NCT06929273

Brief Summary

This is a phase 3, open-label extension study to assess the long-term safety of KarXT for the treatment of mania or mania with mixed features in Bipolar-I disorder (BP-I) The primary objective of the study is to evaluate the long-term safety and tolerability of KarXT in the treatment of participants with mania or mania with mixed features associated with BP-I.

Trial Health

88
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
450

participants targeted

Target at P50-P75 for phase_3

Timeline
24mo left

Started Jul 2025

Typical duration for phase_3

Geographic Reach
20 countries

173 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress31%
Jul 2025Jun 2028

First Submitted

Initial submission to the registry

April 14, 2025

Completed
2 days until next milestone

First Posted

Study publicly available on registry

April 16, 2025

Completed
3 months until next milestone

Study Start

First participant enrolled

July 18, 2025

Completed
2.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 13, 2028

Expected
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

June 13, 2028

Last Updated

June 2, 2026

Status Verified

June 1, 2026

Enrollment Period

2.9 years

First QC Date

April 14, 2025

Last Update Submit

June 1, 2026

Conditions

Keywords

Bipolar-I disorderManiaBipolar-I disorder with Mania

Outcome Measures

Primary Outcomes (1)

  • Number of participants with treatment emergent adverse events (TEAEs)

    Up to week 54

Secondary Outcomes (8)

  • Number of participants with AEs of special interest (AESIs)

    Up to week 54

  • Number of participants with serious AEs (SAEs)

    Up to week 54

  • Number of participants with TEAEs leading to treatment discontinuation

    Up to week 52

  • Number of participants with change in suicidal ideation as assessed by the Columbia-Suicide Severity Rating Scale (C-SSRS)

    Up to week 54

  • Change from baseline in Barnes Akathisia Rating Scale (BARS) score

    Up to week 54

  • +3 more secondary outcomes

Study Arms (1)

KarXT or Adjuvant KarXT

EXPERIMENTAL
Drug: KarXTDrug: LithiumDrug: ValproateDrug: Lamotrigine

Interventions

Therapeutic dose

KarXT or Adjuvant KarXT
KarXTDRUG

Specified dose on specified days

Also known as: BMS-986510, Xanomeline and trospium chloride
KarXT or Adjuvant KarXT

Therapeutic dose

KarXT or Adjuvant KarXT

Therapeutic dose

KarXT or Adjuvant KarXT

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participants who participated in double-blind placebo-controlled study (CN0120036, CN0120037, or CN0120046):
  • a. Participants must have completed treatment period of parent study.
  • De novo participants who did not participate in double-blind placebo-controlled studies:
  • Participants must have primary diagnosis of Bipolar-I disorder established by a comprehensive psychiatric evaluation based on DSM-5-TR criteria and confirmed by the Mini International Neuropsychiatric Interview (MINI, v7.0.2), with symptoms of mania or mixed mania.
  • Participants must have Young Mania Rating Scale (YMRS) score of ≥ 14 at Screening and at baseline.
  • Participants must have CGI-BP score of ≥ 3 at Screening and at baseline.
  • Participants does not require hospitalization for acute mania.

You may not qualify if:

  • Participants who participated in double-blind placebo-controlled study (CN0120036, CN0120037, or CN0120046):
  • a. Discontinuation from any KarXT parent studies.
  • De novo participants who did not participate in double-blind placebo-controlled studies:
  • All participants with a risk for suicidal behavior at baseline as determined by Investigator's clinical assessment or history of suicidal behavior as assessed on C-SSRS.
  • Participants must not have primary diagnosis of BP-I with rapid cycling (ie, ≥ 4 distinct mood episodes in one year).
  • Participants must not have any primary DSM-5-TR disorder other than BP-I with mania or mania with mixed features within 12 months before Screening (confirmed using MINI version 7.0.2 at Screening), including BP-I with depression, (previous 3 months only), Bipolar-II disorder, major depressive disorder, borderline personality disorder, and primary psychotic disorder, with the exception of mild anxiety disorders.
  • Individual has a DSM-5-TR diagnosis of moderate to severe substance use disorder (except tobacco use disorder) within the 12 months before Screening (confirmed using MINI version 7.0.2 at Screening), or current use as determined by urine toxicology screen or alcohol test.
  • Participants must not have history of irritable bowel syndrome (with or without constipation) or serious constipation requiring treatment within the last 6 months.
  • Participants must not have history or high risk of urinary retention, gastric retention, or untreated narrow-angle glaucoma.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (173)

