NCT00807859

Brief Summary

The purpose of this study is to determine if AMG 386 in combination with either paclitaxel and trastuzumab or capecitabine and lapatinib is safe and well tolerated in subjects with HER2-positive locally recurrent or metastatic breast cancer. This is an open-label phase 1b trial and has 2 study parts. Study part 1 is a dose escalation study to determine a tolerable dose of AMG 386 in combination with paclitaxel and trastuzumab (cohort A) or with capecitabine and lapatinib (cohort B). Study part 2 is cohort expansion of the tolerable doses determined in part 1.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
65

participants targeted

Target at P50-P75 for phase_1 breast-cancer

Timeline
Completed

Started Mar 2009

Longer than P75 for phase_1 breast-cancer

Geographic Reach
3 countries

23 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

December 11, 2008

Completed
1 day until next milestone

First Posted

Study publicly available on registry

December 12, 2008

Completed
3 months until next milestone

Study Start

First participant enrolled

March 9, 2009

Completed
5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 27, 2014

Completed
1.6 years until next milestone

Study Completion

Last participant's last visit for all outcomes

October 19, 2015

Completed
Last Updated

November 8, 2022

Status Verified

November 1, 2022

Enrollment Period

5 years

First QC Date

December 11, 2008

Last Update Submit

November 4, 2022

Conditions

Keywords

AMG 386PaclitaxelTrastuzumabCapecitabineLapatinibHER2-positivemetastatic breast cancerlocally recurrent breast cancerTaxolHerceptinXelodaTykerbanti-angiogenic therapy

Outcome Measures

Primary Outcomes (1)

  • Primary objective is to identify the incidence of adverse events and clinical laboratory abnormalities defined as a dose limiting toxicity in subjects treated with AMG 386 plus paclitaxel and trastuzumab or with AMG 386 plus capecitabine and lapatinib

    24 months

Secondary Outcomes (4)

  • To evaluate the incidence of adverse events and clinical laboratory abnormalities not defined as DLTs

    24 months

  • To evaluate the pharmacokinetics (PK) of AMG 386, trastuzumab, and paclitaxel (cohort A) or AMG 386, lapatinib, and capecitabine (and its active metabolite, 5-FU; cohort B) when administered in combination

    24 months

  • To estimate the incidence of anti AMG 386 antibody formation

    24 months

  • To evaluate the treatment effect as measured by the following: objective response rate (ORR), duration of response (DOR), change in tumor burden and progression-free survival (PFS)

    23 months

Study Arms (4)

Cohort A1

EXPERIMENTAL
Drug: AMG 386 10 mgkg, Paclitaxel and Trastuzumab

Cohort A3

EXPERIMENTAL
Drug: AMG 386 30 mg/kg, Paclitaxel and Trastuzumab

Cohort B1

EXPERIMENTAL
Drug: AMG 386 10 mg/kg, Capecitabine and Lapatinib

Cohort B3

EXPERIMENTAL
Drug: AMG 386 30 mg/kg, Capecitabine and Lapatinib

Interventions

AMG 386 30 mg/kg IV QW, paclitaxel 80 mg/m2 IV QW, trastuzumab: initial dose 8 mg/kg IV week 1, then 6 mg/kg IV Q3W

Cohort A3

AMG 386 30 mg/kg IV QW, capecitabine 2000 mg/m2 divided into 2 doses given PO Q12 hrs, days 1-14 every 21 days, lapatinib 1250 mg PO QD

Cohort B3

AMG 386 10 mg/kg IV QW, paclitaxel 80 mg/m2 IV QW, trastuzumab: initial dose 8 mg/kg IV week 1, then 6 mg/kg IV Q3W

Cohort A1

AMG 386 10 mg/kg IV QW, capecitabine 2000 mg/m2 divided into 2 doses given PO Q12 hrs, days 1-14 every 21 days, lapatinib 1250 mg PO QD

Cohort B1

Eligibility Criteria

Age18 Years+
Sexfemale
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • histologically or cytologically confirmed adenocarcinoma of the breast with locally recurrent or metastatic disease not amenable to any local treatment with curative intent.
  • HER2-positive by FISH, CISH, or IHC 3+
  • ECOG performance status 0 or 1
  • Left ventricular ejection fraction greater than or equal to institutional lower limit of normal
  • Adequate laboratory studies (hematological, chemistries and urinalysis)
  • Life expectancy greater than or equal to 3 months
  • Cohort A only:
  • Trastuzumab naïve or trastuzumab in the neo-adjuvant setting
  • No clinically significant drop in cardiac function prior exposure to trastuzumab
  • No prior chemotherapy for metastatic or locally recurrent breast cancer
  • No prior lapatinib therapy
  • At least 3 weeks from enrollment since prior chemotherapeutic agents, including taxanes, in the neoadjuvant or adjuvant setting
  • At least 3 months from enrollment since prior trastuzumab in the neoadjuvant or adjuvant setting
  • Cohort B only:
  • Must have failed trastuzumab in the first-line metastatic setting. Trastuzumab must be discontinued for at least 3 weeks prior to enrollment
  • +4 more criteria

