NCT01120275

Brief Summary

This phase II trial is studying how well gamma-secretase/Notch signalling pathway inhibitor RO4929097 works in treating patients with stage IV melanoma. Gamma-secretase/Notch signalling pathway inhibitor RO4929097 may stop the growth of tumor cells by blocking some of the enzymes needed for cell growth.

Trial Health

57
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
36

participants targeted

Target at P25-P50 for phase_2

Timeline
Completed

Started Oct 2010

Longer than P75 for phase_2

Geographic Reach
1 country

178 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

May 7, 2010

Completed
3 days until next milestone

First Posted

Study publicly available on registry

May 10, 2010

Completed
5 months until next milestone

Study Start

First participant enrolled

October 1, 2010

Completed
2.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 1, 2013

Completed
2.3 years until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2015

Completed
11 months until next milestone

Results Posted

Study results publicly available

June 14, 2016

Completed
Last Updated

June 14, 2016

Status Verified

May 1, 2016

Enrollment Period

2.6 years

First QC Date

May 7, 2010

Results QC Date

October 29, 2015

Last Update Submit

May 6, 2016

Conditions

Outcome Measures

Primary Outcomes (2)

  • Progression-free Survival According to Response Evaluation Criteria in Solid Tumors (RECIST) Version 1.1

    From date of registration to date of first documentation of progression or symptomatic deterioration, or death due to any cause.

    Disease assessments were performed every 6 weeks, up to 3 years.

  • Overall Survival

    From date of registration to date of death due to any cause. Patients last known to be alive are censored at date of last contact.

    Weekly, up to 3 years.

Secondary Outcomes (2)

  • Percentage of Participants With Confirmed and Unconfirmed Complete or Partial Response

    Disease assessments for response were performed every 6 weeks, up to 3 years

  • Number of Patients With Gr 3 Through 5 Adverse Events That Are Related to Study Drugs

    Toxicity assessment was evaluated at least every 3 weeks at the beginning of each cycle, up to 3 years

Study Arms (1)

Treatment (gamma-secretase inhibitor RO4929097)

EXPERIMENTAL

Patients receive gamma-secretase/Notch signalling pathway inhibitor RO4929097 PO on days 1-3, 8-10, and 15-17. Courses repeat every 21 days in the absence of disease progression or unacceptable toxicity.

Drug: gamma-secretase/Notch signalling pathway inhibitor RO4929097Other: laboratory biomarker analysis

Interventions

Given PO

Also known as: R4733, RO4929097
Treatment (gamma-secretase inhibitor RO4929097)

Correlative studies

Treatment (gamma-secretase inhibitor RO4929097)

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Patients must have histologically confirmed melanoma of cutaneous or unknown origin (ocular primary and mucosal primary excluded); patients must have Stage IV disease
  • All patients must undergo a computed tomography (CT) or magnetic resonance imaging (MRI) of the brain within 42 days prior to registration that is negative for brain metastases; patients with a history of brain metastases are ineligible
  • Patients must have measurable disease; all measurable lesions must be assessed (by physical examination, CT, or MRI scan) within 28 days prior to registration; tests to assess non-measurable disease must be performed within 42 days prior to registration; all disease must be assessed and documented on the Baseline Tumor Assessment Form (Response Evaluation Criteria In Solid Tumors \[RECIST\] 1.1); the CT from a combined positron emission tomography (PET)/CT must not be used to document measurable disease unless it is of diagnostic quality
  • Sites must offer all patients participation in translational medicine studies and banking of paraffin embedded tissue and whole blood
  • Patients must not have received any prior systemic therapy for Stage IV disease except for noncytotoxic biologic agents (e.g., vaccines, cytokines, cell therapies that do not require cytotoxic agents); patients may have received prior treatment with up to two prior biological therapies - no cytotoxics or kinase inhibitors - for advanced disease
  • Patients may have had prior adjuvant immunotherapy with biological response modifiers (examples include but are not limited to interferon, vaccines, GM-CSF, and CTLA-4 blocking antibodies); prior adjuvant immunotherapy must have been completed at least 28 days prior to registration
  • Adjuvant therapy containing cytotoxic agents is allowed if completed \>= 180 days prior to registration
  • Patients may have received prior radiation therapy; any side effects the patients had due to prior radiation therapy must have resolved to =\< Grade 1 prior to registration; prior radiation therapy must have completed at least 28 days prior to registration
  • Patients must have Zubrod performance status of 0-1
  • Leukocytes \>= 3,000/mcL
  • Absolute neutrophil count (ANC) \>= 1,500/mcL
  • Platelets \>= 100,000/mcL
  • Hemoglobin \>= 9 g/dL
  • Total bilirubin =\< institutional upper limit of normal (IULN)
  • Aspartate aminotransferase (AST) or alanine aminotransferase (ALT) =\< 2.5 x IULN
  • +19 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (178)

