NCT06597019

Brief Summary

This is a pivotal phase III study designed to evaluate safety, tolerability, and efficacy of inclisiran in children (aged 6 to \<12 years) with heterozygous familial hypercholesterolemia (HeFH) and elevated low density lipoprotein cholesterol (LDLC).

Trial Health

88
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
51

participants targeted

Target at below P25 for phase_3

Timeline
36mo left

Started Dec 2024

Typical duration for phase_3

Geographic Reach
23 countries

66 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress32%
Dec 2024Apr 2029

First Submitted

Initial submission to the registry

September 11, 2024

Completed
8 days until next milestone

First Posted

Study publicly available on registry

September 19, 2024

Completed
3 months until next milestone

Study Start

First participant enrolled

December 9, 2024

Completed
3.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 21, 2028

Expected
1.1 years until next milestone

Study Completion

Last participant's last visit for all outcomes

April 15, 2029

Last Updated

November 21, 2025

Status Verified

November 1, 2025

Enrollment Period

3.3 years

First QC Date

September 11, 2024

Last Update Submit

November 20, 2025

Conditions

Keywords

Heterozygous familial hypercholesterolemia (HeFH),LDL-cholesterol (LDL-C),Children,pediatric,small interfering ribonucleic acid (siRNA),inclisiran,Familial Hypercholesterolemia,Heterozygous FH,Hypercholesterolemia,Lipoprotein(a),Hyperlipidemia,Dyslipidemia,Heart Failure,Cardiovascular Diseases,Cholesterol,Aortic Stenosis

Outcome Measures

Primary Outcomes (1)

  • Percentage change in LDL-C from baseline to Day 330 (Year 1)

    Demonstrate superiority of inclisiran compared to placebo in reducing LDL-C \[percent change\] at Day 330

    Baseline and Day 330

Secondary Outcomes (13)

  • Time-adjusted percent change in LDL-C from baseline after Day 90 and up to Day 330 (Year 1)

    Baseline, after Day 90 up to Day 330

  • Absolute change in LDL-C from baseline to Day 330 (Year 1)

    Baseline and Day 330

  • Percent change in PCSK9 from baseline to Day 330 (Year 1)

    Baseline and Day 330

  • Percent change in total cholesterol, non-HDL-C from baseline to Day 330 (Year 1)

    Baseline and Day 330

  • Percent change in Apo B from baseline to Day 330 (Year 1)

    Baseline and Day 330

  • +8 more secondary outcomes

Study Arms (2)

Inclisiran

EXPERIMENTAL

Year 1 - inclisiran sodium subcutaneous injection (given at Days 1, 90, and 270) Day 360 only - placebo subcutaneous injection Year 2 - inclisiran sodium subcutaneous injection (given at Days 450 and 630)

Drug: Inclisiran

Placebo

PLACEBO COMPARATOR

Year 1 - placebo subcutaneous injection (given at Days 1, 90 and 270) Year 2 - inclisiran sodium subcutaneous injection (given at Days 360, 450, and 630)

Drug: Placebo

Interventions

Inclisiran (inclisiran sodium 300 mg subcutaneous (s.c.) for participants with body weight ≥23 kg and inclisiran sodium 180 mg s.c. for participants with body weight \<23 kg. The dose level is based on the participant's body weight on Day 1 (for Part 1) and Day 360 (for Part 2), respectively.

Also known as: KJX839
Inclisiran

Sterile normal saline (0.9% sodium chloride in water for subcutaneous injection)

Also known as: saline solution
Placebo

Eligibility Criteria

Age6 Years - 11 Years
Sexall
Healthy VolunteersNo
Age GroupsChild (0-17)

You may qualify if:

  • Male or female participants, 6 to \<12 years of age at screening
  • HeFH diagnosed either by genetic testing or on phenotypic criteria
  • Fasting LDL-C \>130 mg/dL (3.4 mmol/L) at screening
  • For participants 8 to \<12 years, on an optimal dose of statin (investigator's discretion) unless statin intolerant, with or without other lipid-lowering therapy (e.g. ezetimibe). For participants \<8 years, the use of background lipid-lowering treatment is based on investigator's discretion.
  • Participants on lipid-lowering therapies (such as statin and/or e.g. ezetimibe) must be on a stable dose for ≥30 days before screening with no planned medication or dose changes during study participation.

