NCT04017832

Brief Summary

This study compares 2 medicines for type 2 diabetes: oral semaglutide (a new medicine) and sitagliptin (a medicine doctors can already prescribe). Participants will either get oral semaglutide or sitagliptin - which treatment is decided by chance. Participants will get 2 tablets a day to take first thing in the morning on an empty stomach. Only 1 tablet has study medicine in it. The other tablet is a dummy medicine (placebo). After taking the semaglutide tablet, participants may not eat or drink anything for at least 30 minutes. After the 30 minutes, participants must take the sitagliptin tablet. Then participants can have their first meal of the day and take any other medicines they may need, including their metformin. The study will last for about 7 months (33 weeks). Participants will have 8 clinic visits and 1 phone call with the study doctor. At all 8 of the clinic visits, participants will have blood samples taken.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
1,441

participants targeted

Target at P75+ for phase_3 diabetes-mellitus-type-2

Timeline
Completed

Started Jul 2019

Typical duration for phase_3 diabetes-mellitus-type-2

Geographic Reach
9 countries

93 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

July 11, 2019

Completed
1 day until next milestone

First Posted

Study publicly available on registry

July 12, 2019

Completed
17 days until next milestone

Study Start

First participant enrolled

July 29, 2019

Completed
2.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 27, 2021

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

October 27, 2021

Completed
1.9 years until next milestone

Results Posted

Study results publicly available

September 29, 2023

Completed
Last Updated

October 1, 2024

Status Verified

September 1, 2024

Enrollment Period

2.2 years

First QC Date

July 11, 2019

Results QC Date

October 26, 2022

Last Update Submit

September 27, 2024

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline to Week 26 in Glycated Haemoglobin (HbA1c) (%)

    Change in HbA1c from baseline to week 26 in percentage (%) point of HbA1c is presented. The outcome data was evaluated based on the on-treatment without rescue medication observation period and in-trial observation period. On-treatment without rescue medication observation period: from date of first dose of trial product following randomization and the end date which was the first date of any of the following: the last dose of trial product plus 3 days or initiation of rescue medication. In-trial observation period: the time period where participants were considered to be in the trial, regardless of discontinuation of trial product or initiation of rescue medication.

    From baseline to week 26

Secondary Outcomes (43)

  • Change From Baseline to Week 26 in Fasting Plasma Glucose (FPG)

    From baseline to week 26

  • Change From Baseline to Week 26 in Self-measured Plasma Glucose (SMPG) Profile: Mean 7-point Profile

    From baseline to week 26

  • Change From Baseline to Week 26 in 7 Point SMPG Profile: Mean Postprandial Increment (Over All Meals)

    From baseline to week 26

  • Number of Participants Who Achieved HbA1c <7.0 % (53 mmol/Mol) (American Diabetes Association [ADA] Target) (Yes/no)

    At week 26

  • Number of Participants Who Achieved HbA1c Equal to or Below 6.5 Percent (48 mmol/Mol) (American Association of Clinical Endocrinologists (AACE) Target) (Yes/no)

    At week 26

  • +38 more secondary outcomes

Study Arms (4)

Oral semaglutide 3 mg and placebo (sitagliptin)

EXPERIMENTAL

Oral semaglutide tablets 3 mg and sitagliptin placebo tablets for 26 weeks

Drug: Oral semaglutideDrug: Placebo (sitagliptin)

Oral semaglutide 7 mg and placebo (sitagliptin)

EXPERIMENTAL

Oral semaglutide tablets and sitagliptin placebo tablets. The dose of oral semaglutide will be escalated over 4 weeks, after which the target dose of 7 mg is taken for 22 weeks

Drug: Oral semaglutideDrug: Placebo (sitagliptin)

Oral semaglutide 14 mg and placebo (sitagliptin)

EXPERIMENTAL

Oral semaglutide tablets and sitagliptin placebo tablets. The dose of oral semaglutide will be escalated over 8 weeks, after which the target dose of 14 mg is taken for 18 weeks

Drug: Oral semaglutideDrug: Placebo (sitagliptin)

Sitagliptin 100 mg and placebo (oral semaglutide)

EXPERIMENTAL

Sitagliptin tablets and oral semaglutide placebo tablets for 26 weeks

Drug: SitagliptinDrug: Placebo (oral semaglutide)

Interventions

Oral semaglutide to be taken every morning in a fasting state, to be followed by sitagliptin placebo after 30 minutes. Only then participants can have their first meal of the day and their pre-study metformin tablets

