NCT01597908

Brief Summary

This was a two-arm, open-label, randomized, Phase III study comparing dabrafenib (GSK2118436) and trametinib (GSK1120212) combination therapy with vemurafenib.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
704

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Jun 2012

Longer than P75 for phase_3

Geographic Reach
27 countries

196 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

May 10, 2012

Completed
4 days until next milestone

First Posted

Study publicly available on registry

May 14, 2012

Completed
21 days until next milestone

Study Start

First participant enrolled

June 4, 2012

Completed
1.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 17, 2014

Completed
8 months until next milestone

Results Posted

Study results publicly available

December 4, 2014

Completed
4.4 years until next milestone

Study Completion

Last participant's last visit for all outcomes

April 25, 2019

Completed
Last Updated

February 24, 2021

Status Verified

February 1, 2021

Enrollment Period

1.9 years

First QC Date

May 10, 2012

Results QC Date

December 1, 2014

Last Update Submit

February 8, 2021

Conditions

Keywords

BRAF inhibitorMetastatic MelanomaCancerMEK inhibitor

Outcome Measures

Primary Outcomes (1)

  • Overall Survival (OS)

    Overall Survival (OS) was defined as the interval of time between the date of randomization and the date of death due to any cause. For patients who did not die, OS was censored at the date of last contact.

    From the date of randomization until date of death due to any cause (up to approximately 6 years)

Secondary Outcomes (3)

  • Progression-Free Survival (PFS), as Assessed by the Investigator

    From randomization until the earliest date of disease progression (PD) or death due to any cause (up to approximately 6 years)

  • Overall Response Rate (ORR) During Randomized Phase, as Assessed by the Investigator

    From randomization until the first documented complete response or partial response (up to approximately 6 years)

  • Duration of Response (DOR), as Assessed by the Investigator

    From the time of the first documented response (CR or PR) until disease progression (up to approximately 6 years)

Study Arms (2)

Dabrafenib plus Trametinib

EXPERIMENTAL

BRAF inhibitor plus MEK inhibitor

Drug: DabrafenibDrug: Trametinib

Vemurafenib

ACTIVE COMPARATOR

BRAF inhibitor

Drug: Vemurafenib

Interventions

Dabrafenib 150 mg twice daily orally

Also known as: GSK2118436
Dabrafenib plus Trametinib

Vemurafenib 960 mg twice daily orally

Also known as: Monotherapy
Vemurafenib

Trametinib 2 mg once daily orally

Also known as: GSK1120212
Dabrafenib plus Trametinib

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • \>= 18 years of age
  • Stage IIIc or Stage IV BRAF V600E/K cutaneous melanoma
  • Measurable disease according to RECIST 1.1
  • Women of childbearing potential with negative serum pregnancy test prior to randomisation
  • Eastern Cooperative Oncology Group (ECOG) Performance Status of 0 or 1
  • Adequate baseline organ function

You may not qualify if:

  • Any prior use of a BRAF or MEK inhibitor
  • Prior systemic anti-cancer treatment in the advanced or metastatic setting; prior systemic treatment in the adjuvant setting is allowed
  • History of another malignancy (except subjects who have been disease free for 3 years or with a history of completely resected non-melanoma skin cancer)
  • Known HIV, HBV, HCV infection (except chronic or cleared HBV and HCV infection which will be allowed)
  • Brain metastases (except if all known lesions were previously treated with surgery or stereotactic radiosurgery and lesions, if still present, are confirmed stable for \>= 12 weeks prior to randomisation or if no longer present are confirmed no evidence of disease for \>= 12 weeks, and are asymptomatic with no corticosteroid requirements for \>= 4 weeks prior to randomisation, and no enzyme inducing anticonvulsants for \>= 4 weeks prior to randomisation
  • History or evidence of cardiovascular risk (LVEF \< LLN; QTcB \>= 480 msec; blood pressure or systolic \>=140 mmHg or diastolic \>= 90 mmHg which cannot be controlled by anti-hypertensive therapy)
  • History or current evidence/risk of retinal vein occlusion (RVO) or central serous retinopathy (CSR)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (205)

