NCT06347133

Brief Summary

This Phase 3 study will evaluate the safety and efficacy of plozasiran injection (ARO-APOC3) in adult participants with hypertriglyceridemia (HTG). After providing informed consent eligible participants will be randomized to receive 4 doses (once every 3 months) of plozasiran or placebo and be evaluated for efficacy and safety.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
1,456

participants targeted

Target at P75+ for phase_3

Timeline
4mo left

Started May 2024

Geographic Reach
15 countries

235 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress86%
May 2024Sep 2026

First Submitted

Initial submission to the registry

March 29, 2024

Completed
6 days until next milestone

First Posted

Study publicly available on registry

April 4, 2024

Completed
2 months until next milestone

Study Start

First participant enrolled

May 21, 2024

Completed
1.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 1, 2026

Completed
4 months until next milestone

Study Completion

Last participant's last visit for all outcomes

September 1, 2026

Expected
Last Updated

October 8, 2025

Status Verified

October 1, 2025

Enrollment Period

1.9 years

First QC Date

March 29, 2024

Last Update Submit

October 3, 2025

Conditions

Outcome Measures

Primary Outcomes (1)

  • Percent Change in Fasting Serum Triglyceride (TG) Levels from Baseline to Month 12 Compared to Placebo

    Baseline, Month 12

Secondary Outcomes (17)

  • Percent Change in Fasting Serum TG Levels from Baseline to Month 10 Compared to Placebo

    Baseline, Month 10

  • Proportion of Participants who Achieve Fasting TG Levels of <150 mg/dL (<1.69 mmol/L) at Month 12 Compared to Placebo

    Month 12

  • Percent change in remnant cholesterol (VLDL-C) from baseline to Month 12 compared to placebo.

    Baseline, Month 12

  • Percent change in non-HDL-C from baseline to Month 12 compared to placebo

    Baseline, Month 12

  • Number of Participants with Adverse Events (AEs) and Serious Adverse Events (SAEs) Over Time through Month 12 as Compared to Placebo

    From first dose of study drug through Month 12

  • +12 more secondary outcomes

Study Arms (2)

Plozasiran Injection

EXPERIMENTAL

4 doses of plozasiran by subcutaneous (sc) injection

Drug: Plozasiran Injection

Placebo

PLACEBO COMPARATOR

calculated volume to match active treatment by sc injection

Drug: Placebo

Interventions

ARO-APOC3 Injection

Also known as: ARO-APOC3
Plozasiran Injection

sterile normal saline (0.9% NaCl)

Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Males, or nonpregnant (who do not plan to become pregnant) nonlactating females, who are ≥18 years of age at screening
  • Established diagnosis of hypertriglyceridemia (HTG) and prior documented evidence (medical history) of mean fasting TG level ≥150 mg/dL (≥1.69 mm/L) and ≤499 mg/dL (≤5.64 mmol/L)
  • Mean fasting TG level ≥150 mg/dL (≥1.69 mmol/L) and ≤499 mg/dL (≤5.64 mmol/L) collected at 2 separate and consecutive visits at least 7 days apart and no more than 17 days apart during the screening period
  • Fasting low density lipoprotein-cholesterol (LDL-C) ≤ 130 mg/dL (≤3.37 mmol/L) at screening
  • Screening HbA1c ≤9.0%
  • Willing to follow diet counseling and maintain a stable low-fat diet
  • Must be on standard of care lipid and TG-lowering medications per local guidelines (unless documented as intolerant as determined by the Investigator, including an inability to safely administer or re-administer a specific drug because of fear, preference, genetic, clinical, or metabolic considerations, or due a previous adverse reaction associated with, attributed to, or caused by specific drug) prior to collection of qualifying TG levels.

