NCT02706847

Brief Summary

The study objective of Period 1 (Day 1 to Week 24) is to compare the safety and efficacy of upadacitinib 30 mg once daily (QD) and 15 mg QD versus placebo for the treatment of signs and symptoms of participants with moderately to severely active rheumatoid arthritis (RA) who are on a stable dose of csDMARDs and had an inadequate response to or intolerance to at least 1 bDMARD. The study objective of Period 2 (Week 24 to Week 260) is to evaluate the long-term safety, tolerability, and efficacy of upadacitinib 15 mg QD and 30 mg QD in participants with RA who completed Period 1.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
499

participants targeted

Target at P50-P75 for phase_3 rheumatoid-arthritis

Timeline
Completed

Started Mar 2016

Longer than P75 for phase_3 rheumatoid-arthritis

Geographic Reach
25 countries

184 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

February 18, 2016

Completed
22 days until next milestone

First Posted

Study publicly available on registry

March 11, 2016

Completed
4 days until next milestone

Study Start

First participant enrolled

March 15, 2016

Completed
1.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 3, 2017

Completed
2.5 years until next milestone

Results Posted

Study results publicly available

October 7, 2019

Completed
2.3 years until next milestone

Study Completion

Last participant's last visit for all outcomes

February 8, 2022

Completed
Last Updated

February 8, 2023

Status Verified

January 1, 2023

Enrollment Period

1.1 years

First QC Date

February 18, 2016

Results QC Date

September 13, 2019

Last Update Submit

January 12, 2023

Conditions

Keywords

Musculoskeletal DiseaseArthritisJoint DiseaseAnti-inflammatory agentsAntirheumatic agentsABT-494upadacitinib

Outcome Measures

Primary Outcomes (2)

  • Percentage of Participants With an American College of Rheumatology 20% (ACR20) Response at Week 12

    The primary endpoint for United States (US)/Food and Drug Administration (FDA) regulatory purposes was ACR 20% response (ACR20) at Week 12. Participants who met the following 3 conditions for improvement from baseline were classified as meeting the ACR20 response criteria: 1. ≥ 20% improvement in 68-tender joint count; 2. ≥ 20% improvement in 66-swollen joint count; and 3. ≥ 20% improvement in at least 3 of the 5 following parameters: * Physician global assessment of disease activity * Patient global assessment of disease activity * Patient assessment of pain * Health Assessment Questionnaire - Disability Index (HAQ-DI) * High-sensitivity C-reactive protein (hsCRP).

    Baseline and Week 12

  • Percentage of Participants Achieving Low Disease Activity (LDA) Based on DAS28(CRP) at Week 12

    The primary endpoint for European Union (EU)/European Medicines Agency (EMA) regulatory purposes was low disease activity, based on a Disease Activity Score 28 (DAS28)-CRP score of ≤ 3.2 at Week 12. The DAS28 is a composite index used to assess rheumatoid arthritis disease activity, calculated based on the tender joint count (out of 28 evaluated joints), swollen joint count (out of 28 evaluated joints), Patient's Global Assessment of Disease Activity (0-100 mm), and hsCRP (in mg/L). Scores on the DAS28 range from 0 to approximately 10, where higher scores indicate more disease activity. A DAS28 score less than or equal to 3.2 indicates low disease activity.

    Week 12

Secondary Outcomes (6)

  • Change From Baseline in in Disease Activity Score 28 (CRP) at Week 12

    Baseline and Week 12

  • Change From Baseline in Health Assessment Questionnaire Disability Index (HAQ-DI) at Week 12

    Baseline and Week 12

  • Change From Baseline in Short-Form 36 (SF-36) Physical Component Score (PCS) at Week 12

    Baseline and Week 12

  • Percentage of Participants With an American College of Rheumatology 50% (ACR50) Response at Week 12

    Baseline and Week 12

  • Percentage of Participants With an American College of Rheumatology 70% (ACR70) Response at Week 12

    Baseline and Week 12

  • +1 more secondary outcomes

Study Arms (4)

Upadacitinib 15 mg

EXPERIMENTAL

Period 1: Participants receive upadacitinib 15 mg once daily for 24 weeks. Period 2: Participants will continue on upadacitinib 15 mg once daily from Week 24 to Week 260.

Drug: Upadacitinib

Upadacitinib 30 mg

EXPERIMENTAL

Period 1: Participants receive upadacitinib 30 mg once daily for 24 weeks. Period 2: Participants continue on upadacitinib 30 mg once daily until implementation of Protocol Amendment 4, then participants begin to receive upadacitinib 15 mg once daily up to Week 260.

