NCT07377578

Brief Summary

Mantle cell lymphoma (MCL) is an aggressive yet often indolent type of B-cell non-Hodgkin lymphoma (NHL). Rocbrutinib (LP-168) is a novel, highly selective, fourth-generation Bruton's tyrosine kinase (BTK) inhibitor that exhibits both covalent (irreversible) and non-covalent (reversible) binding. This unique dual mechanism of action has shown promising efficacy and a favorable safety profile across various B-cell NHL subtypes in prior Phase 1 and 2 studies. This is a Phase 3, randomized, open-label study comparing Rocbrutinib versus investigator's choice of BTK inhibitor (ibrutinib, acalabrutinib, zanubrutinib, or orelabrutinib) in patients with MCL who have received at least one prior line of therapy and are naïve to BTK inhibitor treatment (except for intolerance).

Trial Health

77
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
394

participants targeted

Target at P50-P75 for phase_3

Timeline
82mo left

Started Feb 2026

Longer than P75 for phase_3

Geographic Reach
1 country

2 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress4%
Feb 2026Jan 2033

First Submitted

Initial submission to the registry

January 13, 2026

Completed
17 days until next milestone

First Posted

Study publicly available on registry

January 30, 2026

Completed
6 days until next milestone

Study Start

First participant enrolled

February 5, 2026

Completed
5.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 30, 2031

Expected
1.7 years until next milestone

Study Completion

Last participant's last visit for all outcomes

January 30, 2033

Last Updated

February 6, 2026

Status Verified

February 1, 2026

Enrollment Period

5.3 years

First QC Date

January 13, 2026

Last Update Submit

February 4, 2026

Conditions

Keywords

Mantle Cell LymphomaBTK inhibitorRocbrutinib

Outcome Measures

Primary Outcomes (1)

  • Progression-free survival (PFS) assessed by IRC

    approximately 30 months

Secondary Outcomes (6)

  • PFS assessed by INV

    approximately 30 months

  • Overall Response Rate (ORR) assessed by IRC and INV, respectively

    Up to approximately 24 months

  • Duration of Response (DOR) assessed by IRC and INV, respectively

    approximately 30 months

  • Overall Survival

    approximately 40 months

  • Number of participants with treatment-emergent adverse event as assessed by CTCAE v5.0

    Up to approximately 40 months

  • +1 more secondary outcomes

Study Arms (2)

Arm A (Rocbrutinib)

EXPERIMENTAL
Drug: Rocbrutinib

Arm B (ibrutinib, acalabrutinib, zanubrutinib, or orelabrutinib)

ACTIVE COMPARATOR
Drug: IbrutinibDrug: AcalabrutinibDrug: ZanubrutinibDrug: Orelabrutinib

Interventions

Rocbrutinib at 150 mg once daily orally until disease progression or unacceptable toxicity

Arm A (Rocbrutinib)

Ibrutinib, 560 mg once daily orally and continuously

Arm B (ibrutinib, acalabrutinib, zanubrutinib, or orelabrutinib)

Acalabrutinib, 100 mg twice daily orally and continuously

Arm B (ibrutinib, acalabrutinib, zanubrutinib, or orelabrutinib)

Zanubrutinib, 160 mg twice daily orally and continuously

Arm B (ibrutinib, acalabrutinib, zanubrutinib, or orelabrutinib)

Orelabrutinib, 150 mg once daily orally and continuously

Arm B (ibrutinib, acalabrutinib, zanubrutinib, or orelabrutinib)

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Diagnosed with MCL, who have received at least one prior systemic regimen(s), and have experienced disease progression on the most recent line of therapy.
  • Have at least one measurable lesion according to the Lugano Response Criteria 2014.
  • Eastern Cooperative Oncology Group (ECOG) Performance Status score of 0-2.
  • Life expectancy ≥ 12 weeks.
  • Adequate coagulation function, liver and kidney function, bone marrow hematopoietic function, etc.
  • Toxicities or complications from prior anti-tumor therapy have recovered to Grade ≤1 according to NCI CTCAE v5.0.
  • All male subjects and female subjects of childbearing potential must strictly use medically approved contraception throughout the entire study period. All male subjects must also avoid sperm donation during the above period. For women of childbearing potential, the result of serum pregnancy test must be obtained. Women must be non-lactating.
  • Subject voluntarily enrolls and signs the informed consent form, and agrees to comply with the study treatment plan and visit schedule.

You may not qualify if:

  • Hypersensitivity to Rocbrutinib or any study drug in the control group.
  • Prior treatment with any BTK-targeted therapy (except for intolerance).
  • Central nervous system (CNS) involvement by lymphoma.
  • History of other malignancy (except MCL) within the past 2 years, excluding radically cured skin basal cell carcinoma, cervical carcinoma in situ, breast carcinoma in situ, localized squamous cell carcinoma, etc.
  • History of major cardiovascular events within 6 months prior to randomization.
  • Presence of any severe and/or uncontrolled systemic disease that, in the investigator's judgment, or have poor cardiac function.
  • Uncontrolled active bacterial, fungal, or viral systemic infection, or active tuberculosis infection.
  • Any medical condition that could interfere with the absorption, distribution, metabolism, or excretion (ADME) of the investigational drug or the evaluation of study outcomes.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (2)

Beijing Cancer hospital

Beijing, Beijing Municipality, 100142, China

RECRUITING

The First Affiliated Hospital of Guangxi Medical University

Nanning, Guangxi, 530021, China

NOT YET RECRUITING

MeSH Terms

Conditions

Lymphoma, Mantle-Cell

Interventions

ibrutinibacalabrutinibzanubrutiniborelabrutinib

Condition Hierarchy (Ancestors)

Lymphoma, Non-HodgkinLymphomaNeoplasms by Histologic TypeNeoplasmsLymphoproliferative DisordersLymphatic DiseasesHemic and Lymphatic DiseasesImmunoproliferative DisordersImmune System Diseases

Central Study Contacts

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
SINGLE
Who Masked
INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 13, 2026

First Posted

January 30, 2026

Study Start

February 5, 2026

Primary Completion (Estimated)

May 30, 2031

Study Completion (Estimated)

January 30, 2033

Last Updated

February 6, 2026

Record last verified: 2026-02

Data Sharing

IPD Sharing
Will not share

Locations