NCT01300013

Brief Summary

The primary objective of the study is to evaluate the effect of 48 hours of intravenous (IV) omecamtiv mecarbil compared with placebo on dyspnea in subjects with left ventricular systolic dysfunction hospitalized for acute heart failure. This is a multicenter, randomized, double-blind, placebo-controlled study with 3 dose cohorts enrolled sequentially in order of ascending dose strength of omecamtiv mecarbil. In each cohort, subjects are randomized 1:1 to omecamtiv mecarbil or placebo.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
614

participants targeted

Target at P75+ for phase_2 heart-failure

Timeline
Completed

Started Apr 2011

Typical duration for phase_2 heart-failure

Geographic Reach
19 countries

150 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

February 17, 2011

Completed
4 days until next milestone

First Posted

Study publicly available on registry

February 21, 2011

Completed
1 month until next milestone

Study Start

First participant enrolled

April 1, 2011

Completed
2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 1, 2013

Completed
5 months until next milestone

Study Completion

Last participant's last visit for all outcomes

September 1, 2013

Completed
Last Updated

July 27, 2021

Status Verified

July 1, 2021

Enrollment Period

2 years

First QC Date

February 17, 2011

Last Update Submit

July 25, 2021

Conditions

Keywords

IntravenousIVLeft Ventricular Systolic DysfunctionHospitalizedAcute heart failureHeart failureLeft ventricular ejection fractionpharmacokineticsPharmacodynamicsDyspneahospitalizationIn-patientOmecamtiv mecarbilDouble-blindRandomizedPlacebo-controlled

Outcome Measures

Primary Outcomes (1)

  • The primary objective of the study is to evaluate the effect of 48 hours of intravenous (IV) omecamtiv mecarbil compared with placebo on dyspnea in subjects with left ventricular systolic dysfunction hospitalized for acute heart failure.

    48 hours

Secondary Outcomes (3)

  • To characterize pharmacokinetics of omecamtiv mecarbil including metabolites following IV infusion and to evaluate the relationship between omecamtiv mecarbil plasma concentration and echocardiographic parameters in subjects with AHF

    48 hours

  • To assess the safety and tolerability of 3 dose levels of IV omecamtiv mecarbil compared with placebo in subjects with left ventricular systolic dysfunction hospitalized for acute heart failure

    48 hours

  • To evaluate the effects of 48 hours treatment with IV omecamtiv mecarbil on additional measures of dyspnea, patient global assessment (PGA), change in NT-proBNP, incidence of worsening heart failure, and short term clinical outcomes

    48 hours

Study Arms (2)

Omecamtiv mecarbil

EXPERIMENTAL
Drug: Omecamtiv mecarbil

Placebo

PLACEBO COMPARATOR
Drug: Placebo

Interventions

48-hour infusion of placebo

Placebo

48-hour infusion of omecamtiv mecarbil; dose strength will depend on cohort assignment.

Also known as: CK-1827452, AMG 423
Omecamtiv mecarbil

Eligibility Criteria

Age18 Years - 85 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Male or female 18 - 85 years
  • Hospitalized for worsening heart failure, within 24 hours of initiating IV loop diuretic
  • Dyspnea due to heart failure, at rest or with minimal exertion
  • History of left ventricular ejection fraction (LVEF) ≤ 40%
  • Elevated brain natriuretic peptide (BNP) or N-terminal fragment BNP (NT-proBNP)

You may not qualify if:

  • Receiving IV vasopressor (excluding low dopamine), inotropic or mechanical support
  • Acute coronary syndrome (ACS)
  • Within 30 days prior to enrollment: cardiac resynchronization therapy (CRT) or implantable cardioverter defibrillator (ICD) implantation, ACS, coronary revascularization, transient ischemic attack (TIA) or stroke, sustained ventricular arrhythmia, or major surgery
  • Severe valvular stenosis, hypertrophic obstructive cardiomyopathy, active myocarditis, constrictive pericarditis, or clinically significant congenital heart disease
  • Estimated glomerular filtration rate (eGFR) \< 20 mL/min/1.73m2

