NCT05609370

Brief Summary

This is a Phase 1b/2 study to investigate the efficacy and safety of LBL-007 plus tislelizumab when administered in combination with bevacizumab plus fluoropyrimidine, and LBL-007 in combination with bevacizumab plus fluoropyrimidine versus bevacizumab plus fluoropyrimidine to participants with colorectal cancer.

Trial Health

78
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
113

participants targeted

Target at P75+ for phase_1

Timeline
8mo left

Started Jan 2023

Longer than P75 for phase_1

Geographic Reach
4 countries

76 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress83%
Jan 2023Dec 2026

First Submitted

Initial submission to the registry

October 20, 2022

Completed
19 days until next milestone

First Posted

Study publicly available on registry

November 8, 2022

Completed
3 months until next milestone

Study Start

First participant enrolled

January 29, 2023

Completed
2.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 23, 2025

Completed
1.6 years until next milestone

Study Completion

Last participant's last visit for all outcomes

December 31, 2026

Expected
Last Updated

October 2, 2025

Status Verified

September 1, 2025

Enrollment Period

2.3 years

First QC Date

October 20, 2022

Last Update Submit

September 29, 2025

Conditions

Keywords

Colorectal CancerMicrosatellite StableMismatch Repair ProficientMaintenance Therapy

Outcome Measures

Primary Outcomes (2)

  • Phase 1b: Number of participants with Adverse Events (AEs) and Serious AEs (SAEs)

    Number of participants with AEs and SAEs characterized by type, frequency, severity (as graded by National Cancer Institute Common Terminology Criteria for Adverse Events version 5.0 \[NCI-CTCAE v5.0\]).

    From the first dose of study drug(s) to 30 days after last dose, initiation of new anticancer therapy, death, withdrawal of consent, or loss to follow-up, whichever occurs first (up to approximately 28 months)

  • Phase 2: Progression Free Survival (PFS) as Assessed by The Investigator in PD-L1 Positive Arms A and C

    PFS, as assessed by the investigator per RECIST v1.1 is defined as the time from the date of randomization to the date of first documentation of disease progression or death, whichever occurs first.

    Approximately 28 months

Secondary Outcomes (4)

  • Phase 2: Objective Response rate (ORR) as Assessed by The Investigator in PD-L1 Positive Arms A and C and PD-L1 Negative Arms D and E

    Approximately 28 months

  • Phase 2: Duration of response (DOR) as Assessed by The Investigator in PD-L1 Positive Arms A and C and PD-L1 Negative arms D and E

    Approximately 28 months

  • Phase 2: Progression Free Survival (PFS) as Assessed by The Investigator in PD-L1 Negative Arms D and E

    Approximately 28 months

  • Phase 2: Number of participants with AEs and SAEs

    From the first dose of study drug(s) to 30 days after the last dose, initiation of new anticancer therapy, death, withdrawal of consent, or loss to follow-up, whichever occurs first (up to approximately 28 months)

Study Arms (7)

Phase 1b: Cohort -1: LBL-007 + Tislelizumab + Bevacizumab + Capecitabine

EXPERIMENTAL

LBL-007 (low dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine

Drug: LBL-007Drug: TislelizumabDrug: Bevacizumab or Bevacizumab biosimilarDrug: Capecitabine

Phase 1b: Cohort 1a: LBL-007 + Tislelizumab + Bevacizumab + Capecitabine

EXPERIMENTAL

LBL-007 (medium dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine

Drug: LBL-007Drug: TislelizumabDrug: Bevacizumab or Bevacizumab biosimilarDrug: Capecitabine

Phase 1b: Cohort 1b: LBL-007 + Tislelizumab + Bevacizumab + 5-Fluorouracil (5-FU)

EXPERIMENTAL

LBL-007 (medium dose) + tislelizumab (high dose once every 4 weeks) + bevacizumab (5 mg/kg once every 2 weeks) + 5-FU

Drug: LBL-007Drug: TislelizumabDrug: Bevacizumab or Bevacizumab biosimilarDrug: 5-Fluorouracil

Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + Fluoropyrimidine

EXPERIMENTAL

LBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)

Drug: LBL-007Drug: TislelizumabDrug: Bevacizumab or Bevacizumab biosimilarDrug: CapecitabineDrug: 5-Fluorouracil

Phase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + Fluoropyrimidine

EXPERIMENTAL

LBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)

Drug: LBL-007Drug: TislelizumabDrug: Bevacizumab or Bevacizumab biosimilarDrug: CapecitabineDrug: 5-Fluorouracil

Phase 2: Arm B: LBL-007 + Bevacizumab + Fluoropyrimidine

EXPERIMENTAL

LBL-007 (high dose) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)

Drug: LBL-007Drug: Bevacizumab or Bevacizumab biosimilarDrug: CapecitabineDrug: 5-Fluorouracil

Phase 2: Arm C and Arm E: Bevacizumab + Fluoropyrimidine

ACTIVE COMPARATOR

Bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)

Drug: LBL-007Drug: TislelizumabDrug: Bevacizumab or Bevacizumab biosimilarDrug: CapecitabineDrug: 5-Fluorouracil

Interventions

Administered intravenously.

