NCT02130557

Brief Summary

Phase 3, 2-arm, randomized, open label trial. Patients will be randomized to receive bosutinib or imatinib for the duration of the study.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
536

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Jul 2014

Longer than P75 for phase_3

Geographic Reach
26 countries

189 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

May 1, 2014

Completed
4 days until next milestone

First Posted

Study publicly available on registry

May 5, 2014

Completed
2 months until next milestone

Study Start

First participant enrolled

July 15, 2014

Completed
2.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 11, 2016

Completed
2.3 years until next milestone

Results Posted

Study results publicly available

November 14, 2018

Completed
1.4 years until next milestone

Study Completion

Last participant's last visit for all outcomes

April 17, 2020

Completed
Last Updated

May 18, 2021

Status Verified

April 1, 2021

Enrollment Period

2.1 years

First QC Date

May 1, 2014

Results QC Date

July 13, 2018

Last Update Submit

April 16, 2021

Conditions

Keywords

LeukemiaMyelogenousChronicBCR-ABL PositiveBosutinibLeukemia, MyeloidLeukemia, Myelogenous, Chronic, BCR-ABL PositivePhiladelphia ChromosomeNeoplasms by Histologic TypeBone Marrow DiseasesHematologic DiseasesTranslocation, GeneticPathologic ProcessesImatinibTherapeutic UsesPharmacologic ActionsMolecular Mechanisms of Pharmacological Action

Outcome Measures

Primary Outcomes (1)

  • Percentage of Participants With Major Molecular Response (MMR) at Month 12

    MMR was defined as a ratio of breakpoint cluster region to abelson (BCR-ABL/ABL) less than or equal to (\<=) 0.1 percent (%) on the international scale (IS) (greater than or equal to \[\>=\] 3 log reduction from standardized baseline in ratio of BCR-ABL to ABL transcripts \[\>=3000 ABL required\]) by quantitative reverse transcriptase polymerase chain reaction (RT-qPCR). The percentage of participants with MMR at Month 12 are reported.

    Month 12

Secondary Outcomes (6)

  • Percentage of Participants With Major Molecular Response (MMR) Up to Month 18

    Up to Month 18

  • Kaplan-Meier Estimate of Probability of Retaining Major Molecular Response (MMR) at Month 48

    Month 48

  • Percentage of Participants With Complete Cytogenetic Response (CCyR) Up to Month 12

    Up to Month 12

  • Kaplan-Meier Estimate of Probability of Retaining Complete Cytogenetic Response (CCyR) at Month 48

    Month 48

  • Cumulative Incidence of Event Free Survival (EFS) Events

    Up to Month 60

  • +1 more secondary outcomes

Other Outcomes (9)

  • Summary of Trough Plasma Concentration by Complete Cytogenetic Response (CCyR) of Bosutinib

    Pre-dose on Days 28, 56 and 84

  • Summary of Trough Plasma Concentration by Major Molecular Response (MMR) of Bosutinib

    Pre-dose on Days 28, 56 and 84

  • Summary of Trough Plasma Concentration by Presence of Grade 1 or Higher Adverse Events (AEs) of Bosutinib

    Pre-dose on Days 28, 56 and 84

  • +6 more other outcomes

Study Arms (2)

Bosutinib

EXPERIMENTAL

Bosutinib, 400 mg, oral administration once a day

Drug: Bosutinib

Imatinib

ACTIVE COMPARATOR

Imatinib, 400 mg, oral administration once a day

Drug: Imatinib

Interventions

Bosutinib (Bosulif®) is an orally bioavailable, potent, multi-targeted, dual Src-Abl tyrosine kinase inhibitor (TKI) that has been approved for the treatment of adult patients with Philadelphia positive (Ph+) chronic phase (CP), accelerated phase (AP) and blast phase (BP) chronic myelogenous leukemia (CML) previously treated with other TKI inhibitor therapy.\[1\] This study will investigate the use of bosutinib as first-line treatment for patients with Ph+ CP CML.

Bosutinib

Imatinib mesylate (referred to in this protocol as imatinib) is an inhibitor of the BCR-ABL kinase and been the standard first-line therapy for patients with chronic-phase CML. Imatinib was granted approval by the European Commission in November 2001 and by the FDA in December 2002 for the treatment of newly diagnosed patients with CP Ph+ CML based on results from the IRIS trial. Imatinib is considered the standard of care for both first-line and later line settings, and consequently is an appropriate active comparator.