You may not qualify if:

  • Previous treatment (within 90 days of screening) with monoclonal antibodies directed towards PCSK9
  • Secondary hypercholesterolemia, e.g. hypothyroidism or nephrotic syndrome
  • Homozygous familial hypercholesterolemia (HoFH)
  • Body weight \<16 kg at the screening and/or randomization (Day 1) visit
  • Active liver disease defined as any known current infectious, neoplastic, or metabolic pathology of the liver or unexplained alanine aminotransferase (ALT), aspartate aminotransferase (AST) elevation \>3x ULN, or total bilirubin elevation \>2x ULN (except patients with Gilbert's syndrome)
  • Pregnant or nursing females
  • Recent and/or planned use of other investigational medicinal products or devices

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (66)

UC San Francisco Medical Center

San Francisco, California, 94143, United States

RECRUITING

UC San Francisco Medical Center

San Francisco, California, 94143, United States

RECRUITING

Children's National Hospital

Washington D.C., District of Columbia, 20010, United States

NOT YET RECRUITING

Childrens National Hospital

Washington D.C., District of Columbia, 20010, United States

RECRUITING

Excel Medical Clinical Trials LLC

Boca Raton, Florida, 33434, United States

RECRUITING

Icahn School of Med at Mt Sinai

New York, New York, 10029, United States

RECRUITING

Primary Childrens Medical Center

Salt Lake City, Utah, 84113, United States

NOT YET RECRUITING

Primary Childrens Medical Center

Salt Lake City, Utah, 84113, United States

RECRUITING

Virginia Commonwealth University

Richmond, Virginia, 23298, United States

RECRUITING

West Virginia Childrens Hospital

Morgantown, West Virginia, 26506, United States

RECRUITING

West Virginia Childrens Hospital

Morgantown, West Virginia, 26506, United States

RECRUITING

Novartis Investigative Site

Buenos Aires, C1245AAM, Argentina

RECRUITING

Novartis Investigative Site

CABA, C1181ACH, Argentina

RECRUITING

Novartis Investigative Site

Salzburg, 5020, Austria

RECRUITING

Novartis Investigative Site

Vienna, 1090, Austria

RECRUITING

Novartis Investigative Site

Brussels, 1200, Belgium

RECRUITING

Novartis Investigative Site

Leuven, 3000, Belgium

RECRUITING

Novartis Investigative Site

Fortaleza, Ceará, 60430-275, Brazil

RECRUITING

Novartis Investigative Site

Rio de Janeiro, Rio de Janeiro, 20211-340, Brazil

RECRUITING

Novartis Investigative Site

Porto Alegre, Rio Grande do Sul, 90020-020, Brazil

RECRUITING

Novartis Investigative Site

São Paulo, São Paulo, 05403 000, Brazil

RECRUITING

Novartis Investigative Site

Beijing, Beijing Municipality, 100013, China

RECRUITING

Novartis Investigative Site

Shanghai, 200127, China

RECRUITING

Novartis Investigative Site

Prague, 128 08, Czechia

RECRUITING

Novartis Investigative Site

Prague, 150 06, Czechia

RECRUITING

Novartis Investigative Site

Marseille, 13885, France

RECRUITING

Novartis Investigative Site

Nantes, 44093, France

RECRUITING

Novartis Investigative Site

Paris, 75012, France

RECRUITING

Novartis Investigative Site

Freiburg im Breisgau, Baden-Wurttemberg, 79106, Germany

RECRUITING

Novartis Investigative Site

Frankfurt am Main, Hesse, 60590, Germany

RECRUITING

Novartis Investigative Site

Hanover, 30173, Germany

RECRUITING

Novartis Investigative Site

Athens, 115 27, Greece

RECRUITING

Novartis Investigative Site

Ioannina, 455 00, Greece

RECRUITING

Novartis Investigative Site

Hong Kong, 999077, Hong Kong

RECRUITING

Novartis Investigative Site

Budapest, 1026, Hungary

RECRUITING

Novartis Investigative Site

Jerusalem, 9112001, Israel

RECRUITING

Novartis Investigative Site

Ramat Gan, 5265601, Israel

RECRUITING

Novartis Investigative Site

Milan, MI, 20162, Italy

RECRUITING

Novartis Investigative Site

Roma, RM, 00165, Italy

RECRUITING

Novartis Investigative Site

