NCT01636908

Brief Summary

The purpose of this study is to determine intratumoral concentration of kinase inhibitors upon 2 weeks of treatment in tumor tissue of patients.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
43

participants targeted

Target at P25-P50 for not_applicable cancer

Timeline
Completed

Started Aug 2011

Longer than P75 for not_applicable cancer

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

August 1, 2011

Completed
11 months until next milestone

First Submitted

Initial submission to the registry

July 5, 2012

Completed
5 days until next milestone

First Posted

Study publicly available on registry

July 10, 2012

Completed
5.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 1, 2018

Completed
1.9 years until next milestone

Study Completion

Last participant's last visit for all outcomes

December 1, 2019

Completed
Last Updated

April 15, 2021

Status Verified

April 1, 2021

Enrollment Period

6.4 years

First QC Date

July 5, 2012

Last Update Submit

April 14, 2021

Conditions

Outcome Measures

Primary Outcomes (1)

  • concentrations of intratumoral kinase inhibitors upon 2 weeks of treatment

    2 weeks

Secondary Outcomes (4)

  • kinase inhibitor concentrations in plasma, serum and PBMC's upon 2 weeks of treatment

    2 weeks

  • intra-dermal kinase inhibitor concentrations upon 2 weeks of treatment

    2 weeks

  • To determine per patient whether 2 weeks of treatment with kinase inhibitors induces significant change of phosphoproteomic profiles in tumor tissue

    2 weeks

  • To determine per patient whether 2 weeks of treatment with kinase inhibitors induces significant change of kinase activity in tumor tissue

    2 weeks

Study Arms (1)

Kinase inhibitor

EXPERIMENTAL

Patients are cohort-wise treated with a registered (tyrosine) kinase inhibitor

Drug: SunitinibDrug: SorafenibDrug: ErlotinibDrug: EverolimusDrug: LapatinibDrug: DasatinibDrug: PazopanibDrug: VemurafenibProcedure: tumor biopsyProcedure: skin biopsy (optional)

Interventions

50 mg once daily, oral use, 14 days

Kinase inhibitor

400 mg, twice daily, oral use, 14 days

Kinase inhibitor

150 mg once daily, oral use, 14 days

Kinase inhibitor

10 mg once daily, oral use, 14 days

Kinase inhibitor

1250 mg once daily, oral use, 14 days

Kinase inhibitor

100 mg once daily, oral use, 14 days

Kinase inhibitor

800 mg once daily, oral use, 14 days

Kinase inhibitor

960 mg twice daily, oral use, 15-21 days

Kinase inhibitor
tumor biopsyPROCEDURE
Kinase inhibitor
Kinase inhibitor

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Advanced solid malignancy
  • minimum age 18 years
  • indication for palliative treatment
  • measurable disease with at least one lesion accessable for biopsy

You may not qualify if:

  • Cardiovascular conditions including congestive heartfailure NYHA class \>2
  • recent myocardial infarction or uncontrolled coronary artery disease
  • cardiac arrhythmias requiring anti-arrhythmic therapy
  • uncontrolled hypertension
  • uncontrolled infections
  • serious non-healing wound, ulcer or bone fracture
  • pregnant or breast feeding

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

VUMedical Center

Amsterdam, 1081 HV, Netherlands

Location

MeSH Terms

Conditions

Neoplasms

Interventions

SunitinibSorafenibErlotinib HydrochlorideEverolimusLapatinibDasatinibpazopanibVemurafenib

Intervention Hierarchy (Ancestors)

PyrrolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsIndolesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingPhenylurea CompoundsUreaAmidesOrganic ChemicalsBenzene DerivativesHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsNiacinamideNicotinic AcidsAcids, HeterocyclicPyridinesQuinazolinesSirolimusMacrolidesLactonesThiazolesSulfur CompoundsPyrimidinesSulfonamidesSulfones

Study Officials

  • H.M.W. Verheul, MD, PhD

    VU Medical Center Amsterdam

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
not applicable
Allocation
NA
Masking
NONE
Purpose
DIAGNOSTIC
Intervention Model
SINGLE GROUP
Sponsor Type
OTHER
Responsible Party
PRINCIPAL INVESTIGATOR
PI Title
Medical Oncologist

Study Record Dates

First Submitted

July 5, 2012

First Posted

July 10, 2012

Study Start

August 1, 2011

Primary Completion

January 1, 2018

Study Completion

December 1, 2019

Last Updated

April 15, 2021

Record last verified: 2021-04

Locations