NCT05646381

Brief Summary

The purpose of this study is to evaluate the efficacy, safety and tolerability of pelacarsen (TQJ230) administered subcutaneously once monthly compared to placebo in slowing the progression of calcific aortic valve stenosis.

Trial Health

88
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
502

participants targeted

Target at P75+ for phase_2

Timeline
47mo left

Started Mar 2024

Longer than P75 for phase_2

Geographic Reach
15 countries

139 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress36%
Mar 2024Mar 2030

First Submitted

Initial submission to the registry

December 2, 2022

Completed
10 days until next milestone

First Posted

Study publicly available on registry

December 12, 2022

Completed
1.2 years until next milestone

Study Start

First participant enrolled

March 7, 2024

Completed
6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 12, 2030

Expected
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

March 12, 2030

Last Updated

April 15, 2026

Status Verified

April 1, 2026

Enrollment Period

6 years

First QC Date

December 2, 2022

Last Update Submit

April 10, 2026

Conditions

Keywords

CardiovascularLipoprotein(a)Lp(a)Hyperlipoproteinemia(a)Calcific aortic valve stenosisTQJ230PelacarsenAortic valve stenosisAortic stenosis

Outcome Measures

Primary Outcomes (2)

  • Change in peak aortic jet velocity

    To demonstrate the superiority of pelacarsen (TQJ230) vs. placebo in slowing the progression of calcific aortic valve stenosis by evaluating the change from baseline to month 36 in peak aortic jet velocity by echocardiography

    36 months

  • Change in aortic valve calcium score

    To demonstrate the superiority of pelacarsen (TQJ230) vs. placebo in slowing the progression of calcific aortic valve stenosis by evaluating the change from baseline to month 36 in aortic valve calcium score by computed tomography

    36 months

Secondary Outcomes (3)

  • Change in Lp(a) levels

    12 months

  • Change in fibrocalcific thickening of the aortic valve

    36 months

  • Time from randomization to first occurrence of composite clinical endpoint event

    Up to 36 months

Study Arms (2)

Pelacarsen (TQJ230) 80mg

EXPERIMENTAL

Pelacarsen (TQJ230) 80 mg prefilled syringe injected monthly, administered subcutaneously

Drug: Pelacarsen (TQJ230) 80mg

Matching placebo

PLACEBO COMPARATOR

Placebo to match pelacarsen (TQJ230) prefilled syringe injected monthly, administered subcutaneously

Drug: Matching placebo

Interventions

Pelacarsen (TQJ230) 80mg

Also known as: TQJ230
Pelacarsen (TQJ230) 80mg

Matching placebo

Also known as: Placebo
Matching placebo

Eligibility Criteria

Age50 Years - 80 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Male and female ≥50 to \<80 years of age at Screening Part II
  • Lp(a) ≥175 nmol/L at the screening visit, measured at the Central laboratory
  • Mild or moderate calcific aortic valve stenosis
  • At the randomization visit, participant must be optimally treated for existing CV risk factors

You may not qualify if:

  • Severe calcific aortic valve stenosis
  • Uncontrolled hypertension
  • History of malignancy of any organ system
  • History of hemorrhagic stroke or other major bleeding
  • Platelet count ≤ LLN
  • Active liver disease or hepatic dysfunction
  • Significant kidney disease
  • Pregnant or nursing women

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (139)

