NCT05425745

Brief Summary

This study will be a placebo-controlled, double-blind, randomized, phase 3 study to Evaluate the Efficacy, Safety, and Tolerability of Obicetrapib in Participants with a History of Heterozygous Familial Hypercholesterolemia (HeFH).

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
354

participants targeted

Target at P50-P75 for phase_3

Timeline
Completed

Started Jul 2022

Geographic Reach
10 countries

96 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 15, 2022

Completed
6 days until next milestone

First Posted

Study publicly available on registry

June 21, 2022

Completed
1 month until next milestone

Study Start

First participant enrolled

July 25, 2022

Completed
1.8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 28, 2024

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 28, 2024

Completed
1 year until next milestone

Results Posted

Study results publicly available

June 11, 2025

Completed
Last Updated

June 11, 2025

Status Verified

June 1, 2025

Enrollment Period

1.8 years

First QC Date

June 15, 2022

Results QC Date

May 21, 2025

Last Update Submit

June 10, 2025

Conditions

Keywords

ObicetrapibBROOKLYNCholesteryl ester transfer protein (CETP) inhibitorHeterozygous Familial Hypercholesterolemia (HeFH)LDL-C

Outcome Measures

Primary Outcomes (1)

  • Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) From Baseline to Day 84 [PUC]

    LS mean percent change from baseline to Day 84 in Low-Density Lipoprotein Cholesterol (LDL-C) in the obicetrapib group compared to the placebo group \[PUC\]. LDL-C level was measured by preparative ultracentrifugation (PUC).

    84 Days

Secondary Outcomes (19)

  • Percent Change in Low Density Lipoprotein-Cholesterol (LDL-C) From Baseline to Day 180 [Martin/Hopkins]

    180 Days

  • Percent Change in Low Density Lipoprotein-Cholesterol (LDL-C) From Baseline to Day 365 [PUC]

    365 Days

  • Percent Change in Apolipoprotein B (ApoB) From Baseline to Day 84

    84 Days

  • Percent Change in Apolipoprotein B (ApoB) From Baseline to Day 180

    180 Days

  • Percent Change in Apolipoprotein B (ApoB) From Baseline to Day 365

    365 Days

  • +14 more secondary outcomes

Study Arms (2)

Placebo

PLACEBO COMPARATOR

one placebo tablet once daily

Drug: Placebo

Obicetrapib 10 mg

EXPERIMENTAL

one 10 mg Obicetrapib tablet once daily

Drug: Obicetrapib

Interventions

10 mg Obicetrapib tablet

Also known as: CETP-inhibitor
Obicetrapib 10 mg

placebo tablet made to resemble active

Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Have a history of heterozygous familial hypercholesterolemia (HeFH) by 1) Genotyping (not a screening assessment), WHO Criteria/Dutch Lipid Clinical Network Criteria with a score of \> 8 points; and/or Simon Broome Register Diagnostic Criteria for definite or possible Familial Hypercholesterolemia (FH)
  • Maximally tolerated lipid Modifying therapy for at least 8 weeks prior to screening such as: ATV (40 or 80), or (ROS 20 or 40 mg), Ezetimide, Bempedoic Acid, PCSK9 targeted therapy for at least 4 doses
  • Fasting serum LDL-C ≥70 mg/dL (≥1.80 mmol/L)

You may not qualify if:

  • New York Heart Association class II or IV heart failure or last known left ventricular ejection fraction \< 30%;
  • Hospitalized for heart failure within 5 years prior to Screening
  • Major adverse cardiac event (MACE) within 3 months prior to Screening;
  • HbA1c ≥10%, or fasting glucose
  • Formal diagnosis of homozygous familial hypercholesterolemia (HoFH)
  • Uncontrolled severe hypertension, defined as either systolic blood pressure ≥ 160 mmHg or diastolic blood pressure ≥100 mmHg prior to Randomization

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (96)

