NCT04541225

Brief Summary

At the time of study termination, NUV-422-02 was a first-in-human, open-label, Phase 1 dose escalation study designed to evaluate the safety and efficacy of NUV-422. The study population comprised adults with recurrent or refractory high-grade gliomas (HGGs), metastatic breast cancer (mBC), with and without brain metastases, and recurrent or refractory metastatic castration-resistant prostate cancer (mCRPC). All patients self-administered NUV-422 orally in 28-day cycles until disease progression, toxicity, withdrawal of consent, or termination of the study.

Trial Health

57
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Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
74

participants targeted

Target at P75+ for phase_1

Timeline
Completed

Started Dec 2020

Geographic Reach
1 country

12 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

August 21, 2020

Completed
19 days until next milestone

First Posted

Study publicly available on registry

September 9, 2020

Completed
3 months until next milestone

Study Start

First participant enrolled

December 8, 2020

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 31, 2022

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

August 31, 2022

Completed
Last Updated

July 14, 2023

Status Verified

July 1, 2023

Enrollment Period

1.7 years

First QC Date

August 21, 2020

Last Update Submit

July 12, 2023

Conditions

Keywords

Phase 1malignant gliomametastatic breast cancermetastatic castration-resistant prostate cancer

Outcome Measures

Primary Outcomes (1)

  • Phase 1 Dose Escalation: Safety and tolerability of NUV-422 to determine the recommended Phase 2 dose (RP2D)

    Incidence of treatment-emergent adverse events (TEAEs), serious adverse events (SAEs), and dose-limiting toxicities (DLTs)

    During the DLT period (28 days)

Study Arms (1)

Phase 1 Dose Escalation

EXPERIMENTAL

NUV-422 will be administered at escalating dose levels until the maximum tolerated dose (MTD) is reached.

Drug: NUV-422

Interventions

NUV-422 is an investigational drug for oral dosing.

Phase 1 Dose Escalation

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • For All Cohorts:
  • Recovered from toxicity to prior anti-cancer therapy
  • Adequate bone marrow and organ function
  • Appropriate candidate for NUV-422 monotherapy
  • Life expectancy of \> 3 months
  • High-Grade Glioma:
  • Histologically confirmed diagnosis of high-grade glioma
  • Evidence of recurrence after treatment (ie, surgery, radiation, or temozolomide) or refractory (or intolerant) to treatment
  • Measurable or non-measurable disease
  • Karnofsky Performance Status (KPS) score ≥ 60
  • HR+HER2- Metastatic Breast Cancer:
  • Men and women who are not suitable for surgical resection or radiotherapy for the purpose of cure
  • Diagnosis of locally advanced or HR+HER2- metastatic breast cancer
  • Evidence of progression as determined by the Investigator per standard criteria
  • Patients must have endocrine-resistant disease
  • +9 more criteria

You may not qualify if:

  • Have received chemotherapy, hormonal therapy (with the exception of ongoing LHRH analogs in male patients and premenopausal women), radiation, or biological anti-cancer therapy within 14 days prior to the first dose of NUV-422
  • Has a history of or current use of bevacizumab (glioma and brain metastases only)
  • Received treatment with an investigational agent for any indication within 14 days for non-myelosuppressive agent or 21 days (or \< 5 half-lives) for myelosuppressive agent prior to the first dose of NUV-422
  • Requires systemic corticosteroid therapy \> 4 mg/day (\> 2 mg/day for Expansion Cohort 2) of dexamethasone or equivalent or increasing doses of systemic corticosteroids during the 7 days prior to enrollment
  • Requires anti-seizure medications that are known to be strong inducers of CYP3A4/5 enzymes (carbamazepine, phenytoin) or has a recent history of uncontrolled or intermittent seizures
  • Females who are pregnant or breast feeding

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (12)

Arizona Oncology Associates

Tucson, Arizona, 85711, United States

Location

Miami Cancer Institute

Miami, Florida, 33176, United States

Location

Dana-Farber Cancer Institute

Boston, Massachusetts, 02215, United States

Location

Memorial Sloan Kettering Cancer Center

New York, New York, 10065, United States

Location

Carolina BioOncology Institute

Huntersville, North Carolina, 28078, United States

Location

Prisma Health Cancer Institute

Greenville, South Carolina, 29605, United States

Location

Texas Oncology P.A. Austin

Austin, Texas, 78705, United States

Location

Texas Oncology-Baylor Charles A. Sammons Cancer Center

Dallas, Texas, 75246, United States

Location

The University of Texas MD Anderson Cancer Center

Houston, Texas, 77030, United States

Location

Texas Oncology

Tyler, Texas, 75702, United States

Location

University of Utah Huntsman Cancer Institute

Salt Lake City, Utah, 84112, United States

Location

Virginia Cancer Specialists

Fairfax, Virginia, 22031, United States

Location

MeSH Terms

Conditions

GliomaBreast NeoplasmsProstatic NeoplasmsProstatic Neoplasms, Castration-ResistantGlioblastoma

Condition Hierarchy (Ancestors)

Neoplasms, NeuroepithelialNeuroectodermal TumorsNeoplasms, Germ Cell and EmbryonalNeoplasms by Histologic TypeNeoplasmsNeoplasms, Glandular and EpithelialNeoplasms, Nerve TissueNeoplasms by SiteBreast DiseasesSkin DiseasesSkin and Connective Tissue DiseasesGenital Neoplasms, MaleUrogenital NeoplasmsGenital Diseases, MaleGenital DiseasesUrogenital DiseasesProstatic DiseasesMale Urogenital DiseasesAstrocytoma

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

August 21, 2020

First Posted

September 9, 2020

Study Start

December 8, 2020

Primary Completion

August 31, 2022

Study Completion

August 31, 2022

Last Updated

July 14, 2023

Record last verified: 2023-07

Locations