Oral semaglutide 14 mg and placebo (sitagliptin)Oral semaglutide 3 mg and placebo (sitagliptin)Oral semaglutide 7 mg and placebo (sitagliptin)

Sitagliptin to be taken every morning, 30 minutes after taking the oral semaglutide placebo tablet. Then participants can have their first meal of the day and their pre-study metformin tablets

Sitagliptin 100 mg and placebo (oral semaglutide)

Placebo tablet to be taken first thing in the morning

Sitagliptin 100 mg and placebo (oral semaglutide)

Placebo tablet to be taken 30 minutes after oral semaglutide

Oral semaglutide 14 mg and placebo (sitagliptin)Oral semaglutide 3 mg and placebo (sitagliptin)Oral semaglutide 7 mg and placebo (sitagliptin)

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Informed consent obtained before any trial-related activities. Trial-related activities are any procedures that are carried out as part of the trial, including activities to determine suitability for the trial.
  • Male or female, age above or equal to 18 years at the time of signing informed consent.
  • For Algeria only: Male or female, age above or equal to 19 years at the time of signing informed consent.
  • For Taiwan only: Male or female, age above or equal to 20 years at the time of signing informed consent
  • Diagnosed with type 2 diabetes mellitus 60 days or more prior to day of screening.
  • HbA1c between 7.0-10.5% (53-91 mmol/mol) (both inclusive).
  • Stable daily dose of metformin (equal to or above 1500 mg or maximum tolerated dose as documented in the subject medical record) 60 days or more prior to day of screening

You may not qualify if:

  • Female who is pregnant, breast-feeding or intends to become pregnant or is of child-bearing potential and not using a highly effective contraceptive method (adequate contraceptive measure as required by local regulation or practice).
  • Family or personal history of multiple endocrine neoplasia type 2 (MEN 2) or medullary thyroid carcinoma (MTC). Family is defined as a first degree relative.
  • History or presence of pancreatitis (acute or chronic).
  • History of major surgical procedures involving the stomach potentially affecting absorption of trial product (e.g. subtotal and total gastrectomy, sleeve gastrectomy, gastric bypass surgery).
  • Any of the following: myocardial infarction, stroke, hospitalization for unstable angina or transient ischaemic attack within the past 180 days prior to the day of screening and randomisation.
  • Subjects presently classified as being in New York Heart Association (NYHA) Class IV.
  • Planned coronary, carotid or peripheral artery revascularisation known on the day of screening.
  • Renal impairment measured as estimated glomerular filtration rate (eGFR) below 60 mL/min/1.73 m\^2 as per Chronic Kidney Disease Epidemiology Collaboration formula (CKD-EPI).
  • Subjects with alanine aminotransferase (ALT) above 2.5 x upper limit of the normal (ULN).
  • Uncontrolled and potentially unstable diabetic retinopathy or maculopathy. Verified by a pharmacologically pupil-dilated fundus examination performed by an ophthalmologist or another suitably qualified health care provider within the past 90 days prior to screening or in the period between screening and randomisation. Fundus examination without dilation is only allowed if the digital camera used for fundus photography has this feature.
  • Presence or history of malignant neoplasms within the past 5 years prior to the day of screening. Basal and squamous cell skin cancer and any carcinoma in-situ is allowed.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (93)

Maison des diabétiques El Harrach

Algiers, 16000, Algeria

Location

Department of internal medicine hospital (CHU) of BIRTRARIA

Algiers, 16003, Algeria

Location

Núcleo de Pesquisa Clínica do Rio Grande do Sul Ltda.