Imatinib

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Molecular diagnosis of CP CML of ≤ 6 months (from initial diagnosis).
  • Adequate hepatic, renal and pancreatic function.
  • Age ≥ 18 years.

You may not qualify if:

  • Any prior medical treatment for CML, including tyrosine kinase inhibitors (TKIs), with the exception of hydroxyurea and/or anagrelide treatment, which are permitted for up to 6 months prior to study entry (signature of ICF) if suitably approved for use in the subject's region.
  • Any past or current Central Nervous System (CNS) involvement, including leptomeningeal leukemia.
  • Extramedullary disease only.
  • Major surgery or radiotherapy within 14 days of randomization.
  • History of clinically significant or uncontrolled cardiac disease.
  • Known seropositivity to human immunodeficiency virus (HIV), current acute or chronic hepatitis B (hepatitis B surface-antigen positive), hepatitis C, cirrhosis or evidence of decompensated liver disease. Patients with resolved Hepatitis B can be included.
  • Recent or ongoing clinically significant GI disorder, e.g. Crohn's Disease, Ulcerative Colitis, or prior total or partial gastrectomy.
  • History of another malignancy within 5 years with the exception of basal cell carcinoma or cervical carcinoma in situ or stage 1 or 2 cancer that is considered adequately treated and currently in complete remission for at least l2 months.
  • Current, or recent (within 30 days, or 5 half-lives of investigational product) participation in other clinical trials of investigational agents and/or containing interventional procedures deemed contrary to the objectives and conduct of this trial.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (189)

Pacific Cancer Medical Center, Inc.

