlisib intravenous (IV) per dose level (30 mg, 45 mg, or 60 mg) on day 1 of each 21-day cycle in combination with standard dosing dose adjusted rituximab, etoposide, prednisolone, vincristine, cyclophosphamide, doxorubicin (DA-EPOCH-R) to determine recommended phase 2 dose (RP2D) and maximum tolerated dose (MTD) of copanlisib. Up to 6 cycles total.

Biological: RituximabDrug: EtoposideBiological: CopanlisibDrug: CyclophosphamideDrug: DoxorubicinDrug: VincristineDrug: PrednisoneDiagnostic Test: ECHODiagnostic Test: EKGDiagnostic Test: MRI BrainDiagnostic Test: 18F-FDG - PETDiagnostic Test: CT ScanProcedure: Bone Marrow AspirationProcedure: Bone Marrow BiopsyDiagnostic Test: Lumbar Puncture (LP)

Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)

EXPERIMENTAL

Copanlisib intravenous (IV) at the recommended phase 2 dose (RP2D) or maximum tolerated dose (MTD) on day 1 of each 21-day cycle in combination with standard dosing dose adjusted rituximab, etoposide, prednisolone, vincristine, cyclophosphamide, doxorubicin (DA-EPOCH-R). Up to 6 cycles total.

Biological: RituximabDrug: EtoposideBiological: CopanlisibDrug: CyclophosphamideDrug: DoxorubicinDrug: VincristineDrug: PrednisoneDiagnostic Test: ECHODiagnostic Test: EKGDiagnostic Test: MRI BrainDiagnostic Test: 18F-FDG - PETDiagnostic Test: CT ScanProcedure: Bone Marrow AspirationProcedure: Bone Marrow BiopsyDiagnostic Test: Lumbar Puncture (LP)

Interventions

RituximabBIOLOGICAL

Rituximab 375 mg/m\^2 intravenous (IV) per protocol on Day 1 of each cycle up to 6 cycles

Also known as: Rituxan
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)

Etoposide 50 mg/m\^2/day continuous intravenous infusion (CIVI) on Days 1-4 of each cycle up to 6 cycles

Also known as: Toposar, Etopophos
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)
CopanlisibBIOLOGICAL

Copanlisib intravenous (IV) is administered at a fixed dose (30 mg, 45 mg, or 60 mg) on days 1 and 5 of each 21-day cycle for up to 6 cycles

Also known as: Aliqopa
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)

Cyclophosphamide 750 mg/m\^2 intravenous (IV) on Day 5 of each cycle up to 6 cycles

Also known as: Cytoxan
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)

Doxorubicin 10 mg/m\^2/day continuous intravenous infusion (CIVI) on Days 1-4 of each cycle up to 6 cycles

Also known as: Adriamycin
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)

Vincristine 0.4 mg/m\^2/day (no cap) continuous intravenous infusion (CIVI) on Days 1-4 of each cycle up to 6 cycles

Also known as: Marqibo, Vincasar PFS
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)

Prednisone 60 mg/m\^2 by mouth (PO) twice a day (BID) Days 1-5 (total 120mg/m\^2/day)

Also known as: Deltasone, Rayos, Prednisone Intensol
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)
ECHODIAGNOSTIC_TEST

At screening.

Also known as: Echocardiogram
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)
EKGDIAGNOSTIC_TEST

At screening.

Also known as: Electrocardiogram
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)
MRI BrainDIAGNOSTIC_TEST

At screening.

Also known as: Magnetic resonance imaging of the brain
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)
18F-FDG - PETDIAGNOSTIC_TEST

At screening, baseline, after cycle 1, 3, and 6, and end of treatment.

Also known as: Fludeoxyglucose F18
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)
CT ScanDIAGNOSTIC_TEST

At screening, baseline, after cycle 1, 3, and 6, end of treatment and follow-up.

Also known as: Computed tomography scan
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)

At screening and end of treatment.

Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)

At screening and end of treatment.

Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)
Lumbar Puncture (LP)DIAGNOSTIC_TEST

Baseline and end of treatment.

Also known as: Spinal tap
Arm 1- Dose Escalation, Original Copanlisib Intravenous (IV)Arm 2 - Dose Expansion, Modified Copanlisib Intravenous (IV)

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Subjects must have a histologic diagnosis, confirmed by the Laboratory of Pathology, National Cancer Institute (NCI) with one of the following subtypes and prior therapy, as follows:
  • At least 1 anthracycline-containing regimen:
  • Burkitt lymphoma
  • Burkitt-like lymphoma with 11q aberration
  • High-grade B-cell lymphoma, nor otherwise specified (NOS)
  • High-grade B-cell lymphoma, with myelocytomatosis (MYC) and B-cell lymphoma 2 (BCL2) and/or B-cell lymphoma 6 (BCL6) rearrangements
  • Must have had at least 2 prior regimens, 1 of which must have been anthracycline containing regimen OR be primary refractory to frontline therapy:
  • Diffuse large B-cell lymphoma (DLBCL), NOS, Germinal center B-cell type (GCB) type;
  • NOTE: subjects with coexisting or a history of indolent lymphoma are eligible (i.e., transformed lymphoma)
  • T-cell/histocyte-rich large B-cell lymphoma
  • Measurable or evaluable disease on imaging scans or bone marrow
  • No other current systemic anti-lymphoma therapy. NOTE: Recent short-term (less than or equal to 7 days) use of corticosteroids or prior radiation to sites of disease involvement is permitted.
  • Any human immunodeficiency virus (HIV) status will be included in this study as long as infection is controlled; in the opinion of the investigator. Status must be confirmed at screening and the subject must be willing to take any recommended antiretroviral therapy.
  • Greater than or equal to 18 years of age on day of signing informed consent
  • Eastern Cooperative Oncology Group (ECOG) performance status less than or equal to 2
  • +14 more criteria

You may not qualify if:

  • Subjects previously exposed to, intolerant of, or ineligible for phosphoinositide 3-kinases (PI3K) inhibitors and/or their combination
  • Brain parenchymal involvement
  • Patients who have been treated with prior chimeric antigen receptor (CAR)-T therapy or any regimen containing fludarabine.
  • Cytomegalovirus (CMV)-positive polymerase chain reaction (PCR) at screening
  • History of diabetic ketoacidosis
  • Uncontrolled intercurrent illness including, but not limited to the following that may limit interpretation of results or that could increase risk to the subject at the discretion of the investigator:
  • Any secondary malignancy that requires active systemic therapy
  • Diabetes mellitus with hemoglobin (Hgb) hemoglobin A1C (A1C) \> 8.5
  • Clinically significant interstitial lung disease and/or lung disease that severely impairs lung function
  • Uncontrolled human immunodeficiency virus (HIV)
  • Active hepatitis C infection. NOTE: Subjects who are hepatitis C antibody positive will need to have a negative hepatitis C virus (HCV) PCR result before enrollment. Those with a positive PCR for hepatitis C are excluded.
  • Active hepatitis B infection. NOTE: Patients who are hepatitis B surface antigen (HbsAg) or hepatitis B core antibody (HbcAb) positive will need to have a negative HBV PCR result before enrollment. Those with a positive PCR for hepatitis B are excluded. Those who are hepatitis B surface antigen (HbsAg) or hepatitis B core antibody (HbcAb) positive with a negative PCR for hepatitis B will be treated with antivirals designed to prevent hepatitis B reactivation (e.g., entecavir) throughout therapy and for 12 months after therapy and have monitoring for hepatitis B reactivation with PCR.
  • Clinically significant, uncontrolled heart disease and/or cardiac repolarization abnormalities, including any of the following:
  • History of acute coronary syndromes (including myocardial infarction, unstable angina, coronary artery bypass grafting, coronary angioplasty, or stenting) or symptomatic pericarditis within 6 months prior to screening
  • Congestive heart failure (New York Heart Association functional classification III-IV)
  • +10 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

