NCT05261399

Brief Summary

Clinical study to investigate the efficacy and safety of savolitinib in combination with osimertinib versus platinum-based doublet chemotherapy in participants with EGFR mutated, MET-overexpressed and/or amplified, locally advanced or metastatic NSCLC who have progressed on treatment with Osimertinib.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
341

participants targeted

Target at P50-P75 for phase_3

Timeline
3mo left

Started Aug 2022

Typical duration for phase_3

Geographic Reach
27 countries

214 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress93%
Aug 2022Nov 2026

First Submitted

Initial submission to the registry

February 15, 2022

Completed
15 days until next milestone

First Posted

Study publicly available on registry

March 2, 2022

Completed
5 months until next milestone

Study Start

First participant enrolled

August 3, 2022

Completed
3.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 6, 2026

Completed
5 months until next milestone

Study Completion

Last participant's last visit for all outcomes

November 23, 2026

Expected
Last Updated

August 6, 2026

Status Verified

July 1, 2026

Enrollment Period

3.9 years

First QC Date

February 15, 2022

Last Update Submit

August 5, 2026

Conditions

Keywords

SavolitinibOsimertinibEGFRAmplifiedMetastaticMET DrivencarcinomaNSCLCoverexpressed

Outcome Measures

Primary Outcomes (1)

  • Progression-free survival (PFS) / savolitinib + osimertinib versus platinum doublet chemotherapy in participants with EGFR mutated, MET-overexpressed and/or amplified, locally advanced or metastatic NSCLC who have progressed on osimertinib.

    Defined as time from randomisation until progression per RECIST 1.1 as assessed by BICR, or death due to any cause.

    Approximately 36.5 months post first subject randomized

Secondary Outcomes (13)

  • Overall Survival (OS) /savolitinib + osimertinib versus platinum doublet chemotherapy in participants with EGFR mutated, MET-overexpressed and/or amplified locally advanced or metastatic NSCLC who have progressed on treatment with osimertinib.

    Approximately 36.5+18 months post first subject randomized.

  • Progression-free survival (PFS) / savolitinib + osimertinib versus platinum doublet chemotherapy in participants with EGFR mutated, MET-overexpressed, locally advanced or metastatic NSCLC who have progressed on treatment with osimertinib.

    Approximately 55 months post first subject randomized

  • Overall Survival (OS) / savolitinib in combination with osimertinib versus platinum doublet chemotherapy in participants with EGFR mutated, MET-overexpressed by IHC, locally advanced or metastatic NSCLC who have progressed on treatment with osimertinib.

    Approximately 55 months post first subject randomized

  • Objective response rate (ORR) savolitinib + osimertinib versus platinum doublet chemotherapy in participants with EGFR mutated, MET-overexpressed and/or amplified locally advanced or metastatic NSCLC who have progressed on treatment with osimertinib.

    Approximately 55 months post first subject randomized

  • Savolitinib+osimertinib vs platinum doublet chemotherapy in terms of BICR-assessed CNS endpoints in participants with EGFR mutated, MET overexpressed and/or amplified, locally advanced or metastatic NSCLC progressed on treatment with osimertinib

    Approximately 55 months post first subject randomized

  • +8 more secondary outcomes

Study Arms (2)

Chemotherapy

ACTIVE COMPARATOR

Pemetrexed (500 mg/m2) with either cisplatin (75 mg/m2) or carboplatin (AUC5) on Day 1 of 21-day cycles (Q3W) for 4 cycles, followed by pemetrexed maintenance (500 mg/m2) Q3W

