NCT03785249

Brief Summary

This study will evaluate the safety, tolerability, drug levels, molecular effects, and clinical activity of MRTX849 (adagrasib) in patients with advanced solid tumors that have a KRAS G12C mutation.

Trial Health

78
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
731

participants targeted

Target at P75+ for phase_1

Timeline
8mo left

Started Jan 2019

Longer than P75 for phase_1

Geographic Reach
2 countries

222 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress92%
Jan 2019Dec 2026

First Submitted

Initial submission to the registry

December 18, 2018

Completed
6 days until next milestone

First Posted

Study publicly available on registry

December 24, 2018

Completed
22 days until next milestone

Study Start

First participant enrolled

January 15, 2019

Completed
8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 31, 2026

Expected
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

December 31, 2026

Last Updated

September 30, 2025

Status Verified

September 1, 2025

Enrollment Period

8 years

First QC Date

December 18, 2018

Last Update Submit

September 29, 2025

Conditions

Keywords

KRASNSCLCColorectal CancerColon CancerMetastatic CancerPancreatic CancerAdagrasibSTK11 mutationKRAS G12C

Outcome Measures

Primary Outcomes (3)

  • Characterize the safety of MRTX849 in patients having advanced solid tumor malignancies with KRAS G12C mutation

    Number of participants with treatment related adverse events

    20 months

  • Evaluate the pharmacokinetics of MRTX849

    Blood plasma concentration

    20 months

  • Evaluate clinical activity/efficacy of MRTX849

    Objective response rate in accordance with Response Evaluation Criteria in Solid Tumors (RECIST)

    20 months

Secondary Outcomes (4)

  • Establish maximum tolerated dose

    12 months

  • Characterize safety and tolerability of MRTX849 in combination with selected therapeutic agents

    12 months

  • Evaluate the pharmacokinetics of new MRTX849 oral formulations

    6 months

  • Evaluate the pharmacokinetics of MRTX849 administered with food

    6 months

Study Arms (9)

Phase 1 Dose Exploration

EXPERIMENTAL

Dose escalation of MRTX849 to determine maximum tolerated dose

Drug: MRTX849

Phase 1b Expansion

EXPERIMENTAL

Expansion cohort to ensure sufficient safety experience, pharmacokinetic information, and early evidence of clinical activity of MRTX849 to recommend Phase 2 regimens

Drug: MRTX849

Phase 2

EXPERIMENTAL

Separate cohorts of patients stratified by histological diagnosis, prior treatment history or co-mutation status (e.g., STK11) for evaluation of clinical activity of MRTX849

Drug: MRTX849

Pilot Phase 1b Combination with Pembrolizumab

EXPERIMENTAL

Phase 1 evaluation of the safety, tolerability, PK and clinical activity of MRTX849 in combination with pembrolizumab in patients with NSCLC

Drug: MRTX849Drug: Pembrolizumab

Pilot Phase 1b Combination with Cetuximab

EXPERIMENTAL

Phase 1 evaluation of the safety, tolerability, PK and clinical activity of MRTX849 in combination with cetuximab in patients with CRC

Drug: MRTX849Drug: Cetuximab

Pilot Phase 1b Combination with Afatinib

EXPERIMENTAL

Phase 1 evaluation of the safety, tolerability, PK and clinical activity of MRTX849 in combination with afatinib in patients with NSCLC

Drug: MRTX849Drug: Afatinib

Phase 2 Combination with Cetuximab

EXPERIMENTAL

Phase 2 evaluation of the clinical activity of MRTX849 in combination with cetuximab in patients with CRC

Drug: MRTX849Drug: Cetuximab

Pilot Phase 1b Combination with Cetuximab in NSCLC

EXPERIMENTAL

Phase 1 evaluation of the safety, tolerability, PK and clinical activity of MRTX849 in combination with cetuximab in patients with NSCLC