National Institutes of Health Clinical Center

Bethesda, Maryland, 20892, United States

Location

Related Links

MeSH Terms

Conditions

Burkitt LymphomaLymphoma, Large B-Cell, Diffuse

Interventions

RituximabEtoposideetoposide phosphatecopanlisibCyclophosphamideDoxorubicinVincristinePrednisoneEchocardiographyElectrocardiographyTomography, X-Ray ComputedSpinal Puncture

Condition Hierarchy (Ancestors)

Epstein-Barr Virus InfectionsHerpesviridae InfectionsDNA Virus InfectionsVirus DiseasesInfectionsTumor Virus InfectionsLymphoma, B-CellLymphoma, Non-HodgkinLymphomaNeoplasms by Histologic TypeNeoplasmsLymphoproliferative DisordersLymphatic DiseasesHemic and Lymphatic DiseasesImmunoproliferative DisordersImmune System Diseases

Intervention Hierarchy (Ancestors)

Antibodies, Monoclonal, Murine-DerivedAntibodies, MonoclonalAntibodiesImmunoglobulinsImmunoproteinsBlood ProteinsProteinsAmino Acids, Peptides, and ProteinsSerum GlobulinsGlobulinsPodophyllotoxinTetrahydronaphthalenesNaphthalenesPolycyclic Aromatic HydrocarbonsHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsPolycyclic CompoundsGlucosidesGlycosidesCarbohydratesPhosphoramide MustardsNitrogen Mustard CompoundsMustard CompoundsHydrocarbons, HalogenatedPhosphoramidesOrganophosphorus CompoundsDaunorubicinAnthracyclinesNaphthacenesAminoglycosidesVinca AlkaloidsSecologanin Tryptamine AlkaloidsIndole AlkaloidsAlkaloidsHeterocyclic CompoundsIndolesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingIndolizidinesIndolizinesPregnadienediolsPregnadienesPregnanesSteroidsFused-Ring CompoundsCardiac Imaging TechniquesDiagnostic ImagingDiagnostic Techniques and ProceduresDiagnosisUltrasonographyHeart Function TestsDiagnostic Techniques, CardiovascularElectrodiagnosisImage Interpretation, Computer-AssistedRadiographic Image EnhancementImage EnhancementPhotographyRadiographyTomography, X-RayTomographyBiopsySpecimen HandlingClinical Laboratory TechniquesDiagnostic Techniques, NeurologicalPuncturesTherapeuticsSurgical Procedures, OperativeInvestigative Techniques

Results Point of Contact

Title
Dr. Mark Roschewski
Organization
National Cancer Institute

Study Officials

  • Mark J Roschewski, M.D.

    National Cancer Institute (NCI)

    PRINCIPAL INVESTIGATOR

Publication Agreements

PI is Sponsor Employee
No
Restrictive Agreement
No

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
NIH
Responsible Party
PRINCIPAL INVESTIGATOR
PI Title
Investigator

Study Record Dates

First Submitted

June 18, 2021

First Posted

June 22, 2021

Study Start

March 24, 2022

Primary Completion

November 30, 2023

Study Completion

November 30, 2023

Last Updated

July 9, 2024

Results First Posted

July 9, 2024

Record last verified: 2024-06

Data Sharing

IPD Sharing
Will share

All individual participant data (IPD) recorded in the medical record will be shared with intramural investigators upon request. All large- scale genomic sequencing data will be shared with subscribers to the database of Genotypes and Phenotypes (dbGaP).

Shared Documents
STUDY PROTOCOL, SAP, ICF
Time Frame
Clinical data available during the study and indefinitely. Genomic data are available once genomic data are uploaded per protocol Genomic Data Sharing (GDS) plan for as long as database is active.
Access Criteria
Clinical data will be made available via subscription to Biomedical Translational Research Information System (BTRIS) and with the permission of the study principal investigator (PI). Genomic data are made available via the database of Genotypes and Phenotypes (dbGaP) through requests to the data custodians.

Locations