You may not qualify if:

  • Use of any hepatocyte-targeted small interfering ribonucleic acid (siRNA) that targets lipids and/or triglycerides within 365 days before Day 1 (except inclisiran, which is permitted). Administration of investigational drug and inclisiran must be separated by at least 4 weeks.
  • Use of any other hepatocyte targeted siRNA or antisense Oligonucleotide molecule within 60 days or within 5-half-lives before Day 1 based on plasma pharmacokinetics (PK), whichever is longer
  • Acute pancreatitis within 4 weeks prior to screening
  • Body mass index \>45 kg/m\^2

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (235)

Research Site 1

Birmingham, Alabama, 35205, United States

Location

Research Site 2

Mobile, Alabama, 36604, United States

Location

Research Site 3

Beverly Hills, California, 90211, United States

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Research Site 4

Canoga Park, California, 91303, United States

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Research Site 5

Garden Grove, California, 92844, United States

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Research Site 6

Huntington Beach, California, 92648, United States

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Research Site 7

Lake Forest, California, 92630, United States

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Research Site 8

Lincoln, California, 95648, United States

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Research Site 9

Long Beach, California, 90822, United States

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Research Site 10

Montclair, California, 91763, United States

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Research Site 11

Oxnard, California, 93030, United States

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Research Site 12

Redding, California, 96001, United States

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Research Site 13

Van Nuys, California, 91402, United States

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Research Site 14

Colorado Springs, Colorado, 80909, United States

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Research Site 15

Clearwater, Florida, 33756, United States

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Research Site 16

Hialeah, Florida, 33016, United States

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Research Site 17

Lake City, Florida, 32055, United States

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Research Site 18

Miami Lakes, Florida, 33014, United States

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Research Site 19

Mt. Dora, Florida, 32757, United States

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Research Site 20

North Miami Beach, Florida, 33162, United States

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Research Site 21

Orlando, Florida, 32825, United States

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Research Site 22

Pensacola, Florida, 32503, United States

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Research Site 23

Sarasota, Florida, 34239, United States

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Research Site 24

Tamarac, Florida, 33321, United States

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Research Site 25

Lawrenceville, Georgia, 30044, United States

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Research Site 26

Macon, Georgia, 31210, United States

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Research Site 27

Savannah, Georgia, 31406, United States

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Research Site 28

Sugar Hill, Georgia, 30518, United States

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Research Site 29

Park Ridge, Illinois, 60068, United States

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Research Site 30

Elkhart, Indiana, 46514, United States

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Research Site 31

Indianapolis, Indiana, 46290, United States

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Research Site 32

South Bend, Indiana, 46617, United States

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Research Site 33

Overland Park, Kansas, 66211, United States

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Research Site 34

Topeka, Kansas, 66606, United States

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Research Site 35

Louisville, Kentucky, 40202, United States

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Research Site 36

Zachary, Louisiana, 70791, United States

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Research Site 37

Annapolis, Maryland, 21401, United States

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Research Site 38

Baltimore, Maryland, 21229, United States

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Research Site 39

Flint, Michigan, 48532, United States

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Research Site 40

Minneapolis, Minnesota, 55455, United States

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Research Site 41

Olive Branch, Mississippi, 38654, United States

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Research Site 42

Jefferson City, Missouri, 65109, United States

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Research Site 43

St Louis, Missouri, 63136, United States

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Research Site 44

Norfolk, Nebraska, 68701, United States

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Research Site 46

Omaha, Nebraska, 68114, United States

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Research Site 45

Omaha, Nebraska, 68144, United States

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Research Site 47

Las Vegas, Nevada, 89119, United States

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Research Site 48

Summit, New Jersey, 07901, United States

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Research Site 52

New York, New York, 10016, United States

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Research Site 51

New York, New York, 10029, United States

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Research Site 53

Riverhead, New York, 11901, United States

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Research Site 54

Rochester, New York, 14642, United States