Drug: MRTX849Drug: Cetuximab

Pilot Phase 1b Combination with Cetuximab in PDAC

EXPERIMENTAL

Phase 1 evaluation of the safety, tolerability, PK and clinical activity of MRTX849 in combination with cetuximab in patients with pancreatic adenocarcinoma (PDAC)

Drug: MRTX849Drug: Cetuximab

Interventions

MRTX849 will be administered orally once or twice daily in a continuous regimen

Phase 1 Dose ExplorationPhase 1b ExpansionPhase 2Phase 2 Combination with CetuximabPilot Phase 1b Combination with AfatinibPilot Phase 1b Combination with CetuximabPilot Phase 1b Combination with Cetuximab in NSCLCPilot Phase 1b Combination with Cetuximab in PDACPilot Phase 1b Combination with Pembrolizumab

Pembrolizumab is administered as an intravenous infusion once every 3 weeks

Pilot Phase 1b Combination with Pembrolizumab

Cetuximab will be administered as an intravenous infusion once per week or once every 2 weeks

Phase 2 Combination with CetuximabPilot Phase 1b Combination with CetuximabPilot Phase 1b Combination with Cetuximab in NSCLCPilot Phase 1b Combination with Cetuximab in PDAC

Afatinib will be administered orally once a day in a continuous regimen

Pilot Phase 1b Combination with Afatinib

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Histologically confirmed diagnosis of a solid tumor malignancy with KRAS G12C mutation
  • Unresectable or metastatic disease
  • Standard treatment is not available or patient declines; first-line treatment for NSCLC for certain cohorts
  • Adequate organ function

You may not qualify if:

  • History of intestinal disease or major gastric surgery or inability to swallow oral medications
  • Other active cancer

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (222)