Drug: Upadacitinib

Placebo / Upadacitnib 15 mg

PLACEBO COMPARATOR

Period 1: Participants receive placebo once daily for 12 weeks followed by upadacitinib 15 mg once daily for 12 weeks. Period 2: Participants will continue on upadacitinib 15 mg once daily from Week 24 to Week 260.

Drug: PlaceboDrug: Upadacitinib

Placebo / Upadacitnib 30 mg

PLACEBO COMPARATOR

Period 1: Participants receive placebo once daily for 12 weeks followed by upadacitinib 30 mg once daily for 12 weeks. Period 2: Participants continue on upadacitinib 30 mg once daily until implementation of Protocol Amendment 4, then participants begin to receive upadacitinib 15 mg once daily up to Week 260.

Drug: PlaceboDrug: Upadacitinib

Interventions

Tablet; Oral

Placebo / Upadacitnib 15 mgPlacebo / Upadacitnib 30 mg

Tablet; Oral

Also known as: ABT-494, RINVOQ®
Placebo / Upadacitnib 15 mgPlacebo / Upadacitnib 30 mgUpadacitinib 15 mgUpadacitinib 30 mg

Eligibility Criteria

Age18 Years - 99 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Diagnosis of rheumatoid arthritis (RA) for≥ 3 months.
  • Treated for ≥ 3 months with ≥ 1 bDMARD therapy, but continue to exhibit active RA or had to discontinue due to intolerability or toxicity, irrespective of treatment duration prior to the first dose of study drug.
  • Participant has been receiving csDMARD therapy ≥ 3 months and on a stable dose for ≥ 4 weeks prior to the first dose of study drug. The following csDMARDs are allowed: methotrexate (MTX), sulfasalazine, hydroxychloroquine, chloroquine, and leflunomide. A combination of up to two background csDMARDs is allowed except the combination of MTX and leflunomide.
  • Meets both of the following criteria:
  • ≥ 6 swollen joints (based on 66 joint counts) and ≥ 6 tender joints (based on 68 joint counts) at Screening and Baseline Visits.
  • hsCRP ≥ 3mg/L at Screening Visit.

You may not qualify if:

  • Prior exposure to any Janus kinase (JAK) inhibitor (including but not limited to tofacitinib, baricitinib, and filgotinib).
  • History of any arthritis with onset prior to age 17 years or current diagnosis of inflammatory joint disease other than RA (including but not limited to gout, systemic lupus erythematosus, psoriatic arthritis, axial spondyloarthritis including ankylosing spondylitis and non-radiographic axial spondyloarthritis, reactive arthritis, overlap connective tissue diseases, scleroderma, polymyositis, dermatomyositis, fibromyalgia \[currently with active symptoms\]). Current diagnosis of secondary Sjogren's Syndrome is permitted.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (188)

