NCT04152018

Brief Summary

Open-label, multi-center, non-randomized, multiple dose, safety, tolerability, pharmacokinetic, and pharmacodynamics and clinical activity study of PF-06940434 (Integrin alpha-V/beta-8 Antagonist) in patients with SCCHN (Squamous Cell Carcinoma of the Head and Neck), renal cell carcinoma (RCC - clear cell and papillary), ovarian, gastric, esophageal, esophageal (adeno and squamous), lung squamous cell, pancreatic and biliary duct, endometrial, melanoma and urothelial tumors. This study contains two parts, single agent dose escalation (Part 1A), dose finding of PF 06940434 in combination with anti-PD-1 (Part 1B) and dose expansion (Part 2). Part 2 Dose Combination Expansion will enroll participants into 3 cohorts at doses determined from Part 1B in order to further evaluate the safety of PF-06940434 in combination with anti-PD-1.

Trial Health

63
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
85

participants targeted

Target at P75+ for phase_1

Timeline
Completed

Started Nov 2019

Longer than P75 for phase_1

Geographic Reach
5 countries

31 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 30, 2019

Completed
6 days until next milestone

First Posted

Study publicly available on registry

November 5, 2019

Completed
8 days until next milestone

Study Start

First participant enrolled

November 13, 2019

Completed
5.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 10, 2024

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

December 10, 2024

Completed
Last Updated

May 28, 2025

Status Verified

May 1, 2025

Enrollment Period

5.1 years

First QC Date

October 30, 2019

Last Update Submit

May 23, 2025

Conditions

Outcome Measures

Primary Outcomes (8)

  • Number of participants with Dose-limiting toxicities (DLT) for Dose Escalation and Dose Finding

    Baseline up to 28 Days (Cycle 1)

  • Number of Participants With Clinically Significant Change From Baseline in Laboratory Abnormalities

    Baseline up to approximately 24 months

  • Number of Participants With Adverse Events (AEs) According to Severity

    Baseline up to approximately 24 months

  • Number of Participants With Adverse Events (AEs) According to Seriousness

    Baseline up to up to approximately 24 months

  • Number of Participants With Adverse Events (AEs) by Relationship

    Baseline up to approximately 24 months

  • Progression-Free Survival (PFS) for Dose Expansion

    The period from study entry until disease progression, death or date of last contact.

    Baseline up to 24 Months

  • Objective Response Rate - Percentage of Participants With Objective Response in Dose Expansion

    Baseline up to 24 months

  • Duration of Response (DR) for Dose Expansion

    Baseline up to 24 Months

Secondary Outcomes (20)

  • PF-06940434 after multiple doses PK parameters (Cmax).

    Pre-dose on Cycle 1 Day 1 and on days 3, 8, and 15 of Cycle 1; Day 1 and Day 15 of Cycles 2 and 3; Days 1, 3, 8, and 15 of Cycle 4 and Pre-dose on Day 1 of every cycle thereafter and at end of treatment (each cycle is 28 days).

  • Area under the curve from time zero extrapolated to the last quantifiable dose of PF-06940434.

    Pre-dose on Cycle 1 Day 1 and on days 3, 8, and 15 of Cycle 1; Day 1 and Day 15 of Cycles 2 and 3; Days 1, 3, 8, and 15 of Cycle 4 and Pre-dose on Day 1 of every cycle thereafter and at end of treatment (each cycle is 28 days).

  • Systemic Clearance (CL)

    Pre-dose on Cycle 1 Day 1 and on days 3, 8, and 15 of Cycle 1; Day 1 and Day 15 of Cycles 2 and 3; Days 1, 3, 8, and 15 of Cycle 4 and Pre-dose on Day 1 of every cycle thereafter and at end of treatment (each cycle is 28 days).

  • Volume of Distribution (Vd)

    Pre-dose on Cycle 1 Day 1 and on days 3, 8, and 15 of Cycle 1; Day 1 and Day 15 of Cycles 2 and 3; Days 1, 3, 8, and 15 of Cycle 4 and Pre-dose on Day 1 of every cycle thereafter and at end of treatment (each cycle is 28 days).