Local Institution - 0120

Glendale, Arizona, 85304, United States

NOT YET RECRUITING

Pillar Clinical Research - Richardson

Bentonville, Arkansas, 72712, United States

RECRUITING

Pillar Clinical Research- Little Rock

Little Rock, Arkansas, 72204, United States

RECRUITING

Woodland International Research Group

Little Rock, Arkansas, 72211, United States

RECRUITING

Woodland Research Northwest

Rogers, Arkansas, 72758, United States

RECRUITING

Advanced Research Center Inc.

Anaheim, California, 92805, United States

RECRUITING

Clinical Innovations, Inc. dba CITrials

Bellflower, California, 90706, United States

RECRUITING

Local Institution - 0044

Cerritos, California, 90703, United States

NOT YET RECRUITING

Inland Psychiatric Medical Group - Chino

Chino, California, 91710, United States

RECRUITING

Proscience Research Group

Culver City, California, 90230, United States

RECRUITING

Collaborative Neuroscience Research, LLC

Garden Grove, California, 92845-2506, United States

RECRUITING

Omega Clinical Trials - La Habra

La Habra, California, 90631, United States

RECRUITING

Catalina Research Institute, LLC

Montclair, California, 91763, United States

RECRUITING

NRC Research Institute

Orange, California, 92868, United States

RECRUITING

Clinical Innovations, Inc. dba CITrials

Riverside, California, 92506, United States

RECRUITING

Local Institution - 0136

Santa Ana, California, 92705, United States

NOT YET RECRUITING

Collaborative Neuroscience Research, LLC

Torrance, California, 90504, United States

RECRUITING

Yale New Haven Hospital-Smilow Cancer Center

New Haven, Connecticut, 06510, United States

RECRUITING

Velocity Clinical Research, Hallandale Beach

Hallandale, Florida, 33009, United States

RECRUITING

Local Institution - 0026

Hialeah Gardens, Florida, 33016, United States

NOT YET RECRUITING

Behavioral Clinical Research

Hollywood, Florida, 33021, United States

RECRUITING

Research Centers of America ( Hollywood )

Hollywood, Florida, 33024, United States

RECRUITING

LCC Medical Research Institute

Miami, Florida, 33126, United States

RECRUITING

Advanced Research Institute of Miami

Miami, Florida, 33135, United States

RECRUITING

Innovative Clinical Research, Inc.

Miami Lakes, Florida, 33016, United States

RECRUITING

South Florida Research Phase I-IV

Miami Springs, Florida, 33166, United States

RECRUITING

Local Institution - 0045

St. Petersburg, Florida, 33713, United States

NOT YET RECRUITING

Health Synergy Clinical Research

West Palm Beach, Florida, 33407, United States

RECRUITING

Synexus Clinical Research US, Inc.