Rheum Assoc of North Alabama /ID# 145959

Huntsville, Alabama, 35801, United States

Location

AZ Arthritis and Rheum Assoc /ID# 148593

Mesa, Arizona, 85202, United States

Location

AZ Arthritis and Rheum Researc /ID# 142816

Phoenix, Arizona, 85032-9306, United States

Location

AZ Arthritis and Rheum Researc /ID# 146075

Phoenix, Arizona, 85032-9306, United States

Location

AZ Arthritis and Rheum Researc /ID# 148592

Phoenix, Arizona, 85032-9306, United States

Location

Arizona Research Center, Inc. /ID# 142741

Phoenix, Arizona, 85053-4061, United States

Location

AZ Arthr & Rheum Research /ID# 155256

Prescott, Arizona, 86305, United States

Location

AZ Arthritis & Rheum Research /ID# 156090

Sun City, Arizona, 85351, United States

Location

NEA Baptist Clinic /ID# 149280

Jonesboro, Arkansas, 72401, United States

Location

Covina Arthritis Clinic /ID# 142794

Covina, California, 91722, United States

Location

Rheumatology Ctr of San Diego /ID# 153576

Escondido, California, 92025, United States

Location

St. Joseph Heritage Healthcare /ID# 149273

Fullerton, California, 92835, United States

Location

TriWest Research Associates- La Mesa /ID# 142792

La Mesa, California, 91942, United States

Location

Arthritis & Osteo Medical Ctr /ID# 142770

La Palma, California, 90623-1728, United States

Location

Valerius Med Grp & Res Ctr /ID# 142799

Los Alamitos, California, 90720-5402, United States

Location

Pacific Arthritis Ctr Med Grp /ID# 142783

Los Angeles, California, 90045, United States

Location

University of California, Los Angeles /ID# 148348

Los Angeles, California, 90095, United States

Location

Desert Medical Advances /ID# 142765

Palm Desert, California, 92260, United States

Location

Stanford University School of Med /ID# 142761

Stanford, California, 94305-2200, United States

Location

Robin K. Dore MD, Inc /ID# 150908

Tustin, California, 92780, United States

Location

Inland Rheum Clin Trials Inc. /ID# 142787

Upland, California, 91786, United States

Location

Medvin Clinical Research /ID# 142814

Whittier, California, 90606, United States

Location

Arthritis Assoc & Osteo Ctr /ID# 142809

Colorado Springs, Colorado, 80920, United States

Location

Denver Arthritis Clinic /ID# 142771

Denver, Colorado, 80230, United States

Location

New England Research Associates, LLC /ID# 142763

Bridgeport, Connecticut, 06606-1827, United States

Location

Delaware Arthritis /ID# 142803

Lewes, Delaware, 19958, United States

Location

Lakes Research, LLC /ID# 142755

Miami, Florida, 33014, United States

Location

Medallion Clinical Research Institute, LLC /ID# 142740

Naples, Florida, 34102, United States

Location

Omega Research Consultants /ID# 142780

Orlando, Florida, 32810, United States

Location

Millennium Research /ID# 142782

Ormond Beach, Florida, 32174, United States

Location

Arthritis Research of Florida /ID# 142811

Palm Harbor, Florida, 34684-2672, United States

Location

Arthritis Center, Inc. /ID# 142822

Palm Harbor, Florida, 34684, United States

Location

Advent Clinical Research /ID# 142817

Pinellas Park, Florida, 33781, United States

Location

St. Anthony Comprehsve Res Ins /ID# 148349

St. Petersburg, Florida, 33705, United States

Location

University of South Florida /ID# 145611

Tampa, Florida, 33612, United States

Location

BayCare Medical Group, Inc. /ID# 142747

Tampa, Florida, 33614-7101, United States

Location

Lovelace Scientific Resources /ID# 142779

Venice, Florida, 34292, United States

Location

Jefrey D. Lieberman, MD, P.C. /ID# 151713

Decatur, Georgia, 30033, United States

Location

Marietta Rheumatology Assoc /ID# 151347

Marietta, Georgia, 30060, United States

Location

St. Luke's Clinic - Rheumatolo /ID# 150923

Boise, Idaho, 83702, United States

Location

Institute of Arthritis Res /ID# 142810

Idaho Falls, Idaho, 83404, United States

Location

Advanced Clinical Research /ID# 153089

Meridian, Idaho, 83642, United States

Location

Great Lakes Clinical Trials /ID# 148341

