NCT00890825

Brief Summary

The purpose of this study is to compare the efficacy of AZD6244 in combination with docetaxel versus docetaxel alone in patients with KRAS mutation positive locally advanced or metastatic non small cell lung cancer.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
88

participants targeted

Target at P50-P75 for phase_2

Timeline
Completed

Started Apr 2009

Longer than P75 for phase_2

Geographic Reach
12 countries

63 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

April 20, 2009

Completed
9 days until next milestone

First Submitted

Initial submission to the registry

April 29, 2009

Completed
1 day until next milestone

First Posted

Study publicly available on registry

April 30, 2009

Completed
2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 11, 2011

Completed
5.5 years until next milestone

Study Completion

Last participant's last visit for all outcomes

November 2, 2016

Completed
1.6 years until next milestone

Results Posted

Study results publicly available

June 20, 2018

Completed
Last Updated

June 20, 2018

Status Verified

May 1, 2018

Enrollment Period

2.1 years

First QC Date

April 29, 2009

Results QC Date

June 14, 2017

Last Update Submit

May 22, 2018

Conditions

Keywords

Non small cell lung cancer (NSCLC)KRAS mutation

Outcome Measures

Primary Outcomes (1)

  • Overall Survival

    OS was calculated as the interval from the date of randomisation to the date of patient death (any cause). Patients who had not died at the time of the final analysis, or who withdrew consent, were censored at the last date the patient was known to be alive.

    At least 12 months since start of treatment.

Secondary Outcomes (6)

  • Progression Free Survival

    At least 12 months after start of treatment

  • Objective Response Rate

    At least 12 months after start of treatment

  • Duration of Response

    At least 12 months after start of treatment

  • Change From Baseline in Tumour Size at 6 Week.

    6 weeks after first dose of treatment

  • Change From Baseline in Tumour Size at Week 12

    12 weeks

  • +1 more secondary outcomes

Study Arms (2)

AZD6244 + Docetaxel

ACTIVE COMPARATOR

AZD6244 75 mg bd + Docetaxel 75 mg/m\^2

Drug: AZD6244Drug: docetaxel

Placebo + Docetaxel

PLACEBO COMPARATOR

Placebo + Docetaxel 75 mg/m\^2

Drug: docetaxelDrug: Placebo

Interventions

oral capsules, 75mg twice daily

Also known as: Selumetinib
AZD6244 + Docetaxel

75mg/m2 iv on day 1 of every 21 day cycle

Also known as: Taxotere
AZD6244 + DocetaxelPlacebo + Docetaxel

placebo

Placebo + Docetaxel

Eligibility Criteria

Age18 Years - 130 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Locally advanced or metastatic non small cell lung cancer (IIIB-IV)
  • Failure of first line anti-cancer therapy (either radiological documentation of disease progression or due to toxicity) in advanced disease or subsequent relapse of disease following first line therapy
  • Tumour sample confirmed as KRAS mutation positive (Note: Sample must be available upon enrolment to ship to AZ appointed central laboratory, or mutation status confirmed locally at AstraZeneca agreed local laboratory using agreed methodology, or mutation status confirmed by an accredited (eg CLIA certified) commercial laboratory (eg Genzyme or Lab 21).

You may not qualify if:

  • Received \>1 prior anti-cancer therapy for advanced or metastatic non small cell lung cancer (excluding radiotherapy)
  • Prior treatment with a MEK inhibitor or any docetaxel containing regimen (prior treatment with paclitaxel is acceptable)
  • Having received an investigational drug within 30 days of starting treatment, or have not recovered from side effects of an investigational drug
  • Brain metastases or spinal cord compression unless asymptomatic, treated and stable off steroids and anti-convulsants for at least 1 month

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (63)

Research Site

Los Angeles, California, 90095, United States

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Research Site

Aurora, Colorado, 80045, United States

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Boston, Massachusetts, 02115, United States

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Columbus, Ohio, 43210, United States

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Brussels, 1090, Belgium

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Charleroi, 6000, Belgium

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Edegem, 2650, Belgium

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Leuven, 3000, Belgium

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Liège, 4000, Belgium

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Liège, B-4000, Belgium

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Belo Horizonte, 30180-090, Brazil

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Ijuí, 98700-000, Brazil

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Porto Alegre, 90610-000, Brazil

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Rio de Janeiro, 20230-130, Brazil

