NCT00526617

Brief Summary

This Phase I clinical trial is studying the side effects and best dose of ABT-888 when given together with Temozolomide (chemotherapy) in treating patients with solid tumors, including metastatic melanoma (MM), BRCA deficient breast, ovarian, primary peritoneal, or fallopian tube cancer, and hepatocellular carcinoma (HCC).

Trial Health

100
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
41

participants targeted

Target at P50-P75 for phase_1

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

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Study Timeline

Key milestones and dates

Study Start

First participant enrolled

August 1, 2007

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

September 5, 2007

Completed
5 days until next milestone

First Posted

Study publicly available on registry

September 10, 2007

Completed
2.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 1, 2010

Completed
Last Updated

November 21, 2017

Status Verified

January 1, 2012

Enrollment Period

2.8 years

First QC Date

September 5, 2007

Last Update Submit

November 17, 2017

Conditions

Keywords

Solid TumorMelanomaBreast cancerOvarian cancerPrimary peritoneal cancerFallopian tube cancerHepatocellular carcinomaHCCBRCA deficientBRCA mutationTemozolomideTemodarTMZABT-888PARP inhibitor

Outcome Measures

Primary Outcomes (3)

  • Maximum Tolerated Dose

    Duration of Study

  • Safety and Tolerability

    Duration of Study

  • Pharmacokinetic Profile

    Duration of Study

Study Arms (1)

Open Label

EXPERIMENTAL

Within each dose level, subjects are treated with the same regimen/doses of ABT-888 and TMZ.

Drug: ABT-888Drug: Temozolomide

Interventions

Oral capsules

Open Label

Oral capsules

Also known as: Temodar, TMZ
Open Label

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Dose escalation and expanded safety cohorts
  • Evaluable disease, histologically confirmed malignancy (metastatic or unresectable) and standard curative measures or other therapy that may provide clinical benefit do not exist or are no longer effective
  • ECOG Performance Score less than or equal to 2
  • Adequate hematologic, renal and hepatic function
  • Normal sodium, calcium and magnesium levels
  • Voluntarily signed informed consent
  • Expanded Safety Cohorts Only
  • Population:
  • Metastatic melanoma (MM)
  • Hepatocellular carcinoma (HCC) Child Pugh Category A and B classification only
  • BRCA deficient tumor status\*: advanced breast cancer (with soft tissue disease), or advanced ovarian cancer, or advanced primary peritoneal cancer, or advanced fallopian tube cancer\*
  • \*Patients must have histologically or cytologically confirmed solid tumors with a positive genetic test result documenting BRCA 1 or BRCA 2 mutation status, to be considered eligible.
  • Serial tumor biopsies: Required for all subjects enrolled in one of the Expanded Low Dose Safety Cohorts.

You may not qualify if:

  • Dose Escalation and Expanded Safety Cohorts
  • Known central nervous system (CNS) metastases or CNS primary cancer.
  • Previous or current malignancies at other sites, except: adequately treated in situ carcinoma of cervix uteri; basal/squamous cell carcinoma of skin; previous malignancy considered cured.
  • Previous history or current seizure disorder.
  • Clinically significant and uncontrolled major medical condition(s) or any medical condition that places the subject at an unacceptably high risk for toxicities.
  • Transplant recipients and patients receiving combination anti-retroviral therapy for HIV due to the use of immunosuppressant therapies.
  • Lactating or pregnant female.
  • Chemotherapy, immunotherapy, radiotherapy, biologic or any investigational therapy will not be allowed within either 4 weeks, or 5 half lives of a targeted therapy prior to study drug administration (Study Day 1).
  • Prior therapy with regimens containing dacarbazine (DTIC) or TMZ is not permitted.
  • Anti-cancer therapy is not permitted during the treatment portion of the study.
  • Hormone therapy, bisphosphonates or LHRH-agonists for prostate cancer are permitted prior to and during the study.
  • Significant adverse event or toxicity due to previous anti-cancer treatment that has not recovered to within one grade level (not to exceed Grade 2) of baseline.
  • Expanded Safety Cohorts Only:
  • MM Only: Prior treatment with DNA damaging agents or cytotoxic chemotherapy including carboplatin, cisplatin, fotemustine, paclitaxel, vincristine, TMZ and DTIC.
  • Prior therapy with biologic agents (including IL-2, interferon, bevacizumab, vaccines and immunostimulants) and signal transduction inhibitors (including sorafenib, erlotinib, sutent and elesclomol) are allowed.
  • +2 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Related Publications (1)

  • Nuthalapati S, Munasinghe W, Giranda V, Xiong H. Clinical Pharmacokinetics and Mass Balance of Veliparib in Combination with Temozolomide in Subjects with Nonhematologic Malignancies. Clin Pharmacokinet. 2018 Jan;57(1):51-58. doi: 10.1007/s40262-017-0547-z.

MeSH Terms

Conditions

MelanomaBreast NeoplasmsOvarian NeoplasmsFallopian Tube NeoplasmsCarcinoma, Hepatocellular

Interventions

veliparibTemozolomide

Condition Hierarchy (Ancestors)

Neuroendocrine TumorsNeuroectodermal TumorsNeoplasms, Germ Cell and EmbryonalNeoplasms by Histologic TypeNeoplasmsNeoplasms, Nerve TissueNevi and MelanomasSkin NeoplasmsNeoplasms by SiteSkin DiseasesSkin and Connective Tissue DiseasesBreast DiseasesEndocrine Gland NeoplasmsOvarian DiseasesAdnexal DiseasesGenital Diseases, FemaleFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesGenital Neoplasms, FemaleUrogenital NeoplasmsGenital DiseasesEndocrine System DiseasesGonadal DisordersFallopian Tube DiseasesAdenocarcinomaCarcinomaNeoplasms, Glandular and EpithelialLiver NeoplasmsDigestive System NeoplasmsDigestive System DiseasesLiver Diseases

Intervention Hierarchy (Ancestors)

DacarbazineTriazenesOrganic ChemicalsImidazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Officials

  • Bhardwaj Desai, MD

    Abbott

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 5, 2007

First Posted

September 10, 2007

Study Start

August 1, 2007

Primary Completion

June 1, 2010

Last Updated

November 21, 2017

Record last verified: 2012-01