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (150)

Research Site

Mobile, Alabama, 36608, United States

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Inglewood, California, 90301, United States

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La Jolla, California, 92037, United States

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San Francisco, California, 94121, United States

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Danbury, Connecticut, 06810, United States

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Newark, Delaware, 19718, United States

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Atlantis, Florida, 33462, United States

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Clearwater, Florida, 33756, United States

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Fort Lauderdale, Florida, 33308, United States

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Miami, Florida, 33133, United States

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Orlando, Florida, 32803, United States

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Atlanta, Georgia, 30322, United States

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Chicago, Illinois, 60611, United States

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Peoria, Illinois, 61636, United States

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Baltimore, Maryland, 21201, United States

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Detroit, Michigan, 48201, United States

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Detroit, Michigan, 48202, United States

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Novi, Michigan, 48374, United States

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Minneapolis, Minnesota, 55417, United States

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St Louis, Missouri, 63110, United States

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Lincoln, Nebraska, 68506, United States

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Newark, New Jersey, 07103, United States

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Cortlandt Manor, New York, 10567, United States

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Roslyn, New York, 11576, United States

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The Bronx, New York, 10467, United States

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Chapel Hill, North Carolina, 27599, United States

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Charlotte, North Carolina, 28204, United States

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Durham, North Carolina, 27705, United States

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Winston-Salem, North Carolina, 27103, United States

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Cincinnati, Ohio, 45219, United States

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Cincinnati, Ohio, 45220, United States

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Cincinnati, Ohio, 45267, United States

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Cleveland, Ohio, 44109, United States

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Columbus, Ohio, 43210, United States

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Fairfield, Ohio, 45014, United States

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Oklahoma City, Oklahoma, 73120, United States

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Portland, Oregon, 97239, United States

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Charleston, South Carolina, 29425, United States

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Greenville, South Carolina, 29605, United States

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Memphis, Tennessee, 38120, United States

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Nashville, Tennessee, 37203, United States

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Nashville, Tennessee, 37232-8802, United States

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Tullahoma, Tennessee, 37388, United States

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Houston, Texas, 77030, United States

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Murray, Utah, 84107, United States

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Darlinghurst, New South Wales, 2010, Australia

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Woolloongabba, Queensland, 4102, Australia

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Bedford Park, South Australia, 5042, Australia

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Prahran, Victoria, 3181, Australia

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Richmond, Victoria, 3121, Australia

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Aalst, 9300, Belgium

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Bonheiden, 2820, Belgium

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Ghent, 9000, Belgium

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Roeselare, 8800, Belgium

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Blagoevgrad, 2700, Bulgaria

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Kazanlak, 6100, Bulgaria

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Pazardzhik, 4700, Bulgaria

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Plovdiv, 4002, Bulgaria

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Sandanski, 2800, Bulgaria

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Smolyan, 4400, Bulgaria

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Sofia, 1309, Bulgaria

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Sofia, 1431, Bulgaria

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Sofia, 1527, Bulgaria

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Calgary, Alberta, T2N 4Z6, Canada

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Edmonton, Alberta, T6G 2B7, Canada

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Edmonton, Alberta, T6L 5X8, Canada

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Halifax, Nova Scotia, B3H 3A7, Canada

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Ottawa, Ontario, K1Y 4W7, Canada

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Toronto, Ontario, M5B 1W8, Canada

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Toronto, Ontario, M5G 1X5, Canada

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Montreal, Quebec, H3G 1A4, Canada

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Québec, Quebec, G1V 4G5, Canada

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Sherbrooke, Quebec, J1H 5N4, Canada

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Brno, 625 00, Czechia

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Brno, 656 91, Czechia

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Prague, 128 08, Czechia

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Prague, 150 06, Czechia

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Ústí nad Labem, 401 13, Czechia