Providence Hospital

Mobile, Alabama, 36608, United States

Location

Fairbanks Memorial Hospital

Fairbanks, Alaska, 99701, United States

Location

University of Arizona Health Sciences Center

Tucson, Arizona, 85724, United States

Location

Saint Edward Mercy Medical Center

Fort Smith, Arkansas, 72903, United States

Location

University of Arkansas for Medical Sciences

Little Rock, Arkansas, 72205, United States

Location

Loma Linda University Medical Center

Loma Linda, California, 92354, United States

Location

Fremont - Rideout Cancer Center

Marysville, California, 95901, United States

Location

University of California Medical Center At Irvine-Orange Campus

Orange, California, 92868, United States

Location

University of California at Davis Cancer Center

Sacramento, California, 95817, United States

Location

Tahoe Forest Cancer Center

Truckee, California, 96161, United States

Location

University of Colorado Cancer Center - Anschutz Cancer Pavilion

Aurora, Colorado, 80045, United States

Location

Denver Veterans Administration Medical Center

Denver, Colorado, 80220, United States

Location

Poudre Valley Hospital

Fort Collins, Colorado, 80524, United States

Location

Saint Mary's Hospital and Regional Medical Center

Grand Junction, Colorado, 81502, United States

Location

Saint Francis Hospital and Medical Center

Hartford, Connecticut, 06105, United States

Location

Northeast Georgia Medical Center

Gainesville, Georgia, 30501, United States

Location

Oncare Hawaii Inc-POB II

Honolulu, Hawaii, 96813, United States

Location

Queen's Medical Center

Honolulu, Hawaii, 96813, United States

Location

Straub Clinic and Hospital

Honolulu, Hawaii, 96813, United States

Location

University of Hawaii

Honolulu, Hawaii, 96813, United States

Location

Oncare Hawaii Inc-Kuakini

Honolulu, Hawaii, 96817, United States

Location

The Cancer Center of Hawaii-Liliha

Honolulu, Hawaii, 96817, United States

Location

Kapiolani Medical Center for Women and Children

Honolulu, Hawaii, 96826, United States

Location

Castle Medical Center

Kailua, Hawaii, 96734, United States

Location

Wilcox Memorial Hospital and Kauai Medical Clinic

Lihue, Hawaii, 96766, United States

Location

Maui Memorial Medical Center

Wailuku, Hawaii, 96793, United States

Location

Pali Momi Medical Center

‘Aiea, Hawaii, 96701, United States

Location

Saint Anthony's Health

Alton, Illinois, 62002, United States

Location

University of Chicago

Chicago, Illinois, 60637, United States

Location

Decatur Memorial Hospital

Decatur, Illinois, 62526, United States

Location

Loyola University Medical Center

Maywood, Illinois, 60153, United States

Location

Good Samaritan Regional Health Center

Mount Vernon, Illinois, 62864, United States

Location

Memorial Medical Center

Springfield, Illinois, 62781-0001, United States

Location

Saint Francis Hospital and Health Centers

Beech Grove, Indiana, 46107, United States

Location

Reid Hospital and Health Care Services

Richmond, Indiana, 47374, United States

Location

Genesis Medical Center - East Campus

Davenport, Iowa, 52803, United States

Location

Hays Medical Center

Hays, Kansas, 67601, United States

Location

Promise Regional Medical Center-Hutchinson

Hutchinson, Kansas, 65702, United States

Location

University of Kansas Medical Center

Kansas City, Kansas, 66160, United States

Location

Lawrence Memorial Hospital

Lawrence, Kansas, 66044, United States

Location

Menorah Medical Center

Overland Park, Kansas, 66209, United States

Location

Saint Luke's South Hospital

Overland Park, Kansas, 66213, United States

Location

Via Christi Hospital-Pittsburg

Pittsburg, Kansas, 66762, United States

Location

Kansas City CCOP

Prairie Village, Kansas, 66208, United States

Location

Salina Regional Health Center

Salina, Kansas, 67401, United States

Location

Shawnee Mission Medical Center

Shawnee Mission, Kansas, 66204, United States

Location

Saint Francis Hospital and Medical Center - Topeka

Topeka, Kansas, 66606, United States

Location

Wesley Medical Center

Wichita, Kansas, 67214, United States

