NCT04940052

Brief Summary

The purpose of this study is to assess the efficacy and safety of dabrafenib in combination with trametinib for treating adult patients with locally advanced or metastatic Differentiated Thyroid Cancer (DTC) harboring the BRAFV600E mutation, who are refractory to radioactive iodine (RAI) therapy and have experienced disease progression following one or two prior VEGFR-targeted treatments.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
153

participants targeted

Target at P25-P50 for phase_3

Timeline
13mo left

Started Nov 2021

Longer than P75 for phase_3

Geographic Reach
11 countries

41 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress81%
Nov 2021Jun 2027

First Submitted

Initial submission to the registry

June 22, 2021

Completed
3 days until next milestone

First Posted

Study publicly available on registry

June 25, 2021

Completed
5 months until next milestone

Study Start

First participant enrolled

November 15, 2021

Completed
3.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 22, 2025

Completed
2.4 years until next milestone

Study Completion

Last participant's last visit for all outcomes

June 4, 2027

Expected
Last Updated

December 2, 2025

Status Verified

November 1, 2025

Enrollment Period

3.2 years

First QC Date

June 22, 2021

Last Update Submit

November 24, 2025

Conditions

Keywords

Differentiated Thyroid Cancer (DTC)Locally advanced or metastatic differentiated thyroid cancerradio active iodine refractorypreviously targeted therapyB-Raf proto-oncogene, serine/threonine kinase (BRAF)BRAFV600E mutationDabrafenib (DRB436)trametinib (TMT212)

Outcome Measures

Primary Outcomes (1)

  • Progression Free Survival (PFS)

    Progression Free Survival (PFS) was defined as the time from the date of randomization to the date of the first documented progression according to RECIST 1.1 based on Blinded Independent Review Committee (BIRC) assessment, or death due to any cause.

    From randomization to first documented progression or deaths, whichever comes first, assessed up to approximately 2 years

Secondary Outcomes (5)

  • Overall Response Rate (ORR)

    From randomization up to approximately 2 years

  • Overall Survival (OS)

    From randomization to death assessed up to approximately 5 years

  • Duration of Response (DOR)

    From the start date of the first documented response of complete response or partial response and the date defined as the date of the first documented progression or death due to any cause up to 2 years

  • Number of participants with Adverse Events (AEs) and Serious Adverse Events (SAEs)

    Throughout study completion, an average 5 years

  • Number of participants with trametinib associated serous retinopathy ocular events

    screening, week 4, week 8, week 12, week 20 and every 12 weeks after week 20, up to approximately 2 years

Study Arms (2)

Dabrafenib plus Trametinib

EXPERIMENTAL

Eligible participants will receive Dabrafenib 150 mg twice a day (BID) and Trametinib 2 mg once a day (QD) until disease progression as per RECIST 1.1 as confirmed by blinded independent review committee (BIRC), unacceptable toxicity, pregnancy, loss of clinical benefit as determined by the investigator, withdrawal of consent, lost to follow-up, death, or study termination by the sponsor.

Drug: DabrafenibDrug: Trametinib

Dabrafenib Placebo plus Trametinib Placebo

PLACEBO COMPARATOR

Eligible participants will receive matching placebo for Dabrafenib 150 mg twice a day (BID) and matching placebo for Trametinib 2 mg once a day (QD) until disease progression as per RECIST 1.1 as confirmed by blinded independent review committee (BIRC), unacceptable toxicity, pregnancy, loss of clinical benefit as determined by the investigator, withdrawal of consent, lost to follow-up, death, or study termination by the sponsor.

Drug: Trametinib PlaceboDrug: Dabrafenib placebo

Interventions

Dabrafenib 150 mg capsule administered orally twice a day (BID)

Also known as: DRB436
Dabrafenib plus Trametinib

Trametinib 2 mg tablet administered once a day (QD)

Also known as: TMT212
Dabrafenib plus Trametinib

matching placebo tablet for Trametinib 2 mg will be administered orally once a day (QD)

Dabrafenib Placebo plus Trametinib Placebo

matching placebo capsule for Dabrafenib 150 mg will be administered orally twice a day (BID)

Dabrafenib Placebo plus Trametinib Placebo

Eligibility Criteria

Age18 Years - 99 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Signed informed consent
  • Male or female ≥ 18 years of age at time of informed consent
  • Histologically or cytologically confirmed diagnosis of advanced/metastatic differentiated thyroid carcinoma
  • Radioactive-iodine refractory disease
  • BRAF V600E mutation-positive tumor sample as per central laboratory result
  • Has progressed on at least 1 but not more than 2 prior VEGFR targeted therapies
  • Eastern Cooperative Oncology Group (ECOG) performance status ≤ 2
  • At least one measurable lesion as defined by RECIST v1.1.