Chicago, Illinois, 60640, United States

Location

Clinical Investigation Special /ID# 149270

Skokie, Illinois, 60076, United States

Location

Springfield Clinic /ID# 142818

Springfield, Illinois, 62702-3749, United States

Location

Deerbrook Medical Associates /ID# 151712

Vernon Hills, Illinois, 60061, United States

Location

The Arthritis & Diabetes Clinic, Inc. /ID# 142793

Monroe, Louisiana, 71203, United States

Location

Vanguard Medical Research, LLC /ID# 153123

Shreveport, Louisiana, 71011, United States

Location

MMP Women's Health /ID# 145612

Portland, Maine, 04102, United States

Location

The Center for Rheumatology & /ID# 142742

Wheaton, Maryland, 20902, United States

Location

Mansfield Health Center /ID# 147628

Mansfield, Massachusetts, 02048, United States

Location

Clinical Pharmacology Study Gr /ID# 142744

Worcester, Massachusetts, 01605, United States

Location

June DO, PC /ID# 142756

Lansing, Michigan, 48910, United States

Location

North Mississippi Med Clinics /ID# 142781

Tupelo, Mississippi, 38801, United States

Location

Clayton Medical Associates dba Saint Louis Rheumatology /ID# 142745

St Louis, Missouri, 63119-3845, United States

Location

Barbara Caciolo, MD /ID# 142749

St Louis, Missouri, 63139-2338, United States

Location

Westroads Clinical Research /ID# 142802

Omaha, Nebraska, 68114, United States

Location

Dartmouth-Hitchcock Medical Center /ID# 145958

Lebanon, New Hampshire, 03756, United States

Location

Atlantic Coast Research /ID# 148347

Toms River, New Jersey, 08755, United States

Location

Ocean Rheumatology, PA /ID# 142785

Toms River, New Jersey, 08755, United States

Location

The Center for Rheumatology /ID# 142784

Albany, New York, 12206, United States

Location

North Shore University Hospital /ID# 142772

New Hyde Park, New York, 11040, United States

Location

Buffalo Rheumatology /ID# 142766

Orchard Park, New York, 14127, United States

Location

Joint & Muscle Research Instit /ID# 142797

Charlotte, North Carolina, 28204, United States

Location

DJL Clinical Research, PLLC /ID# 142769

Charlotte, North Carolina, 28210-8508, United States

Location

Cape Fear Arthritis Care /ID# 148344

Leland, North Carolina, 28451, United States

Location

Coastal Carolina Health Care /ID# 148351

New Bern, North Carolina, 28562, United States

Location

Shanahan Rheuma & Immuno /ID# 142812

Raleigh, North Carolina, 27617, United States

Location

Trinity Health Med Arts Clinic /ID# 142754

Minot, North Dakota, 58701, United States

Location

Cincinnati Rheumatic Disease Study Group, Inc. /ID# 142791

Cincinnati, Ohio, 45242-4468, United States

Location

STAT Research, Inc. /ID# 142821

Vandalia, Ohio, 45377-9464, United States

Location

Health Research Oklahoma /ID# 142751

Oklahoma City, Oklahoma, 73103-2400, United States

Location

Healthcare Research Consultant /ID# 142815

Tulsa, Oklahoma, 74135, United States

Location

East Penn Rheumatology Assoc /ID# 142790

Bethlehem, Pennsylvania, 18015, United States

Location

Clinical Research Ctr Reading /ID# 151714

Wyomissing, Pennsylvania, 19610, United States

Location

Columbia Arthritis Center /ID# 153728

Columbia, South Carolina, 29204, United States

Location

West Tennessee Research Inst /ID# 142739

Jackson, Tennessee, 38305, United States

Location

Arthritis Associates, PLLC /ID# 142774

Kingsport, Tennessee, 37660, United States

Location

Arthritis Associates, PLLC /ID# 155462

Kingsport, Tennessee, 37660, United States

Location

Dr. Ramesh Gupta /ID# 142767

Memphis, Tennessee, 38119, United States

Location

Tekton Research, Inc. /ID# 142805

Austin, Texas, 78745, United States

Location

Diagnostic Group Integrated He /ID# 148340

Beaumont, Texas, 77701, United States

Location

Arth and Osteo Clin Brazo Valley /ID# 148343

College Station, Texas, 77845, United States

Location

Arthritis Care and Diagnostic /ID# 151344

Dallas, Texas, 75231, United States

Location

Metroplex Clinical Research /ID# 142758

Dallas, Texas, 75231, United States