Torino, TO, 10126, Italy

RECRUITING

Novartis Investigative Site

Verona, VR, 3712, Italy

RECRUITING

Novartis Investigative Site

Kuala Lumpur, Kuala Lumpur, 50586, Malaysia

RECRUITING

Novartis Investigative Site

Amsterdam, North Holland, 1105 AZ, Netherlands

RECRUITING

Novartis Investigative Site

Bialystok, 15-274, Poland

RECRUITING

Novartis Investigative Site

Gdansk, 80 952, Poland

RECRUITING

Novartis Investigative Site

Lodz, Łódź Voivodeship, 93-338, Poland

RECRUITING

Novartis Investigative Site

Coimbra, 3000-602, Portugal

RECRUITING

Novartis Investigative Site

Lisbon, 1649-035, Portugal

RECRUITING

Novartis Investigative Site

Porto, 4050-651, Portugal

RECRUITING

Novartis Investigative Site

Porto, 4200 319, Portugal

RECRUITING

Novartis Investigative Site

Bloemfontein, Free State, 9301, South Africa

RECRUITING

Novartis Investigative Site

Elche, Alicante, 03203, Spain

RECRUITING

Novartis Investigative Site

Cadiz, Andalusia, 11009, Spain

RECRUITING

Novartis Investigative Site

Esplugues, Barcelona, 08950, Spain

RECRUITING

Novartis Investigative Site

Badalona, Catalonia, 08916, Spain

RECRUITING

Novartis Investigative Site

Pamplona, Navarre, 31008, Spain

RECRUITING

Novartis Investigative Site

Barcelona, 08041, Spain

RECRUITING

Novartis Investigative Site

Málaga, 29011, Spain

RECRUITING

Novartis Investigative Site

Seville, 41013, Spain

RECRUITING

Novartis Investigative Site

Taipei, 111045, Taiwan

RECRUITING

Novartis Investigative Site

Taipei, 11217, Taiwan

RECRUITING

Novartis Investigative Site

Adana, Saricam, 01330, Turkey (Türkiye)

RECRUITING

Novartis Investigative Site

Ankara, Yenimahalle, 06500, Turkey (Türkiye)

RECRUITING

Novartis Investigative Site

Izmir, 35100, Turkey (Türkiye)

RECRUITING

Novartis Investigative Site

West Midlands, Birmingham, B4 6NH, United Kingdom

RECRUITING

Novartis Investigative Site

London, NW3 2QG, United Kingdom

RECRUITING

MeSH Terms

Conditions

Hyperlipoproteinemia Type IIHypercholesterolemiaHyperlipidemiasDyslipidemiasHeart FailureCardiovascular DiseasesAortic Valve Stenosis

Interventions

ALN-PCSSaline Solution

Condition Hierarchy (Ancestors)

Lipid Metabolism, Inborn ErrorsMetabolism, Inborn ErrorsGenetic Diseases, InbornCongenital, Hereditary, and Neonatal Diseases and AbnormalitiesHyperlipoproteinemiasLipid Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesHeart DiseasesAortic Valve DiseaseHeart Valve DiseasesVentricular Outflow Obstruction

Intervention Hierarchy (Ancestors)

Crystalloid SolutionsIsotonic SolutionsSolutionsPharmaceutical Preparations

Study Officials

  • Novartis Pharmaceuticals

    Novartis Pharmaceuticals

    STUDY DIRECTOR

Central Study Contacts

Novartis Pharmaceuticals

CONTACT

Novartis Pharmaceuticals

CONTACT

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Masking Details
Masked (Year 1) to No Masking (Year 2)
Purpose
TREATMENT
Intervention Model
PARALLEL
Model Details: Parallel (Year 1) to single-group (Year 2)
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 11, 2024

First Posted

September 19, 2024

Study Start

December 9, 2024

Primary Completion (Estimated)

March 21, 2028

Study Completion (Estimated)

April 15, 2029

Last Updated

November 21, 2025

Record last verified: 2025-11

Data Sharing

IPD Sharing
Will share

Novartis is committed to sharing with qualified external researchers, access to patient-level data and supporting clinical documents from eligible studies. These requests are reviewed and approved by an independent review panel on the basis of scientific merit. All data provided is anonymized to respect the privacy of patients who have participated in the trial in line with applicable laws and regulations. This trial data availability is according to the criteria and process described on www.clinicalstudydatarequest.com.

Locations