NCT00754988

Brief Summary

This 4 arm study will assess the efficacy, safety and tolerability of taspoglutide compared to sitagliptin and placebo in patients with type 2 diabetes mellitus inadequately controlled with metformin. Patients will be randomized to receive taspoglutide (10mg once weekly or 10mg once weekly for 4 weeks followed by 20mg once weekly), sitagliptin 100mg once daily or placebo, in a ratio of 2:2:2:1, in addition to their continued prestudy metformin treatment. After 24 weeks of treatment, patients on active treatment will continue on the same treatment and patients on placebo will be switched to taspoglutide 10mg once weekly or taspoglutide 20mg once weekly (after 4 weeks of taspoglutide 10mg once weekly). The anticipated time on study treatment is 2+ years, and the target sample size is 500+ individuals.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
666

participants targeted

Target at P50-P75 for phase_3 diabetes-mellitus-type-2

Timeline
Completed

Started Oct 2008

Typical duration for phase_3 diabetes-mellitus-type-2

Geographic Reach
23 countries

148 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 17, 2008

Completed
1 day until next milestone

First Posted

Study publicly available on registry

September 18, 2008

Completed
13 days until next milestone

Study Start

First participant enrolled

October 1, 2008

Completed
2.4 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 1, 2011

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

March 1, 2011

Completed
Last Updated

November 4, 2016

Status Verified

November 1, 2016

Enrollment Period

2.4 years

First QC Date

September 17, 2008

Last Update Submit

November 3, 2016

Conditions

Outcome Measures

Primary Outcomes (1)

  • Mean changes in HbA1c

    24 weeks

Secondary Outcomes (2)

  • Change from baseline in fasting plasma glucose; change from baseline in body weight; responder rates for HbA1c (target <=7.0%, <=6.5%); responder rates for body weight; change from baseline in lipid profile; beta cell function.

    24 weeks

  • Safety: Adverse events, vital signs, physical examination, clinical laboratory tests, ECG and anti-taspoglutide antibodies.

    Throughout study

Study Arms (4)

Placebo

PLACEBO COMPARATOR

Once daily oral administration of placebo (matching sitagliptin). Once weekly sc injection of placebo (matching taspoglutide). Continued treatment with metformin at prescribed doses.

Drug: MetforminDrug: Placebo (matching sitagliptin)Drug: Placebo (matching taspoglutide)

Sitagliptin

ACTIVE COMPARATOR

Once daily oral administration of 100 mg of sitagliptin. Once weekly sc injection of placebo (matching taspoglutide). Continued treatment with metformin at prescribed doses.

Drug: MetforminDrug: Placebo (matching taspoglutide)Drug: Sitagliptin

Taspoglutide 10 mg

EXPERIMENTAL

Once weekly subcutaneous (sc) injection of 10 mg of taspoglutide. Once daily oral administration of placebo (matching sitagliptin). Continued treatment with metformin at prescribed doses.

Drug: MetforminDrug: Placebo (matching sitagliptin)Drug: Taspoglutide

Taspoglutide up-titrated to 20 mg

EXPERIMENTAL

Once weekly sc injection of 10 mg of taspoglutide for the first 4 weeks, then up-titrated to once weekly sc injection of 20 mg of taspoglutide from week 5 onwards. Once daily oral administration of placebo (matching sitagliptin). Continued treatment with metformin at prescribed doses.

Drug: MetforminDrug: Placebo (matching sitagliptin)Drug: Taspoglutide

Interventions

As prescribed

PlaceboSitagliptinTaspoglutide 10 mgTaspoglutide up-titrated to 20 mg

Once daily oral administration of placebo (matching sitagliptin).

PlaceboTaspoglutide 10 mgTaspoglutide up-titrated to 20 mg

Once weekly subcutaneous (sc) injection of placebo (matching taspoglutide).

PlaceboSitagliptin

Once daily oral administration of 100 mg of sitagliptin.

Sitagliptin

Once weekly subcutaneous (sc) injection of 10 mg or 20 mg of taspoglutide.