Local Institution - 001-826

Birmingham, Alabama, 35294, United States

Location

Local Institution - 001-965

Anchorage, Alaska, 99508, United States

Location

Local Institution - 001-821

Phoenix, Arizona, 85054, United States

Location

Local Institution - 001-873-A

Tucson, Arizona, 85704, United States

Location

Local Institution - 001-873

Tucson, Arizona, 85704, United States

Location

Local Institution - 001-840-B

Bellflower, California, 90706, United States

Location

Local Institution - 001-834

Beverly Hills, California, 90211, United States

Location

Local Institution - 001-843

Duarte, California, 91010, United States

Location

Local Institution - 001-850-K

Dublin, California, 94568, United States

Location

Local Institution - 001-851

Fullerton, California, 92835, United States

Location

Local Institution - 001-840-C

Harbor City, California, 90710, United States

Location

Local Institution - 001-805

La Jolla, California, 92093, United States

Location

Local Institution - 001-779

Los Alamitos, California, 90720, United States

Location

Local Institution - 001-840

Los Angeles, California, 90027, United States

Location

Local Institution - 001-578

Los Angeles, California, 90067, United States

Location

Local Institution - 001-847

Newport Beach, California, 92663, United States

Location

Local Institution - 001-850-B

Oakland, California, 94611, United States

Location

Local Institution - 001-803

Orange, California, 92868, United States

Location

Local Institution - 001-850-C

Roseville, California, 95661, United States

Location

Local Institution - 001-850-J

Sacramento, California, 95814, United States

Location

Local Institution - 001-850-D

Sacramento, California, 95825, United States

Location

Local Institution - 001-845

San Diego, California, 92111, United States

Location

Local Institution - 001-840-A

San Diego, California, 92120, United States

Location

Local Institution - 001-850-H

San Francisco, California, 94080, United States

Location

Local Institution - 001-850-E

San Francisco, California, 94115, United States

Location

Local Institution - 001-850-F

San Jose, California, 95119, United States

Location

Local Institution - 001-850-A

San Leandro, California, 94577, United States

Location

Local Institution - 001-884

Santa Barbara, California, 93105, United States

Location

Local Institution - 001-850-I

Santa Clara, California, 95051, United States

Location

Local Institution - 001-884-A

Solvang, California, 93463, United States

Location

Local Institution - 001-850

Vallejo, California, 94589, United States

Location

Local Institution - 001-850-G

Walnut Creek, California, 94596, United States

Location

Local Institution - 001-872

Aurora, Colorado, 80012, United States

Location

Local Institution - 001-810

Aurora, Colorado, 80045, United States

Location

Local Institution - 001-872-H

Boulder, Colorado, 80303, United States

Location

Local Institution - 001-872-E

Colorado Springs, Colorado, 80907, United States

Location

Local Institution - 001-872-L

Colorado Springs, Colorado, 80920, United States

Location

Local Institution - 001-872-B

Denver, Colorado, 80218, United States

Location

Local Institution - 001-951 - A

Denver, Colorado, 80218, United States

Location

Local Institution - 001-951 - B

Denver, Colorado, 80218, United States

Location

Local Institution - 001-846

Grand Junction, Colorado, 81501, United States

Location

Local Institution - 001-951

Lafayette, Colorado, 80026, United States

Location

Local Institution - 001-872-A

Lakewood, Colorado, 80228, United States

Location

Local Institution - 001-872-D

Littleton, Colorado, 80218, United States

Location

Local Institution - 001-872-K

Lone Tree, Colorado, 80124, United States

Location

Local Institution - 001-872-C

Longmont, Colorado, 80501, United States

Location

Local Institution - 001-872-J

Parker, Colorado, 80138, United States

Location

Local Institution - 001-872-F

Pueblo, Colorado, 81008, United States

Location

Local Institution - 001-872-G

Pueblo, Colorado, 81008, United States

Location

Local Institution - 001-872-I

Thornton, Colorado, 80260, United States

Location

Local Institution - 001-816

New Haven, Connecticut, 06510, United States

Location

Local Institution - 001-871

Newark, Delaware, 19713-2055, United States

Location

Local Institution - 001-929i

Altamonte Springs, Florida, 32701, United States

Location

Local Institution - 001-839

Boca Raton, Florida, 33432, United States

Location

Local Institution - 001-922A

Bonita Springs, Florida, 34135, United States

Location

Local Institution - 001-922D