You may not qualify if:

  • Anaplastic or medullary carcinoma of the thyroid
  • Previous treatment with a BRAF inhibitor and/or a MEK inhibitor
  • Concomitant RET Fusion-Positive Thyroid Cancer
  • Treatment with any type of small molecule kinase inhibitor (including investigational kinase inhibitor) within 2 weeks before randomization
  • Treatment with any type of anticancer antibody (including investigational antibody) or systemic chemotherapy within 4 weeks before randomization
  • Treatment with radiation therapy for bone metastasis within 2 weeks or any other radiation therapy within 4 weeks before randomization
  • A history or current evidence/risk of retinal vein occlusion (RVO) or central serous retinopathy

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (41)

Northwestern University Med School

Chicago, Illinois, 60611, United States

Location

Massachusetts General Hospital

Boston, Massachusetts, 02114, United States

Location

Novartis Investigative Site

CABA, Buenos Aires, C1417DTB, Argentina

Location

Novartis Investigative Site

Rio de Janiero, Rio de Janeiro, 20231-050, Brazil

Location

Novartis Investigative Site

Blumenau, Santa Catarina, 89015-200, Brazil

Location

Novartis Investigative Site

São Paulo, São Paulo, 01246-000, Brazil

Location

Novartis Investigative Site

Edmonton, Alberta, T6G 1Z2, Canada

Location

Novartis Investigative Site

London, Ontario, N6A 5W9, Canada

Location

Novartis Investigative Site

Fuzhou, Fujian, 350014, China

Location

Novartis Investigative Site

Zhengzhou, Henan, 450008, China

Location

Novartis Investigative Site

Wuhan, Hubei, 430022, China

Location

Novartis Investigative Site

Changsha, Hunan, 410013, China

Location

Novartis Investigative Site

Nanjing, Jiangsu, 210006, China

Location

Novartis Investigative Site

Nanjing, Jiangsu, 210009, China

Location

Novartis Investigative Site

Xuzhou, Jiangsu, 221003, China

Location

Novartis Investigative Site

Changchun, Jilin, 130033, China

Location

Novartis Investigative Site

Chengdu, Sichuan, 610041, China

Location

Novartis Investigative Site

Tianjin, Tianjin Municipality, 300121, China

Location

Novartis Investigative Site

Beijing, 100036, China

Location

Novartis Investigative Site

Beijing, 100730, China

Location

Novartis Investigative Site

Guangzhou, 510060, China

Location

Novartis Investigative Site

Shanghai, 200233, China

Location

Novartis Investigative Site

Tianjin, 300052, China

Location

Novartis Investigative Site

Tianjin, 300480, China

Location

Novartis Investigative Site

Hisar, Haryana, 125005, India

Location

Novartis Investigative Site

New Delhi, National Capital Territory of Delhi, 110029, India

Location

Novartis Investigative Site

Chennai, 600 020, India

Location

Novartis Investigative Site

George Town, Pulau Pinang, 10450, Malaysia

Location

Novartis Investigative Site

Kuching, Sarawak, 93586, Malaysia

Location

Novartis Investigative Site

Kuala Lumpur, 59100, Malaysia

Location

Novartis Investigative Site

Seoul, Korea, 03080, South Korea

Location

Novartis Investigative Site

Seoul, 05505, South Korea

Location

Novartis Investigative Site

Seoul, 06351, South Korea

Location

Novartis Investigative Site

Seoul, 06591, South Korea

Location

Novartis Investigative Site

Tainan, 70403, Taiwan

Location

Novartis Investigative Site

Taipei, 10002, Taiwan

Location

Novartis Investigative Site

Istanbul, Fatih, 34098, Turkey (Türkiye)

Location

Novartis Investigative Site

Edirne, Merkez, 22030, Turkey (Türkiye)

Location

Novartis Investigative Site

Ankara, Yenimahalle, 06500, Turkey (Türkiye)

Location

Novartis Investigative Site

Adana, Yuregir, 01250, Turkey (Türkiye)

Location

Novartis Investigative Site

Hanoi, 100000, Vietnam

Location

MeSH Terms

Interventions

dabrafenibtrametinib

Study Officials

  • Novartis Pharmaceuticals

    Novartis Pharmaceuticals

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
CROSSOVER
Model Details: Patients will be randomized in a 2:1 ratio to either dabrafenib plus trametinib or placebo. Patients will be stratified by number of prior VEGFR targeted therapy (1 versus 2) and prior Lenvatinib treatment (yes versus no).
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 22, 2021

First Posted

June 25, 2021

Study Start

November 15, 2021

Primary Completion

January 22, 2025

Study Completion (Estimated)

June 4, 2027

Last Updated

December 2, 2025

Record last verified: 2025-11

Data Sharing

IPD Sharing
Will share

Novartis is committed to sharing with qualified external researchers, access to patient-level data and supporting clinical documents from eligible studies. These requests are reviewed and approved by an independent review panel on the basis of scientific merit. All data provided is anonymized to respect the privacy of patients who have participated in the trial in line with applicable laws and regulations. This trial data availability is according to the criteria and process described on www.clinicalstudydatarequest.com.

Locations