NCT02996500

Brief Summary

This is a Phase 2, multicenter, randomized, double blind, double dummy, placebo and active-controlled, parallel group study to assess the efficacy and safety of PF 06650833 at Week 12 in subjects with moderate-severe, active, RA who have had an inadequate response to MTX. PF-06650833 or matching placebo tablets will be administered orally QD under fasting conditions, and tofacitinib or matching tofacitinib placebo tablets will be administered orally BID for 12 weeks in a blinded fashion.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
269

participants targeted

Target at P75+ for phase_2 rheumatoid-arthritis

Timeline
Completed

Started Nov 2016

Geographic Reach
19 countries

103 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 13, 2016

Completed
28 days until next milestone

Study Start

First participant enrolled

November 10, 2016

Completed
1 month until next milestone

First Posted

Study publicly available on registry

December 19, 2016

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 15, 2018

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

August 15, 2018

Completed
1.5 years until next milestone

Results Posted

Study results publicly available

February 27, 2020

Completed
Last Updated

February 27, 2020

Status Verified

February 1, 2020

Enrollment Period

1.8 years

First QC Date

October 13, 2016

Results QC Date

July 29, 2019

Last Update Submit

February 12, 2020

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline in the Simplified Disease Activity Index (SDAI) at Week 12

    The SDAI is a continuous composite measure derived from components of the American College of Rheumatology (ACR) Core Dataset.The SDAI was calculated using the following formula: SDAI = Tender / Painful Joint Count(TJC) (using 28 joints) + Swollen Joint Count (SJC) (using 28 joints) + Patient Global Assessment of Arthritis (PtGA) (0-10 cm scale) + Physician's Global Assessment of Arthritis (PhGA) (0-10 cm scale) + high sensitivity C-reactive protein (hsCRP) (mg/dL). SDAI total score= 0-86. SDAI \<=3.3 indicates disease remission, \>3.4 to 11 = low disease activity, \>11 to 26 = moderate disease activity, and \>26 = high disease activity. The primary analysis utilized a Bayesian ANCOVA model with an informative placebo prior distribution with borrowing from tofacitinib historical placebo data. The confidence interval was credible interval in this statistical analysis. The efficacy endpoint for the tofatinicib arm was an exploratory endpoint and neither primary nor secondary endpoints.

    Baseline and Week 12

Secondary Outcomes (33)

  • Change From Baseline in SDAI at Weeks 4 and 8

    Baseline, Weeks 4 and 8

  • Percentage of Participants With SDAI Low Disease Activity Score (LDAS) (SDAI <=11) at 4, 8, and 12 Weeks

    Weeks 4, 8 and 12

  • Percentage of Participants With SDAI Remission (SDAI <=3.3) at 4, 8, and 12 Weeks

    Weeks 4, 8 and 12

  • Percentage of Participants With Disease Activity Score-28 (4 Components Based on Erythrocyte Sedimentation Rate) (DAS28-4 [ESR]) LDAS (DAS28 <3.2) at 4, 8, and 12 Weeks

    Weeks 4, 8 and 12

  • Percentage of Participants With DAS28-3 (ESR) LDAS (DAS28 <3.2) at 4, 8, and 12 Weeks

    Weeks 4, 8 and 12

  • +28 more secondary outcomes

Study Arms (6)

Arm 1: 20 mg QD

EXPERIMENTAL

PF-06650833 , 20 mg QD

Drug: PF-06650833

Arm 2: 60 mg QD

EXPERIMENTAL

PF-06650833, 60 mg QD

Drug: PF-06650833

Arm 3: 200 mg QD

EXPERIMENTAL

Pf-06650833, 200 mg QD

Drug: PF-06650833

Arm 4: 400 mg QD

EXPERIMENTAL

PF-06650833, 400 mg QD

Drug: PF-06650833

Placebo

PLACEBO COMPARATOR

Placebo, 0 mg BID

Drug: Placebo

Arm 5: Tofacitinib

ACTIVE COMPARATOR

Tofacitinib 5 mg BID

Drug: Tofacitinib

Interventions

Investigational

Arm 1: 20 mg QDArm 2: 60 mg QDArm 3: 200 mg QDArm 4: 400 mg QD

Placebo

Placebo

Investigational

Also known as: Xeljanz
Arm 5: Tofacitinib

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Male and female (including WOCBP) subjects between the ages of 18 and 75 years, inclusive.
  • Diagnosis of RA and meeting the 2010 American College of Rheumatology (ACR)/European League Against Rheumatism (EULAR) classification criteria for RA with a Total Score ≥6/10.
  • The subject has active disease at both Screening and Baseline, as defined by both:
  • joints tender or painful on motion, AND
  • joints swollen; and fulfills 1 of the following 2 criteria at Screening:
  • High sensitivity C reactive protein (hsCRP) \>7 mg/L at screening
  • Erythrocyte sedimentation rate (ESR) (Westergren method) \>28 mm/hr;
  • Meets Class I, II or III of the ACR 1991 Revised Criteria for Global Functional Status in RA.
  • Subjects must be ACPA positive between screening and randomization.
  • Subjects must have been taking oral MTX for at least 3 months at an adequate dose to determine that the subject had an inadequate response to MTX
  • Up to 50 % of subjects may have received one (and only one) approved TNF-inhibiting biologic agent administered that was inadequately effective and/or not tolerated. The anti-TNF biologic could also have been discontinued due to lack of continued access.