Heart Center Research Llc

Huntsville, Alabama, 35801, United States

RECRUITING

Cardiovascular Res Found

Beverly Hills, California, 90210, United States

RECRUITING

National Heart Institute

Beverly Hills, California, 90211, United States

RECRUITING

Flourish Clinical Resrch Covin

Covina, California, 91723, United States

RECRUITING

Valley Clinical Trials

Northridge, California, 91325, United States

RECRUITING

Stanford University Medical Center

Palo Alto, California, 94304, United States

RECRUITING

University Of California San Diego

San Diego, California, 92103-8415, United States

RECRUITING

UC San Francisco Medical Center

San Francisco, California, 94143, United States

RECRUITING

Excel Medical Clinical Trials LLC

Boca Raton, Florida, 33434, United States

WITHDRAWN

Nova Clinical Research LLC

Bradenton, Florida, 34209, United States

RECRUITING

Flourish Res Acq LLC North Miami

Miami, Florida, 33138, United States

RECRUITING

Inpatient Research Clinical LLC

Miami Lakes, Florida, 33014, United States

RECRUITING

Advanced Research for Health Improvement LLC

Naples, Florida, 34102, United States

ACTIVE NOT RECRUITING

Midwest Heart and Vascular Spec

Overland Park, Kansas, 66211, United States

RECRUITING

Tufts Medical Center

Boston, Massachusetts, 02111, United States

RECRUITING

Massachusetts General Hospital

Boston, Massachusetts, 02114, United States

RECRUITING

Massachusetts General Hospital

Boston, Massachusetts, 02114, United States

RECRUITING

Brigham and Womens Hosp Harvard Med School

Boston, Massachusetts, 02115, United States

RECRUITING

Brigham and Womens Hosp Harvard Med School

Boston, Massachusetts, 02115, United States

RECRUITING

Henry Ford Hospital

Detroit, Michigan, 48202, United States

RECRUITING

Henry Ford Hospital

Detroit, Michigan, 48202, United States

RECRUITING

AA Medical Research Center

Flint, Michigan, 48504, United States

RECRUITING

William Beaumont Hospital

Royal Oak, Michigan, 48073-4192, United States

RECRUITING

Minneapolis Heart Institute

Minneapolis, Minnesota, 55407, United States

WITHDRAWN

University Of Minnesota

Minneapolis, Minnesota, 55455, United States

RECRUITING

Overlook Medical Center

Summit, New Jersey, 07901, United States

RECRUITING

Capital Cardiology Associates

Albany, New York, 12211, United States

RECRUITING

New York Presbyterian Hospital

New York, New York, 10021, United States

ACTIVE NOT RECRUITING

Icahn School of Med at Mt Sinai

New York, New York, 10029, United States

RECRUITING

Strong Memorial Hospital

Rochester, New York, 14642, United States

RECRUITING

Wake Forest University Baptist Medical Center

Winston-Salem, North Carolina, 27157, United States

RECRUITING

Lindner Ctr At The Christ Hosp

Cincinnati, Ohio, 45219, United States

RECRUITING

Ohio State University

Columbus, Ohio, 43210, United States

WITHDRAWN

Perelman School of Medicine

Philadelphia, Pennsylvania, 19104, United States

RECRUITING

Orion Medical

Houston, Texas, 77034, United States

RECRUITING

Virginia Heart

Falls Church, Virginia, 22042, United States

RECRUITING

Carient Heart and Vascular

Manassas, Virginia, 20109, United States

RECRUITING

Novartis Investigative Site

Innsbruck, Tyrol, 6020, Austria

RECRUITING

Novartis Investigative Site

Linz, 4021, Austria

WITHDRAWN

Novartis Investigative Site

Vienna, 1100, Austria

RECRUITING

Novartis Investigative Site

Vienna, 1190, Austria

RECRUITING

Novartis Investigative Site

Vienna, A 1090, Austria

RECRUITING

Novartis Investigative Site

Genk, Limburg, 3600, Belgium

RECRUITING

Novartis Investigative Site

Yvoir, Namur, 5530, Belgium

RECRUITING

Novartis Investigative Site

Aalst, Oost Vlaanderen, 9300, Belgium

RECRUITING

Novartis Investigative Site

Kortrijk, West-Vlaanderen, 8500, Belgium

RECRUITING

Novartis Investigative Site

Roeselare, West-Vlaanderen, 8800, Belgium

RECRUITING

Novartis Investigative Site

Cambridge, Ontario, N1R 6V6, Canada

RECRUITING

Novartis Investigative Site