Atlanta, Georgia, 30328, United States

RECRUITING

Atlanta Center for Medical Research

Atlanta, Georgia, 30331, United States

RECRUITING

CenExel iResearch, LLC

Decatur, Georgia, 30030, United States

RECRUITING

CenExel iResearch, LLC

Savannah, Georgia, 31405, United States

RECRUITING

Local Institution - 0031

Chicago, Illinois, 60640, United States

NOT YET RECRUITING

Pillar Clinical Research -Chicago

Chicago, Illinois, 60641, United States

RECRUITING

CBH Health

Gaithersburg, Maryland, 20877, United States

RECRUITING

Precise Research Centers

Flowood, Mississippi, 39232, United States

RECRUITING

Arch Clinical Trials

St Louis, Missouri, 63141, United States

RECRUITING

Local Institution - 0121

North Las Vegas, Nevada, 89030, United States

NOT YET RECRUITING

Local Institution - 0122

North Las Vegas, Nevada, 89030, United States

WITHDRAWN

Hassman Research Institute Marlton Site

Marlton, New Jersey, 08053, United States

RECRUITING

Local Institution - 0058

Marlton, New Jersey, 08053, United States

WITHDRAWN

Richmond Behavioral Associates

Staten Island, New York, 10314, United States

RECRUITING

Local Institution - 0124

Charlotte, North Carolina, 28211, United States

WITHDRAWN

University of Cincinnati Medical Center

Cincinnati, Ohio, 45219, United States

RECRUITING

Neuro-Behavioral Clinical Research

North Canton, Ohio, 44720, United States

RECRUITING

Community Clinical Research

Austin, Texas, 78754, United States

RECRUITING

InSite Clinical Research

DeSoto, Texas, 75115, United States

RECRUITING

Local Institution - 0046

Houston, Texas, 77021, United States

WITHDRAWN

Elevate Clinical Research-Houston

Houston, Texas, 77058, United States

RECRUITING

Local Institution - 0036

Irving, Texas, 75062, United States

WITHDRAWN

Prime Clinical Research - Mansfield

Mansfield, Texas, 76063, United States

RECRUITING

Pillar Clinical Research - Richardson

Richardson, Texas, 75080, United States

RECRUITING

Local Institution - 0128

ABB, Buenos Aires F.D., C1199ABB, Argentina

NOT YET RECRUITING

Local Institution - 0127

Córdoba, 5000, Argentina

NOT YET RECRUITING

Local Institution - 0126

Mendoza, 5502, Argentina

NOT YET RECRUITING

Ramsay Clinic Northside

St Leonards, New South Wales, 2065, Australia

RECRUITING

Ramsay Clinic New Farm

Brisbane, Queensland, 4005, Australia

RECRUITING

Center for Mental Health Prof. Dr. Ivan Temkov

Burgas, 8001, Bulgaria

RECRUITING

State Psychiatric Hospital Sv. Ivan Rilski Novi Iskar

Novi Iskar, 1282, Bulgaria

RECRUITING

"University Multiprofile Hospital for Active Treatment - Dr. Georgi Stranski" EAD

Pleven, 5800, Bulgaria

RECRUITING

MHAT "Dr. Ival Seliminski"

Sliven, 8800, Bulgaria

RECRUITING

Mental Health Center - Vratsa

Vratsa, 3000, Bulgaria

RECRUITING

Local Institution - 0177

Beijing, Beijing Municipality, 100088, China

NOT YET RECRUITING

Local Institution - 0174

Beijing, Beijing Municipality, 100096, China

NOT YET RECRUITING

Local Institution - 0175

Guangzhou, Guangdong, 510370, China

NOT YET RECRUITING

Local Institution - 0181

Baoding, Hebei, 71000, China

NOT YET RECRUITING

Local Institution - 0185

Shijiazhuang, Hebei, 050031, China

NOT YET RECRUITING

Local Institution - 0184

Changsha, Hunan, 410011, China

NOT YET RECRUITING

Local Institution - 0180

Nanjing, Jiangsu, 210029, China

NOT YET RECRUITING

Local Institution - 0176

Xi'an, Shaanxi, 710061, China

NOT YET RECRUITING

Local Institution - 0179

Chengdu, Sichuan, 610036, China

NOT YET RECRUITING

Local Institution - 0183

Tianjin, Tianjin Municipality, 300022, China

NOT YET RECRUITING

Local Institution - 0182

Ningbo, Zhejiang, 315201, China

NOT YET RECRUITING

Local Institution - 0018

Zagreb, City of Zagreb, 10090, Croatia

WITHDRAWN

Klinika za psihijatriju "Vrapče"