You may not qualify if:

  • Subjects with a known immunodeficiency disorder or a first degree relative with a hereditary immunodeficiency.
  • Subjects with any of the following infections or infections history:
  • Any infection requiring treatment within 2 weeks prior to screening (Visit 1).
  • Any infection requiring hospitalization, parenteral antimicrobial therapy within 60 days, or as otherwise judged to be an opportunistic infection or clinically significant by the investigator, within the past 6 months.
  • Infected joint prosthesis at any time with the prosthesis still in situ.
  • Recurrent (more than one episode) herpes zoster or disseminated (a single episode) herpes zoster or disseminated (a single episode) herpes simplex.
  • Subjects will be screened for HIV. Subjects who test positive for HIV will be excluded from the study.
  • Subjects will be screened for hepatitis B virus infection and will be excluded if positive for hepatitis B surface antigen (HBsAg). Subjects with HBsAg negative testing but who test positive for hepatitis B core antibody (HBcAb) must have further testing for hepatitis B surface antibody (HBsAb). If HBsAb is negative, the subject will be excluded from the study.
  • Subjects with clinically significant active hepatic disease or hepatic impairment by laboratory assessment.
  • Subjects will be screened for hepatitis C virus (HCV Ab). Subjects with positive HCV Ab tests will be reflex tested for HCV ribonucleic acid (HCV RNA). Only subjects with negative HCV Ab or HCV RNA will be allowed to enroll in the study.
  • Evidence of active or latent, untreated or inadequately treated infection with Mycobacterium tuberculosis (TB)
  • Pre-existing chronic autoimmune disease.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (103)

Clinical and Translational Research Center of Alabama, PC

Tuscaloosa, Alabama, 35406, United States

Location

Dory Hardy, PharmD

Tucson, Arizona, 85723, United States

Location

Southern Arizona VA Health care System

Tucson, Arizona, 85723, United States

Location

Robert W. Levin, MD,PA

Clearwater, Florida, 33765, United States

Location

Millennium Research

Ormond Beach, Florida, 32174, United States

Location

Arthritis & Rheumatic Care Center

South Miami, Florida, 33143, United States

Location

Qps-Mra, Llc

South Miami, Florida, 33143, United States

Location

Medical Associates of North Georgia

Canton, Georgia, 30115, United States

Location

Graves Gilbert Clinic

Bowling Green, Kentucky, 42101, United States

Location

Arthritis and Diabetes Clinic, Inc.

Monroe, Louisiana, 71203, United States

Location

Ramesh C Gupta, M.D.

Memphis, Tennessee, 38119, United States

Location

Accurate Clinical Management, LLC

Baytown, Texas, 77521, United States

Location

Accurate Clinical Management, LLC

Houston, Texas, 77004, United States

Location

Accurate Clinical Management, LLC

Houston, Texas, 77084, United States

Location

DM Clinical Research

Tomball, Texas, 77375, United States

Location

Canberra Hospital

Garran, Australian Capital Territory, 2605, Australia

Location

Genesis Research Services

Broadmeadow, New South Wales, 2292, Australia

Location

General Hospital "Prim.dr.Abdulah Nakas"

Sarajevo, Kanton Sarajevo, 71000, Bosnia and Herzegovina

Location

University Clinical Center Republic of Srpska

Banja Luka, Republika Srpska, 78000, Bosnia and Herzegovina

Location

Health Center Gradiska

Gradiška, Republika Srpska, 78400, Bosnia and Herzegovina

Location

UMHAT Kaspela

Plovdiv, 4001, Bulgaria

Location

MHAT Liulin

Sofia, 1336, Bulgaria

Location

UMHAT "Sv.Ivan Rilski", Clinic of rheumatology

Sofia, 1612, Bulgaria

Location

Medical Center Synexus Sofia EOOD

Sofia, 1784, Bulgaria

Location

Specialized Hospital for Active Treatment of Oncology Diseases EAD, Department of Imaging Diagnostic

Sofia, 1784, Bulgaria

Location

Poliklinika K-centar

Zagreb, City of Zagreb, 10000, Croatia

Location

Medicinski centar Kuna&Peric

Zagreb, 10000, Croatia

Location

CCBR Ostrava s.r.o.