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Santo André, 09060-650, Brazil

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São Paulo, 01221-020, Brazil

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São Paulo, 04023-062, Brazil

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São Paulo, 04530-001, Brazil

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Plovdiv, 4000, Bulgaria

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Sofia, 1233, Bulgaria

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Sofia, 1527, Bulgaria

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Sofia, 1756, Bulgaria

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Sofia, 1784, Bulgaria

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Varna, 9010, Bulgaria

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Oshawa, Ontario, L1G 2B9, Canada

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Ottawa, Ontario, K1H 8L6, Canada

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Toronto, Ontario, M5G 2M9, Canada

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Ostrava, 708 52, Czechia

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Prague, 180 81, Czechia

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Znojmo, 669 02, Czechia

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Brest, 29609, France

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Clermont-Ferrand, 63003, France

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Dijon, 21034, France

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Lyon, 69373, France

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Marseille, 13015, France

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Rennes, 35033, France

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Budapest, 1032, Hungary

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Budapest, 1121, Hungary

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Budapest, 1122, Hungary

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Budapest, 1125, Hungary

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Győr, 9024, Hungary

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Mosdós, 7257, Hungary

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Székesfehérvár, 8000, Hungary

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Törökbálint, 2045, Hungary

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Bologna, 40131, Italy

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Genova, 16100, Italy

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Milan, 20162, Italy

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Orbassano, 10043, Italy

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Perugia, 06132, Italy

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Roma, 00144, Italy

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Rozzano, 20089, Italy

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México, 14080, Mexico

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Morelia, 58000, Mexico

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Zacatecas City, 98000, Mexico

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Lima, LIMA 11, Peru

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Lima, LIMA 27, Peru

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Lima, LIMA 33, Peru

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Lima, LIMA 41, Peru

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A Coruña, 15006, Spain

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Badalona(Barcelona), 08916, Spain

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Research Site

Barcelona, 08028, Spain

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Madrid, 28041, Spain

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Research Site

Málaga, 29010, Spain

Location

Related Publications (2)

  • Janne PA, Smith I, McWalter G, Mann H, Dougherty B, Walker J, Orr MC, Hodgson DR, Shaw AT, Pereira JR, Jeannin G, Vansteenkiste J, Barrios CH, Franke FA, Crino L, Smith P. Impact of KRAS codon subtypes from a randomised phase II trial of selumetinib plus docetaxel in KRAS mutant advanced non-small-cell lung cancer. Br J Cancer. 2015 Jul 14;113(2):199-203. doi: 10.1038/bjc.2015.215. Epub 2015 Jun 30.

  • Janne PA, Shaw AT, Pereira JR, Jeannin G, Vansteenkiste J, Barrios C, Franke FA, Grinsted L, Zazulina V, Smith P, Smith I, Crino L. Selumetinib plus docetaxel for KRAS-mutant advanced non-small-cell lung cancer: a randomised, multicentre, placebo-controlled, phase 2 study. Lancet Oncol. 2013 Jan;14(1):38-47. doi: 10.1016/S1470-2045(12)70489-8. Epub 2012 Nov 28.

Related Links

MeSH Terms

Conditions

Carcinoma, Non-Small-Cell Lung

Interventions

AZD 6244Docetaxel

Condition Hierarchy (Ancestors)

Carcinoma, BronchogenicBronchial NeoplasmsLung NeoplasmsRespiratory Tract NeoplasmsThoracic NeoplasmsNeoplasms by SiteNeoplasmsLung DiseasesRespiratory Tract Diseases

Intervention Hierarchy (Ancestors)

TaxoidsCyclodecanesCycloparaffinsHydrocarbons, AlicyclicHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsDiterpenesTerpenes

Results Point of Contact

Title
Tracy Cunningham
Organization
AstraZeneca

Study Officials

  • Dr. Pasi Janne

    Dana-Farber Cancer Institute, Boston, USA

    PRINCIPAL INVESTIGATOR
  • Dr. Gabriella Mariani

    AstraZeneca, Hertfordshire, UK

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
LTE60
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 29, 2009

First Posted

April 30, 2009

Study Start

April 20, 2009

Primary Completion

May 11, 2011

Study Completion

November 2, 2016

Last Updated

June 20, 2018

Results First Posted

June 20, 2018

Record last verified: 2018-05

Locations