Also known as: Alcestobart
Phase 1b: Cohort -1: LBL-007 + Tislelizumab + Bevacizumab + CapecitabinePhase 1b: Cohort 1a: LBL-007 + Tislelizumab + Bevacizumab + CapecitabinePhase 1b: Cohort 1b: LBL-007 + Tislelizumab + Bevacizumab + 5-Fluorouracil (5-FU)Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm B: LBL-007 + Bevacizumab + FluoropyrimidinePhase 2: Arm C and Arm E: Bevacizumab + Fluoropyrimidine

Administered intravenously.

Also known as: BGB-A317
Phase 1b: Cohort -1: LBL-007 + Tislelizumab + Bevacizumab + CapecitabinePhase 1b: Cohort 1a: LBL-007 + Tislelizumab + Bevacizumab + CapecitabinePhase 1b: Cohort 1b: LBL-007 + Tislelizumab + Bevacizumab + 5-Fluorouracil (5-FU)Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm C and Arm E: Bevacizumab + Fluoropyrimidine

Administered intravenously

Phase 1b: Cohort -1: LBL-007 + Tislelizumab + Bevacizumab + CapecitabinePhase 1b: Cohort 1a: LBL-007 + Tislelizumab + Bevacizumab + CapecitabinePhase 1b: Cohort 1b: LBL-007 + Tislelizumab + Bevacizumab + 5-Fluorouracil (5-FU)Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm B: LBL-007 + Bevacizumab + FluoropyrimidinePhase 2: Arm C and Arm E: Bevacizumab + Fluoropyrimidine

Administered in accordance with relevant local guidelines and/or prescribing information

Phase 1b: Cohort -1: LBL-007 + Tislelizumab + Bevacizumab + CapecitabinePhase 1b: Cohort 1a: LBL-007 + Tislelizumab + Bevacizumab + CapecitabinePhase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm B: LBL-007 + Bevacizumab + FluoropyrimidinePhase 2: Arm C and Arm E: Bevacizumab + Fluoropyrimidine

Administered in accordance with relevant local guidelines and/or prescribing information

Phase 1b: Cohort 1b: LBL-007 + Tislelizumab + Bevacizumab + 5-Fluorouracil (5-FU)Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidinePhase 2: Arm B: LBL-007 + Bevacizumab + FluoropyrimidinePhase 2: Arm C and Arm E: Bevacizumab + Fluoropyrimidine

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participant must have measurable disease as defined per RECIST version 1.1
  • Has a histologically confirmed colorectal adenocarcinoma with metastatic or unresectable disease (Stage IV as defined by American Joint Committee on Cancer \[AJCC\] 8th edition)
  • No prior systemic therapy for colorectal cancer (CRC) in the metastatic setting except for the induction treatment of first-line therapy. Note: Local regional treatment performed during induction systemic treatment is allowed
  • Participants who have completed the first-line induction treatment, with an overall response of stable disease or better. The duration of induction treatment should be completed within approximately 6 months. The first dose of study treatment needs to occur within 2 weeks (for 2-week regimen) or 3 weeks (for 3-week regimen) to 6 weeks after Day 1 of the last cycle of induction therapy

You may not qualify if:

  • Participants whose disease has become resectable at the investigator's discretion during or after induction treatment are not eligible
  • Progressive disease occurred less than 6 months from completion of any prior neoadjuvant therapy (ie, chemotherapy with or without radiotherapy) or adjuvant therapy (ie, chemotherapy with or without radiotherapy), whichever occurred later
  • Participants who have been treated with anti-epidermal growth factor receptor (EGFR) antibody in the induction treatment
  • Any prior therapy targeting T-cell stimulation or checkpoint pathways
  • Participants with B-raf proto-oncogene, serine/threonine kinase (BRAF)V600E mutations
  • Have locally or centrally confirmed microsatellite instability-high (MSI-H) by polymerase chain reaction (PCR) method or dMMR by immunohistochemistry (IHC) method
  • Note: Other protocol defined criteria may apply.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (76)