Zagreb, 10090, Croatia

RECRUITING

Klinika za psihijatriju "Vrapče"

Zagreb, 10090, Croatia

RECRUITING

Klinika za psihijatriju "Vrapče"

Zagreb, 10090, Croatia

RECRUITING

Psihijatrijska bolnica "Sveti Ivan"

Zagreb, 10090, Croatia

RECRUITING

Local Institution - 0153

Aalborg, North Denmark, 9000, Denmark

NOT YET RECRUITING

Local Institution - 0154

Glostrup Municipality, 2600, Denmark

NOT YET RECRUITING

Local Institution - 0170

Nice, Alpes-Maritimes, 06000, France

NOT YET RECRUITING

Local Institution - 0171

Clermont-Ferrand, 63000, France

NOT YET RECRUITING

Local Institution - 0172

Montpellier, 34295, France

NOT YET RECRUITING

Petz Aladar Egyetemi Oktato Korhaz

Győr, Győr-Moson-Sopron, 9024, Hungary

RECRUITING

Local Institution - 0110

Budapest, 0, Hungary

NOT YET RECRUITING

Semmelweis Egyetem

Budapest, 1083, Hungary

RECRUITING

Local Institution - 0111

Vadodara, Gujarat, 390021, India

NOT YET RECRUITING

Local Institution - 0132

Belagavi, Karnataka, 590010, India

NOT YET RECRUITING

Local Institution - 0159

Mangalore, Karnataka, 575003, India

NOT YET RECRUITING

Local Institution - 0190

Mangaluru, Karnataka, 574143, India

NOT YET RECRUITING

Local Institution - 0079

Kozhikode, Kerala, 673009, India

NOT YET RECRUITING

Local Institution - 0077

Ludhiana, Punjab, 141001, India

NOT YET RECRUITING

Local Institution - 0158

Madurai, Tamil Nadu, 625020, India

NOT YET RECRUITING

Local Institution - 0078

Hyderabad, Telangana, 500034, India

NOT YET RECRUITING

Local Institution - 0080

Hyderabad, Telangana, 500082, India

NOT YET RECRUITING

Local Institution - 0076

Kolkata, West Bengal, 700014, India

NOT YET RECRUITING

Local Institution - 0160

Kolkata, West Bengal, 700025, India

NOT YET RECRUITING

Shalvata Mental Health Center

Hod HaSharon, Central District, 4534708, Israel

RECRUITING

Ness Ziona Mental Health Center

Ness Ziona, Central District, 7410001, Israel

RECRUITING

Local Institution - 0084

Petah Tikva, Central District, 4910002, Israel

NOT YET RECRUITING

Sheba Medical Center

Ramat Gan, Central District, 5265601, Israel

RECRUITING

Be'er Sheva Mental Health Center

Beersheba, Southern District, 8461144, Israel

RECRUITING

Local Institution - 0173

Ashkelon, 78306, Israel

NOT YET RECRUITING

Local Institution - 0187

Bnei Brak, 5154475, Israel

NOT YET RECRUITING

Local Institution - 0168

Jerusalem, 91120, Israel

NOT YET RECRUITING

Kfar Shaul Mental Health Center

Jerusalem, 9546105, Israel

RECRUITING

Local Institution - 0066

Milan, Lombardy, 20122, Italy

NOT YET RECRUITING

Local Institution - 0083

Pisa, Tuscany, 56126, Italy

NOT YET RECRUITING

Local Institution - 0065

Siena, Tuscany, 53100, Italy

NOT YET RECRUITING

Local Institution - 0070

Ancona, 60126, Italy

NOT YET RECRUITING

Local Institution - 0069

Genova, 16132, Italy

NOT YET RECRUITING

Hotei Hospital

Kōnan, Aichi-ken, 4838248, Japan

RECRUITING

Okehazama Hospital

Toyoake, Aichi-ken, 470-1168, Japan

RECRUITING

National Kohnodai Medical Center.