You may not qualify if:

  • Inflammatory breast cancer
  • Central nervous system metastasis
  • Clinically significant cardiovascular disease
  • Radiation therapy ≤ 14 days prior to enrollment.
  • Concurrent anticoagulation therapy, excluding aspirin, anti-platelet agents, low molecular weight heparin or low dose warfarin per protocol.
  • Uncontrolled hypertension defined as diastolic blood pressure \> 90 mmHg OR systolic blood pressure \> 140 mmHg.
  • Subjects with a history of prior malignancy, except:
  • For Cohort B only:
  • Current or prior history of long QT syndrome
  • Baseline ECG report of QTc interval of \> 480 milliseconds
  • Severe chronic liver disease (Child Pugh C)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (23)

Research Site

Tucson, Arizona, 85724, United States

Location

Research Site

Boca Raton, Florida, 33428, United States

Location

Research Site

Iowa City, Iowa, 52242, United States

Location

Research Site

Boston, Massachusetts, 02111, United States

Location

Research Site

Minneapolis, Minnesota, 55407, United States

Location

Research Site

Lebanon, New Hampshire, 03756-0001, United States

Location

Research Site

Lebanon, New Hampshire, 03756, United States

Location

Research Site

Albuquerque, New Mexico, 87131, United States

Location

Research Site

Great Neck, New York, 11021, United States

Location

Research Site

New City, New York, 10956, United States

Location

Research Site

New York, New York, 10032, United States

Location

Research Site

Nyack, New York, 10960, United States

Location

Research Site

Middletown, Ohio, 45042, United States

Location

Research Site

Leuven, 3000, Belgium

Location

Research Site

Liège, 4000, Belgium

Location

Research Site

Wilrijk, 2610, Belgium

Location

Research Site

Bordeaux, 33075, France

Location

Research Site

Caen, 14076, France

Location

Research Site

La Roche-sur-Yon, 85925, France

Location

Research Site

Marseille, 13009, France

Location

Research Site

Nantes, 44202, France

Location

Research Site

Pierre Bénite Cedex, 69495, France

Location

Research Site

Toulouse, 31052, France

Location

Related Publications (1)

  • Kaufman PA, Wildiers H, Freyer G, Kemeny M, Goncalves A, Jerusalem G, Stopeck A, Vrindavanam N, Dalenc F, Nanayakkara N, Wu B, Pickett CA. Phase 1b Study of Trebananib Plus Paclitaxel and Trastuzumab in Patients With HER2-Positive Locally Recurrent or Metastatic Breast Cancer. Clin Breast Cancer. 2019 Feb;19(1):47-57. doi: 10.1016/j.clbc.2018.09.012. Epub 2018 Oct 9.

    PMID: 30420181BACKGROUND

Related Links

MeSH Terms

Conditions

Breast NeoplasmsNeoplasmsNeoplasm Metastasis

Interventions

trebananibPaclitaxelTrastuzumabCapecitabineLapatinib

Condition Hierarchy (Ancestors)

Neoplasms by SiteBreast DiseasesSkin DiseasesSkin and Connective Tissue DiseasesNeoplastic ProcessesPathologic ProcessesPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

TaxoidsCyclodecanesCycloparaffinsHydrocarbons, AlicyclicHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsDiterpenesTerpenesAntibodies, Monoclonal, HumanizedAntibodies, MonoclonalAntibodiesImmunoglobulinsImmunoproteinsBlood ProteinsProteinsAmino Acids, Peptides, and ProteinsSerum GlobulinsGlobulinsDeoxycytidineCytidinePyrimidine NucleosidesPyrimidinesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsFluorouracilUracilPyrimidinonesDeoxyribonucleosidesNucleosidesNucleic Acids, Nucleotides, and NucleosidesQuinazolinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-Ring

Study Officials

  • MD

    Amgen

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

December 11, 2008

First Posted

December 12, 2008

Study Start

March 9, 2009

Primary Completion

February 27, 2014

Study Completion

October 19, 2015

Last Updated

November 8, 2022

Record last verified: 2022-11

Locations