Novartis Investigative Site

Birmingham, Alabama, 35243, United States

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Novartis Investigative Site

Gilbert, Arizona, 85234, United States

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Novartis Investigative Site

Beverly Hills, California, 90211, United States

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Novartis Investigative Site

San Francisco, California, 94115, United States

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Novartis Investigative Site

Vallejo, California, 94589, United States

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Novartis Investigative Site

Aurora, Colorado, 80010, United States

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Novartis Investigative Site

Jacksonville, Florida, 32204, United States

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Novartis Investigative Site

Miami Beach, Florida, 33140, United States

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Novartis Investigative Site

Orlando, Florida, 32804, United States

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Novartis Investigative Site

Atlanta, Georgia, 30322, United States

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Novartis Investigative Site

Atlanta, Georgia, 30341, United States

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Novartis Investigative Site

Iowa City, Iowa, 52242, United States

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Novartis Investigative Site

Ann Arbor, Michigan, 48109, United States

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Novartis Investigative Site

Fridley, Minnesota, 55432, United States

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Novartis Investigative Site

St Louis, Missouri, 63110, United States

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Novartis Investigative Site

Las Vegas, Nevada, 89148, United States

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Novartis Investigative Site

Hackensack, New Jersey, 07601, United States

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Novartis Investigative Site

New Brunswick, New Jersey, 08901, United States

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Novartis Investigative Site

New York, New York, 10029, United States

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Novartis Investigative Site

Chapel Hill, North Carolina, 27599-7600, United States

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Novartis Investigative Site

Charlotte, North Carolina, 28204, United States

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Novartis Investigative Site

Durham, North Carolina, 27710, United States

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Novartis Investigative Site

Cincinnati, Ohio, 45219, United States

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Novartis Investigative Site

Columbus, Ohio, 43210, United States

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Novartis Investigative Site

Bend, Oregon, 97701, United States

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Novartis Investigative Site

Portland, Oregon, 97213, United States

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Novartis Investigative Site

Portland, Oregon, 97239, United States

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Novartis Investigative Site

Charleston, South Carolina, 29425, United States

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Novartis Investigative Site

Greenville, South Carolina, 29605, United States

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Nashville, Tennessee, 37232, United States

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Novartis Investigative Site

Dallas, Texas, 75246, United States

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Salt Lake City, Utah, 84106, United States

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Novartis Investigative Site

Salt Lake City, Utah, 84112-5550, United States

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Novartis Investigative Site

Burlington, Vermont, 05403, United States

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Novartis Investigative Site

Charlottesville, Virginia, 22903, United States

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Novartis Investigative Site

Milwaukee, Wisconsin, 53226, United States

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Novartis Investigative Site

Capital Federal, Buenos Aires, C1426ANZ, Argentina

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Novartis Investigative Site

Viedma, Río Negro Province, R8500ACE, Argentina

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Novartis Investigative Site

Rosario, Santa Fe Province, S2000KZE, Argentina

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Novartis Investigative Site

Buenos Aires, C1121ABE, Argentina

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Novartis Investigative Site

San Miguel de Tucumán, T4000IAK, Argentina

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Santa Fe, 3000, Argentina

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North Sydney, New South Wales, 2060, Australia

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Westmead, New South Wales, 2145, Australia

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Novartis Investigative Site

Greenslopes, Queensland, 4120, Australia

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Novartis Investigative Site

Herston, Queensland, 4029, Australia

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Novartis Investigative Site

South Brisbane, Queensland, 4101, Australia

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Novartis Investigative Site

Woodville, South Australia, 5011, Australia

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Novartis Investigative Site

Box Hill, Victoria, 3128, Australia

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Novartis Investigative Site

Melbourne, Victoria, 3004, Australia

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Novartis Investigative Site

Nedlands, Western Australia, 6009, Australia

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Novartis Investigative Site

Graz, A-8036, Austria

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Innsbruck, 6020, Austria

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Novartis Investigative Site

Salzburg, A-5020, Austria

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Novartis Investigative Site

Vienna, 1090, Austria

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Novartis Investigative Site

Vienna, A-1030, Austria

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Novartis Investigative Site

Brasschaat, 2930, Belgium

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Brussels, 1090, Belgium

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Novartis Investigative Site

Brussels, 1200, Belgium

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Novartis Investigative Site

Ghent, 9000, Belgium

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Novartis Investigative Site

Kortrijk, 8500, Belgium

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Leuven, 3000, Belgium

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Novartis Investigative Site

Namur, 5000, Belgium

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Wilrijk, 2610, Belgium

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Ijuí, Rio Grande do Sul, 98700-000, Brazil

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Novartis Investigative Site

Itajaí, Santa Catarina, 88301-215, Brazil

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Novartis Investigative Site

Sao Paulo - SP, 01323-900, Brazil

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Novartis Investigative Site

Calgary, Alberta, T2N 4N2, Canada

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Kelowna, British Columbia, V1Y 5L3, Canada