Location

Rheumatic Disease Clin Res Ctr /ID# 150914

Houston, Texas, 77004, United States

Location

Baylor College of Medicine /ID# 142753

Houston, Texas, 77030-3411, United States

Location

Rheumatology Clinic of Houston /ID# 150915

Houston, Texas, 77065, United States

Location

Houston Institute for Clin Res /ID# 142768

Houston, Texas, 77074, United States

Location

Pioneer Research Solutions, Inc. /ID# 151346

Houston, Texas, 77098-5294, United States

Location

Arthritis & Osteoporosis Assoc /ID# 147567

Lubbock, Texas, 79424, United States

Location

P&I Clinical Research /ID# 151345

Lufkin, Texas, 75904-3132, United States

Location

SW Rheumatology Res. LLC /ID# 142813

Mesquite, Texas, 75150, United States

Location

Trinity Universal Research Association /ID# 149278

Plano, Texas, 75024-5283, United States

Location

Arthritis & Osteo Ctr of S. TX /ID# 142773

San Antonio, Texas, 78232, United States

Location

Arthritis Clinic of Central TX /ID# 148346

San Marcos, Texas, 78666, United States

Location

DM Clinical Research /ID# 151007

Tomball, Texas, 77375, United States

Location

Arthritis & Osteoporosis Clinic /ID# 142760

Waco, Texas, 76710, United States

Location

Western Washington Arthritis C /ID# 142776

Bothell, Washington, 98021, United States

Location

Arthritis Northwest, PLLC /ID# 150924

Spokane, Washington, 99204, United States

Location

The Vancouver Clinic, INC. PS /ID# 147946

Vancouver, Washington, 98664, United States

Location

West Virginia Research Inst /ID# 153087

South Charleston, West Virginia, 25309, United States

Location

Aurora Rheumatology and Immunotherapy Center /ID# 142820

Franklin, Wisconsin, 53132, United States

Location

The Queen Elizabeth Hospital /ID# 142419

Woodville, South Australia, 5011, Australia

Location

Emeritus Research /ID# 142416

Camberwell, Victoria, 3124, Australia

Location

Medizinische Universität Wien /ID# 142424

Vienna, Vienna, 1090, Austria

Location

Universitaetsklinik fuer Inner /ID# 142423

Graz, 8036, Austria

Location

Rheuma Zentrum Favoriten GmbH /ID# 142421

Vienna, 1100, Austria

Location

Rheuma-Zentrum Wien-Oberlaa /ID# 142425

Vienna, 1100, Austria

Location

Wilhelminenspital der Stadt Wien /ID# 142422

Vienna, 1160, Austria

Location

Cliniques Universitaires Saint Luc /ID# 142426

Woluwe-Saint-Lambert, Brussels Capital, 1200, Belgium

Location

Rhumaconsult SPRL /ID# 151378

Charleroi, Hainaut, 6000, Belgium

Location

UZ Gent /ID# 142429

Ghent, Oost-Vlaanderen, 9000, Belgium

Location

ReumaClinic Genk /ID# 142431

Genk, 3600, Belgium

Location

AZ Damiaan /ID# 142427

Ostend, 8400, Belgium

Location

Ciads /Id# 142526

Winnipeg, Manitoba, R3N 0K6, Canada

Location

Revmatologie MUDr. Klara Sirova /ID# 142536

Ostrava, 702 00, Czechia

Location

Medical Plus, s.r.o. /ID# 148345

Uherské Hradište, 686 01, Czechia

Location

MediTrials /ID# 151777

Tartu, Tartu, 50406, Estonia

Location

East Tallinn Central Hospital /ID# 142543

Tallinn, 10138, Estonia

Location

Kiljava Medical Research /ID# 142546

Hyvinkää, 05800, Finland

Location

Paijat-Hame Central Hospital /ID# 149185

Lahti, 15850, Finland

Location

CHR Orleans - Hopital de la Source /ID# 142557

Orléans, Centre-Val de Loire, 45067, France

Location

Hopital Universitaire Purpan /ID# 144697

Toulouse, Haute-Garonne, 31059, France

Location

Hopital Saint Eloi /ID# 142552

Montpellier, Herault, 34295, France

Location

Centre Hospitalier Le Mans /ID# 145956

Le Mans, Sarthe, 72037, France

Location

CHU Bordeaux-Hopital Pellegrin /ID# 144700

Bordeaux, 33076, France

Location

Centre Hospitalier Jean Rougie /ID# 142556

Cahors, 46005, France

Location

Hopital Edouard Herriot /ID# 144698

Lyon, 69437, France

Location

Uniklinik Koln /ID# 142563

Cologne, North Rhine-Westphalia, 50937, Germany

Location

Rheumazentrum Ruhrgebiet /ID# 145600

Herne, North Rhine-Westphalia, 44649, Germany

Location

Charité Universitätsmedizin Campus Mitte /ID# 142559

Berlin, 10117, Germany