Anaheim, California, 92801, United States

Location

Emory University Hospital

Atlanta, Georgia, 30322, United States

Location

The Emory Clinic

Atlanta, Georgia, 30322, United States

Location

Winship Cancer Institute, Emory University

Atlanta, Georgia, 30322, United States

Location

Kaiser Permanente Hawaii

Honolulu, Hawaii, 96819, United States

Location

Saint Alphonsus Regional Medical Center, Cancer Care Center

Boise, Idaho, 83706, United States

Location

Saint Alphonsus Regional Medical Center

Boise, Idaho, 83706, United States

Location

Saint Alphonsus Caldwell Cancer Care Center

Caldwell, Idaho, 83605, United States

Location

Saint Alphonsus Medical Center Nampa

Nampa, Idaho, 83686, United States

Location

University of Illinois Cancer Center

Chicago, Illinois, 60612, United States

Location

John H. Stroger, Jr. Hospital of Cook County

Chicago, Illinois, 60621, United States

Location

Indiana Blood and Marrow Transplantation

Indianapolis, Indiana, 46237, United States

Location

PHARMACY Department Franciscan St. Francis Health ATTN:Jill Leslie, Pharm D

Indianapolis, Indiana, 46237, United States

Location

Cancer Center of Acadiana at Lafayette General Medical Center

Lafayette, Louisiana, 70503, United States

Location

Lafayette General Medical Center

Lafayette, Louisiana, 70503, United States

Location

LSU Health Sciences Center-Shreveport

Shreveport, Louisiana, 71103, United States

Location

University Health Shreveport

Shreveport, Louisiana, 71103, United States

Location

Rcca Md Llc

Bethesda, Maryland, 20817, United States

Location

University of Massachusetts Memorial Medical Center, ONC/Research Pharmacy

Worcester, Massachusetts, 01655, United States

Location

University of Massachusetts Memorial Medical Center

Worcester, Massachusetts, 01655, United States

Location

St. Joseph Mercy Hospital - Inpatient Pharmacy

Ann Arbor, Michigan, 48106, United States

Location

St. Joseph Mercy Hospital

Ann Arbor, Michigan, 48106, United States

Location

St. Joseph Mercy-Brighton

Brighton, Michigan, 48114, United States

Location

St. Joseph Mercy-Canton

Canton, Michigan, 48188, United States

Location

Chelsea Community Hospital

Chelsea, Michigan, 48118-1370, United States

Location

St. John Hospital&Medical Center

Detroit, Michigan, 48236, United States

Location

St. John Hospital&Medical Center-Van Elslander Cancer Center

Grosse Pointe Woods, Michigan, 48236, United States

Location

Van Elslander Cancer Center, Pharmacy

Grosse Pointe Woods, Michigan, 48236, United States

Location

Minnesota Oncology Hematology, PA

Edina, Minnesota, 55435, United States

Location

Park Nicollet Frauenshuh Cancer center

Saint Louis Park, Minnesota, 55426, United States

Location

Lakeview Hospital

Stillwater, Minnesota, 55082, United States

Location

North Mississippi Medical Center Hematology and Oncology Clinic

Tupelo, Mississippi, 38801, United States

Location

Nebraska Methodist Hospital

Omaha, Nebraska, 68114, United States

Location

Hackensack University Medical Center

Hackensack, New Jersey, 07601, United States

Location

John Theurer Cancer Center at Hackensack University Medical Center

Hackensack, New Jersey, 07601, United States

Location

San Juan Oncology Associates

Farmington, New Mexico, 87401, United States

Location

NYU Winthrop Hospital - Oncology / Hematology department

Mineola, New York, 11501, United States

Location

NYU Winthrop Hospital - Pharmacy Department

Mineola, New York, 11501, United States

Location

Beth Israel Medical Center

New York, New York, 10003, United States

Location

University of Rochester Investigational Drug Pharmacy

Rochester, New York, 14642, United States

Location

University of Rochester

Rochester, New York, 14642, United States

Location

FirstHealth Moore Regional Hospital

Pinehurst, North Carolina, 28374, United States

Location

FirstHealth Outpatient Cancer Center

Pinehurst, North Carolina, 28374, United States

Location

University of Cincinnati Medical Center

Cincinnati, Ohio, 45219, United States

Location

UC Health Physicians Office South,

West Chester, Ohio, 45069, United States

Location

MUSC University Hospital

Charleston, South Carolina, 29425, United States

Location

MUSC University of South Carolina, Investigational Drug Services

Charleston, South Carolina, 29425, United States

Location

MUSC-Hollings Cancer Center

Charleston, South Carolina, 29425, United States

Location

GHS Cancer Institute

Easley, South Carolina, 29640, United States

Location

GHS Cancer Institute

Greenville, South Carolina, 29605, United States

Location

GHS Cancer Institute

Greenville, South Carolina, 29615, United States

Location

GHS Cancer Institute

Greer, South Carolina, 29650, United States

Location

GHS Cancer Institute

Seneca, South Carolina, 29672, United States

Location

GHS Cancer Institute

Spartanburg, South Carolina, 29307, United States

Location

The University of Texas, MD Anderson Cancer Center

Houston, Texas, 77030, United States

Location

Utah Cancer Specialists

Murray, Utah, 84157, United States

Location

Utah Cancer Specialists

Salt Lake City, Utah, 84106, United States

Location

Huntsman Cancer Hospital

Salt Lake City, Utah, 84112, United States

Location

Huntsman Cancer Institute

Salt Lake City, Utah, 84112, United States

Location

Virginia Mason Medical Center

Seattle, Washington, 98101, United States

Location

Seattle Cancer Care Alliance

Seattle, Washington, 98109, United States

Location

HSHS St. Vincent Hospital Regional Cancer Center at HSHS St. Vincent Hospital

Green Bay, Wisconsin, 54301, United States

Location

HSHS St. Vincent Hospital

Green Bay, Wisconsin, 54301, United States

Location

HSHS St. Vincent Hospital Regional Cancer Center at HSHS St. Mary's Hospital Medical Center

Green Bay, Wisconsin, 54303, United States

Location

Froedtert Hospital and the Medical College of Wisconsin

Milwaukee, Wisconsin, 53226, United States

Location

St George Hospital - Hematology Department

Kogarah, New South Wales, 2217, Australia

Location

Eastern Clinical Research Unit, Level 2

Box Hill, Victoria, 3128, Australia

Location

UZ Ghent (University Hospital Ghent)

Ghent, 9000, Belgium

Location

Department of Haematology at UZ Leuven (7 th Floor)