Porto Alegre, Rio Grande do Sul, 90430-001, Brazil

Location

CPQuali Pesquisa Clínica Ltda

São Paulo, São Paulo, 01228-000, Brazil

Location

CPCLIN - Centro de Pesquisas Clínicas

São Paulo, São Paulo, 01228-200, Brazil

Location

Anhui Provincial Hospital

Hefei, Anhui, 230001, China

Location

The First Affiliated Hospital of Anhui Medical University

Hefei, Anhui, 230061, China

Location

Peking University People's Hospital

Beijing, Beijing Municipality, 100044, China

Location

Peking University Shougang Hospital

Beijing, Beijing Municipality, 100144, China

Location

Beijing Pinggu Hospital

Beijing, Beijing Municipality, 101200, China

Location

Second Affliated Hospital of Chongqing Medical University

Chongqing, Chongqing Municipality, 400010, China

Location

900th Hospital of Joint Logistics Support Force

Fuzhou, Fujian, 350025, China

Location

The Second Affiliated Hospital of Fujian Medical University

Quanzhou, Fujian, 362000, China

Location

Shunde Hospital of Southern Medical University

Foshan, Guangdong, 528399, China

Location

Sun Yat-sen Memorial Hospital, Sun Yat-sen Universtiy

Guangzhou, Guangdong, 510120, China

Location

Guangzhou Panyu Central Hospital

Guangzhou, Guangdong, 511400, China

Location

Huizhou Central People's Hospital

Huizhou, Guangdong, 516001, China

Location

The 2nd Affiliated Hospital of Shantou Uni Medical College

Shantou, Guangdong, 515065, China

Location

Cangzhou People's Hospital

Cangzhou, Hebei, 061000, China

Location

Harrison International Peace Hospital

Hengshui, Hebei, 053000, China

Location

The Second Hospital of Hebei Medical University

Shijiazhuang, Hebei, 050000, China

Location

Huaihe Hospital of Henan University

Kaifeng, Henan, 475000, China

Location

The First Affiliated Hospital of Henan university of Science

Luoyang, Henan, 471003, China

Location

Zhengzhou First People's Hospital

Zhengzhou, Henan, 450004, China

Location

Taihe Hospital

Shiyan, Hubei, 442008, China

Location

Wuhan Puai Hosptial

Wuhan, Hubei, 430034, China

Location

Changsha Central Hospital

Changsha, Hunan, 410018, China

Location

Chenzhou No.1 People's Hospital

Chenzhou, Hunan, 423000, China

Location

The First Affiliated Hospital Of University Of South China

Hengyang, Hunan, 421001, China

Location

Zhuzhou Central Hospital

Zhuzhou, Hunan, 412007, China

Location

Changzhou No.2 People's Hospital, Yanghu Branch

Changzhou, Jiangsu, 213003, China

Location

The First People's Hospital of Changzhou

Changzhou, Jiangsu, 213003, China

Location

The Second Affiliated Hospital of Nanjing Medical University

Nanjing, Jiangsu, 210011, China

Location

Nanjing Jiangning Hospital

Nanjing, Jiangsu, 211106, China

Location

Sir Run Run Hospital Nanjing Medical University

Nanjing, Jiangsu, 211166, China

Location

The Second Affiliated Hospital of Soochow University

Suzhou, Jiangsu, 215004, China

Location

The First Affiliated Hospital of Soochow University

Suzhou, Jiangsu, 215006, China

Location

Wuxi People's Hospital

Wuxi, Jiangsu, 214023, China

Location

The Affiliated Hospital of Xuzhou Medical University

Xuzhou, Jiangsu, 221002, China

Location

The Affiliated Hospital of Jiangsu University

Zhenjiang, Jiangsu, 212001, China

Location

Pingxiang People's Hospital

Pingxiang, Jiangxi, 337055, China

Location

Jilin Province People's Hospital

Changchun, Jilin, 130021, China

Location

China-Japan Union Hospital of Jilin University

Changchun, Jilin, 130033, China

Location

The Second Hospital of Jilin University

Changchun, Jilin, 130041, China

Location

General Hospital of Ningxia Medical University

Yinchuan, Ningxia, 750004, China

Location

Qinghai Provincial People's Hospital

Xining, Qinghai, 810007, China

Location

The second Affiliated Hospital of Xi'an Jiaotong University

Xi'an, Shaanxi, 710004, China

Location

Jinan Central Hospital Affiliated to Shandong University

Jinan, Shandong, 250013, China

Location

The Affiliated Hospital of Qingdao Medical College

Qingdao, Shandong, 266003, China

Location

Weifang People's Hospital

Weifang, Shandong, 261041, China

Location

Shanghai Pudong New Area People's Hospital

Pudong New District, Shanghai Municipality, 201200, China

Location

Shanghai Huashan Hospital, Affiliated to Fudan University

Shanghai, Shanghai Municipality, 200040, China

Location

Tongji Hospital of Tongji university

Shanghai, Shanghai Municipality, 200065, China

Location

Shanghai Tenth People's Hsopital, Tongji University