Bradenton, Florida, 34211, United States

Location

Local Institution - 001-929c

Brandon, Florida, 33511, United States

Location

Local Institution - 001-922E

Cape Coral, Florida, 33909, United States

Location

Local Institution - 001-929g

Clearwater, Florida, 33761, United States

Location

Local Institution - 001-926b

Daytona Beach, Florida, 32117, United States

Location

Local Institution - 001-922

Fort Myers, Florida, 33901, United States

Location

Local Institution - 001-922B

Fort Myers, Florida, 33905, United States

Location

Local Institution - 001-922C

Fort Myers, Florida, 33908, United States

Location

Local Institution - 001-929b

Gainesville, Florida, 32605, United States

Location

Local Institution - 001-829

Jacksonville, Florida, 32224, United States

Location

Local Institution - 001-929m

Lady Lake, Florida, 32159, United States

Location

Local Institution - 001-929e

Largo, Florida, 33770, United States

Location

Local Institution - 001-929n

Lecanto, Florida, 34461, United States

Location

Local Institution - 001-870

Miami, Florida, 33176, United States

Location

Local Institution - 001-825

Miami Beach, Florida, 33140, United States

Location

Local Institution - 001-922F

Naples, Florida, 34102, United States

Location

Local Institution - 001-922G

Naples, Florida, 34102, United States

Location

Local Institution - 001-538

Ocala, Florida, 34474, United States

Location

Local Institution - 001-929p

Ocala, Florida, 34474, United States

Location

Local Institution - 001-914

Orange City, Florida, 32763, United States

Location

Local Institution - 001-929j

Orange City, Florida, 32763, United States

Location

Local Institution - 001-929l

Orlando, Florida, 32806, United States

Location

Local Institution - 001-877

Pensacola, Florida, 32503, United States

Location

Local Institution - 001-922H

Port Charlotte, Florida, 33980, United States

Location

Local Institution - 001-922I

Sarasota, Florida, 34232, United States

Location

Local Institution - 001-922J

Sarasota, Florida, 34236, United States

Location

Local Institution - 001-929h

Spring Hill, Florida, 34608, United States

Location

Local Institution - 001-929a

St. Petersburg, Florida, 33705, United States

Location

Local Institution - 001-929

St. Petersburg, Florida, 33705, United States

Location

Local Institution - 001-926d

Stuart, Florida, 34994, United States

Location

Local Institution - 001-929d

Tampa, Florida, 33607, United States

Location

Local Institution - 001-929k

Tavares, Florida, 32778, United States

Location

Local Institution - 001-929f

Trinity, Florida, 34655, United States

Location

Local Institution - 001-922K

Venice, Florida, 34285, United States

Location

Local Institution - 001-922L

Venice, Florida, 34292, United States

Location

Local Institution - 001-926c

Vero Beach, Florida, 32960, United States

Location

Local Institution - 001-926a

Wellington, Florida, 33414, United States

Location

Local Institution - 001-926

West Palm Beach, Florida, 33401, United States

Location

Local Institution - 001-929o

Winter Park, Florida, 32789, United States

Location

Local Institution - 001-967

Athens, Georgia, 30607, United States

Location

Local Institution - 001-835-C

Austell, Georgia, 30106, United States

Location

Local Institution - 001-835-E

Austell, Georgia, 30106, United States

Location

Local Institution - 001-835-D

Carrollton, Georgia, 30117, United States

Location

Local Institution - 001-835-F

Carrollton, Georgia, 30117, United States

Location

Local Institution - 001-835-A

Cartersville, Georgia, 30121, United States

Location

Local Institution - 001-835-B

Douglasville, Georgia, 30134, United States

Location

Local Institution - 001-835

Marietta, Georgia, 30060, United States

Location

Local Institution - 001-862

Chicago Ridge, Illinois, 60415, United States

Location

Local Institution - 001-883

Niles, Illinois, 60714, United States

Location

Local Institution - 001-781

South Bend, Indiana, 46601, United States

Location

Local Institution - 001-831

Iowa City, Iowa, 52242, United States

Location

Local Institution - 001-820

Westwood, Kansas, 66205, United States

Location

Local Institution - 001-844

Lexington, Kentucky, 40536, United States

Location

Local Institution - 001-920

Baton Rouge, Louisiana, 70809, United States

Location

Local Institution - 001-827

Biddeford, Maine, 04005, United States

Location

Local Institution - 001-881-B

Brandywine, Maryland, 20613, United States

Location

Local Institution - 001-881

Columbia, Maryland, 21044, United States

Location

Local Institution - 001-881-A