Location

University of Kentucky

Lexington, Kentucky, 40536, United States

Location

Louisiana State University Sciences Center- Monroe

Monroe, Louisiana, 71210, United States

Location

Highland Clinic

Shreveport, Louisiana, 71105, United States

Location

Louisiana State University Health Sciences Center Shreveport

Shreveport, Louisiana, 71130, United States

Location

Sinai Hospital of Baltimore

Baltimore, Maryland, 21215, United States

Location

Saint Joseph Mercy Hospital

Ann Arbor, Michigan, 48106-0995, United States

Location

Michigan Cancer Research Consortium Community Clinical Oncology Program

Ann Arbor, Michigan, 48106, United States

Location

University of Michigan

Ann Arbor, Michigan, 48109, United States

Location

Bronson Battle Creek

Battle Creek, Michigan, 49017, United States

Location

Spectrum Health Big Rapids Hospital

Big Rapids, Michigan, 49307, United States

Location

Oakwood Hospital

Dearborn, Michigan, 48124, United States

Location

Wayne State University/Karmanos Cancer Institute

Detroit, Michigan, 48201, United States

Location

Saint John Hospital and Medical Center

Detroit, Michigan, 48236, United States

Location

Hurley Medical Center

Flint, Michigan, 48502, United States

Location

Genesys Regional Medical Center-West Flint Campus

Flint, Michigan, 48532, United States

Location

Grand Rapids Clinical Oncology Program

Grand Rapids, Michigan, 49503, United States

Location

Mercy Health Saint Mary's

Grand Rapids, Michigan, 49503, United States

Location

Spectrum Health at Butterworth Campus

Grand Rapids, Michigan, 49503, United States

Location

Allegiance Health

Jackson, Michigan, 49201, United States

Location

Sparrow Hospital

Lansing, Michigan, 48912, United States

Location

Saint Mary Mercy Hospital

Livonia, Michigan, 48154, United States

Location

Mercy Health Mercy Campus

Muskegon, Michigan, 49444, United States

Location

Saint Joseph Mercy Oakland

Pontiac, Michigan, 48341-2985, United States

Location

Saint Joseph Mercy Port Huron

Port Huron, Michigan, 48060, United States

Location

William Beaumont Hospital-Royal Oak

Royal Oak, Michigan, 48073, United States

Location

Saint Mary's of Michigan

Saginaw, Michigan, 48601, United States

Location

Munson Medical Center

Traverse City, Michigan, 49684, United States

Location

Saint John Macomb-Oakland Hospital

Warren, Michigan, 48093, United States

Location

Metro Health Hospital

Wyoming, Michigan, 49519, United States

Location

Central Care Cancer Center-Carrie J Babb Cancer Center

Bolivar, Missouri, 65613, United States

Location

CoxHealth Cancer Center

Branson, Missouri, 65616, United States

Location

Saint Francis Medical Center

Cape Girardeau, Missouri, 63703, United States

Location

Truman Medical Center

Kansas City, Missouri, 64108, United States

Location

Saint Luke's Cancer Institute

Kansas City, Missouri, 64111, United States

Location

Saint Luke's Hospital of Kansas City

Kansas City, Missouri, 64111, United States

Location

Saint Joseph Health Center

Kansas City, Missouri, 64114, United States

Location

North Kansas City Hospital

Kansas City, Missouri, 64116, United States

Location

Research Medical Center

Kansas City, Missouri, 64132, United States

Location

Saint Luke's East - Lee's Summit

Lee's Summit, Missouri, 64086, United States

Location

Liberty Hospital

Liberty, Missouri, 64068, United States

Location

Heartland Regional Medical Center

Saint Joseph, Missouri, 64506, United States

Location

Ozark Health Ventures LLC dba Cancer Research for The Ozarks Springfield

Springfield, Missouri, 65802, United States

Location

Mercy Hospital Springfield

Springfield, Missouri, 65804, United States

Location

CoxHealth South Hospital

Springfield, Missouri, 65807, United States

Location

Saint Louis Cancer and Breast Institute-South City

St Louis, Missouri, 63109, United States

Location

Saint John's Mercy Medical Center

St Louis, Missouri, 63141, United States

Location

Saint Louis-Cape Girardeau CCOP

St Louis, Missouri, 63141, United States

Location

Montana Cancer Consortium CCOP