Ostrava, 702 00, Czechia

Location

Revmatologicka ambulance

Prague, 140 00, Czechia

Location

Medical Plus s.r.o.

Uherské Hradiště, 68601, Czechia

Location

LTD Israeli-Georgian Medical Research Clinic HELSICORE

Tbilisi, 0112, Georgia

Location

LTD " Diagnostic Service "

Tbilisi, 0159, Georgia

Location

Ltd Institute of Clinical Cardiology

Tbilisi, 0159, Georgia

Location

LTD Unimedi Kakheti

Tbilisi, 0159, Georgia

Location

LTD "MediClubGeorgia"

Tbilisi, 0160, Georgia

Location

Ltd "Medicore"

Tbilisi, 0186, Georgia

Location

Unimedi Kakheti LTD

Telavi, 2200, Georgia

Location

Knappschaftsklinikum Saar GmbH

Püttlingen, 66346, Germany

Location

Revita Reumatologiai Rendelo

Budapest, 1027, Hungary

Location

Pest Megyei Flor Ferenc Korhaz

Kistarcsa, 2143, Hungary

Location

CRU Hungary Ltd.

Miskolc, 3529, Hungary

Location

Szegedi Tudomanyegyetem Szent-Gyorgyi Albert Klinikai Kozpont

Szeged, 6725, Hungary

Location

Csongrad Megyei Dr. Bugyi Istvan Korhaz, Mozgasszervi Rehabilitacios Osztaly

Szentes, 6600, Hungary

Location

VITAL MEDICAL CENTER Orvosi es Fogorvosi Kozpont

Veszprém, 8200, Hungary

Location

Private Practice - Dr. Miguel Cortes Hernandez

Cuernavaca, Morelos, 62290, Mexico

Location

Centro Peninsular de Investigacion Clinica S.C.P

Mérida, Yucatán, 97000, Mexico

Location

Kohler & Milstein Research S.A de C.V

Mérida, Yucatán, 97070, Mexico

Location

Centro de Alta Especialidad en Reumatología e Investigación del Potosi, S.C.

San Luis Potosí City, 78213, Mexico

Location

Szpital Specjalistyczny nr 1 w Bytomiu

Bytom, 41-902, Poland

Location

Synexus Polska Sp. z o.o. Oddzial w Gdansku

Gdansk, 80-382, Poland

Location

Synexus Polska Sp z o.o. Oddzial w Gdyni

Gdynia, 81-537, Poland

Location

McBk S.C.

Grodzisk Mazowiecki, 05-825, Poland

Location

Synexus Polska Sp.Zo.o.

Katowice, 40-040, Poland

Location

Prywatna Praktyka Lekarska Prof. UM Dr hab. Med. Pawel Hrycaj

Poznan, 61-397, Poland

Location

Synexus Polska Sp. z o.o.

Warsaw, 01-192, Poland

Location

Reumatika Centrum Reumatologii NZOZ

Warsaw, 02-691, Poland

Location

Synexus Polska Sp. z o.o. Oddział we Wroclawiu

Wroclaw, 50-381, Poland

Location

Centrul Medical Unirea

Bucharest, 010306, Romania

Location

Med Life

Bucharest, 010719, Romania

Location

Centrul Medical Sana

Bucharest, 011025, Romania

Location

Euroclinic Hospital

Bucharest, 014461, Romania

Location

Spitalul Clinic de Recuperare Iasi

Iași, 700661, Romania

Location

Spitalul Clinic Judetean de Urgenta Tirgu Mures

Târgu Mureş, 540136, Romania

Location

FSBEI HE "Kazan State Medical University" MoH of RF

Kazan', 420064, Russia

Location

FSBEI HE "Kazan State Medical University" MoH of RF

Kazan', 420103, Russia

Location

FSBSI "Scientific Research Institute of Rheumatology n.a. V.A. Nasonova"

Moscow, 115522, Russia

Location

SBHI of Moscow City Clinical Hospital # 1 n.a. N.I. Pirogov of Moscow Healthcare Department

Moscow, 119049, Russia

Location

FSBHI Central Clinical Hospital of Russian Academy of Sciences

Moscow, 119333, Russia

Location

State Budgetary Institution of Ryazan Region "Regional clinical cardiology dispensary"

Ryazan, 390026, Russia

Location

LLC "Sanavita"

Saint Petersburg, 190031, Russia

Location

Saint Petersburg State Budgetary Institution of Health Care "Clinical Rheumatology Hospital #25"

Saint Petersburg, 190068, Russia

Location

LLC "Sanavita"

Saint Petersburg, 195257, Russia

Location

SBHI of VR "Regional Clinical Hospital"

Vladimir, 600023, Russia

Location

Institute of Rheumatology

Belgrade, 11000, Serbia

Location

Military Medical Academy

Belgrade, 11000, Serbia

Location

Institute for Treatment and Rehabilitation "Niska Banja"

Niška Banja, 18205, Serbia

Location

Special Hospital for Rheumatic Diseases Novi Sad

Novi Sad, 21112, Serbia

Location

Reumacentrum s.r.o.