Leuven, 3000, Belgium

Location

Hematology Department of CHU de Liège

Liège, 4000, Belgium

Location

Hematology Department CHR Verviers

Verviers, 4800, Belgium

Location

Horizon Health Network - The Moncton Hospital

Moncton, New Brunswick, E1C 6Z8, Canada

Location

Juravinski Cancer Centre

Hamilton, Ontario, L8V 5C2, Canada

Location

Lakeridge Health

Oshawa, Ontario, L1G 2B9, Canada

Location

Princess Margaret Cancer Centre

Toronto, Ontario, M5G 2M9, Canada

Location

Hopital Maisonneuve-Rosemont

Montreal, Quebec, H1T 2M4, Canada

Location

Saskatoon Cancer Centre

Saskatoon, Saskatchewan, S7N 4H4, Canada

Location

CHU de Québec - Université Laval

Québec, G1J 1Z4, Canada

Location

Fakultní Nemocnice Brno

Brno, 625 00, Czechia

Location

Fakultní Nemocnice Hradec Králové

Hradec Králové, 500 05, Czechia

Location

Fakultní nemocnice Olomouc

Olomouc, 775 20, Czechia

Location

Všeobecná fakultní Nemocnice v Praze

Prague, 128 08, Czechia

Location

Aalborg University Hospital

Aalborg, 9000, Denmark

Location

Aarhus University Hospital

Aarhus, 8000, Denmark

Location

Roskilde Hospital

Roskilde, 4000, Denmark

Location

Helsinki University Central Hospital

Helsinki, 00029 HUS, Finland

Location

Oncologie Centre de Radiotherapie

Strasbourg, NC, 67000, France

Location

Institut Bergonié

Bordeaux, 33076, France

Location

private Practice of Pr Philippe Rousselot

Le Chesnay, 78157, France

Location

private Practice of Dr. Viviane Dubruille

Nantes, 44093, France

Location

Hôpital L'Archet 1-CHU Nice

Nice, 06202, France

Location

Institut de Cancérologie du Gard - Hématologie Clinique

Nîmes, 30029, France

Location

Pr Mauricette Michallet Centre Hospitalier Lyon Sud

Pierre-Bénite, 69495, France

Location

INSERM CIC 1402 - CHU Poitiers

Poitiers, 86021, France

Location

Institut Universitaire du Cancer de Toulouse - Oncopole

Toulouse, 31059, France

Location

Universitätsklinikum Bonn

Bonn, Rhineland-Palatinate, 53105, Germany

Location

Uniklinikum Aachen

Aachen, 52074, Germany

Location

Charité, CVK, Med. Klinik m.S Hämatologie und Onkologie

Berlin, 13353, Germany

Location

Universitätsklinikum Freiburg, Klinik für Innere Medizin I

Freiburg im Breisgau, 79106, Germany

Location

Universitätsklinikum Hamburg-Eppendorf, Onkologisches Zentrum

Hamburg, 20251, Germany

Location

Universitätsklinikum Jena, Klinik für Innere Medizin II

Jena Lobeda-Ost, 07747, Germany

Location

Schwerpunktpraxis für Hämatologie und Onkologie

Magdeburg, 39104, Germany

Location

Semmelweis Egyetem I. Belgyógyászat

Budapest, 1083, Hungary

Location

Debreceni Egyetem Klinikai Központ, Belgyógyászati Inézet Hematológiai Tanszék

Debrecen, 4032, Hungary

Location

Petz Aladár Megyei OktatóKórház, II. Belgyógyászati Osztály és Haematológiai Részleg

Győr, 9023, Hungary

Location

Somogy Megyei Kaposi Mór Oktató Kórház

Kaposvár, 7400, Hungary

Location

Szegedi Tudományegyetem, AOK, Szent-Györgyi Albert Klinikai Központ, II. sz.

Szeged, 6725, Hungary

Location

Jász-Nagykun-Szolnok Megyei Hetényi, Géza Kórház-Rendelőintézet

Szolnok, 5000, Hungary

Location

Hematology Department, Rambam Medical Centre

Haifa, 31096, Israel

Location

Hematology Div. Davidoff Cancer Center, Rabin Medical Center

Petah Tikva, 49100, Israel

Location

Azienda Ospedaliero-Universitaria "Policlinico - Vittorio Emanuele" - P.O. G. Rodolico