Drug: PemetrexedDrug: CisplatinDrug: Carboplatin

Savolitinib + Osimertinib

EXPERIMENTAL

300 mg savolitinib BID plus 80 mg osimertinib QD

Drug: SavolitinibDrug: Osimertinib

Interventions

300 mg savolitinib (3 × 100 mg tablets twice daily) Administrative route : oral

Also known as: AZD6094, HMPL-504, volitinib
Savolitinib + Osimertinib

80 mg osimertinib (1 × 80 mg tablet once daily) Administrative route : oral

Also known as: AZD9291, Tagrisso
Savolitinib + Osimertinib

Pemetrexed (500 mg/m2) Administrative route : IV infusion

Also known as: NAP
Chemotherapy

Cisplatin (75 mg/m2) Administrative route : IV infusion

Also known as: NAP
Chemotherapy

Carboplatin (AUC5) Administrative route : IV infusion

Also known as: NAP
Chemotherapy

Eligibility Criteria

Age18 Years - 130 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Provision of signed and dated written ICF prior to any mandatory and non-mandatory study-specific procedures, sampling and analyses.
  • Participant must be ≥18 years (≥ 19 years of age in South Korea) at the time of signing the informed consent. All genders are permitted.
  • Histologically or cytologically confirmed locally advanced or metastatic NSCLC which is not amenable to curative therapy.
  • Must have at least one documented sensitising EGFR mutation: exon19 deletion, L858R mutation, and/or T790M.
  • Documented radiologic progression on first- or second-line treatment with osimertinib as the most recent anti-cancer therapy.
  • Mandatory provision of FFPE tumour tissue.
  • MET overexpression and/or amplification in tumour specimen collected following progression on prior osimertinib treatment.
  • Measurable disease as defined by RECIST 1.1.
  • Adequate haematological, liver, renal and cardiac functions, and coagulation parameters.
  • ECOG performance status of 0 or 1.

You may not qualify if:

  • Predominant squamous NSCLC, and small cell lung cancer.
  • Prior or current treatment with a third-generation EGFR-TKI other than Osimertinib.
  • Prior or current treatment with savolitinib or another MET inhibitors.
  • Spinal cord compression or brain metastases, unless asymptomatic and are stable.
  • History or active leptomeningeal carcinomatosis.
  • Unresolved toxicities from any prior therapy greater than CTCAE Grade 1 and prior platinum-therapy related Grade 2 neuropathies with the exception of alopecia and haemoglobin ≥ 9.0 g/dL.
  • Active/unstable cardiac diseases currently or within the last 6 months, clinically significant ECG abnormalities, and/or factors/medications that may affect QTc intervals.
  • History of liver cirrhosis of any origin and clinical stage; or history of other serious liver disease or chronic disease with relevant liver involvement.
  • Known serious active infection including, but not limited to, tuberculosis, or HIV, HBV or HCV or gastrointestinal disease.
  • Receipt of live attenuated vaccine (including against COVID-19) within 30 days prior to the first dose of study intervention.
  • Past medical history of ILD, drug-induced ILD, radiation pneumonitis, which required steroid treatment, or any evidence of clinically active ILD.
  • Participants currently receiving medications or herbal supplements known to be strong inducers of cytochrome P450 (CYP)3A4 or strong inhibitors of CYP1A2.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (214)

Research Site

Orlando, Florida, 32804, United States

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Honolulu, Hawaii, 96819, United States

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New Brunswick, New Jersey, 08903, United States

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New York, New York, 10032, United States

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Nashville, Tennessee, 37232, United States

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Buenos Aires, C1125ABD, Argentina

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CABA, C1019ABS, Argentina

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Florida, B1602DQD, Argentina

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La Rioja, F5300COE, Argentina

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Rosario, 2000, Argentina

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Rosario, 2123, Argentina

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San Miguel de Tucumán, 4000, Argentina

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Viedma, R8500ACE, Argentina

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Fremantle, 6160, Australia

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Southport, 4215, Australia

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Waratah NSW, 2298, Australia

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Westmead, 2145, Australia

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Brussels, 1000, Belgium

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Ghent, 9000, Belgium

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Roeselare, 8800, Belgium

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Belo Horizonte, 30110-022, Brazil

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Cachoeiro de Itapemirim, 29308-014, Brazil

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Ijuí, 98700-000, Brazil

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Porto Alegre, 90035-903, Brazil

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Porto Alegre, 90050-170, Brazil

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Salvador, 41253-190, Brazil

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Salvador, 41950-610, Brazil

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São Paulo, 04014-002, Brazil

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São Paulo, 04538-132, Brazil

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São Paulo, 04556-100, Brazil

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Vitória, 29043-260, Brazil

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Toronto, Ontario, M4N 3M5, Canada

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Toronto, Ontario, M5G 2M9, Canada

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Montreal, Quebec, H3T 1E2, Canada

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Montreal, Quebec, H3T 1M5, Canada