  • Incidence and titers of anti-drug antibodies (ADA) against PF-06940434.

    Pre-dose on Days 1 and 15 of Cycle 1, pre-dose on Day 1 of Cycles 2 and 3, pre-dose on Day 1 of Cycle 4, pre-dose on Day 1 of every cycle thereafter and at end of treatment (each cycle is 28 days).

  • +15 more secondary outcomes

Study Arms (5)

Dose Escalation

EXPERIMENTAL

Single Agent Dose Escalation

Drug: PF-06940434

Dose Finding Anti-PD-1 Combination 1

EXPERIMENTAL

Part 1B PF-06940434 plus anti-PD-1

Drug: PF-06940434Drug: PF-06801591

Dose Expansion Arm A

EXPERIMENTAL

PF-06940434 with anti-PD-1 in SCCHN

Drug: PF-06940434Drug: PF-06801591

Dose Expansion Arm B

EXPERIMENTAL

PF-06940434 with anti-PD-1 in RCC

Drug: PF-06940434Drug: PF-06801591

Dose Expansion, Arm C

EXPERIMENTAL

PF-06940434 with anti-PD-1 (both Q3W)

Drug: PF-06940434Drug: PF-06801591

Interventions

PF-06940434 is given intravenously (IV) every 2 or 4 weeks in a 28 day cycle or every 3 weeks in a 21 day cycle. Multiple dose levels will be evaluated

Dose EscalationDose Expansion Arm ADose Expansion Arm BDose Expansion, Arm CDose Finding Anti-PD-1 Combination 1

PF-06801591 will be administered subcutaneously on Day 1 of each 28 day cycle or Day 1 of each 21 day cycle.

Also known as: Anti-PD-1
Dose Expansion Arm ADose Expansion Arm BDose Expansion, Arm CDose Finding Anti-PD-1 Combination 1

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • \- Histological or cytological diagnosis of SCCHN, RCC (clear cell and papillary cell), ovarian, gastric, esophageal (adeno and squamous), lung squamous cell, pancreatic and biliary duct, endometrial, melanoma, or urothelial cancer.
  • Part 2:
  • Arm A SCCHN:
  • Primary tumor location of the oral cavity, oropharynx, hypopharynx or larynx.
  • PDL-1 expression positive and CPS ≥1. No prior systemic therapy administered in the recurrent or metastatic setting (except for systemic therapy given as part of a multimodal treatment for locally advanced disease).
  • Arm B RCC (clear cell):
  • or 2 prior lines of therapy including PD-L1/PD-1 immunotherapy in combination or sequentially with antiangiogenic directed treatment
  • Adequate bone marrow, kidney and liver function.
  • Performance status of 0 or 1.

You may not qualify if:

  • Participant disease status is suitable for local therapy administered with curative intent.
  • Hypertension that cannot be controlled by medications.
  • Active or prior autoimmune disease
  • Active, uncontrolled bacterial, fungal, or viral infection, including (but not limited to) Hepatitis B, Hepatitis C, and known Human Immunodeficiency Virus infection or Acquired Immunodeficiency Syndrome-related illness

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (31)