Taspoglutide 10 mgTaspoglutide up-titrated to 20 mg

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • adult patients, 18-75 years of age;
  • type 2 diabetes receiving metformin (\>=1500mg/day) for at least 12 weeks;
  • HbA1c \>=7.0% and \<=10.0% at screening;
  • BMI \>=25 (\>23 for Asians) and \<=45kg/m2 at screening;
  • stable weight +/- 5% for at least 12 weeks prior to screening.

You may not qualify if:

  • history of type 1 diabetes mellitus or acute metabolic diabetic complications such as ketoacidosis or hyperosmolar coma in the previous 6 months;
  • evidence of clinically significant diabetic complications;
  • clinically symptomatic gastrointestinal disease;
  • myocardial infarction, coronary artery bypass surgery, post-transplantation cardiomyopathy or stroke within the previous 6 months;
  • known hemoglobinopathy or chronic anemia.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (148)

Unknown Facility

Birmingham, Alabama, 35233, United States

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Huntsville, Alabama, 35802, United States

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Tallassee, Alabama, 36078, United States

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Scottsdale, Arizona, 85254, United States

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Little Rock, Arkansas, 72205, United States

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Huntington Beach, California, 92646, United States

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La Jolla, California, 92037, United States

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Los Angeles, California, 90017, United States

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Roseville, California, 95661, United States

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San Francisco, California, 94109, United States

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Tacoma, California, 98405, United States

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Colorado Springs, Colorado, 80904, United States

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New London, Connecticut, 06320, United States

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Manati, District of Columbia, 00674, United States

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Daytona Beach, Florida, 32117, United States

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Hialeah, Florida, 33012, United States

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Jacksonville, Florida, 32205, United States

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Miami, Florida, 33186, United States

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Panama City, Florida, 32401, United States

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Tampa, Florida, 33606, United States

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Augusta, Georgia, 30904, United States

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Conyers, Georgia, 30094, United States

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Snellville, Georgia, 30029, United States

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Honolulu, Hawaii, 96813, United States

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Indianapolis, Indiana, 46229, United States

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Indianapolis, Indiana, 46254, United States

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Lafayette, Indiana, 47905, United States

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South Bend, Indiana, 46628, United States

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Baltimore, Maryland, 21229, United States

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Brockton, Massachusetts, 02301, United States

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Cadillac, Michigan, 49601, United States

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Brooklyn Center, Minnesota, 55430, United States

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Minneapolis, Minnesota, 55416, United States

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City of Saint Peters, Missouri, 63376, United States

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Fulton, New York, 13069, United States

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Hudson, New York, 12534, United States

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Rochester, New York, 14609, United States

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Charlotte, North Carolina, 28211, United States

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Raleigh, North Carolina, 27609, United States

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Shelby, North Carolina, 28150, United States

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Statesville, North Carolina, 28625, United States

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Winston-Salem, North Carolina, 27103, United States

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Columbus, Ohio, 43213, United States

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Delaware, Ohio, 43015, United States

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Marion, Ohio, 43302, United States

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Corvallis, Oregon, 97330, United States

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Eugene, Oregon, 97401, United States

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Aliquippa, Pennsylvania, 15001, United States

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Beaver, Pennsylvania, 15009, United States

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Erie, Pennsylvania, 16508, United States

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Reading, Pennsylvania, 17601, United States

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Reading, Pennsylvania, 19606, United States

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Shippensburg, Pennsylvania, 17257, United States

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Warminster, Pennsylvania, 18974, United States

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Anderson, South Carolina, 29621, United States

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Kingsport, Tennessee, 37660, United States

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Dallas, Texas, 75230, United States

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Houston, Texas, 77030, United States

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South Burlington, Vermont, 05403, United States

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Hampton, Virginia, 23666, United States

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Norfolk, Virginia, 23502, United States

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Richmond, Virginia, 23249, United States

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Richmond, Virginia, 23294, United States

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Federal Way, Washington, 98003, United States

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Buenos Aires, C1012, Argentina

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Buenos Aires, C1213AAH, Argentina