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Santiago, 7500713, Chile

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Baoding, 71030, China

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Beijing, 100036, China

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Beijing, 101149, China

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Bengbu, 233004, China

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Changchun, 130012, China

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Changsha, 410011, China

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Changsha, 41003, China

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Chengdu, 610041, China

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Chongqing, 400016, China

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Fuzhou, 350001, China

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Fuzhou, 350011, China

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Hangzhou, 310022, China

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Harbin, 150040, China

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Hefei, 230031, China

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Jinan, 250022, China

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Linyi, 276000, China

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Nanchang, 330006, China

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Qingdao, 266035, China

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Shanghai, 200030, China

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Shenyang, 110001, China

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Shenzhen, 518020, China

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Wuhan, 430022, China

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Wuhan, 430079, China

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Xi'an, 710061, China

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Xi'an, 710100, China

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Xiangfan, 441021, China

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Yichang, 443003, China

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Zhengzhou, 450008, China

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Bobigny, 93000, France

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Brest, 29200, France

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Créteil, 94010, France

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Dijon, 21079, France

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Marseille, 13915, France

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Paris, 75005, France

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Poitiers, 86021, France

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Rennes, 35033, France

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Rouen, 76000, France

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Saint-Herblain, 44800, France

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Saint-Quentin, 02321, France

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Strasbourg, 67091, France

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Suresnes, 92151, France

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Berlin, 14165, Germany

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Chemnitz, 09113, Germany

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Frankfurt A. Main, 60590, Germany

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Gauting, 82131, Germany

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Immenhausen, 34376, Germany

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Löwenstein, 74245, Germany

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München, 81925, Germany

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Münster, 48149, Germany

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Wangen, 88239, Germany

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Athens, 115 27, Greece

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Athens, 11527, Greece

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Chaïdári, 124 62, Greece

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Heraklion, 71110, Greece

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Larissa, 41110, Greece

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Rio, 265 04, Greece

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Thessaloniki, 546 39, Greece

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Thessaloniki, 54622, Greece

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Hong Kong, 999077, Hong Kong

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Kowloon, Hong Kong

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Afula, 18341, Israel

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Ashdod, 7747629, Israel

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Be’er Ya‘aqov, 70300, Israel

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Hadera, 38100, Israel

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Jerusalem, 91031, Israel

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Tel Aviv, 6423906, Israel

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Avellino, 83100, Italy

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Aviano, 33081, Italy

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Catania, 95123, Italy

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Meldola, 47014, Italy

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Milan, 20133, Italy

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Milan, 20141, Italy

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Modena, 41124, Italy

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Monserrato, 09042, Italy

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Naples, 80138, Italy

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Orbassano, 10043, Italy

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Padova, 35128, Italy

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Parma, 43126, Italy

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Perugia, 6124, Italy

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Peschiera del Garda, 37019, Italy

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Roma, 00144, Italy

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Roma, 00152, Italy

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Treviso, 31100, Italy

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Bunkyō City, 113-8603, Japan

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Chūōku, 104-0045, Japan

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Fukuoka, 812-8582, Japan

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Hirosaki-shi, 036-8563, Japan

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Hiroshima, 730-8518, Japan

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Iwakuni-shi, 740-8510, Japan

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Kanazawa, 920-8641, Japan

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Kashiwa, 277-8577, Japan

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Kobe, 650-0017, Japan

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Kobe, 650-0046, Japan

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Kumamoto, 860-8556, Japan

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Kurume-shi, 830-0011, Japan

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Nagasaki, 852-8501, Japan

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Okayama, 700-8558, Japan

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Osaka, 534-0021, Japan

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Osakasayama-shi, 589-8511, Japan

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Sakaishi, 591-8555, Japan

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Sapporo, 003-0804, Japan

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Sapporo, 060-8638, Japan

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Sendai, 980-0873, Japan

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Sunto-gun, 411-8777, Japan

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Utsunomiya, 320-0834, Japan

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Wakayama, 641-8510, Japan

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Yokohama, 241-8515, Japan

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Kota Bharu, 15586, Malaysia

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Kuala Lumpur, 59100, Malaysia

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Petaling Jaya, 47500, Malaysia

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Pulau Pinang, 10990, Malaysia

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Sabak Bernam, 88996, Malaysia

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Bacolod, 6100, Philippines

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Davao City, 8000, Philippines

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Manila, 1000, Philippines

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Quezon City, 1100, Philippines

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Quezon City, 1112, Philippines

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San Juan City, 1502, Philippines

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Lodz, 93-338, Poland

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Olsztyn, 10-357, Poland

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Singapore, 169610, Singapore

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Singapore, 308433, Singapore

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Goyang-si, 10408, South Korea

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Gyeonggi-do, 13620, South Korea