Catania, CT, 95123, Italy

Location

USC Ematologia, A. O. Papa Giovanni XXIII

Bergamo, 24127, Italy

Location

Policlinico S. Orsola - Malpighi,

Bologna, 40138, Italy

Location

A.O. Brozu - P.O. Armando Businco

Cagliari, 09121, Italy

Location

Azienda Ospedaliero Universitaria Careggi

Florence, 50134, Italy

Location

IRCCS - AOU San Martino_IST, Ematologia 1

Genova, 16132, Italy

Location

Istituto Scientifico San Raffaele

Milan, 20132, Italy

Location

Unità di Ricerca Clinica, U.O. Ematologia Adulti

Monza, 20900, Italy

Location

A.O.U. Policlinico Università degli Studi di Napoli "Federico II"

Napoli, 80131, Italy

Location

Dipartimento di ematologia

Reggio Calabria, 89124, Italy

Location

ASL Roma 2 - Ospedale Sant'Eugenio

Roma, 00144, Italy

Location

Hospital Angeles del Pedregal (S.A. de C.V.)

Mexico City, Mexico City, 10700, Mexico

Location

Monterrey International Research Center

Monterrey, Nuevo León, 64000, Mexico

Location

Klinische Farrnacologie en Apotheek

Amsterdam, North Holland, 1081 BT, Netherlands

Location

VU University Medical Center

Amsterdam, North Holland, 1081 HV, Netherlands

Location

Haukeland University Hospital Department of Hematology

Bergen, 5021, Norway

Location

St. Olavs Hospital

Trondheim, 7006, Norway

Location

Klinika Hematologii i Transplantologii Uniwersyteckie Centrum Kliniczne

Gdansk, Pomeranian Voivodeship, 80-214, Poland

Location

SPZOZ ZSM w Chorzowie Oddzial Hematologiczny

Chorzów, 41-500, Poland

Location

Samodzielny Publiczny Szpital Kliniczny im. A Mielęckiego, ŚUM w Katowicach

Katowice, 40032, Poland

Location

Szpital Uniwersytecki w Krakowie, Oddział Kliniczny Hematologii

Krakow, 31501, Poland

Location

Wojewódzki Szpital Specjalistyczny im M. Kopernika, Klinika Hematologii Uniwersytetu Medycznego

Lodz, 93510, Poland

Location

SPSK, Klinika Hematoonkologii i Transplantacji Szpiku w Lublinie

Lublin, 20081, Poland

Location

Universytet Medyczny im. Piastów Śląskich we Wrocławiu Katedra i

Wroclaw, 50-367, Poland

Location

National University Hospital, Main Building

Singapore, 119228, Singapore

Location

Singapore General Hospital

Singapore, 169608, Singapore

Location

Tan Tock Seng Hospital

Singapore, 308433, Singapore

Location

Univerzitná Nemocnica Bratislava-Nemocnica sv. Cyrila a Metoda

Bratislava, 851 07, Slovakia

Location

The Medical Oncology Centre of Rosebank

Johannesburg, Gauteng, 2196, South Africa

Location

Department of Medical Oncology, University of Pretoria and Steve Biko

Pretoria, Gauteng, 0002, South Africa

Location

Groenkloof Life hospital.