Partizánske, Trenčín Region, 958 01, Slovakia

Location

AAGS s.r.o., Reumatologicka ambulancia

Dunajská Streda, 92901, Slovakia

Location

Nemocnica Kosice-Saca, a.s.1.sukromna nemocnica

Kosice-Saca, 040 15, Slovakia

Location

Neštátna Reumatologická ambulancia

Považská Bystrica, 017 01, Slovakia

Location

REUMEX s.r.o. Reumatologicka ambulancia

Rimavská Sobota, 979 01, Slovakia

Location

Reumatologicka ambulancia, MUDr. Pavol Polak s.r.o.

Žilina, 010 01, Slovakia

Location

Seoul National University hospital

Seoul, 03080, South Korea

Location

Hanyang University Seoul hospital

Seoul, 04763, South Korea

Location

Konkuk University Medical Center

Seoul, 05030, South Korea

Location

The Catholic University of Korea, Seoul St.Mary's Hospital

Seoul, 06591, South Korea

Location

Complejo Hospitalario Universitario de Santiago de Compostela

Santiago de Compostela, A Coruna, 15706, Spain

Location

HM Hospital Nuestra Señora de La Esperanza

Santiago de Compostela, A Coruña, 15705, Spain

Location

Hospital Universitario Cruces

Barakaldo, Vizcaya, 48903, Spain

Location

Hospital Universitario A Coruña

A Coruña, 15006, Spain

Location

Hospital Quironsalud Infanta Luisa

Seville, 41010, Spain

Location

China Medical University Hospital

Taichung, 40447, Taiwan

Location

National Taiwan University Hospital

Taipei, 10043, Taiwan

Location

Taipei Medical University Hospital

Taipei, 110, Taiwan

Location

Komunalnyi likuvalno-profilaktychnyi zaklad "Chernihivska oblasna likarnia",

Chernihiv, 14029, Ukraine

Location

Derzhavna ustanova "Natsionalnyi instytut terapii imeni L.T. Maloi

Kharkiv, 61039, Ukraine

Location

Komunalne nekomertsiine pidpryiemstvo "Konsultatyvno-diahnostychnyi tsentr"

Kyiv, 01103, Ukraine

Location

Medychnyi tsentr tovarystva z obmezhenoiu vidpovidalnistiu "Revmotsentr", m. Kyiv

Kyiv, 04070, Ukraine

Location

Derzhavna ustanova "Instytut herontolohii imeni D.F. Chebotarova

Kyiv, 04114, Ukraine

Location

Poltavska oblasna klinichna likarnia im. M.V. Sklifosovskoho,

Poltava, 36011, Ukraine

Location

Ternopilska universytetska likarnia, revmatolohichne viddilennia, Derzhavnyi vyshchyi navchalnyi

Ternopil, 46002, Ukraine

Location

Vinnytska oblasna klinichna likarnia im. M.I.Pyrohova, revmatolohichne viddilennia

Vinnytsia, 21018, Ukraine

Location

Related Links

MeSH Terms

Conditions

Arthritis, Rheumatoid

Interventions

1-(((2S,3S,4S)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl)methoxy)-7-methoxyisoquinoline-6-carboxamidetofacitinib

Condition Hierarchy (Ancestors)

ArthritisJoint DiseasesMusculoskeletal DiseasesRheumatic DiseasesConnective Tissue DiseasesSkin and Connective Tissue DiseasesAutoimmune DiseasesImmune System Diseases

Results Point of Contact

Title
Pfizer ClinicalTrials.gov Call Center
Organization
Pfizer, Inc.

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 13, 2016

First Posted

December 19, 2016

Study Start

November 10, 2016

Primary Completion

August 15, 2018

Study Completion

August 15, 2018

Last Updated

February 27, 2020

Results First Posted

February 27, 2020

Record last verified: 2020-02

Data Sharing

IPD Sharing
Will share

Pfizer will provide access to individual de-identified participant data and related study documents (e.g. protocol, Statistical Analysis Plan (SAP), Clinical Study Report (CSR)) upon request from qualified researchers, and subject to certain criteria, conditions, and exceptions. Further details on Pfizer's data sharing criteria and process for requesting access can be found at: https://www.pfizer.com/science/clinical\_trials/trial\_data\_and\_results/data\_requests.

More information

Locations