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Jinju, 660-702, South Korea

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Seoul, 06273, South Korea

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Seoul, 06351, South Korea

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Seoul, 08308, South Korea

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Seoul, 138-736, South Korea

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Seoul, 6591, South Korea

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Suwon, 16247, South Korea

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Badajoz, 6006, Spain

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Badalona, 8916, Spain

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Barcelona, 08036, Spain

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Barcelona, 8035, Spain

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Córdoba, 14004, Spain

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Girona, 17007, Spain

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Madrid, 28040, Spain

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Madrid, 28041, Spain

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Majadahonda, 28222, Spain

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Málaga, 29010, Spain

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Pontevedra, 36312, Spain

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Sabadell, 08208, Spain

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Seville, 41009, Spain

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Valencia, 46026, Spain

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Zaragoza, 50009, Spain

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Baden, CH-5405, Switzerland

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Zurich, 8063, Switzerland

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Chiayi City, 62247, Taiwan

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Hsinchu, 300, Taiwan

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Kaohsiung City, 83301, Taiwan

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Liuying, 736, Taiwan

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Taichung, 404, Taiwan

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Taichung, 40705, Taiwan

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Taipei, 100, Taiwan

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Taipei, 11259, Taiwan

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Taipei, 112, Taiwan

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Bangkok, 10210, Thailand

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Bangkok, 10700, Thailand

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Chanthaburi, 22000, Thailand

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Chiang Mai, 50200, Thailand

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Dusit, 10300, Thailand

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Hat Yai, 90110, Thailand

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Muang, 40002, Thailand

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Adana, 1370, Turkey (Türkiye)

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Ankara, 6800, Turkey (Türkiye)

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Edirne, 22030, Turkey (Türkiye)

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Istanbul, 34214, Turkey (Türkiye)

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Istanbul, 34722, Turkey (Türkiye)

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Izmir, 35100, Turkey (Türkiye)

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London, SE1 9RT, United Kingdom

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Manchester, M20 4BX, United Kingdom

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Wolverhampton, WV10 0QP, United Kingdom

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Can Tho, 900000, Vietnam

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Hanoi, 100000, Vietnam

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Hanoi, 10000, Vietnam

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Ho Chi Minh City, 700000, Vietnam

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Ho Chi Minh City, 70000, Vietnam

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Related Links

MeSH Terms

Conditions

CarcinomaNeoplasm Metastasis

Interventions

1-(1-(imidazo(1,2-a)pyridin-6-yl)ethyl)-6-(1-methyl-1H-pyrazol-4-yl)-1H-(1,2,3)triazolo(4,5-b)pyrazineosimertinibPemetrexedCisplatinCarboplatin

Condition Hierarchy (Ancestors)

Neoplasms, Glandular and EpithelialNeoplasms by Histologic TypeNeoplasmsNeoplastic ProcessesPathologic ProcessesPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

GuanineHypoxanthinesPurinonesPurinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic CompoundsGlutamatesAmino Acids, AcidicAmino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, DicarboxylicChlorine CompoundsInorganic ChemicalsNitrogen CompoundsPlatinum CompoundsCoordination ComplexesOrganic Chemicals

Study Officials

  • Shun Lu, Prof,MD,PhD,

    Shanghai Chest Hospital, Shanghai JiaoTong University, #241 Huai Hai Road (west), Shanghai, China.

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Model Details: Parallel Assignment
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

February 15, 2022

First Posted

March 2, 2022

Study Start

August 3, 2022

Primary Completion

July 6, 2026

Study Completion (Estimated)

November 23, 2026

Last Updated

August 6, 2026

Record last verified: 2026-07

Data Sharing

IPD Sharing
Will share

Qualified researchers can request access to anonymized individual patient-level data from AstraZeneca group of companies sponsored clinical trials via the request portal Vivli.org. All request will be evaluated as per the AZ disclosure commitment: https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure. Yes, indicates that AZ are accepting requests for IPD, but this does not mean all requests will be shared.

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
AstraZeneca will meet or exceed data availability as per the commitments made to the EFPIA Pharma Data Sharing Principles. For details of our timelines, please rerefer to our disclosure commitment at https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure.
Access Criteria
When a request has been approved AstraZeneca will provide access to the anonymized individual patient-level data via secure research environment Vivli.org. Signed Data Usage Agreement (non-negotiable contract for data accessors) must be in place before accessing requested information.
More information

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