Location

Rheumaforschungszentrum II /ID# 142560

Hamburg, 20095, Germany

Location

Schoen Klinikum Hamburg Eilbek /ID# 142566

Hamburg, 22081, Germany

Location

Asklepios Klinik Altona /ID# 142561

Hamburg, 22763, Germany

Location

LMU Klinikum der Universität München /ID# 142564

Munich, 80337, Germany

Location

MVZ Planegg /ID# 142565

Planegg, 82152, Germany

Location

Knappschaftsklinikum Saar /ID# 142562

Püttlingen, 66346, Germany

Location

General Hospital of Athens Laiko /ID# 142579

Athens, Attica, 115 27, Greece

Location

Vital Medical Center Orvosi es /ID# 142586

Veszprém, Veszprém megye, 8200, Hungary

Location

Revita Reumatologiai Rendelo /ID# 142590

Budapest, 1027, Hungary

Location

Debreceni Egyetem Kenezy Gyula Egyetemi Korhaz /ID# 142587

Debrecen, 4031, Hungary

Location

Bekes Megyei Pandy Kalman Korh /ID# 142588

Gyula, 5700, Hungary

Location

St Vincent's University Hosp /ID# 142593

Dublin, D04 T6F4, Ireland

Location

Tel Aviv Sourasky Medical Ctr /ID# 142597

Tel Aviv, Tel Aviv, 6423906, Israel

Location

Bnai Zion Medical Center /ID# 151945

Haifa, 3339419, Israel

Location

The Lady Davis Carmel MC /ID# 142599

Haifa, 3436212, Israel

Location

LTD M+M Centers /ID# 142624

Ādaži, 2164, Latvia

Location

P. Stradins Clinical Univ Hosp /ID# 142623

Riga, LV-1002, Latvia

Location

Arthritis Clinic Ltd /ID# 153560

Riga, LV-1050, Latvia

Location

Timaru Medical Specialists Ltd /ID# 142657

Timaru, 7910, New Zealand

Location

Pratia MCM Krakow /ID# 142664

Krakow, Lesser Poland Voivodeship, 30-510, Poland

Location

WroMedica I. Bielicka, A. Strzalkowska s.c. /ID# 142665

Wroclaw, Lower Silesian Voivodeship, 51-685, Poland

Location

Centrum Medyczne Pratia Warszawa /ID# 142667

Warsaw, Masovian Voivodeship, 01-869, Poland

Location

Centrum Medyczne AMED Warszawa Targowek /ID# 142663

Warsaw, Masovian Voivodeship, 03-291, Poland

Location

Centrum Medyczne Pratia Gdynia /ID# 142666

Gdynia, Pomeranian Voivodeship, 81-338, Poland

Location

Centro Hospitalar De Vila Nova /ID# 142670

Vila Nova de Gaia, Porto District, 4434-502, Portugal

Location

Centro Hospitalar Lisboa Norte, EPE /ID# 142668

Lisbon, 1649-035, Portugal

Location

GCM Medical Group /ID# 142671

San Juan, 00909, Puerto Rico

Location

Family Outpatient clinic#4,LLC /ID# 150910

Korolev, Moscow, 141060, Russia

Location

ARTROMAC n.o. /ID# 142692

Košice, 040 11, Slovakia

Location

Nemocnica Kosice Saca, a.s. /ID# 142693

Košice, 040 15, Slovakia

Location

Narodny ustav reumatickych chorob Piestany /ID# 142691

Pieštany, 921 12, Slovakia

Location

Hanyang University Seoul Hospi /ID# 150883

Seoul, Seongdong-gu, 04763, South Korea

Location

Inha University Hospital /ID# 150881

Incheon, 22332, South Korea

Location

Seoul National University Hospital /ID# 142622

Seoul, 03080, South Korea

Location

H. Un. Marques de Valdecilla /ID# 142706

Santander, Cantabria, 39008, Spain

Location

Hospital Regional de Malaga /ID# 142707

Málaga, Malaga, 29009, Spain

Location

Comple Hosp Univ de A Coruna /ID# 142708

A Coruña, 15006, Spain

Location

Hospital Clin Univ San Carlos /ID# 142711

Madrid, 28040, Spain

Location

Clinica Gaias /ID# 142709

Santiago de Compostela, 15702, Spain

Location

Hospital Universitario La Fe /ID# 142716

Valencia, 46026, Spain

Location

Sahlgrenska University Hosp /ID# 142720

Gothenburg, 413 45, Sweden

Location

Capio Movement Halmstad /ID# 148236

Halmstad, 302 33, Sweden

Location

Orebro Universitetssjukhuset /ID# 142718

Örebro, 70185, Sweden

Location

Vastmanlands Sjukhus /ID# 142721

Västerås, 72189, Sweden

Location

Universitaetsspital Basel /ID# 145610

Basel, 4031, Switzerland

Location

HFR Fribourg - Hopital Canton /ID# 142723

Fribourg, 1708, Switzerland

Location

Hacettepe University Medical Faculty /ID# 142729

Ankara, 06100, Turkey (Türkiye)

Location

Ankara Ataturk Training & Res /ID# 142727

Ankara, 06800, Turkey (Türkiye)

Location

Ondokuz mayis University Facul /ID# 142728

Samsun, 55139, Turkey (Türkiye)