Ichikawa, Chiba, 272-8516, Japan

RECRUITING

Local Institution - 0166

Iizuka, Fukuoka, 820-8505, Japan

WITHDRAWN

Local Institution - 0063

Kitakyushu, Fukuoka, 803-0831, Japan

WITHDRAWN

Obihiro Kosei Hospital

Obihiro, Hokkaido, 080-0024, Japan

RECRUITING

Goryokai Medical Corporation - Goryokai Hospital

Sapporo, Hokkaido, 002-8029, Japan

RECRUITING

Local Institution - 0165

Yokohama, Kanagawa, 234-0051, Japan

NOT YET RECRUITING

Kansai Medical University Medical Center

Moriguchi, Osaka, 570-8507, Japan

RECRUITING

Local Institution - 0007

Sakai-shi, Osaka, 590-0018, Japan

NOT YET RECRUITING

Rainbow and Sea Hospital

Karatsu-shi, Saga-ken, 847-0031, Japan

RECRUITING

Local Institution - 0016

Iruma, Saitama, 350-0495, Japan

WITHDRAWN

Saitama Konan Hospital

Kumagaya, Saitama, 360-0114, Japan

RECRUITING

Local Institution - 0163

Bunkyo-ku, Tokyo, 113-8431, Japan

NOT YET RECRUITING

Nippon Medical School Hospital

Bunkyo-ku, Tokyo, 1138603, Japan

RECRUITING

National Center of Neurology and Psychiatry

Kodaira, Tokyo, 187-8551, Japan

RECRUITING

Narimasu Kosei Hospital

tabashi City, Tokyo, 175-0091, Japan

RECRUITING

Kuramitsu Hospital

Fukuoka, 819-0037, Japan

RECRUITING

Kochi Health Sciences Center

Kochi, 781-8555, Japan

RECRUITING

Miyazaki Prefectural Miyazaki Hospital

Miyazaki, 880-8510, Japan

RECRUITING

Osaka Metropolitan University Hospital

Osaka, 545-8586, Japan

RECRUITING

Showa Medical University Karasuyama Hospital

Tokyo, 157-8577, Japan

RECRUITING

Wakayama Medical University Hospital

Wakayama, 641-8510, Japan

RECRUITING

Yamagata Sakuracho Hospital

Yamagata, 990-0045, Japan

RECRUITING

North Shore Hospital

Auckland, 0622, New Zealand

RECRUITING

Centrum Medyczne HCP

Poznan, Greater Poland Voivodeship, 61-485, Poland

RECRUITING

Instytut Psychiatrii i Neurologii

Warsaw, Masovian Voivodeship, 02-957, Poland

RECRUITING

Klinika Psychiatrii Uniwersytet Medyczny w Białymstoku

Bialystok, Podlaskie Voivodeship, 15-272, Poland

RECRUITING

Local Institution - 0093

Gdansk, Pomeranian Voivodeship, 80-214, Poland

NOT YET RECRUITING

M2M Med

Rybnik, Silesian Voivodeship, 44-200, Poland

RECRUITING

Clinica Inventiva

Tuszyn, 95-080, Poland

RECRUITING

Local Institution - 0095

Bucharest, Bucharest, 041914, Romania

NOT YET RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041914, Romania

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041914, Romania

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041914, Romania

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041914, Romania

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041914, Romania

RECRUITING

Local Institution - 0167

Bucharest, 011241, Romania

NOT YET RECRUITING

Centrul de Evaluare și Tratament a Toxicodependenței pentru Tineri Sf.Stelian

Bucharest, 060222, Romania

RECRUITING

Spitalul Universitar de Urgenta Militar Central Dr. Carol Davila

Bucharest, 0, Romania

RECRUITING

Local Institution - 0097

Iași, 700282, Romania

NOT YET RECRUITING

Spitalul de Psihiatrie și Neurologie Brașov

Sanpetru /Brasov, 507190, Romania

RECRUITING

Local Institution - 0118

Košice, Košice Region, 040 01, Slovakia

NOT YET RECRUITING