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Research Site 49

The Bronx, New York, 10455, United States

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Research Site 50

The Bronx, New York, 10461, United States

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Research Site 55

Vestal, New York, 13850, United States

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Research Site 56

Asheboro, North Carolina, 27203, United States

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Research Site 57

Morehead City, North Carolina, 28557, United States

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Research Site 58

Wilmington, North Carolina, 28412, United States

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Research Site 59

Winston-Salem, North Carolina, 27157, United States

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Research Site 60

Beavercreek, Ohio, 45431, United States

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Research Site 61

Cincinnati, Ohio, 45267, United States

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Research Site 63

Columbus, Ohio, 43210, United States

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Research Site 62

Columbus, Ohio, 43214, United States

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Research Site 64

Norman, Oklahoma, 73072, United States

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Research Site 66

Oklahoma City, Oklahoma, 73111, United States

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Research Site 65

Oklahoma City, Oklahoma, 73112, United States

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Research Site 67

Horsham, Pennsylvania, 19044, United States

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Research Site 68

Newport, Pennsylvania, 17074, United States

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Research Site 69

Newport, Pennsylvania, 17074, United States

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Research Site 70

Philadelphia, Pennsylvania, 19104, United States

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Research Site 71

Wilkes-Barre, Pennsylvania, 18711, United States

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Research Site 72

Fort Mill, South Carolina, 29707, United States

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Research Site 73

Greenville, South Carolina, 29607, United States

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Research Site 74

Chattanooga, Tennessee, 37411, United States

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Research Site 75

Powell, Tennessee, 37849, United States

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Research Site 76

El Paso, Texas, 79905, United States

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Research Site 77

Fort Worth, Texas, 76132, United States

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Research Site 86

Houston, Texas, 77029, United States

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Research Site 84

Houston, Texas, 77030, United States

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Research Site 85

Houston, Texas, 77030, United States

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Research Site 78

Houston, Texas, 77040, United States

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Research Site 80

Houston, Texas, 77061, United States

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Research Site 83

Houston, Texas, 77074, United States

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Research Site 82

Houston, Texas, 77079, United States

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Research Site 79

Houston, Texas, 77090, United States

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Research Site 81

Houston, Texas, 77095, United States

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Research Site 87

Laredo, Texas, 78041, United States

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Research Site 88

Missouri City, Texas, 77459, United States

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Research Site 89

Plano, Texas, 75093, United States

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Research Site 90

San Antonio, Texas, 78230, United States

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Research Site 91

Sugar Land, Texas, 77479, United States

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Research Site 92

Tomball, Texas, 77375, United States

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Research Site 93

Victoria, Texas, 77901, United States

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Research Site 94

Bountiful, Utah, 84010, United States

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Research Site 95

St. George, Utah, 84790, United States

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Research Site 96

Manassas, Virginia, 20110, United States

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Research Site 97

Seattle, Washington, 98109, United States

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Research Site 102

CABA, Buenos Aires, 1128, Argentina

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Research Site 100

CABA, Buenos Aires, 1417, Argentina

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Research Site 103

Ciudad Autonoma Buenos Aires, Buenos Aires, C1430CKE, Argentina

Location

Research Site 104

Córdoba, Córdoba Province, 5000, Argentina

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Research Site 98

Córdoba, Córdoba Province, 5006, Argentina

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Research Site 101

Godoy Cruz, Mendoza Province, 5501, Argentina

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Research Site 105

Rosario, Santa Fe Province, 2000, Argentina

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Research Site 99

Rosario, Santa Fe Province, 2000, Argentina

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Research Site 106

Córdoba, 5000, Argentina

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Research Site 107

Blacktown, New South Wales, 2148, Australia

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Research Site 108

Merewether, New South Wales, 2291, Australia

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Research Site 110

Clayton, Victoria, 3168, Australia