Location

Whipps Cross Univ Hospital /ID# 145957

London, London, City of, E11 1NR, United Kingdom

Location

The Royal Free Hospital /ID# 142733

London, London, City of, NW3 2QG, United Kingdom

Location

Mid Essex Hospitals NHS Trust /ID# 148992

Chelmsford, CM1 7ET, United Kingdom

Location

Western General Hospital /ID# 142732

Edinburgh, EH4 2XU, United Kingdom

Location

West Suffolk Hospital /ID# 148993

Ipswich, IP33 2QZ, United Kingdom

Location

Arrowe Park Hospital /ID# 148991

Metropolitan Borough of Wirral, CH49 5PE, United Kingdom

Location

Queen Alexandra Hospital /ID# 142735

Portsmouth, PO6 3LY, United Kingdom

Location

Related Publications (14)

  • Genovese MC, Fleischmann R, Combe B, Hall S, Rubbert-Roth A, Zhang Y, Zhou Y, Mohamed MF, Meerwein S, Pangan AL. Safety and efficacy of upadacitinib in patients with active rheumatoid arthritis refractory to biologic disease-modifying anti-rheumatic drugs (SELECT-BEYOND): a double-blind, randomised controlled phase 3 trial. Lancet. 2018 Jun 23;391(10139):2513-2524. doi: 10.1016/S0140-6736(18)31116-4. Epub 2018 Jun 18.

    PMID: 29908670BACKGROUND
  • Burmester GR, Deodhar A, Irvine AD, Panaccione R, Winthrop KL, Vleugels RA, Levy G, Suravaram S, Palac H, Wegrzyn L, Ford S, Meerwein S, Guttman-Yassky E. Safety Profile of Upadacitinib: Descriptive Analysis in Over 27,000 Patient-Years Across Rheumatoid Arthritis, Psoriatic Arthritis, Axial Spondyloarthritis, Atopic Dermatitis, and Inflammatory Bowel Disease. Adv Ther. 2025 Oct;42(10):5215-5237. doi: 10.1007/s12325-025-03328-y. Epub 2025 Aug 28.

  • van Vollenhoven RF, Hall S, Wells AF, Meerwein S, Song Y, Tanjinatus O, Fleischmann R. Long-term sustainability of response to upadacitinib among patients with active rheumatoid arthritis refractory to biological treatments: results up to 5 years from SELECT-BEYOND. RMD Open. 2024 Jul 24;10(3):e004037. doi: 10.1136/rmdopen-2023-004037.

  • Rubbert-Roth A, Kakehasi AM, Takeuchi T, Schmalzing M, Palac H, Coombs D, Liu J, Anyanwu SI, Lippe R, Curtis JR. Malignancy in the Upadacitinib Clinical Trials for Rheumatoid Arthritis, Psoriatic Arthritis, Ankylosing Spondylitis, and Non-radiographic Axial Spondyloarthritis. Rheumatol Ther. 2024 Feb;11(1):97-112. doi: 10.1007/s40744-023-00621-6. Epub 2023 Nov 20.

  • Charles-Schoeman C, Choy E, McInnes IB, Mysler E, Nash P, Yamaoka K, Lippe R, Khan N, Shmagel AK, Palac H, Suboticki J, Curtis JR. MACE and VTE across upadacitinib clinical trial programmes in rheumatoid arthritis, psoriatic arthritis and ankylosing spondylitis. RMD Open. 2023 Nov;9(4):e003392. doi: 10.1136/rmdopen-2023-003392.

  • Fleischmann R, Curtis JR, Charles-Schoeman C, Mysler E, Yamaoka K, Richez C, Palac H, Dilley D, Liu J, Strengholt S, Burmester G. Safety profile of upadacitinib in patients at risk of cardiovascular disease: integrated post hoc analysis of the SELECT phase III rheumatoid arthritis clinical programme. Ann Rheum Dis. 2023 Sep;82(9):1130-1141. doi: 10.1136/ard-2023-223916. Epub 2023 Jun 12.

  • Conaghan PG, Pavelka K, Hsieh SC, Bonnington TL, Kent TC, Marchbank K, Edwards CJ. Evaluating the efficacy of upadacitinib in patients with moderate rheumatoid arthritis: a post-hoc analysis of the SELECT phase 3 trials. Rheumatol Adv Pract. 2023 Feb 8;7(1):rkad017. doi: 10.1093/rap/rkad017. eCollection 2023.

  • Burmester GR, Cohen SB, Winthrop KL, Nash P, Irvine AD, Deodhar A, Mysler E, Tanaka Y, Liu J, Lacerda AP, Palac H, Shaw T, Mease PJ, Guttman-Yassky E. Safety profile of upadacitinib over 15 000 patient-years across rheumatoid arthritis, psoriatic arthritis, ankylosing spondylitis and atopic dermatitis. RMD Open. 2023 Feb;9(1):e002735. doi: 10.1136/rmdopen-2022-002735.

