NCT04079179

Brief Summary

This is a research study of a drug called cobimetinib in children and adults diagnosed with Langerhans cell histiocytosis (LCH), and other histiocytic disorders that has returned or does not respond to treatment. Cobimetinib blocks activation of a protein called Mitogen-activated protein kinase (MEK) that is part of incorrect growth signals in histiocytosis cells. Four different groups of patients will be enrolled.

Trial Health

77
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
90

participants targeted

Target at P50-P75 for phase_2

Timeline
44mo left

Started Apr 2021

Longer than P75 for phase_2

Geographic Reach
1 country

12 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress59%
Apr 2021Dec 2029

First Submitted

Initial submission to the registry

August 10, 2019

Completed
27 days until next milestone

First Posted

Study publicly available on registry

September 6, 2019

Completed
1.6 years until next milestone

Study Start

First participant enrolled

April 19, 2021

Completed
4.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 1, 2025

Completed
4 years until next milestone

Study Completion

Last participant's last visit for all outcomes

December 1, 2029

Expected
Last Updated

September 18, 2025

Status Verified

September 1, 2025

Enrollment Period

4.6 years

First QC Date

August 10, 2019

Last Update Submit

September 12, 2025

Conditions

Keywords

CobimetinibLangerhans Cell Histiocytosis (LCH)

Outcome Measures

Primary Outcomes (1)

  • Overall Response Rates using modified RECiST criteria

    Proportion of participants with (complete response, partial response, stable disease, progressive disease) by 1 year of therapy with Cobimetinib. It is assumed that at each protocol-specified timepoint, a response assessment occurs. Status calculation will occur at each timepoint for patients who have measurable disease at baseline per the criteria defined in the protocol.

    12 months

Secondary Outcomes (2)

  • Progression Free Survival

    12 months

  • Nature and Severity of Adverse Events

    12 months

Other Outcomes (1)

  • Response assessment (Modified RECIST) of histiocytic lesions with specific mutations

    12 months

Study Arms (4)

Patients < 21 years with recurrent LCH (Grp1)

EXPERIMENTAL

Children (≥ 6 months) and young adults (\<21 years) with recurrent active LCH lesions (may also have LCH-ND).

Drug: Cobimetinib

Patients of any age with LCH-ND (Grp2)

EXPERIMENTAL

Patients of any age (≥ 6 months) with progressive LCH Neurodegenerative Disease (LCH-ND) without other sites of active LCH.

Drug: Cobimetinib

Patients <21 years with other histiocytic disorders (Grp3)

EXPERIMENTAL

Newly diagnosed or relapsed/refractory children (≥ 6 months) and young adults (\<21 years) with other histiocytic disorders including juvenile xanthogranuloma, Erdheim-Chester disease, histiocytic sarcoma and Rosai-Dorfman disease.

Drug: Cobimetinib

Patients ≥ 21 years with LCH/histiocytic disorders (Grp4)

EXPERIMENTAL

Adults (≥21 years) with LCH or other histiocytic disorder with recurrent active lesions (may also have LCH-ND).

Drug: Cobimetinib

Interventions

Cobimetinib will be administered at a maximal dose of 60 mg daily for patients \<18 years old and a flat dose of 40 mg daily for patients ≥18 years for 21 days on, then 7 days off, in a 28-day treatment cycle for a total of 12 cycles (approximately 12 months).

Also known as: COTELLIC, RO5514041
Patients < 21 years with recurrent LCH (Grp1)Patients <21 years with other histiocytic disorders (Grp3)Patients of any age with LCH-ND (Grp2)Patients ≥ 21 years with LCH/histiocytic disorders (Grp4)

Eligibility Criteria

Sexall
Healthy VolunteersNo
Age GroupsChild (0-17), Adult (18-64), Older Adult (65+)

You may qualify if:

  • Age at study entry
  • For Group 1: Participant must be at least 6 months of age and less than 21 years of age at the time of enrollment
  • For Group 2: Participant may be at least 6 months of age at the time of enrollment
  • For Group 3: Participant must be at least 6 months of age and less than 21 years of age at the time of enrollment
  • For Group 4: Participant must be 21 years of age or older at the time of enrollment
  • Participant must be able to take an enteral dose and formulation of medication. Study medication is only available as an oral suspension or tablet which may be taken by mouth or other enteral route such as nasogastric or gastric tube.
  • Biopsy proven LCH -AND
  • Failure of at least front-line therapy for LCH with evaluable disease. -OR
  • Diagnosis of LCH-associated neurodegenerative disease with radiologic or clinical progression within the past 3 months. -OR
  • Biopsy proven JXG, ECD, RDD, histiocytic sarcoma, or other histiocytic lesion (newly diagnosed or relapsed/refractory disease) with evaluable active disease.
  • Performance Level:
  • Karnofsky ≥ 50% for patients \> 16 years of age and Lansky ≥ 50% for patients ≤ 16 years of age.
  • Adequate Hematologic Function Defined as:
  • ANC ≥ 0.75 x 10\^9/L (unsupported/without growth factor stimulant)
  • Platelet count ≥ 75 x 10\^9/L (unsupported/without transfusion within the past 7 days).
  • +17 more criteria

You may not qualify if:

  • \- Prior and Concomitant Use of Drugs with CYP3A4 inducing/inhibiting activity: Patient taking strong inducers or inhibitors of CYP3A4 within 14 days prior to study enrollment, including but not limited to the following: erythromycin, clarithromycin, ketoconazole, azithromycin, itraconazole, grapefruit juice or St. John's wort.
  • Prior Therapy Restrictions Completion of previous chemotherapy, immunotherapy, radiotherapy, or targeted therapy for LCH (or other histiocytic disorder) at least 28 days (except where specified below) prior to study enrollment, with resolution of all associated toxicity to ≤ Grade 1 prior to study enrollment (exception for alopecia and ototoxicity which do not need to be resolved ≤ Grade 1). Patients must have fully recovered from the acute toxic effects of all prior anti-cancer therapy and must meet the following minimum duration from prior anti-cancer directed therapy prior to enrollment. If after the required timeframe, the laboratory eligibility criteria are met, the patient is considered to have recovered adequately. See below for specific consideration of prednisone and corticosteroids prior to enrollment.
  • Radiation therapy within the 14 days prior to enrollment.
  • Any prior treatment with Cobimetinib.
  • Treatment with a long-acting hematopoietic growth factor within 14 days prior to initiation of study drug or a short-acting hematopoietic growth factor within 7 days prior to enrollment.
  • Treatment with hormonal therapy (except hormone replacement therapy or oral contraceptives), immunotherapy, biologic therapy, investigational therapy, or herbal cancer therapy within 28 days or \< 5 half-lives, whichever is longer, prior to study enrollment.
  • Treatment with high-dose chemotherapy and stem-cell rescue (autologous stem cell transplant) or allogeneic stem cell transplant within 90 days prior to enrollment. Anti-GVHD agents post-transplant: Patients who are receiving cyclosporine, tacrolimus or other agents to prevent graft-versus-host disease post bone marrow transplant are not eligible for this trial.
  • For patients with brain tumors (intracranial masses), use of anticoagulants within 7 days prior to enrollment.
  • Corticosteroid therapy less than or equal to 0.5 mg/kg/day averaged during the 28 days prior to study enrollment is permissible. Patients receiving corticosteroids must be on a stable or decreasing dose for 14 days prior to enrollment and discontinue once study treatment has started.
  • Patient has received treatment with investigational therapy within 4 weeks prior to initiation of study drug.
  • Patients taking anticoagulants or have a pre-existing bleeding disorder unrelated to histiocytic disease.
  • Other active malignancy or history of secondary malignancy.
  • Refractory nausea and vomiting, malabsorption, external biliary shunt
  • Infection: Patients who have a known active infection (excluding documented fungal infection of the nail beds) within 28 days prior to enrollment that has not completely resolved.
  • Major surgical procedure or significant traumatic injury within 28 days prior to enrollment, or anticipation of need for major surgical procedure during the course of the study. Placement of a vascular access device or minor surgery is permitted within fourteen (14) days prior to study enrollment (provided that the wound has healed).
  • +14 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (12)

Phoenix Children's Hospital

Phoenix, Arizona, 85016, United States

RECRUITING

Arkansas Children's Hospital

Little Rock, Arkansas, 72202, United States

RECRUITING

Children's Hospital of Orange County

Orange, California, 92868, United States

RECRUITING

UCSF Benioff Children's Hospital

San Francisco, California, 94158, United States

RECRUITING

Children's National Hospital

Washington D.C., District of Columbia, 20010, United States

RECRUITING

John Hopkins University School of Medicine

Baltimore, Maryland, 21287, United States

RECRUITING

Dana Farber Cancer Institute, Boston Children's

Boston, Massachusetts, 02215, United States

RECRUITING

Memorial Sloan Kettering Cancer Center

New York, New York, 10065, United States

RECRUITING

NACHO Consortium

Memphis, Tennessee, 38105, United States

NOT YET RECRUITING

Children's Medical Center- UTSW

Dallas, Texas, 75235, United States

RECRUITING

Texas Children's Hospital

Houston, Texas, 77030, United States

RECRUITING

University of Wisconsin-American Family Children's Hospital

Madison, Wisconsin, 53792, United States

TERMINATED

MeSH Terms

Conditions

Histiocytosis, Langerhans-CellXanthogranuloma, JuvenileErdheim-Chester DiseaseHistiocytosis, SinusHistiocytic SarcomaHistiocytic Disorders, Malignant

Interventions

cobimetinib

Condition Hierarchy (Ancestors)

Lung Diseases, InterstitialLung DiseasesRespiratory Tract DiseasesHistiocytosisLymphatic DiseasesHemic and Lymphatic DiseasesHistiocytosis, Non-Langerhans-CellSkin DiseasesSkin and Connective Tissue DiseasesNeoplasms by Histologic TypeNeoplasms

Study Officials

  • Carl E Allen, MD, PhD

    Baylor College of Medicine

    STUDY CHAIR

Central Study Contacts

Carl E Allen, MD, PhD

CONTACT

Olive Eckstein, MD

CONTACT

Study Design

Study Type
interventional
Phase
phase 2
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Model Details: Participants are assigned to one of 4 groups in parallel for the duration of the study.
Sponsor Type
OTHER
Responsible Party
SPONSOR INVESTIGATOR
PI Title
Associate Professor

Study Record Dates

First Submitted

August 10, 2019

First Posted

September 6, 2019

Study Start

April 19, 2021

Primary Completion

December 1, 2025

Study Completion (Estimated)

December 1, 2029

Last Updated

September 18, 2025

Record last verified: 2025-09

Locations