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Research Site 109

Heidelberg Heights, Victoria, 3081, Australia

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Research Site 111

Blagoevgrad, 2700, Bulgaria

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Research Site 112

Burgas, 8000, Bulgaria

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Research Site 113

Byala, 7100, Bulgaria

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Research Site 114

Dimitrovgrad, 6400, Bulgaria

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Research Site 115

Haskovo, 6300, Bulgaria

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Research Site 116

Kyustendil, 2500, Bulgaria

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Research Site 117

Pleven, 5800, Bulgaria

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Research Site 118

Pleven, 5800, Bulgaria

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Research Site 120

Plovdiv, 4001, Bulgaria

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Research Site 119

Plovdiv, 4002, Bulgaria

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Research Site 121

Plovdiv, 4004, Bulgaria

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Research Site 122

Rousse, 7013, Bulgaria

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Research Site 123

Sevlievo, 5400, Bulgaria

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Research Site 137

Sofia, 1202, Bulgaria

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Research Site 133

Sofia, 1336, Bulgaria

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Research Site 126

Sofia, 1431, Bulgaria

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Research Site 129

Sofia, 1431, Bulgaria

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Research Site 132

Sofia, 1431, Bulgaria

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Research Site 130

Sofia, 1510, Bulgaria

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Research Site 131

Sofia, 1527, Bulgaria

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Research Site 135

Sofia, 1527, Bulgaria

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Research Site 124

Sofia, 1616, Bulgaria

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Research Site 125

Sofia, 1618, Bulgaria

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Research Site 127

Sofia, 1680, Bulgaria

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Research Site 134

Sofia, 1680, Bulgaria

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Research Site 128

Sofia, 1750, Bulgaria

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Research Site 136

Stara Zagora, 6010, Bulgaria

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Research Site 140

North Vancouver, British Columbia, V7M 2H4, Canada

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Research Site 141

Victoria, British Columbia, V8T 5G4, Canada

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Research Site 142

Brampton, Ontario, L6S 0C6, Canada

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Research Site 143

Sarnia, Ontario, N7T 4X3, Canada

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Research Site 144

Waterloo, Ontario, N2T0C1, Canada

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Research Site 145

Chicoutimi, Quebec, G7H 7K9, Canada

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Research Site 146

Laval, Quebec, H7T 2P5, Canada

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Research Site 149

Montreal, Quebec, H2W 1R7, Canada

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Research Site 139

Québec, Quebec, G1G 3Y8, Canada

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Research Site 147

Québec, Quebec, G1V 4W2, Canada

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Research Site 148

Québec, Quebec, J6X 4P7, Canada

Location

Research Site 138

Halifax, B3H 1V7, Canada

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Research Site 151

Prague, Prague, 140 21, Czechia

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Research Site 157

Brno, 602 00, Czechia

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Research Site 154

Hodonín, 69501, Czechia

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Research Site 159

Hradec Králové, 500 05, Czechia

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Research Site 160

Náchod, 547 01, Czechia

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Research Site 162

Olomouc, 779 00, Czechia

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Research Site 155

Ostrava, 702 00, Czechia

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Research Site 152

Prague, 101 00, Czechia

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Research Site 156

Praha 4-Krc, 140 59, Czechia

Location

Research Site 150

Slaný, 27401, Czechia

Location

Research Site 163

Teplice, 41501, Czechia

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Research Site 158

Trutnov, 541 01, Czechia

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Research Site 161

Uherské Hradiště, 686 01, Czechia

Location

Research Site 153

Ústí nad Labem, 40113, Czechia

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Research Site 164

Marseille, Bouches du Rhone, 13005, France

Location

Research Site 167

Pessac, Gironde, 33604, France

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Research Site 166

Lyon, Rhone, 69007, France

Location

Research Site165

Paris, 75013, France

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Research Site 170

Deggingen, Baden-Wurttemberg, 73326, Germany

Location

Research Site 169

Wallerfing, Bavaria, 94574, Germany

Location

Research Site 168

Magdeburg, Saxony-Anhalt, 39120, Germany

Location

Research Site 171

Békéscsaba, 5600, Hungary

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Research Site 175

Budapest, 1033, Hungary

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Research Site 183

Budapest, 1051, Hungary

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Research Site 179

Budapest, 1132, Hungary

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Research Site 184

Budapest, 1135, Hungary

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Research Site 180

Budapest, 1152, Hungary

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Research Site 182