Pretoria, Gauteng, 0181, South Africa

Location

Department of Haematology

Cape Town, Western Cape, 7935, South Africa

Location

Hallym University Sacred Heart Hospital

Anyang-si, 14068, South Korea

Location

Dong A University Hospital

Busan, 49201, South Korea

Location

Keimyung University Dongsan Hospital

Daegu, 41931, South Korea

Location

Chonbuk National University Hospital

Jeonju, 54907, South Korea

Location

Kangbuk Samsung Hospital

Seoul, 03181, South Korea

Location

Seoul St. Mary's Hospital of the Catholic University of Korea

Seoul, 06591, South Korea

Location

Hospital (Universitari(o)) Germans Trias i Pujol

Badalona, Barcelona, 08916, Spain

Location

Hospital Universitario La Princesa

Madrid, Málaga, 28006, Spain

Location

Hospital Vall d'Hebron

Barcelona, 08035, Spain

Location

Hospital Clínic

Barcelona, 08036, Spain

Location

Hospital Universitario Gregorio Marañón

Madrid, 28007, Spain

Location

Hospital Ramón y Cajal

Madrid, 28034, Spain

Location

Hospital Clinico San Carlos

Madrid, 28040, Spain

Location

Hospital Universitario de Salamanca

Salamanca, 37007, Spain

Location

Hospital Virgen de la Salud

Toledo, 45004, Spain

Location

Hospital Clínico Universitario de Valencia

Valencia, 46010, Spain

Location

Linköping University Hospital

Linköping, SE-581 85, Sweden

Location

Skåne University Hospital

Lund, SE-221 85, Sweden

Location

Karolinska University Hospital Solna

Stockholm, SE-171 76, Sweden

Location

Norrlands University Hospital

Umeå, SE-901 85, Sweden

Location

Akademiska Hospital

Uppsala, SE-751 85, Sweden

Location

China Medical University Hospital

Taichung, R.o.c., 40447, Taiwan

Location

Chi-Mei Medical Center

Tainan, R.o.c., 710, Taiwan

Location

Mackay Memorial Hospital

Taipei, R.o.c., 10449, Taiwan

Location

Kaohsiung Medical University Chung-Ho Memorial Hospital

Kaohsiung City, 807, Taiwan

Location

Division of Hematology, Department of Internal Medicine, Maharaj Nakorn Chiang Mai Hospital

Muang, Chiang Mai, 50200, Thailand

Location

King Chulalongkorn Memorial Hospital

Bangkok, 10330, Thailand

Location

Phramongkutklao Hospital

Bangkok, 10400, Thailand

Location

Division of Hematology, Department of Medicine, Faculty of Medicine Siriraj Hospital

Bangkok, 10700, Thailand

Location

MI "Cherkasy Regional Oncological Dispensary " of Cherkasy Regional Council

Cherkasy, 18009, Ukraine

Location

Regional Clinical Hospital in Ivano-Frankivsk, Hematology Department

Ivano-Frankivsk, 76008, Ukraine

Location

Khmelnytskyi Regional Hospital, Hematology Department

Khmelnytskyi, 29000, Ukraine

Location

State Institution "National research center for radiation medicine of NAMS of Ukraine",

Kyiv, 03115, Ukraine

Location

State Institution "National research center for radiation medicine of NAMS of Ukraine"

Kyiv, 03115, Ukraine

Location

transplantation department of hemotology and transplantology division within Clinical Radiology

Kyiv, 03115, Ukraine

Location

Chair of internal medicine #2.

Kyiv, 04112, Ukraine

Location

Kyiv City Clinical Hospital #9, Hematology department #1,

Kyiv, 04112, Ukraine

Location

State Institution "Institute of Blood Pathology and Transfusion Medicine NAMS of Ukraine"

Lviv, 79044, Ukraine

Location

Catherine Lewis Centre, Hammersmith Hospital

London, Greater London, W12 0HS, United Kingdom

Location

Linda McCartney Centre

Liverpool, Merseyside, L7 8XP, United Kingdom

Location

Department of Clinical Haematology

Nottingham, Nottinghamshire, NG5 1PB, United Kingdom

Location

Cancer & Haematology Centre, Churchill Hospital

Oxford, Oxfordshire, OX3 7LE, United Kingdom

Location

Department of Haematology The Royal Hallamshire Hospital

Sheffield, South Yorkshire, S10 2JF, United Kingdom

Location

Heartlands Hospital

Birmingham, WEST Midlands, B9 5SS, United Kingdom

Location

St James's Institute of Oncology

Leeds, WEST Yorkshire, LS9 7TF, United Kingdom

Location

Department of Haematology

Cardiff, CF14 4XW, United Kingdom

Location

The Hope Clinical Trials Facility

Leicester, LE1 5WW, United Kingdom

Location

Related Publications (5)

  • Garrett M, Knight B, Cortes JE, Deininger MW. Population modeling of bosutinib exposure-response in patients with newly diagnosed chronic phase chronic myeloid leukemia. Cancer Med. 2023 Sep;12(17):17981-17992. doi: 10.1002/cam4.6439. Epub 2023 Aug 8.

  • Brummendorf TH, Cortes JE, Milojkovic D, Gambacorti-Passerini C, Clark RE, le Coutre P, Garcia-Gutierrez V, Chuah C, Kota V, Lipton JH, Rousselot P, Mauro MJ, Hochhaus A, Hurtado Monroy R, Leip E, Purcell S, Yver A, Viqueira A, Deininger MW; BFORE study investigators. Bosutinib versus imatinib for newly diagnosed chronic phase chronic myeloid leukemia: final results from the BFORE trial. Leukemia. 2022 Jul;36(7):1825-1833. doi: 10.1038/s41375-022-01589-y. Epub 2022 May 28.