Alaska Oncology and Hematology, Llc

Anchorage, Alaska, 99508, United States

Location

Banner Md Anderson Cancer Center

Gilbert, Arizona, 85234, United States

Location

Toi Clinical Research

Cerritos, California, 90703, United States

Location

Usc Norris Comprehensive Cancer Center (Nccc)

Los Angeles, California, 90033, United States

Location

Valkyrie Clinical Trials

Los Angeles, California, 90067, United States

Location

UCLA

Los Angeles, California, 90095, United States

Location

Hoag Memorial Presbyterian

Newport, California, 92663, United States

Location

Kaiser Permanente Northern California

Vallejo, California, 94510, United States

Location

Baptist Md Anderson Cancer Center

Jacksonville, Florida, 32207, United States

Location

Fort Wayne Medical Oncology and Hematology

Fort Wayne, Indiana, 46804, United States

Location

Baptist Health Lexington

Lexington, Kentucky, 40503, United States

Location

University of Kentucky Markey Cancer Center

Lexington, Kentucky, 40536, United States

Location

Norton Cancer Institute

Louisville, Kentucky, 40217, United States

Location

Pontchartrain Cancer Center

Covington, Louisiana, 70433, United States

Location

Ochsner Clinic Foundation

New Orleans, Louisiana, 70121, United States

Location

Washington University School of Medicine

St Louis, Missouri, 63110, United States

Location

St Vincent Frontier Cancer Center

Billings, Montana, 59102, United States

Location

Comprehensive Cancer Centers of Nevada

Las Vegas, Nevada, 89169, United States

Location

Cancer Care Specialists

Reno, Nevada, 89511, United States

Location

University of New Mexico Cancer Center

Albuquerque, New Mexico, 87102, United States

Location

Perlmutter Cancer Center At Winthrop Oncology Hematology Associatesnyu Winthrop Hospital

Mineola, New York, 11501, United States

Location

Laura and Isaac Perlmutter Cancer Center At Nyu Langone Health

New York, New York, 10016, United States

Location

Columbia University Medical Center

New York, New York, 10032, United States

Location

Duke Cancer Center

Durham, North Carolina, 27710, United States

Location

University of Tennessee Medical Center

Knoxville, Tennessee, 37920, United States

Location

Ut Southwestern Medical Center

Dallas, Texas, 75390, United States

Location

Ut Health San Antonio Mays Cancer Center

San Antonio, Texas, 78229, United States

Location

Virginia Cancer Specialists

Fairfax, Virginia, 22031, United States

Location

Cancer Care Northwest

Spokane Valley, Washington, 99216, United States

Location

Multicare Health System Institute For Research and Innovation

Tacoma, Washington, 98405, United States

Location

Blacktown Cancer and Haematology Centre

Blacktown, New South Wales, 2148, Australia

Location

Orange Health Service (Central West Cancer Care Centre)

Orange, New South Wales, 2800, Australia

Location

Riverina Cancer Care Centre

Wagga Wagga, New South Wales, 2650, Australia

Location

Calvary Mater Newcastle

Waratah, New South Wales, 2298, Australia

Location

Pindara Private Hospital

Benowa, Queensland, 4217, Australia

Location

Icon Cancer Centre South Brisbane

South Brisbane, Queensland, 4101, Australia

Location

Flinders Centre For Innovation in Cancer (Fcic)

Bedford Park, South Australia, 5042, Australia

Location

Lyell McEwin Hospital

Elizabeth Vale, South Australia, 5112, Australia

Location

Monash Health

Clayton, Victoria, 3168, Australia

Location

Austin Health

Heidelberg, Victoria, 3084, Australia

Location

The Alfred Hospital

Melbourne, Victoria, 3004, Australia

Location

St John of God, Murdoch

Murdoch, Western Australia, 6150, Australia

Location

One Clinical Research

Nedlands, Western Australia, 6009, Australia

Location

The Second Hospital of Anhui Medical University

Hefei, Anhui, 230601, China

Location

Peking University First Hospital

Beijing, Beijing Municipality, 100034, China

Location

Beijing Tsinghua Changgung Hospital

Beijing, Beijing Municipality, 102218, China

Location

Fujian Medical University Union Hospital

Fuzhou, Fujian, 350001, China

Location

Quanzhou First Affliated Hospital of Fujian Medical University

Quanzhou, Fujian, 362000, China

Location

The First Affiliated Hospital of Xiamen University

Xiamen, Fujian, 361003, China

Location

Gansu Provincial Hospital

Lanzhou, Gansu, 730000, China

Location

Sun Yat Sen Memorial Hospital, Sun Yat Sen University (North)

