NCT04720976

Brief Summary

To evaluate the safety and tolerability of JAB-3312 administered in investigational regimens in adult participants with advanced solid tumors.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
58

participants targeted

Target at P50-P75 for phase_1

Timeline
Completed

Started Mar 2021

Typical duration for phase_1

Geographic Reach
1 country

15 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

January 18, 2021

Completed
4 days until next milestone

First Posted

Study publicly available on registry

January 22, 2021

Completed
2 months until next milestone

Study Start

First participant enrolled

March 23, 2021

Completed
2.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 19, 2023

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

December 19, 2023

Completed
Last Updated

April 11, 2025

Status Verified

March 1, 2025

Enrollment Period

2.7 years

First QC Date

January 18, 2021

Last Update Submit

April 9, 2025

Conditions

Keywords

KRAS G12C, EGFR

Outcome Measures

Primary Outcomes (7)

  • Number of participants with dose limiting toxicities

    Incidence of dose limiting toxicities (DLTs) in the dose escalation phase. A DLT is defined as an adverse event or abnormal laboratory value assessed as unrelated to disease, disease progression, inter-current illness, or concomitant medications that occurs within the first treatment cycle. (Dose escalation phase)

    24 months

  • Objective response rate (ORR)

    ORR is defined as the proportion of participants with complete response or partial response (CR+PR). (Dose expansion phase)

    24 months

  • Duration of response (DOR)

    DOR is defined as the time from the participant's initial objective response (CR or PR) to study drug therapy, to disease progression or death due to any cause, whichever occurs first. (Dose expansion phase)

    24 months

  • Duration of response (DCR)

    DCR is defined as proportion of participants with complete response, partial response, stable disease(CR+PR+SD). (Dose expansion phase)

    24 months

  • Progression-free survival (PFS)

    PFS is defined as the interval of time between the date of first treatment to the earliest date of disease progression or death which occurs first. (Dose expansion phase)

    24 months

  • Overall survival (OS)

    OS is defined as the interval of time between the date of first treatment until death, loss to follow up or termination of the study by the sponsor. (Dose expansion phase)

    24 months

  • Number of participants with adverse events

    All patients participating in this study will be assessed for incidence and severity of adverse events (AEs) and serious AEs, including changes in laboratory values, vital signs, electrocardiograms, cardiac imaging and ophthalmological assessments (Dose escalation phase)

    24 months

Secondary Outcomes (9)

  • Objective response rate (ORR)

    24 months

  • Duration of response (DOR)

    24 months

  • Duration of response (DCR)

    24 months

  • Progression-free survival (PFS)

    24 months

  • Overall survival (OS)

    24 months

  • +4 more secondary outcomes

Study Arms (8)

JAB-3312+Pembrolizumab dose escalation

EXPERIMENTAL

Dose escalation

Drug: JAB-3312Drug: Pembrolizumab

JAB-3312+ Binimetinib dose escalation

EXPERIMENTAL

Dose escalation

Drug: JAB-3312Drug: Binimetinib

JAB-3312+Pembrolizumab dose expansion

EXPERIMENTAL

Dose expansion

Drug: JAB-3312Drug: Pembrolizumab

JAB-3312+Binimetinib dose expansion

EXPERIMENTAL

Dose expansion

Drug: JAB-3312Drug: Binimetinib

JAB-3312+Sotorasib dose escalation

EXPERIMENTAL

Dose escalation

Drug: JAB-3312Drug: Sotorasib

JAB-3312+ Osimertinib dose escalation

EXPERIMENTAL

Dose escalation

Drug: JAB-3312Drug: Osimertinib

JAB-3312+ Sotorasib dose expansion

EXPERIMENTAL

Dose expansion

Drug: JAB-3312Drug: Sotorasib

JAB-3312+ Osimertinib dose expansion

EXPERIMENTAL

Dose expansion

Drug: JAB-3312Drug: Osimertinib

Interventions

JAB-3312 will be administered orally, variable dose.

JAB-3312+ Binimetinib dose escalationJAB-3312+ Osimertinib dose escalationJAB-3312+ Osimertinib dose expansionJAB-3312+ Sotorasib dose expansionJAB-3312+Binimetinib dose expansionJAB-3312+Pembrolizumab dose escalationJAB-3312+Pembrolizumab dose expansionJAB-3312+Sotorasib dose escalation

Binimetinib will be administered orally.

JAB-3312+ Binimetinib dose escalationJAB-3312+Binimetinib dose expansion

Pembrolizumab will be administered as an intravenous infusion.

JAB-3312+Pembrolizumab dose escalationJAB-3312+Pembrolizumab dose expansion

Sotorasib will be administered orally.

JAB-3312+ Sotorasib dose expansionJAB-3312+Sotorasib dose escalation

Osimertinib will be administered orally.

JAB-3312+ Osimertinib dose escalationJAB-3312+ Osimertinib dose expansion

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Must have histologically or cytologically confirmed metastatic or locally advanced solid tumor. Some cohorts must meet specific expression or gene mutation where indicated
  • Sufficient organ function
  • Participants must have at least 1 measurable lesion as defined by RECIST v1.1
  • Must be able to provide an archived tumor sample
  • ECOG performance status score of 0 or 1.

You may not qualify if:

  • History of cancer that is histologically distinct from the cancers under study
  • Active or untreated central nervous system (CNS) metastases
  • History of pneumonitis or interstitial lung disease (ILD)
  • Has active hepatitis B, hepatitis C infection, HIV
  • Any severe and/or uncontrolled medical conditions
  • LVEF ≤50%
  • QTcF \>470 msec

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (15)

Research Site

Phoenix, Arizona, 85054, United States

Location

Research Site

Scottsdale, Arizona, 85259, United States

Location

Research Site

Los Angeles, California, 90033, United States

Location

Research Site

New Haven, Connecticut, 06510, United States

Location

Research Site

Jacksonville, Florida, 32224, United States

Location

Research Site

Orange City, Florida, 32763, United States

Location

Research Site

Chicago, Illinois, 60637, United States

Location

Research Site

Indianapolis, Indiana, 46202, United States

Location

Research Site

Detroit, Michigan, 48202, United States

Location

Research Site

Rochester, Minnesota, 55902, United States

Location

Research Site

St Louis, Missouri, 63130, United States

Location

Research Site

New York, New York, 10016, United States

Location

Research Site

Oklahoma City, Oklahoma, 73104, United States

Location

Research Site

Houston, Texas, 77030, United States

Location

Research Site

Salt Lake City, Utah, 84112, United States

Location

Related Publications (1)

  • Kang D, Wang Y, Lin Y, Ma WW, Morgensztern D, Leventakos K, Bi C, Ding Y, Xiong J, Yan M, Sun X, Wang P, Ma C, Wang Y. JAB-3312, a Potent Allosteric SHP2 Inhibitor That Enhances the Efficacy of RTK/RAS/MAPK and PD-1 Blockade Therapies. Clin Cancer Res. 2025 Jul 15;31(14):3019-3032. doi: 10.1158/1078-0432.CCR-24-3691.

MeSH Terms

Interventions

binimetinibpembrolizumabsotorasibosimertinib

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 18, 2021

First Posted

January 22, 2021

Study Start

March 23, 2021

Primary Completion

December 19, 2023

Study Completion

December 19, 2023

Last Updated

April 11, 2025

Record last verified: 2025-03

Locations