Site 01022

Jonesboro, Arkansas, 72401, United States

Location

Site 01015

Toluca Lake, California, 91602, United States

Location

Site 01009

Sarasota, Florida, 34230, United States

Location

Site 01023

Boise, Idaho, 83702, United States

Location

Site 01018

Chicago, Illinois, 60602, United States

Location

Site 01012

Iowa City, Iowa, 52240, United States

Location

Site 01007

Baton Rouge, Louisiana, 70809, United States

Location

Site 01005

Port Gibson, Mississippi, 39105, United States

Location

Site 01006

St Louis, Missouri, 63130, United States

Location

Site 01011

Lincoln, Nebraska, 68510, United States

Location

Site 01004

Norfolk, Nebraska, 68701, United States

Location

Site 01002

Morristown, New Jersey, 07960, United States

Location

Site 01010

New Providence, New Jersey, 07901, United States

Location

Site 01001

North Massapequa, New York, 11758, United States

Location

Site 01020

Morganton, North Carolina, 28655, United States

Location

Site 01019

Winston-Salem, North Carolina, 27157, United States

Location

Site 01008

Chattanooga, Tennessee, 37405, United States

Location

Site 01016

El Paso, Texas, 79905, United States

Location

Site 01013

Houston, Texas, 76706, United States

Location

Site 01014

Suffolk, Virginia, 23434, United States

Location

Site 06007

Brampton, L6Z 4N5, Canada

Location

Site 06008

Chicoutimi, G7H 7K9, Canada

Location

Site 06005

Halifax, B3H 3A7, Canada

Location

Site 06003

Montreal, H2W 1R7, Canada

Location

Site 06009

Montreal, H3A 1A1, Canada

Location

Site 06004

Québec, G1V 4W2, Canada

Location

Site 06006

Sherbrooke, J1H 5N4, Canada

Location

Site 06001

Vancouver, V6Z 2C7, Canada

Location

Site 06002

Victoria, V8T 5G4, Canada

Location

Site 02006

Brno, 65691, Czechia

Location

Site 02002

Hradec Králové, 500 05, Czechia

Location

Site 02003

Prague, 128 08, Czechia

Location

Site 02005

Prague, 140 21, Czechia

Location

Site 02004

Prague, 15006, Czechia

Location

Site 02001

Uherské Hradiště, 686 01, Czechia

Location

Site 022001

Batumi, 6000, Georgia

Location

Site 022003

Tbilisi, 112, Georgia

Location

Site 022004

Tbilisi, 131, Georgia

Location

Site 022010

Tbilisi, 144, Georgia

Location

Site 022006

Tbilisi, 159, Georgia

Location

Site 022007

Tbilisi, 159, Georgia

Location

Site 022008

Tbilisi, 159, Georgia

Location

Site 022002

Tbilisi, 186, Georgia

Location

Site 022005

Tbilisi, 186, Georgia

Location

Site 022009

Tbilisi, 579, Georgia

Location

Site 04001

Amsterdam, 1105AZ, Netherlands

Location

Site 04003

Arnhem, 6815 AD, Netherlands

Location

Site 04002

Deventer, 7416 SE, Netherlands

Location

Site 04004

Eindhoven, 5631 BM, Netherlands

Location

Site 04005

Roosendaal, 4708 AE, Netherlands

Location

Site 04006

Rotterdam, 3015 GD, Netherlands

Location

Site 023003

Bodø, 8008, Norway

Location

Site 023002

Oslo, 587, Norway

Location

Site 05002

Bialystok, 15-276, Poland

Location

Site 05003

Lodz, 92-213, Poland

Location

Site 05004

Lodz, 93-338, Poland

Location

Site 05005

Zabrze, 41-800, Poland

Location

Site 05001

Zamość, 22-400, Poland

Location

Site 018001

Bloemfontein, 9301, South Africa

Location

Site 018002

Cape Town, 7530, South Africa

Location

Site 018009

Centurion, 154, South Africa

Location

Site 018006

Centurion, 157, South Africa

Location

Site 018004