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Vancouver, British Columbia, V5Z 4E6, Canada

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Novartis Investigative Site

Winnipeg, Manitoba, R3E 0V9, Canada

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Novartis Investigative Site

Halifax, Nova Scotia, B3H 2Y9, Canada

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Kingston, Ontario, K7L 5P9, Canada

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Oshawa, Ontario, L1G 2B9, Canada

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Ottawa, Ontario, K1H 8L6, Canada

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Novartis Investigative Site

Toronto, Ontario, M4N 3M5, Canada

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Toronto, Ontario, M5G 2M9, Canada

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Novartis Investigative Site

Montreal, Quebec, H2L 4M1, Canada

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Novartis Investigative Site

Québec, Quebec, G1R 2J6, Canada

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Novartis Investigative Site

Olomouc, 775 20, Czechia

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Novartis Investigative Site

Ostrava, 708 52, Czechia

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Novartis Investigative Site

Prague, 100 34, Czechia

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Novartis Investigative Site

Prague, 128 08, Czechia

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Novartis Investigative Site

Zlín, 76275, Czechia

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Novartis Investigative Site

Arhus C, 8000, Denmark

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Novartis Investigative Site

Herlev, 2730, Denmark

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Novartis Investigative Site

Odense, 5000 C, Denmark

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Novartis Investigative Site

Helsinki, 00029, Finland

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Novartis Investigative Site

Jyväskylä, 40620, Finland

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Novartis Investigative Site

Tampere, 33520, Finland

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Novartis Investigative Site

Turku, 20520, Finland

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Novartis Investigative Site

Bordeaux, 33075, France

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Novartis Investigative Site

Grenoble, 38043, France

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Novartis Investigative Site

Lille, 59037, France

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Marseille, 13385, France

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Montpellier, 34295, France

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Nantes, 44093, France

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Novartis Investigative Site

Nice, 06202, France

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Paris, 75475, France

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Novartis Investigative Site

Reims, 51092, France

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Rennes, 35042, France

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Novartis Investigative Site

Villejuif, 94805, France

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Novartis Investigative Site

Heidelberg, Baden-Wurttemberg, 69120, Germany

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Novartis Investigative Site

Heilbronn, Baden-Wurttemberg, 74078, Germany

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Mannheim, Baden-Wurttemberg, 68167, Germany

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Novartis Investigative Site

Tübingen, Baden-Wurttemberg, 72076, Germany

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Novartis Investigative Site

Erlangen, Bavaria, 91054, Germany

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Munich, Bavaria, 80337, Germany

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Munich, Bavaria, 80802, Germany

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Novartis Investigative Site

Munich, Bavaria, 80804, Germany

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Novartis Investigative Site

Nuremberg, Bavaria, 90419, Germany

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Regensburg, Bavaria, 93053, Germany

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Novartis Investigative Site

Würzburg, Bavaria, 97080, Germany

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Novartis Investigative Site

Buxtehude, Lower Saxony, 21614, Germany

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Novartis Investigative Site

Hanover, Lower Saxony, 30625, Germany

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Bonn, North Rhine-Westphalia, 53127, Germany

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Cologne, North Rhine-Westphalia, 50937, Germany

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Essen, North Rhine-Westphalia, 45122, Germany

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Novartis Investigative Site

Ludwigshafen am Rhein, Rhineland-Palatinate, 67063, Germany

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Mainz, Rhineland-Palatinate, 55131, Germany

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Dresden, Saxony, 01307, Germany

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Leipzig, Saxony, 04103, Germany

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Novartis Investigative Site

Magdeburg, Saxony-Anhalt, 39120, Germany

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Novartis Investigative Site

Kiel, Schleswig-Holstein, 24105, Germany

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Novartis Investigative Site

Lübeck, Schleswig-Holstein, 23538, Germany

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Novartis Investigative Site

Erfurt, Thuringia, 99089, Germany

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Novartis Investigative Site

Gera, Thuringia, 07548, Germany

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Novartis Investigative Site

Budapest, 1062, Hungary

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Budapest, H-1122, Hungary

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Novartis Investigative Site

Debrecen, 4032, Hungary

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Győr, H-9024, Hungary

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Kaposvár, 7400, Hungary

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Miskolc, 3526, Hungary

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Novartis Investigative Site

Szeged, 6720, Hungary

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Novartis Investigative Site

Co.Cork, Ireland

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Dublin, 4, Ireland

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Dublin, 7, Ireland

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Dublin, 9, Ireland

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Galway, Ireland

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Jerusalem, Israel

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Ramat Gan, 52621, Israel

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Napoli, Campania, 80131, Italy