  • Kakehasi AM, Radominski SC, Baravalle MD, Palazuelos FCI, Garcia-Garcia C, Arruda MS, Curi M, Liu J, Qiao M, Velez-Sanchez P, Vargas JI. Safety of upadacitinib in Latin American patients with rheumatoid arthritis: an integrated safety analysis of the SELECT phase 3 clinical program. Clin Rheumatol. 2023 May;42(5):1249-1258. doi: 10.1007/s10067-023-06513-y. Epub 2023 Jan 30.

  • Bergman M, Buch MH, Tanaka Y, Citera G, Bahlas S, Wong E, Song Y, Zueger P, Ali M, Strand V. Routine Assessment of Patient Index Data 3 (RAPID3) in Patients with Rheumatoid Arthritis Treated with Long-Term Upadacitinib Therapy in Five Randomized Controlled Trials. Rheumatol Ther. 2022 Dec;9(6):1517-1529. doi: 10.1007/s40744-022-00483-4. Epub 2022 Sep 20.

  • Yamaoka K, Tanaka Y, Kameda H, Khan N, Sasaki N, Harigai M, Song Y, Zhang Y, Takeuchi T. The Safety Profile of Upadacitinib in Patients with Rheumatoid Arthritis in Japan. Drug Saf. 2021 Jun;44(6):711-722. doi: 10.1007/s40264-021-01067-x. Epub 2021 May 27.

  • Cohen SB, van Vollenhoven RF, Winthrop KL, Zerbini CAF, Tanaka Y, Bessette L, Zhang Y, Khan N, Hendrickson B, Enejosa JV, Burmester GR. Safety profile of upadacitinib in rheumatoid arthritis: integrated analysis from the SELECT phase III clinical programme. Ann Rheum Dis. 2021 Mar;80(3):304-311. doi: 10.1136/annrheumdis-2020-218510. Epub 2020 Oct 28.

  • Strand V, Schiff M, Tundia N, Friedman A, Meerwein S, Pangan A, Ganguli A, Fuldeore M, Song Y, Pope J. Effects of upadacitinib on patient-reported outcomes: results from SELECT-BEYOND, a phase 3 randomized trial in patients with rheumatoid arthritis and inadequate responses to biologic disease-modifying antirheumatic drugs. Arthritis Res Ther. 2019 Dec 2;21(1):263. doi: 10.1186/s13075-019-2059-8.

  • Nader A, Mohamed MF, Winzenborg I, Doelger E, Noertersheuser P, Pangan AL, Othman AA. Exposure-Response Analyses of Upadacitinib Efficacy and Safety in Phase II and III Studies to Support Benefit-Risk Assessment in Rheumatoid Arthritis. Clin Pharmacol Ther. 2020 Apr;107(4):994-1003. doi: 10.1002/cpt.1671. Epub 2019 Nov 30.

Related Links

MeSH Terms

Conditions

Arthritis, RheumatoidMusculoskeletal DiseasesArthritisJoint Diseases

Interventions

upadacitinib

Condition Hierarchy (Ancestors)

Rheumatic DiseasesConnective Tissue DiseasesSkin and Connective Tissue DiseasesAutoimmune DiseasesImmune System Diseases

Results Point of Contact

Title
Global Medical Services
Organization
AbbVie

Study Officials

  • AbbVie Inc.

    AbbVie

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

February 18, 2016

First Posted

March 11, 2016

Study Start

March 15, 2016

Primary Completion

April 3, 2017

Study Completion

February 8, 2022

Last Updated

February 8, 2023

Results First Posted

October 7, 2019

Record last verified: 2023-01

Data Sharing

IPD Sharing
Will share

AbbVie is committed to responsible data sharing regarding the clinical trials we sponsor. This includes access to anonymized, individual and trial-level data (analysis data sets), as well as other information (e.g., protocols and clinical study reports), as long as the trials are not part of an ongoing or planned regulatory submission. This includes requests for clinical trial data for unlicensed products and indications.

Shared Documents
STUDY PROTOCOL, SAP, CSR, ANALYTIC CODE
Time Frame
For details on when studies are available for sharing, please refer to the link below.
Access Criteria
Access to this clinical trial data can be requested by any qualified researchers who engage in rigorous, independent scientific research, and will be provided following review and approval of a research proposal and Statistical Analysis Plan (SAP) and execution of a Data Sharing Agreement (DSA). For more information on the process, or to submit a request, visit the following link.
More information

Locations