Local Institution - 0119

Košice, Košice Region, 040 01, Slovakia

NOT YET RECRUITING

Local Institution - 0117

Vranov nad Topľou, Presov, 093 01, Slovakia

NOT YET RECRUITING

Hospital Universitari Vall d'Hebron

Barcelona, Barcelona [Barcelona], 08035, Spain

RECRUITING

Osi Bilbao-Basurto

Bilbao, Basque Country, 48013, Spain

RECRUITING

Hospital Clínic de Barcelona

Barcelona, Catalunya [Cataluña], 08036, Spain

RECRUITING

Nacka Local Hospital

Nacka, Stockholms Län [se-01], 131 45, Sweden

RECRUITING

Local Institution - 0112

Uppsala, Uppsala Län [se-03], 751 85, Sweden

WITHDRAWN

Local Institution - 0116

Gothenburg, Västra Götalands Län [se-14], 413 45, Sweden

WITHDRAWN

Local Institution - 0152

Smila, Cherkasy Oblast, 20708, Ukraine

NOT YET RECRUITING

Local Institution - 0146

Skarzhyntsi, Khmelnytskyi Oblast, 32120, Ukraine

NOT YET RECRUITING

Local Institution - 0143

Hlevakha, Kyivska Oblast, 08631, Ukraine

NOT YET RECRUITING

Local Institution - 0147

Lviv, Lviv Oblast, 79021, Ukraine

NOT YET RECRUITING

Local Institution - 0145

Oleksandrivka, Odesa Oblast, 67513, Ukraine

NOT YET RECRUITING

Local Institution - 0189

Ternopil, Ternopil Oblast, 460027, Ukraine

NOT YET RECRUITING

Local Institution - 0148

Vinnytsia, Vinnytsia Oblast, 21037, Ukraine

NOT YET RECRUITING

Local Institution - 0149

Dnipro, 49115, Ukraine

NOT YET RECRUITING

Local Institution - 0151

Kropyvnytskyi, 25491, Ukraine

NOT YET RECRUITING

Local Institution - 0150

Kyiv, 04080, Ukraine

NOT YET RECRUITING

Local Institution - 0141

Poltava, 36013, Ukraine

NOT YET RECRUITING

Related Links

MeSH Terms

Conditions

Mania

Interventions

xanomelinetrospium chlorideLithiumValproic AcidLamotrigine

Condition Hierarchy (Ancestors)

Neurobehavioral ManifestationsNeurologic ManifestationsNervous System DiseasesSigns and SymptomsPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

Metals, AlkaliElementsInorganic ChemicalsMetals, LightMetalsPentanoic AcidsValeratesAcids, AcyclicCarboxylic AcidsOrganic ChemicalsFatty Acids, VolatileFatty AcidsLipidsTriazinesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Officials

  • Bristol-Myers Squibb

    Bristol-Myers Squibb

    STUDY DIRECTOR

Central Study Contacts

BMS Clinical Trials Contact Center www.BMSClinicalTrials.com

CONTACT

First line of the email MUST contain NCT # and Site #.

CONTACT

Study Design

Study Type
interventional
Phase
phase 3
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 14, 2025

First Posted

April 16, 2025

Study Start

July 18, 2025

Primary Completion (Estimated)

June 13, 2028

Study Completion (Estimated)

June 13, 2028

Last Updated

June 2, 2026

Record last verified: 2026-06

Data Sharing

IPD Sharing
Will share

BMS will provide access to individual anonymized participant data upon request from qualified researchers, and subject to certain criteria. Additional information regarding Bristol Myer Squibb's data sharing policy and process can be found at https://www.bms.com/researchers-and-partners/clinical-trials-and-research.html

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
See Plan Description
Access Criteria
See Plan Description
More information

Locations