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Rome, Lazio, 00167, Italy

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Genoa, Liguria, 16132, Italy

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Bergamo, Lombardy, 24128, Italy

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Novartis Investigative Site

Milan, Lombardy, 20133, Italy

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Milan, Lombardy, 20141, Italy

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Pisa, Tuscany, 56126, Italy

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Padua, Veneto, 35128, Italy

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Novartis Investigative Site

Amsterdam, 1066 CX, Netherlands

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Amsterdam, 1081 HV, Netherlands

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Novartis Investigative Site

Groningen, 9713 GZ, Netherlands

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Novartis Investigative Site

Leeuwarden, 8934 AD, Netherlands

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Novartis Investigative Site

Leiden, 2333 ZA, Netherlands

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Rotterdam, 3015 GD, Netherlands

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Novartis Investigative Site

Christchurch, 8011, New Zealand

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Novartis Investigative Site

Newtown, Wellington, 6002, New Zealand

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Novartis Investigative Site

Kristiansand, 4604, Norway

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Novartis Investigative Site

Lorenskog, 1478, Norway

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Novartis Investigative Site

Oslo, 0310, Norway

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Novartis Investigative Site

Gdansk, 80-215, Poland

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Novartis Investigative Site

Konin, 62-500, Poland

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Poznan, 60-693, Poland

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Novartis Investigative Site

Warsaw, 02-781, Poland

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Novartis Investigative Site

Chelyabinsk, 454087, Russia

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Novartis Investigative Site

Magnitogorsk, 455001, Russia

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Moscow, 115478, Russia

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Novartis Investigative Site

Moscow, 143423, Russia

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Novartis Investigative Site

Nizhny Novgorod, 603081, Russia

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Novartis Investigative Site

Ryazan, 390011, Russia

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Novartis Investigative Site

Saint Petersburg, 197758, Russia

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Novartis Investigative Site

Goyang-si, Gyeonggi-Do, 410-769, South Korea

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Novartis Investigative Site

Seoul, 03080, South Korea

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Novartis Investigative Site

Seoul, 135-710, South Korea

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Novartis Investigative Site

Barcelona, 08036, Spain

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Novartis Investigative Site

Hospitalet de Llobregat, Barcelona, 08907, Spain

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Novartis Investigative Site

Las Palmas de Gran Canaria, 35016, Spain

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Novartis Investigative Site

Madrid, 28007, Spain

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Novartis Investigative Site

Madrid, 28050, Spain

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Novartis Investigative Site

Palma de Mallorca, 07010, Spain

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Pamplona, 31008, Spain

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Novartis Investigative Site

Valencia, 46009, Spain

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Novartis Investigative Site

Valencia, 46014, Spain

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Novartis Investigative Site

Linköping, SE-581 85, Sweden

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Novartis Investigative Site

Umeå, SE-901 85, Sweden

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Novartis Investigative Site

Basel, 4031, Switzerland

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Novartis Investigative Site

Lausanne, 1011, Switzerland

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Zurich, 8091, Switzerland

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Novartis Investigative Site

Tainan, 704, Taiwan

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Taipei, 100, Taiwan

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Novartis Investigative Site

Taoyuan District, 333, Taiwan

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Dnipropetrovsk, 49102, Ukraine

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Donetsk, 83092, Ukraine

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Kharkiv, 61070, Ukraine

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Kyiv, 03022, Ukraine

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Lviv, 79031, Ukraine

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Sumy, 40005, Ukraine

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Uzhhorod, 88017, Ukraine

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Cambridge, CB2 0QQ, United Kingdom

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Glasgow, G12 0YN, United Kingdom

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Novartis Investigative Site

London, NW3 2QG, United Kingdom

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Novartis Investigative Site

London, SE1 7EH, United Kingdom

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Novartis Investigative Site

Manchester, M20 4BX, United Kingdom

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Novartis Investigative Site

Southampton, SO16 6YD, United Kingdom

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Novartis Investigative Site

Swansea, SA2 8QA, United Kingdom

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Related Publications (5)

  • Schadendorf D, Robert C, Dummer R, Flaherty KT, Tawbi HA, Menzies AM, Banerjee H, Lau M, Long GV. Pyrexia in patients treated with dabrafenib plus trametinib across clinical trials in BRAF-mutant cancers. Eur J Cancer. 2021 Aug;153:234-241. doi: 10.1016/j.ejca.2021.05.005. Epub 2021 Jul 2.