North York, Ontario, M6B 3H7, Canada

RECRUITING

Novartis Investigative Site

Ottawa, Ontario, K1Y 4W7, Canada

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Novartis Investigative Site

Montreal, Quebec, H1T 1C8, Canada

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Novartis Investigative Site

Montreal, Quebec, H3T 1E2, Canada

RECRUITING

Novartis Investigative Site

Montreal, Quebec, H4A 3J1, Canada

RECRUITING

Novartis Investigative Site

Québec, Quebec, G1V 4G5, Canada

RECRUITING

Novartis Investigative Site

Hradec Králové, 500 02, Czechia

RECRUITING

Novartis Investigative Site

Jaroměř, 551 01, Czechia

RECRUITING

Novartis Investigative Site

Prague, 128 08, Czechia

RECRUITING

Novartis Investigative Site

Prague, 14021, Czechia

RECRUITING

Novartis Investigative Site

Prague, 150 06, Czechia

RECRUITING

Novartis Investigative Site

Esbjerg, 6700, Denmark

RECRUITING

Novartis Investigative Site

Hvidovre, 2650, Denmark

RECRUITING

Novartis Investigative Site

Roskilde, 4000, Denmark

RECRUITING

Novartis Investigative Site

Viborg, 8800, Denmark

RECRUITING

Novartis Investigative Site

Paris, 75012, France

RECRUITING

Novartis Investigative Site

Paris, 75013, France

RECRUITING

Novartis Investigative Site

Paris, 75015, France

RECRUITING

Novartis Investigative Site

Pessac, 33604, France

RECRUITING

Novartis Investigative Site

Poitiers, 86021, France

RECRUITING

Novartis Investigative Site

Rennes, 35033, France

RECRUITING

Novartis Investigative Site

Frankfurt am Main, Hesse, 60594, Germany

RECRUITING

Novartis Investigative Site

Kaiserslautern, Rhineland-Palatinate, 67655, Germany

RECRUITING

Novartis Investigative Site

Dresden, Saxony, 01099, Germany

RECRUITING

Novartis Investigative Site

Leipzig, Saxony, 04289, Germany

RECRUITING

Novartis Investigative Site

Ahaus, 48683, Germany

RECRUITING

Novartis Investigative Site

Berlin, 13353, Germany

RECRUITING

Novartis Investigative Site

Bonn, 53105, Germany

RECRUITING

Novartis Investigative Site

Essen, 45147, Germany

RECRUITING

Novartis Investigative Site

Hamburg, 20246, Germany

RECRUITING

Novartis Investigative Site

Hamburg, 22763, Germany

RECRUITING

Novartis Investigative Site

Lüneburg, 21339, Germany

WITHDRAWN

Novartis Investigative Site

Mannheim, 68165, Germany

RECRUITING

Novartis Investigative Site

München, 80636, Germany

RECRUITING

Novartis Investigative Site

Münster, 48149, Germany

RECRUITING

Novartis Investigative Site

Oldenburg, 26133, Germany

RECRUITING

Novartis Investigative Site

Beersheba, 8457108, Israel

RECRUITING

Novartis Investigative Site

Haifa, 3104802, Israel

RECRUITING

Novartis Investigative Site

Haifa, 3109601, Israel

RECRUITING

Novartis Investigative Site

Jerusalem, 9103102, Israel

RECRUITING

Novartis Investigative Site

Jerusalem, 9112001, Israel

RECRUITING

Novartis Investigative Site

Nahariya, 2210001, Israel

RECRUITING

Novartis Investigative Site

Petah Tikva, 4941492, Israel

RECRUITING

Novartis Investigative Site

Ramat Gan, 5265601, Israel

RECRUITING

Novartis Investigative Site

Tel Aviv, 6423906, Israel

RECRUITING

Novartis Investigative Site

Ancona, AN, 60126, Italy

RECRUITING

Novartis Investigative Site

Bergamo, BG, 24127, Italy

RECRUITING

Novartis Investigative Site

Bologna, BO, 40138, Italy

WITHDRAWN

Novartis Investigative Site

Brescia, BS, 25123, Italy

RECRUITING

Novartis Investigative Site

Caserta, CE, 81100, Italy

RECRUITING

Novartis Investigative Site

Cona, FE, 44124, Italy

RECRUITING

Novartis Investigative Site

Pozzilli, IS, 86077, Italy

RECRUITING

Novartis Investigative Site

Milan, MI, 20138, Italy

RECRUITING

Novartis Investigative Site

Milan, MI, 20157, Italy

RECRUITING

Novartis Investigative Site

Milan, MI, 20162, Italy

RECRUITING

Novartis Investigative Site

Padova, PD, 35128, Italy

RECRUITING

Novartis Investigative Site

Pordenone, PN, 33170, Italy

RECRUITING

Novartis Investigative Site

Amsterdam, North Holland, 1090 HM, Netherlands