Shanghai, Shanghai Municipality, 200072, China

Location

Dongfang Hospital Affiliated to Shanghai Tongji University

Shanghai, Shanghai Municipality, 200120, China

Location

The Fifth People's Hospital of Shanghai

Shanghai, Shanghai Municipality, 200240, China

Location

Tongren Hospital Shanghai Jiao Tong Univ. School of Medicine

Shanghai, Shanghai Municipality, 200336, China

Location

General Hospital of Tianjin Medical University

Tianjin, Tianjin Municipality, 300052, China

Location

The Second Hospital of Tianjin Medical University

Tianjin, Tianjin Municipality, 300211, China

Location

First Affiated Hospital of Kunming Medical University

Kunming, Yunnan, 650032, China

Location

The First People's Hospital of Yunnan Province

Kunming, Yunnan, 650032, China

Location

The Second Affiliated Hospital of Kunming Medical University

Kunming, Yunnan, 650101, China

Location

The 2nd Affi Hosp of Zhejiang Univer School of Medicine

Hangzhou, Zhejiang, 310009, China

Location

The Third Xiangya Hospital of Central South University

Changsha, 410013, China

Location

Nemocnice milosrdnych bratri

Brno, 63900, Czechia

Location

DIAMIN

Chrudim, 537 01, Czechia

Location

Interna a diabetologie MUDr. Vodickova

Liberec, 46001, Czechia

Location

CCR Prague

Prague, 130 00, Czechia

Location

MUDr. Michala Pelikanova

Prague, 140 00, Czechia

Location

Prince of Wales Hospital

Shatin, New Territories, Hong Kong

Location

SC Grand Med SRL

Oradea, Bihor County, 410025, Romania

Location

S.C. Endodigest S.R.L.

Oradea, Bihor County, 410151, Romania

Location

SC Centru Medical Dr. Negrisanu SRL

Timișoara, Timiș County, 300456, Romania

Location

SC Nutrilife SRL

Bucharest, 13682, Romania

Location

Clinic of Diabetes Constanta

Constanța, 900591, Romania

Location

Clinical County Emergency Hosp

Oradea, 410169, Romania

Location

Clinical Hospital Centre Dragisa Misovic

Belgrade, 11000, Serbia

Location

Endocrinology, Diabetes and Metabolism Diseases Clinic

Belgrade, 11000, Serbia

Location

Clinical Hospital Centre Zemun

Belgrade, 11080, Serbia

Location

GCT

Arcadia, Gauteng, 0083, South Africa

Location

Dr R Dulabh

Johannesburg, Gauteng, 1812, South Africa

Location

Newtown Clinical Research

Johannesburg, Gauteng, 2001, South Africa

Location

WITS Clinical Research

Johannesburg, Gauteng, 2193, South Africa

Location

Clinresco Centres (Pty) Ltd

Kempton Park, Gauteng, 1619, South Africa

Location

Setshaba Research Centre

Soshanguve, Gauteng, 0152, South Africa

Location

Armansis Medical Centre

Brits, North West, 0250, South Africa

Location

Cape Town Medical Research Centre

Kuilsriver, Western Cape, 7580, South Africa

Location

Paarl Reserch Centre

Paarl, Western Cape, 7646, South Africa

Location

Union Hospital

Alberton, 1449, South Africa

Location

National Taiwan University Hospital

Taipei, 100, Taiwan

Location

Taipei Veterans General Hospital

Taipei, 112, Taiwan

Location

Tri-Service General Hospital

Taipei, 114, Taiwan

Location

Chang Gung Medical Foundation - Linko Branch

Taoyuan, 333, Taiwan

Location

Related Publications (1)

  • Ji L, Agesen RM, Bain SC, Fu F, Gabery S, Geng J, Li Y, Lu Y, Luo B, Pang W, Tao Y; PIONEER 12 investigators. Efficacy and safety of oral semaglutide vs sitagliptin in a predominantly Chinese population with type 2 diabetes uncontrolled with metformin: PIONEER 12, a double-blind, Phase IIIa, randomised trial. Diabetologia. 2024 Sep;67(9):1800-1816. doi: 10.1007/s00125-024-06133-4. Epub 2024 Jul 10.

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

semaglutideSitagliptin Phosphate

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

TriazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPyrazines

Results Point of Contact

Title
Clinical Reporting Anchor and Disclosure (2834)
Organization
Novo Nordisk A/S

Study Officials

  • Clinical Reporting Anchor and Disclosure (1452)

    Novo Nordisk A/S

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Masking Details
Sponsor staff involved in the clinical trial is masked according to company standard procedures
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

July 11, 2019

First Posted

July 12, 2019

Study Start

July 29, 2019

Primary Completion

October 27, 2021

Study Completion

October 27, 2021

Last Updated

October 1, 2024

Results First Posted

September 29, 2023

Record last verified: 2024-09

Data Sharing

IPD Sharing
Will share

According to the Novo Nordisk disclosure commitment on novonordisk-trials.com

Locations