Silver Spring, Maryland, 20904, United States

Location

Local Institution - 001-808

Boston, Massachusetts, 02215, United States

Location

Local Institution - 001-842

Detroit, Michigan, 48201, United States

Location

Local Institution - 001-811

Detroit, Michigan, 48202, United States

Location

Local Institution - 001-842-A

Farmington Hills, Michigan, 48334, United States

Location

Local Institution - 001-838-F

Coon Rapids, Minnesota, 55433, United States

Location

Local Institution - 001-838-E

Edina, Minnesota, 55435, United States

Location

Local Institution - 001-875 - D

Edina, Minnesota, 55435, United States

Location

Local Institution - 001-838-D

Maplewood, Minnesota, 55109, United States

Location

Local Institution - 001-875 - A

Maplewood, Minnesota, 55109, United States

Location

Local Institution - 001-838-C

Minneapolis, Minnesota, 55404, United States

Location

Local Institution - 001-875

Minneapolis, Minnesota, 55404, United States

Location

Local Institution - 001-838-G

Minneapolis, Minnesota, 55415, United States

Location

Local Institution - 001-822-A

Minneapolis, Minnesota, 55455, United States

Location

Local Institution - 001-822

Minneapolis, Minnesota, 55455, United States

Location

Local Institution - 001-830

Rochester, Minnesota, 55905, United States

Location

Local Institution - 001-838

Saint Louis Park, Minnesota, 55416, United States

Location

Local Institution - 001-838-B

Saint Louis Park, Minnesota, 55426-5000, United States

Location

Local Institution - 001-838-A

Saint Paul, Minnesota, 55101, United States

Location

Local Institution - 001-875 - B

Saint Paul, Minnesota, 55102, United States

Location

Local Institution - 001-875 - C

Woodbury, Minnesota, 55125, United States

Location

Local Institution - 001-952

Bolivar, Missouri, 65613, United States

Location

Local Institution - 001-950

Jefferson City, Missouri, 65109, United States

Location

Local Institution - 001-841

Billings, Montana, 59102, United States

Location

Local Institution - 001-544B

Omaha, Nebraska, 68105-1850, United States

Location

Local Institution - 001-959

Omaha, Nebraska, 68114, United States

Location

Local Institution - 001-544A

Omaha, Nebraska, 68118, United States

Location

Local Institution - 001-544

Omaha, Nebraska, 68198, United States

Location

Local Institution - 001-860A

Henderson, Nevada, 89052, United States

Location

Local Institution - 001-860C

Henderson, Nevada, 89052, United States

Location

Local Institution - 001-860B

Henderson, Nevada, 89074, United States

Location

Local Institution - 001-860

Henderson, Nevada, 89074, United States

Location

Local Institution - 001-860E

Las Vegas, Nevada, 89128, United States

Location

Local Institution - 001-860D

Las Vegas, Nevada, 89144, United States

Location

Local Institution - 001-860F

Las Vegas, Nevada, 89148, United States

Location

Local Institution - 001-861

Albany, New York, 12206, United States

Location

Local Institution - 001-815

Buffalo, New York, 14203, United States

Location

Local Institution - 001-813

New York, New York, 10016, United States

Location

Local Institution - 001-806

New York, New York, 10065, United States

Location

Local Institution - 001-812

Chapel Hill, North Carolina, 27514, United States

Location

Local Institution - 001-971

Pinehurst, North Carolina, 28374, United States

Location

Local Institution - 001-966

Cincinnati, Ohio, 45219, United States

Location

Local Institution - 001-823

Cincinnati, Ohio, 45267, United States

Location

Local Institution - 001-818

Cleveland, Ohio, 44195, United States

Location

Local Institution - 001-833 - H

Columbus, Ohio, 43201, United States

Location

Local Institution - 001-833 - C

Columbus, Ohio, 43203, United States

Location

Local Institution - 001-833 - J

Columbus, Ohio, 43203, United States

Location

Local Institution - 001-833 - A

Columbus, Ohio, 43210, United States

Location

Local Institution - 001-833 - F

Columbus, Ohio, 43210, United States

Location

Local Institution - 001-833

Columbus, Ohio, 43210, United States

Location

Local Institution - 001-833 - D

Columbus, Ohio, 43212, United States

Location

Local Institution - 001-833 - I

Columbus, Ohio, 43212, United States

Location

Local Institution - 001-930

Columbus, Ohio, 43219, United States

Location

Local Institution - 001-833 - B

Columbus, Ohio, 43221, United States

Location

Local Institution - 001-833 - G

Columbus, Ohio, 43221, United States

Location

Local Institution - 001-833 - E

Gahanna, Ohio, 43230, United States

Location

Local Institution - 001-836-A

Kettering, Ohio, 45429, United States

Location