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Helsinki, 00029, Finland

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Turku, 20521, Finland

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Caen, 14033, France

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Lille, 59037, France

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Montpellier, 34295, France

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Paris, 75010, France

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Paris, 75651, France

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Strasbourg, 67091, France

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Toulouse, 31403, France

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Bad Nauheim, 61231, Germany

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Dortmund, 44137, Germany

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Dresden, 01307, Germany

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Frankfurt, 60488, Germany

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Frankfurt, 60590, Germany

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Greifswald, 17475, Germany

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Halle, 06097, Germany

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Hamburg, 20246, Germany

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Homburg, 66421, Germany

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Langen, 63225, Germany

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Regensburg, 93053, Germany

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Stuttgart, 70376, Germany

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Würzburg, 97080, Germany

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Athens, 11528, Greece

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Athens, 16673, Greece

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Haidari, 12462, Greece

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Heraklion, 71110, Greece

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Pátrai, 26500, Greece

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Budapest, 1023, Hungary

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Budapest, 1122, Hungary

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Budapest, 1125, Hungary

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Budapest, 1134, Hungary

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Pécs, 7624, Hungary

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Szolnok, 5004, Hungary

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Brescia, 25125, Italy

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Cagliari, 09134, Italy

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Pavia, 27100, Italy

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Udine, 33100, Italy

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Kaunas, 50009, Lithuania

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Vilnius, 08661, Lithuania

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Delft, 2625 AD, Netherlands

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Deventer, 7416 SE, Netherlands

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Utrecht, 3584 CX, Netherlands

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Oslo, 0424, Norway

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Stavanger, 4011, Norway

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Bialystok, 15-276, Poland

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Gdansk, 80-952, Poland

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Krakow, 31-202, Poland

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Krakow, 31-501, Poland

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Lodz, 91-347, Poland

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Lublin, 20-954, Poland

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Wroclaw, 50-981, Poland

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Moscow, 109240, Russia

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Moscow, 111539, Russia

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Moscow, 115093, Russia

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Moscow, 117292, Russia

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Moscow, 119620, Russia

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Moscow, 119991, Russia

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Moscow, 127299, Russia

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Moscow, 127473, Russia

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Saint Petersburg, 195067, Russia

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Saint Petersburg, 197341, Russia

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Saint Petersburg, 198205, Russia

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Saint Petersburg, 199106, Russia

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St.-Petrsburg, 196247, Russia

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Bratislava, 826 06, Slovakia

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Bratislava, 851 07, Slovakia

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Košice, 040 66, Slovakia

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Nitra, 949 01, Slovakia

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Bristol, BS2 8HW, United Kingdom

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Cottingham, HU16 5JQ, United Kingdom

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Glasgow, G11 6NT, United Kingdom

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Harrow, HA1 3UJ, United Kingdom

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Related Publications (1)

  • Teerlink JR, Felker GM, McMurray JJV, Ponikowski P, Metra M, Filippatos GS, Ezekowitz JA, Dickstein K, Cleland JGF, Kim JB, Lei L, Knusel B, Wolff AA, Malik FI, Wasserman SM; ATOMIC-AHF Investigators. Acute Treatment With Omecamtiv Mecarbil to Increase Contractility in Acute Heart Failure: The ATOMIC-AHF Study. J Am Coll Cardiol. 2016 Mar 29;67(12):1444-1455. doi: 10.1016/j.jacc.2016.01.031.

Related Links

MeSH Terms

Conditions

Heart FailureVentricular Dysfunction, LeftDyspnea

Interventions

omecamtiv mecarbil

Condition Hierarchy (Ancestors)

Heart DiseasesCardiovascular DiseasesVentricular DysfunctionRespiration DisordersRespiratory Tract DiseasesSigns and Symptoms, RespiratorySigns and SymptomsPathological Conditions, Signs and Symptoms

Study Officials

  • MD

    Amgen

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

February 17, 2011

First Posted

February 21, 2011

Study Start

April 1, 2011

Primary Completion

April 1, 2013

Study Completion

September 1, 2013

Last Updated

July 27, 2021

Record last verified: 2021-07

Locations