Billings, Montana, 59101, United States

Location

Saint Vincent Healthcare

Billings, Montana, 59101, United States

Location

Hematology-Oncology Centers of the Northern Rockies PC

Billings, Montana, 59102, United States

Location

Billings Clinic

Billings, Montana, 59107-7000, United States

Location

Bozeman Deaconess Cancer Center

Bozeman, Montana, 59715, United States

Location

Bozeman Deaconess Hospital

Bozeman, Montana, 59715, United States

Location

Benefis Healthcare- Sletten Cancer Institute

Great Falls, Montana, 59405, United States

Location

Great Falls Clinic

Great Falls, Montana, 59405, United States

Location

Saint Peter's Community Hospital

Helena, Montana, 59601, United States

Location

Glacier Oncology PLLC

Kalispell, Montana, 59901, United States

Location

Kalispell Regional Medical Center

Kalispell, Montana, 59901, United States

Location

Montana Cancer Specialists

Missoula, Montana, 59802, United States

Location

Saint Patrick Hospital - Community Hospital

Missoula, Montana, 59802, United States

Location

University Medical Center of Southern Nevada

Las Vegas, Nevada, 89102, United States

Location

Nevada Cancer Research Foundation CCOP

Las Vegas, Nevada, 89106, United States

Location

University of Rochester

Rochester, New York, 14642, United States

Location

Mission Hospital-Memorial Campus

Asheville, North Carolina, 28801, United States

Location

Novant Health Presbyterian Medical Center

Charlotte, North Carolina, 28204, United States

Location

Wayne Memorial Hospital

Goldsboro, North Carolina, 27534, United States

Location

Margaret R Pardee Memorial Hospital

Hendersonville, North Carolina, 28791, United States

Location

Iredell Memorial Hospital

Statesville, North Carolina, 28677, United States

Location

Mary Rutan Hospital

Bellefontaine, Ohio, 43311, United States

Location

Adena Regional Medical Center

Chillicothe, Ohio, 45601, United States

Location

Good Samaritan Hospital - Cincinnati

Cincinnati, Ohio, 45220, United States

Location

University of Cincinnati

Cincinnati, Ohio, 45267, United States

Location

Riverside Methodist Hospital

Columbus, Ohio, 43214, United States

Location

Columbus CCOP

Columbus, Ohio, 43215, United States

Location

Grant Medical Center

Columbus, Ohio, 43215, United States

Location

Mount Carmel Health Center West

Columbus, Ohio, 43222, United States

Location

Doctors Hospital

Columbus, Ohio, 43228, United States

Location

Grandview Hospital

Dayton, Ohio, 45405, United States

Location

Good Samaritan Hospital - Dayton

Dayton, Ohio, 45406, United States

Location

Miami Valley Hospital

Dayton, Ohio, 45409, United States

Location

Samaritan North Health Center

Dayton, Ohio, 45415, United States

Location

Dayton CCOP

Dayton, Ohio, 45420, United States

Location

Grady Memorial Hospital

Delaware, Ohio, 43015, United States

Location

Blanchard Valley Hospital

Findlay, Ohio, 45840, United States

Location

Atrium Medical Center-Middletown Regional Hospital

Franklin, Ohio, 45005-1066, United States

Location

Wayne Hospital

Greenville, Ohio, 45331, United States

Location

Kettering Medical Center

Kettering, Ohio, 45429, United States

Location

Fairfield Medical Center

Lancaster, Ohio, 43130, United States

Location

Marietta Memorial Hospital

Marietta, Ohio, 45750, United States

Location

Knox Community Hospital

Mount Vernon, Ohio, 43050, United States

Location

Licking Memorial Hospital

Newark, Ohio, 43055, United States

Location

Springfield Regional Medical Center

Springfield, Ohio, 45505, United States

Location

Upper Valley Medical Center

Troy, Ohio, 45373, United States

Location

Saint Ann's Hospital

Westerville, Ohio, 43081, United States

Location

Clinton Memorial Hospital

Wilmington, Ohio, 45177, United States

Location

Greene Memorial Hospital

Xenia, Ohio, 45385, United States

Location

Genesis HealthCare System

Zanesville, Ohio, 43701, United States

Location

Adventist Medical Center

Portland, Oregon, 97216, United States

Location

SWOG

Portland, Oregon, 97239, United States

Location

AnMed Health Hospital