HonorHealth Research Institute

Scottsdale, Arizona, 85258, United States

Location

HonorHealth Scottsdale Shea Medical Center

Scottsdale, Arizona, 85260, United States

Location

Ronald Reagan UCLA Medical Center

Los Angeles, California, 90095, United States

Location

UCLA Hematology Oncology

Los Angeles, California, 90095, United States

Location

UCLA Hematology/Oncology

Santa Monica, California, 90404, United States

Location

Greenebaum Comprehensive Cancer Center

Baltimore, Maryland, 21201, United States

Location

Siteman Cancer Center - St. Peters

City of Saint Peters, Missouri, 63376, United States

Location

Siteman Cancer Center - West County

Creve Coeur, Missouri, 63141, United States

Location

Siteman Cancer Center - North County

Florissant, Missouri, 63031, United States

Location

Barnes-Jewish Hospital

St Louis, Missouri, 63110, United States

Location

Washington University School of Medicine Siteman Cancer Center

St Louis, Missouri, 63110, United States

Location

Siteman Cancer Center - South County

St Louis, Missouri, 63129, United States

Location

Duke Univ. Medical Center/Duke Cancer Center

Durham, North Carolina, 27710, United States

Location

Investigational Chemotherapy Service

Durham, North Carolina, 27710, United States

Location

The University of Texas MD Anderson Cancer Center

Houston, Texas, 77030, United States

Location

NEXT Oncology

San Antonio, Texas, 78229, United States

Location

Fred Hutchinson Cancer Center

Seattle, Washington, 98109, United States

Location

University of Washington Medical Center

Seattle, Washington, 98195, United States

Location

Southern Medical Day Care Centre

Wollongong, New South Wales, 2500, Australia

Location

Onkologicky ustav sv. Alzbety, s.r.o.

Bratislava, 812 50, Slovakia

Location

Univerzitna nemocnica Bratislava

Bratislava, 82101, Slovakia

Location

Narodny ustav srdcovych a cievnych chorob, a.s.

Bratislava, 833 48, Slovakia

Location

MR Poprad s.r.o.

Komárno, 945 01, Slovakia

Location

KARDIO, s.r.o.

Poprad, 058 01, Slovakia

Location

POKO Poprad, s.r.o., Ambulancia klinickej onkologie

Poprad, 058 01, Slovakia

Location

Nemocnica Poprad a.s.

Poprad, 058 45, Slovakia

Location

Asan Medical Center

Seoul, Seoul-teukbyeolsi [seoul], 05505, South Korea

Location

Severance Hospital, Yonsei University Health System

Seoul, 03722, South Korea

Location

National Cheng Kung University Hospital

Tainan, 70403, Taiwan

Location

National Taiwan University Hospital

Taipei, 100, Taiwan

Location

Taipei Veterans General Hospital

Taipei, 11217, Taiwan

Location

Related Links

MeSH Terms

Conditions

Squamous Cell Carcinoma of Head and NeckCarcinoma, Renal CellOvarian NeoplasmsStomach NeoplasmsEsophageal NeoplasmsPancreatic NeoplasmsBile Duct NeoplasmsEndometrial Neoplasms

Interventions

spartalizumab

Condition Hierarchy (Ancestors)

Carcinoma, Squamous CellCarcinomaNeoplasms, Glandular and EpithelialNeoplasms by Histologic TypeNeoplasmsHead and Neck NeoplasmsNeoplasms by SiteAdenocarcinomaKidney NeoplasmsUrologic NeoplasmsUrogenital NeoplasmsFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesKidney DiseasesUrologic DiseasesMale Urogenital DiseasesEndocrine Gland NeoplasmsOvarian DiseasesAdnexal DiseasesGenital Diseases, FemaleGenital Neoplasms, FemaleGenital DiseasesEndocrine System DiseasesGonadal DisordersGastrointestinal NeoplasmsDigestive System NeoplasmsDigestive System DiseasesGastrointestinal DiseasesStomach DiseasesEsophageal DiseasesPancreatic DiseasesBiliary Tract NeoplasmsBile Duct DiseasesBiliary Tract DiseasesUterine NeoplasmsUterine Diseases

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 30, 2019

First Posted

November 5, 2019

Study Start

November 13, 2019

Primary Completion

December 10, 2024

Study Completion

December 10, 2024

Last Updated

May 28, 2025

Record last verified: 2025-05

Data Sharing

IPD Sharing
Will not share

Pfizer will provide access to individual de-identified participant data and related study documents (e.g. protocol, Statistical Analysis Plan (SAP), Clinical Study Report (CSR)) upon request from qualified researchers, and subject to certain criteria, conditions, and exceptions. Further details on Pfizer's data sharing criteria and process for requesting access can be found at: https://www.pfizer.com/science/clinical\_trials/trial\_data\_and\_results/data\_requests.

Locations