Guangzhou, Guangdong, 510000, China

Location

Zhujiang Hospital of Southern Medical University

Guangzhou, Guangdong, 510000, China

Location

The First Affiliated Hospital of Shantou University Medical College

Shantou, Guangdong, 515041, China

Location

Nanyang Central Hospital

Nanyang, Henan, 473000, China

Location

Henan Cancer Hospital

Zhengzhou, Henan, 450000, China

Location

Hubei Cancer Hospital

Wuhan, Hubei, 430079, China

Location

Hunan Cancer Hospital

Changsha, Hunan, 410013, China

Location

The First Peoples Hospital of Changzhou

Changzhou, Jiangsu, 213000, China

Location

Nantong First Peoples Hospital

Nantong, Jiangsu, 215124, China

Location

Affiliated Hospital of Jiangnan University South Campus

Wuxi, Jiangsu, 214122, China

Location

The First Hospital of Jilin University

Changchun, Jilin, 130021, China

Location

General Hospital of Ningxia Medical University

Yinchuan, Ningxia, 750004, China

Location

Shandong Cancer Hospital

Jinan, Shandong, 250117, China

Location

Jining No.1 Peoples Hospital West Branch

Jining, Shandong, 272000, China

Location

Linyi Peoples Hospital

Linyi, Shandong, 276000, China

Location

Qingdao Municipal Hospital

Qingdao, Shandong, 266000, China

Location

Renji Hospital Shanghai Jiao Tong University School of Medicine

Shanghai, Shanghai Municipality, 200000, China

Location

Shanghai 10Th Peoples Hospital

Shanghai, Shanghai Municipality, 200072, China

Location

Shanghai East Hospital Branch Hospital

Shanghai, Shanghai Municipality, 200123, China

Location

Shanxi Provincial Cancer Hospital

Taiyuan, Shanxi, 030013, China

Location

Tianjin Medical University Cancer Institute and Hospital

Tianjin, Tianjin Municipality, 300060, China

Location

Tianjin Union Medical Center (Nankai University Affiliated Hospital)

Tianjin, Tianjin Municipality, 300121, China

Location

Karamay Central Hospital of Xinjiang

Karamay, Xinjiang, 834009, China

Location

The Xinjiang Uygur Autonomous Region Peoples Hospital

Ürümqi, Xinjiang, 830001, China

Location

The Second Affiliated Hospital of Zhejiang University School of Medicine

Hangzhou, Zhejiang, 310009, China

Location

Pan American Oncology Trials, Llc

Rio Piedras, 00935, Puerto Rico

Location

MeSH Terms

Conditions

Colorectal Neoplasms

Interventions

tislelizumabBevacizumabCapecitabineFluorouracil

Condition Hierarchy (Ancestors)

Intestinal NeoplasmsGastrointestinal NeoplasmsDigestive System NeoplasmsNeoplasms by SiteNeoplasmsDigestive System DiseasesGastrointestinal DiseasesColonic DiseasesIntestinal DiseasesRectal Diseases

Intervention Hierarchy (Ancestors)

Antibodies, Monoclonal, HumanizedAntibodies, MonoclonalAntibodiesImmunoglobulinsImmunoproteinsBlood ProteinsProteinsAmino Acids, Peptides, and ProteinsSerum GlobulinsGlobulinsDeoxycytidineCytidinePyrimidine NucleosidesPyrimidinesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsUracilPyrimidinonesDeoxyribonucleosidesNucleosidesNucleic Acids, Nucleotides, and Nucleosides

Study Officials

  • Study Director

    BeiGene

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 20, 2022

First Posted

November 8, 2022

Study Start

January 29, 2023

Primary Completion

May 23, 2025

Study Completion (Estimated)

December 31, 2026

Last Updated

October 2, 2025

Record last verified: 2025-09

Data Sharing

IPD Sharing
Will share

BeiGene shares data on completed studies responsibly and provides qualified scientific and medical researchers access to data and supporting documentation for clinical trials in dossiers for medicines and indications after submission and approval in the United States, China, and Europe. Clinical trials supporting subsequent local approvals, new indications, or combination products are eligible for sharing once corresponding regulatory approvals are achieved. BeiGene shares data only when permitted by applicable data privacy and security laws and regulations, when it is feasible to do so without compromising the privacy of study participants, and other considerations. Qualified researchers with appropriate competencies who are engaged in novel scientific research may submit a request for participant-level data with a research proposal for BeiGene review. Research teams must include a biostatistician and sign a Data Sharing Agreement prior to receiving access to clinical trial data.

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
See plan description
Access Criteria
See plan description
More information

Locations