Anderson, South Carolina, 29621, United States

Location

McLeod Regional Medical Center

Florence, South Carolina, 29506, United States

Location

Spartanburg Regional Medical Center

Spartanburg, South Carolina, 29303, United States

Location

Upstate Carolina CCOP

Spartanburg, South Carolina, 29303, United States

Location

Wellmont Holston Valley Hospital and Medical Center

Kingsport, Tennessee, 37660, United States

Location

Thompson Cancer Survival Center

Knoxville, Tennessee, 37916, United States

Location

Danville Regional Medical Center

Danville, Virginia, 24541, United States

Location

Memorial Hospital Of Martinsville

Martinsville, Virginia, 24115, United States

Location

Cancer Care Center at Island Hospital

Anacortes, Washington, 98221, United States

Location

PeaceHealth Saint Joseph Medical Center

Bellingham, Washington, 98225, United States

Location

Harrison HealthPartners Hematology and Oncology-Bremerton

Bremerton, Washington, 98310, United States

Location

Highline Medical Center-Main Campus

Burien, Washington, 98166, United States

Location

Columbia Basin Hematology and Oncology PLLC

Kennewick, Washington, 99336, United States

Location

Evergreen Hospital Medical Center

Kirkland, Washington, 98033, United States

Location

Skagit Valley Hospital

Mount Vernon, Washington, 98274, United States

Location

Harrison HealthPartners Hematology and Oncology-Poulsbo

Poulsbo, Washington, 98370, United States

Location

Virginia Mason CCOP

Seattle, Washington, 98101, United States

Location

Harborview Medical Center

Seattle, Washington, 98104, United States

Location

Minor and James Medical PLLC

Seattle, Washington, 98104, United States

Location

Pacific Medical Center-First Hill

Seattle, Washington, 98104, United States

Location

Fred Hutchinson Cancer Research Center/University of Washington Cancer Consortium

Seattle, Washington, 98109, United States

Location

Group Health Cooperative-Seattle

Seattle, Washington, 98112, United States

Location

Swedish Medical Center-First Hill

Seattle, Washington, 98122-4307, United States

Location

The Polyclinic

Seattle, Washington, 98122, United States

Location

University of Washington Medical Center

Seattle, Washington, 98195, United States

Location

United General Hospital

Sedro-Woolley, Washington, 98284, United States

Location

Cancer Care Northwest - Spokane South

Spokane, Washington, 99202, United States

Location

Evergreen Hematology and Oncology PS

Spokane, Washington, 99218, United States

Location

Wenatchee Valley Medical Center

Wenatchee, Washington, 98801, United States

Location

Rocky Mountain Oncology

Casper, Wyoming, 82609, United States

Location

Welch Cancer Center

Sheridan, Wyoming, 82801, United States

Location

Related Publications (1)

  • Lee SM, Moon J, Redman BG, Chidiac T, Flaherty LE, Zha Y, Othus M, Ribas A, Sondak VK, Gajewski TF, Margolin KA. Phase 2 study of RO4929097, a gamma-secretase inhibitor, in metastatic melanoma: SWOG 0933. Cancer. 2015 Feb 1;121(3):432-440. doi: 10.1002/cncr.29055. Epub 2014 Sep 23.

MeSH Terms

Conditions

Melanoma

Interventions

2,2-dimethyl-N-(6-oxo-6,7-dihydro-5H-dibenzo(b,d)azepin-7-yl)-N'-(2,2,3,3,3-pentafluoropropyl)malonamide

Condition Hierarchy (Ancestors)

Neuroendocrine TumorsNeuroectodermal TumorsNeoplasms, Germ Cell and EmbryonalNeoplasms by Histologic TypeNeoplasmsNeoplasms, Nerve TissueNevi and MelanomasSkin NeoplasmsNeoplasms by SiteSkin DiseasesSkin and Connective Tissue Diseases

Results Point of Contact

Title
Melanoma Committee Statistician
Organization
SWOG Statistical Center

Study Officials

  • Kim Margolin

    SWOG Cancer Research Network

    PRINCIPAL INVESTIGATOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
LTE60
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
NIH
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 7, 2010

First Posted

May 10, 2010

Study Start

October 1, 2010

Primary Completion

May 1, 2013

Study Completion

August 1, 2015

Last Updated

June 14, 2016

Results First Posted

June 14, 2016

Record last verified: 2016-05

Locations