Local Institution - 001-836

Kettering, Ohio, 45429, United States

Location

Local Institution - 001-600

Lawton, Oklahoma, 73505, United States

Location

Local Institution - 001-584

Tulsa, Oklahoma, 74146, United States

Location

Local Institution - 001-586-A

Bend, Oregon, 97701, United States

Location

Local Institution - 001-586

Bend, Oregon, 97701, United States

Location

Local Institution - 001-889

Eugene, Oregon, 97401, United States

Location

Local Institution - 001-837

Allentown, Pennsylvania, 18103, United States

Location

Local Institution - 001-837-A

Bethlehem, Pennsylvania, 18017, United States

Location

Local Institution - 001-817

Hershey, Pennsylvania, 17033-0850, United States

Location

Local Institution - 001-783

Media, Pennsylvania, 19063, United States

Location

Local Institution - 001-887

Charleston, South Carolina, 29414, United States

Location

Local Institution - 001-819

Charleston, South Carolina, 29425, United States

Location

Local Institution - 001-801-G

Gallatin, Tennessee, 37066, United States

Location

Local Institution - 001-801-A

Hendersonville, Tennessee, 37075, United States

Location

Local Institution - 001-801-D

Hermitage, Tennessee, 37076, United States

Location

Local Institution - 001-801-F

Murfreesboro, Tennessee, 37129, United States

Location

Local Institution - 001-801-B

Nashville, Tennessee, 37203, United States

Location

Local Institution - 001-801

Nashville, Tennessee, 37203, United States

Location

Local Institution - 001-801-E

Nashville, Tennessee, 37207, United States

Location

Local Institution - 001-801-C

Nashville, Tennessee, 37211, United States

Location

Local Institution - 001-888-B

Arlington, Texas, 76012, United States

Location

Local Institution - 001-888

Arlington, Texas, 76012, United States

Location

Local Institution - 001-880

Austin, Texas, 78731, United States

Location

Local Institution - 001-848a

Conroe, Texas, 77384, United States

Location

Local Institution - 001-809

Dallas, Texas, 75230, United States

Location

Local Institution - 001-886

Dallas, Texas, 75231, United States

Location

Local Institution - 001-879

Dallas, Texas, 75246, United States

Location

Local Institution - 001-785

Denison, Texas, 75020, United States

Location

Local Institution - 001-876

Fort Worth, Texas, 76104, United States

Location

Local Institution - 001-848

Houston, Texas, 77030, United States

Location

Local Institution - 001-969

Houston, Texas, 77030, United States

Location

Local Institution - 001-935A

Houston, Texas, 77090, United States

Location

Local Institution - 001-999

Irving, Texas, 75063, United States

Location

Local Institution - 001-935D

Kingwood, Texas, 77339, United States

Location

Local Institution - 001-935

Kingwood, Texas, 77339, United States

Location

Local Institution - 001-554

Midland, Texas, 79701, United States

Location

Local Institution - 001-802

San Antonio, Texas, 78229, United States

Location

Local Institution - 001-935B

Shenandoah, Texas, 77380, United States

Location

Local Institution - 001-935C

Spring, Texas, 77389, United States

Location

Local Institution - 001-874

Sugar Land, Texas, 77479, United States

Location

Local Institution - 001-935E

Tomball, Texas, 77375, United States

Location

Local Institution - 001-878

Tyler, Texas, 75702, United States

Location

Local Institution - 001-890

Waco, Texas, 76712, United States

Location

Local Institution - 001-814

Fairfax, Virginia, 22031, United States

Location

Local Institution - 001-597

Fredericksburg, Virginia, 24408, United States

Location

Local Institution - 001-882

Newport News, Virginia, 23606, United States

Location

Local Institution - 001-882-A

Norfolk, Virginia, 23502, United States

Location

Local Institution - 001-890-A

Norfolk, Virginia, 23502, United States

Location

Local Institution - 001-968

Richmond, Virginia, 23229, United States

Location

Local Institution - 001-824

Seattle, Washington, 98109, United States

Location

Local Institution - 001-885

Vancouver, Washington, 98684, United States

Location

Local Institution - 001-804

Madison, Wisconsin, 53792, United States

Location

Local Institution - 001-900

San Juan, PR, 00935, Puerto Rico

Location

Related Publications (7)

  • Negrao MV, Spira AI, Heist RS, Janne PA, Pacheco JM, Weiss J, Gadgeel SM, Velastegui K, Yang W, Der-Torossian H, Christensen JG, Sabari JK. Intracranial Efficacy of Adagrasib in Patients From the KRYSTAL-1 Trial With KRASG12C-Mutated Non-Small-Cell Lung Cancer Who Have Untreated CNS Metastases. J Clin Oncol. 2023 Oct 1;41(28):4472-4477. doi: 10.1200/JCO.23.00046. Epub 2023 Jun 16.