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Mar del Plata, B7600DHK, Argentina

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Freemantle, Queensland, 6959, Australia

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Adelaide, South Australia, 5000, Australia

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London, Ontario, N6A 4V2, Canada

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Thornhill, Ontario, L4J 8L7, Canada

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Toronto, Ontario, M9W 4L6, Canada

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Montreal, Quebec, H2W 1T8, Canada

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Pointe-Claire, Quebec, H9R 4S3, Canada

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Bondy, 93143, France

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Nantes, 44093, France

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Poitiers, 86021, France

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Rennes, 35203, France

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Saint-Mandé, 94163, France

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Berlin, 10115, Germany

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Dormagen, 41539, Germany

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Dresden, 01307, Germany

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Kiel Kronshagen, 24119, Germany

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München, 80336, Germany

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Sulzbach-Rosenberg, 92237, Germany

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Villingen-Schwenningen, 78048, Germany

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Larissa, 41110, Greece

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Cuernavaca, 62250, Mexico

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Hermosillo, 83200, Mexico

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Jalisco, 44690, Mexico

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Mexico City, 06700, Mexico

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Mexico City, 11520, Mexico

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Monterrey, 64000, Mexico

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Pachuca, 42086, Mexico

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Elverum, 2401, Norway

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Oslo, 0027, Norway

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Oslo, 0176, Norway

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Oslo, 0407, Norway

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Lima, Lima 33, Peru

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Lima, Lima 9, Peru

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Bialystok, 15-445, Poland

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Gdansk, 80-858, Poland

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Kamieniec Ząbkowicki, 57-230, Poland

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Rzeszów, 35-073, Poland

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Skierniewice, 96-100, Poland

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Sobótka, 55-050, Poland

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Wroclaw, 51-124, Poland

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Caguas, 00725, Puerto Rico

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Carolina, 00983, Puerto Rico

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Bucharest, 020359, Romania

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Buzău, 120203, Romania

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Cluj-Napoca, 400006, Romania

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Ploieşti, 100163, Romania

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Ploieşti, 100342, Romania

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Levice, 93405, Slovakia

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Prešov, 080 01, Slovakia

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Šamorín, 931 01, Slovakia

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Trebišov, 07501, Slovakia

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Trenčín, 911 01, Slovakia

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Cape Town, 7130, South Africa

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Pretoria, 0002, South Africa

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Gyeonggi-do, 443-380, South Korea

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Gyeonggi-do, South Korea

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Seoul, 152-703, South Korea

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Seoul, South Korea

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Wŏnju, 220-701, South Korea

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Bacarot Alicant, Alicante, 03114, Spain

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Almería, Almeria, 04001, Spain

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Seville, Sevilla, 41010, Spain

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Valencia, Valencia, 46014, Spain

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Ljungby, 34182, Sweden

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Örebro, 701 85, Sweden

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Stockholm, 14186, Sweden

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Basel, 4031, Switzerland

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Geneva, 1211, Switzerland

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Zurich, 8063, Switzerland

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Taichung, 407, Taiwan

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Taipei, 114, Taiwan

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Taipei, 220, Taiwan

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Taoyuan, 333, Taiwan

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Bangkok, 10330, Thailand

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Songkhla, 90112, Thailand

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Istanbul, 34390, Turkey (Türkiye)

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Bexhill-on-Sea, TN39 4SP, United Kingdom

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Crawley, RH10 7DX, United Kingdom

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Glasgow, G46 8NY, United Kingdom

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Hinckley, LE10 2SE, United Kingdom

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Reading, RG7 3SQ, United Kingdom

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MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

MetforminSitagliptin Phosphatetaspoglutide

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

BiguanidesGuanidinesAmidinesOrganic ChemicalsTriazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPyrazines

Study Officials

  • Clinical Trials

    Hoffmann-La Roche

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 17, 2008

First Posted

September 18, 2008

Study Start

October 1, 2008

Primary Completion

March 1, 2011

Study Completion

March 1, 2011

Last Updated

November 4, 2016

Record last verified: 2016-11

Locations