Kaposvár, 7400, Hungary

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Research Site 176

Miskolc, 3530, Hungary

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Research Site 172

Pécs, 7623, Hungary

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Research Site 177

Pécs, 7635, Hungary

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Research Site 178

Szeged, 6725, Hungary

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Research Site 173

Veszprém, 8200, Hungary

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Research Site 174

Zalaegerszeg, 8900, Hungary

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Research Site 186

Rozzano, Milano, 20089, Italy

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Research Site 187

Palermo, Sicily, 90127, Italy

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Research Site 189

Bologna, 40138, Italy

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Research Site 185

Brescia, 25123, Italy

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Research Site 188

Milan, 20162, Italy

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Research Site 200

Bydgoszcz, 85-065, Poland

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Research Site 202

Bydgoszcz, 85-231, Poland

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Research Site 192

Elblag, 82-300, Poland

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Research Site 193

Gdynia, 81-338, Poland

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Research Site 190

Katowice, 40-156, Poland

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Research Site 197

Krakow, 30-727, Poland

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Research Site 204

Krakow, 31-501, Poland

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Research Site 201

Lodz, 91-363, Poland

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Research Site 191

Lodz, 94-255, Poland

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Research Site 194

Malbork, 82-200, Poland

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Research Site 199

Szczecin, 71-500, Poland

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Research Site 207

Torun, 87-100, Poland

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Research Site 205

Warsaw, 00-215, Poland

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Research Site 198

Warsaw, 03-291, Poland

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Research Site 196

Wroclaw, 51-314, Poland

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Research Site 208

Wroclaw, 53-030, Poland

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Research Site 206

Wroclaw, 53-673, Poland

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Research Site 195

Zamość, 22-400, Poland

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Research Site 203

Żarów, 58-130, Poland

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Research Site 214

Banská Bystrica, 97401, Slovakia

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Research Site 212

Bardejov, 8501, Slovakia

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Research Site 217

Bratislava, 81109, Slovakia

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Research Site 216

Bratislava, 83101, Slovakia

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Research Site 210

Košice, 040 01, Slovakia

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Research Site 213

Moldava nad Bodvou, 045 01, Slovakia

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Research Site 209

Nové Zámky, 94002, Slovakia

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Research Site 211

Prešov, 8001, Slovakia

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Research Site 215

Rožňava, 4801, Slovakia

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Research Site 218

Žilina, 01001, Slovakia

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Research Site 221

Centurion, Gauteng, 0157, South Africa

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Research Site 222

Krugersdorp, Gauteng, 1739, South Africa

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Research Site 228

Pretoria, Gauteng, 0181, South Africa

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Research Site 224

Durban, KwaZulu-Natal, 4449, South Africa

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Research Site 227

Cape Town, Western Cape, 7500, South Africa

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Research Site 219

Cape Town, Western Cape, 7530, South Africa

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Research Site 223

Cape Town, Western Cape, 7550, South Africa

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Research Site 225

Cape Town, Western Cape, 7925, South Africa

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Research Site 220

Somerset West, Western Cape, 7130, South Africa

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Research Site 226

Pretoria, 0184, South Africa

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Research Site 234

Barcelona, Barcelona, 08035, Spain

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Research Site 229

A Coruña, La Coruña, 15006, Spain

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Research Site 230

Barcelona, 08023, Spain

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Research Site 232

Madrid, 28041, Spain

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Research Site 231

Valencia, 46010, Spain

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Research Site 233

Zaragoza, 50009, Spain

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Research Site 236

Plymouth, Devon, PL5 3JB, United Kingdom

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Research Site 235

London, EC1M 6BQ, United Kingdom

Location

MeSH Terms

Conditions

Hypertriglyceridemia

Interventions

plozasiran

Condition Hierarchy (Ancestors)

HyperlipidemiasDyslipidemiasLipid Metabolism DisordersMetabolic DiseasesNutritional and Metabolic Diseases

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 29, 2024

First Posted

April 4, 2024

Study Start

May 21, 2024

Primary Completion

May 1, 2026

Study Completion (Estimated)

September 1, 2026

Last Updated

October 8, 2025

Record last verified: 2025-10

Data Sharing

IPD Sharing
Will not share

Locations