  • Robert C, Grob JJ, Stroyakovskiy D, Karaszewska B, Hauschild A, Levchenko E, Chiarion Sileni V, Schachter J, Garbe C, Bondarenko I, Gogas H, Mandala M, Haanen JBAG, Lebbe C, Mackiewicz A, Rutkowski P, Nathan PD, Ribas A, Davies MA, Flaherty KT, Burgess P, Tan M, Gasal E, Voi M, Schadendorf D, Long GV. Five-Year Outcomes with Dabrafenib plus Trametinib in Metastatic Melanoma. N Engl J Med. 2019 Aug 15;381(7):626-636. doi: 10.1056/NEJMoa1904059. Epub 2019 Jun 4.

  • Long GV, Grob JJ, Nathan P, Ribas A, Robert C, Schadendorf D, Lane SR, Mak C, Legenne P, Flaherty KT, Davies MA. Factors predictive of response, disease progression, and overall survival after dabrafenib and trametinib combination treatment: a pooled analysis of individual patient data from randomised trials. Lancet Oncol. 2016 Dec;17(12):1743-1754. doi: 10.1016/S1470-2045(16)30578-2. Epub 2016 Nov 16.

  • Grob JJ, Amonkar MM, Karaszewska B, Schachter J, Dummer R, Mackiewicz A, Stroyakovskiy D, Drucis K, Grange F, Chiarion-Sileni V, Rutkowski P, Lichinitser M, Levchenko E, Wolter P, Hauschild A, Long GV, Nathan P, Ribas A, Flaherty K, Sun P, Legos JJ, McDowell DO, Mookerjee B, Schadendorf D, Robert C. Comparison of dabrafenib and trametinib combination therapy with vemurafenib monotherapy on health-related quality of life in patients with unresectable or metastatic cutaneous BRAF Val600-mutation-positive melanoma (COMBI-v): results of a phase 3, open-label, randomised trial. Lancet Oncol. 2015 Oct;16(13):1389-98. doi: 10.1016/S1470-2045(15)00087-X.

  • Robert C, Karaszewska B, Schachter J, Rutkowski P, Mackiewicz A, Stroiakovski D, Lichinitser M, Dummer R, Grange F, Mortier L, Chiarion-Sileni V, Drucis K, Krajsova I, Hauschild A, Lorigan P, Wolter P, Long GV, Flaherty K, Nathan P, Ribas A, Martin AM, Sun P, Crist W, Legos J, Rubin SD, Little SM, Schadendorf D. Improved overall survival in melanoma with combined dabrafenib and trametinib. N Engl J Med. 2015 Jan 1;372(1):30-9. doi: 10.1056/NEJMoa1412690. Epub 2014 Nov 16.

MeSH Terms

Conditions

MelanomaNeoplasms

Interventions

dabrafenibVemurafenibtrametinib

Condition Hierarchy (Ancestors)

Neuroendocrine TumorsNeuroectodermal TumorsNeoplasms, Germ Cell and EmbryonalNeoplasms by Histologic TypeNeoplasms, Nerve TissueNevi and MelanomasSkin NeoplasmsNeoplasms by SiteSkin DiseasesSkin and Connective Tissue Diseases

Intervention Hierarchy (Ancestors)

SulfonamidesAmidesOrganic ChemicalsSulfonesSulfur CompoundsIndolesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic Compounds

Results Point of Contact

Title
Clinical Disclosure Office
Organization
Novartis Pharmaceuticals

Study Officials

  • Novartis Pharmaceuticals

    Novartis Pharmaceuticals

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 10, 2012

First Posted

May 14, 2012

Study Start

June 4, 2012

Primary Completion

April 17, 2014

Study Completion

April 25, 2019

Last Updated

February 24, 2021

Results First Posted

December 4, 2014

Record last verified: 2021-02

Data Sharing

IPD Sharing
Will share

Novartis is committed to sharing with qualified external researchers, access to patient-level data and supporting clinical documents from eligible studies. These requests are reviewed and approved by an independent review panel on the basis of scientific merit. All data provided is anonymized to respect the privacy of patients who have participated in the trial in line with applicable laws and regulations. This trial data availability is according to the criteria and process described on www.clinicalstudydatarequest.com.

Locations