Parow, 7500, South Africa

Location

Site 018003

Somerset West, 7130, South Africa

Location

Site 018005

Somerset West, 7130, South Africa

Location

Site 018007

Tongaat, 4400, South Africa

Location

Site 018008

Umhlanga, 4321, South Africa

Location

Site 17004

A Coruña, 15001, Spain

Location

Site 017001

Barcelona, 8036, Spain

Location

Site 17002

Barcelona, 8907, Spain

Location

Site 17003

Córdoba, 14004, Spain

Location

Site 17018

Figueras, 17600, Spain

Location

Site 17011

Granada, 18014, Spain

Location

Site 17017

Huelva, 21007, Spain

Location

Site 17012

Huesca, 22002, Spain

Location

Site 17008

Las Palmas de Gran Canaria, 35016, Spain

Location

Site 17010

Madrid, 28034, Spain

Location

Site 17016

Madrid, 28041, Spain

Location

Site 17007

Málaga, 29010, Spain

Location

Site 17013

Sabadell, 8208, Spain

Location

Site 17015

Santiago de Compostela, 15706, Spain

Location

Site 17009

Seville, 41009, Spain

Location

Site 17006

Seville, 41013, Spain

Location

Site 17014

Valencia, 46014, Spain

Location

Site 17005

Zaragoza, 50009, Spain

Location

Site 014006

Birmingham, B21 9RY, United Kingdom

Location

Site 014012

Bristol, BS2 8HW, United Kingdom

Location

Site 014009

Cardiff, CF14 4XW, United Kingdom

Location

Site 014010

Chichester, PO19 6SE, United Kingdom

Location

Site 014001

Dundee, DD1 9SY, United Kingdom

Location

Site 014002

London, NW3 2QG, United Kingdom

Location

Site 014003

Manchester, M23 9LT, United Kingdom

Location

Site 014008

Metropolitan Borough of Wirral, CH62 6EE, United Kingdom

Location

Site 014011

Penzance, TR19 7HU, United Kingdom

Location

Site 014005

Stevenage, SG14AB, United Kingdom

Location

Site 014004

West Bromwich, B71 4HJ, United Kingdom

Location

Related Publications (1)

  • Nicholls SJ, Nelson AJ, Ditmarsch M, Kastelein JJP, Ballantyne CM, Ray KK, Navar AM, Nissen SE, Goldberg AC, Brunham LR, Curcio D, Wuerdeman E, Neild A, Kling D, Hsieh A, Dicklin MR, Ference BA, Laufs U, Banach M, Mehran R, Catapano AL, Davidson MH. Obicetrapib on top of maximally tolerated lipid-modifying therapies in participants with or at high risk for atherosclerotic cardiovascular disease: rationale and designs of BROADWAY and BROOKLYN. Am Heart J. 2024 Aug;274:32-45. doi: 10.1016/j.ahj.2024.05.002. Epub 2024 May 4.

MeSH Terms

Conditions

DyslipidemiasHypercholesterolemiaHyperlipoproteinemia Type IILipid Metabolism DisordersMetabolic DiseasesLipid Metabolism, Inborn ErrorsGenetic Diseases, InbornHyperlipoproteinemias

Condition Hierarchy (Ancestors)

Nutritional and Metabolic DiseasesHyperlipidemiasMetabolism, Inborn ErrorsCongenital, Hereditary, and Neonatal Diseases and Abnormalities

Results Point of Contact

Title
Study Director
Organization
NewAmsterdam Pharma

Study Officials

  • Marc Ditmarsch

    NewAmsterdam Pharma

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Masking Details
placebo tablet made to resemble active
Purpose
TREATMENT
Intervention Model
PARALLEL
Model Details: Placebo-Controlled, double-blind, randomized
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 15, 2022

First Posted

June 21, 2022

Study Start

July 25, 2022

Primary Completion

May 28, 2024

Study Completion

May 28, 2024

Last Updated

June 11, 2025

Results First Posted

June 11, 2025

Record last verified: 2025-06

Data Sharing

IPD Sharing
Will not share

Locations