  • Takahashi N, Cortes JE, Sakaida E, Ishizawa K, Ono T, Doki N, Matsumura I, Garcia-Gutierrez V, Rosti G, Ono C, Ohkura M, Tanetsugu Y, Viqueira A, Brummendorf TH. Safety profile of bosutinib in Japanese versus non-Japanese patients with chronic myeloid leukemia: a pooled analysis. Int J Hematol. 2022 Jun;115(6):838-851. doi: 10.1007/s12185-022-03314-y. Epub 2022 Mar 2.

  • Chuah C, Koh LP, Numbenjapon T, Zang DY, Ong KH, Do YR, Ohkura M, Ono C, Viqueira A, Cortes JE, Brummendorf TH. Efficacy and safety of bosutinib versus imatinib for newly diagnosed chronic myeloid leukemia in the Asian subpopulation of the phase 3 BFORE trial. Int J Hematol. 2021 Jul;114(1):65-78. doi: 10.1007/s12185-021-03144-4. Epub 2021 Apr 13.

  • Cortes JE, Gambacorti-Passerini C, Deininger MW, Mauro MJ, Chuah C, Kim DW, Dyagil I, Glushko N, Milojkovic D, le Coutre P, Garcia-Gutierrez V, Reilly L, Jeynes-Ellis A, Leip E, Bardy-Bouxin N, Hochhaus A, Brummendorf TH. Bosutinib Versus Imatinib for Newly Diagnosed Chronic Myeloid Leukemia: Results From the Randomized BFORE Trial. J Clin Oncol. 2018 Jan 20;36(3):231-237. doi: 10.1200/JCO.2017.74.7162. Epub 2017 Nov 1.

MeSH Terms

Conditions

LeukemiaBronchiolitis Obliterans SyndromeLeukemia, MyeloidLeukemia, Myelogenous, Chronic, BCR-ABL PositivePhiladelphia ChromosomeNeoplasms by Histologic TypeBone Marrow DiseasesHematologic DiseasesTranslocation, GeneticPathologic Processes

Interventions

bosutinibImatinib Mesylate

Condition Hierarchy (Ancestors)

NeoplasmsHemic and Lymphatic DiseasesOrganizing PneumoniaBronchiolitis ObliteransBronchiolitisBronchitisBronchial DiseasesRespiratory Tract DiseasesLung Diseases, ObstructiveLung DiseasesGraft vs Host DiseaseImmune System DiseasesMyeloproliferative DisordersChronic DiseaseDisease AttributesPathological Conditions, Signs and SymptomsChromosome Aberrations

Intervention Hierarchy (Ancestors)

BenzamidesAmidesOrganic ChemicalsBenzoatesAcids, CarbocyclicCarboxylic AcidsBenzene DerivativesHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsPiperazinesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPyrimidines

Results Point of Contact

Title
Pfizer ClinicalTrials.gov Call Center
Organization
Pfizer Inc.

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Masking Details
NOTE: Value was Open Label in old format; This study has an open-label design. Although most efficacy studies have a double blind design, this is not feasible in this trial, due to the complexity of the dose reduction and dose escalation schemes with tablets of various sizes, dosage strengths, as well as the number of tablets that would be required daily. However, the opportunity for bias is mitigated by the use of objective outcome measures (MMR, CCyR, CHR). The Investigators will be instructed to ensure that laboratory/pathology personnel are blinded to treatment information. For these reasons, an open-label, randomized study is appropriate.
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 1, 2014

First Posted

May 5, 2014

Study Start

July 15, 2014

Primary Completion

August 11, 2016

Study Completion

April 17, 2020

Last Updated

May 18, 2021

Results First Posted

November 14, 2018

Record last verified: 2021-04

Data Sharing

IPD Sharing
Will share

Pfizer will provide access to individual de-identified participant data and related study documents (e.g. protocol, Statistical Analysis Plan (SAP), Clinical Study Report (CSR)) upon request from qualified researchers, and subject to certain criteria, conditions, and exceptions. Further details on Pfizer's data sharing criteria and process for requesting access can be found at: https://www.pfizer.com/science/clinical\_trials/trial\_data\_and\_results/data\_requests.

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