  • Bekaii-Saab TS, Yaeger R, Spira AI, Pelster MS, Sabari JK, Hafez N, Barve M, Velastegui K, Yan X, Shetty A, Der-Torossian H, Pant S. Adagrasib in Advanced Solid Tumors Harboring a KRASG12C Mutation. J Clin Oncol. 2023 Sep 1;41(25):4097-4106. doi: 10.1200/JCO.23.00434. Epub 2023 Apr 26.

  • Yaeger R, Weiss J, Pelster MS, Spira AI, Barve M, Ou SI, Leal TA, Bekaii-Saab TS, Paweletz CP, Heavey GA, Christensen JG, Velastegui K, Kheoh T, Der-Torossian H, Klempner SJ. Adagrasib with or without Cetuximab in Colorectal Cancer with Mutated KRAS G12C. N Engl J Med. 2023 Jan 5;388(1):44-54. doi: 10.1056/NEJMoa2212419. Epub 2022 Dec 21.

  • Janne PA, Riely GJ, Gadgeel SM, Heist RS, Ou SI, Pacheco JM, Johnson ML, Sabari JK, Leventakos K, Yau E, Bazhenova L, Negrao MV, Pennell NA, Zhang J, Anderes K, Der-Torossian H, Kheoh T, Velastegui K, Yan X, Christensen JG, Chao RC, Spira AI. Adagrasib in Non-Small-Cell Lung Cancer Harboring a KRASG12C Mutation. N Engl J Med. 2022 Jul 14;387(2):120-131. doi: 10.1056/NEJMoa2204619. Epub 2022 Jun 3.

  • Sabari JK, Velcheti V, Shimizu K, Strickland MR, Heist RS, Singh M, Nayyar N, Giobbie-Hurder A, Digumarthy SR, Gainor JF, Rajan AP, Nieblas-Bedolla E, Burns AC, Hallin J, Olson P, Christensen JG, Kurz SC, Brastianos PK, Wakimoto H. Activity of Adagrasib (MRTX849) in Brain Metastases: Preclinical Models and Clinical Data from Patients with KRASG12C-Mutant Non-Small Cell Lung Cancer. Clin Cancer Res. 2022 Aug 2;28(15):3318-3328. doi: 10.1158/1078-0432.CCR-22-0383.

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Related Links

MeSH Terms

Conditions

Neoplasm MetastasisNeoplasmsColorectal NeoplasmsColonic NeoplasmsPancreatic Neoplasms

Interventions

adagrasibpembrolizumabCetuximabAfatinib

Condition Hierarchy (Ancestors)

Neoplastic ProcessesPathologic ProcessesPathological Conditions, Signs and SymptomsIntestinal NeoplasmsGastrointestinal NeoplasmsDigestive System NeoplasmsNeoplasms by SiteDigestive System DiseasesGastrointestinal DiseasesColonic DiseasesIntestinal DiseasesRectal DiseasesEndocrine Gland NeoplasmsPancreatic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

Antibodies, Monoclonal, HumanizedAntibodies, MonoclonalAntibodiesImmunoglobulinsImmunoproteinsBlood ProteinsProteinsAmino Acids, Peptides, and ProteinsSerum GlobulinsGlobulinsAmidesOrganic ChemicalsQuinazolinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic Compounds

Study Officials

  • Bristol-Myers Squibb

    Bristol-Myers Squibb

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR
Expanded Access
Yes

Study Record Dates

First Submitted

December 18, 2018

First Posted

December 24, 2018

Study Start

January 15, 2019

Primary Completion (Estimated)

December 31, 2026

Study Completion (Estimated)

December 31, 2026

Last Updated

September 30, 2025

Record last verified: 2025-09

Data Sharing

IPD Sharing
Will not share

Locations