RECRUITING

Novartis Investigative Site

Amsterdam, North Holland, 1105 AZ, Netherlands

RECRUITING

Novartis Investigative Site

Rotterdam, South Holland, 3015 GD, Netherlands

RECRUITING

Novartis Investigative Site

Rotterdam, South Holland, 3079 DZ, Netherlands

RECRUITING

Novartis Investigative Site

Nieuwegein, Utrecht, 3435 CM, Netherlands

RECRUITING

Novartis Investigative Site

Alcabideche, 2755-009, Portugal

RECRUITING

Novartis Investigative Site

Braga, 4710243, Portugal

RECRUITING

Novartis Investigative Site

Coimbra, 3004-561, Portugal

RECRUITING

Novartis Investigative Site

Vila Nova de Gaia, 4434 502, Portugal

RECRUITING

Novartis Investigative Site

Cáceres, Extremadura, 10003, Spain

RECRUITING

Novartis Investigative Site

Córdoba, 14004, Spain

RECRUITING

Novartis Investigative Site

Madrid, 28034, Spain

RECRUITING

Novartis Investigative Site

Madrid, 28040, Spain

WITHDRAWN

Novartis Investigative Site

Madrid, 28041, Spain

RECRUITING

Novartis Investigative Site

Madrid, 28046, Spain

RECRUITING

Novartis Investigative Site

Salamanca, 37007, Spain

RECRUITING

Novartis Investigative Site

Valencia, 46010, Spain

RECRUITING

Novartis Investigative Site

Basel, 4031, Switzerland

RECRUITING

Novartis Investigative Site

Geneva, 1211, Switzerland

RECRUITING

Novartis Investigative Site

Lausanne, 1011, Switzerland

RECRUITING

Novartis Investigative Site

Lugano, 6900, Switzerland

RECRUITING

Novartis Investigative Site

Zurich, 8091, Switzerland

RECRUITING

Novartis Investigative Site

Reading, Berkshire, RG1 5AN, United Kingdom

RECRUITING

Novartis Investigative Site

Portadown, Nothern Ireland, BT63 5QQ, United Kingdom

RECRUITING

Novartis Investigative Site

Edinburgh, ED16 4SA, United Kingdom

RECRUITING

Novartis Investigative Site

Leicester, LE3 9QP, United Kingdom

RECRUITING

Novartis Investigative Site

Liverpool, L14 3PE, United Kingdom

RECRUITING

Novartis Investigative Site

London, EC1A 7BE, United Kingdom

RECRUITING

Novartis Investigative Site

London, SE1 7EH, United Kingdom

RECRUITING

Novartis Investigative Site

Londonderry, BT47 6SB, United Kingdom

RECRUITING

Novartis Investigative Site

Manchester, M23 9LT, United Kingdom

RECRUITING

Novartis Investigative Site

Middlesbrough, TS4 3BW, United Kingdom

RECRUITING

Novartis Investigative Site

Norwich, NR4 7UY, United Kingdom

RECRUITING

Novartis Investigative Site

Tyne and Wear, NE29 8NH, United Kingdom

RECRUITING

Related Publications (1)

  • Nicholls SJ, Nelson AJ, Michael LF. Oral agents for lowering lipoprotein(a). Curr Opin Lipidol. 2024 Dec 1;35(6):275-280. doi: 10.1097/MOL.0000000000000953. Epub 2024 Sep 25.

MeSH Terms

Conditions

Aortic Valve Stenosis

Interventions

pelacarsen

Condition Hierarchy (Ancestors)

Aortic Valve DiseaseHeart Valve DiseasesHeart DiseasesCardiovascular DiseasesVentricular Outflow Obstruction

Study Officials

  • Novartis Pharmaceuticals

    Novartis Pharmaceuticals

    STUDY DIRECTOR

Central Study Contacts

Novartis Pharmaceuticals

CONTACT

Novartis Pharmaceuticals

CONTACT

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Masking Details
Double-blind study
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR
Expanded Access
Yes

Study Record Dates

First Submitted

December 2, 2022

First Posted

December 12, 2022

Study Start

March 7, 2024

Primary Completion (Estimated)

March 12, 2030

Study Completion (Estimated)

March 12, 2030

Last Updated

April 15, 2026

Record last verified: 2026-04

Data Sharing

IPD Sharing
Will share

Novartis is committed to sharing with qualified external researchers, access to patient-level data and supporting clinical documents from eligible studies. These requests are reviewed and approved by an independent review panel on the basis of scientific merit. All data provided is anonymized to respect the privacy of patients who have participated in the trial in line with the applicable laws and regulations.

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