NCT04398329

Brief Summary

This is a Phase 1b/2, randomized, blinded, active-controlled study. Phase 1b will evaluate escalating doses of HTX-034 compared with bupivacaine HCl. Phase 2 will be a dose-expansion phase to evaluate additional subjects treated with the HTX-034 dose selected based on Phase 1b compared with bupivacaine HCl.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
73

participants targeted

Target at P75+ for phase_1

Timeline
Completed

Started May 2020

Geographic Reach
1 country

4 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

May 18, 2020

Completed
Same day until next milestone

Study Start

First participant enrolled

May 18, 2020

Completed
3 days until next milestone

First Posted

Study publicly available on registry

May 21, 2020

Completed
1.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 1, 2021

Completed
1 month until next milestone

Study Completion

Last participant's last visit for all outcomes

August 3, 2021

Completed
Last Updated

February 15, 2022

Status Verified

January 1, 2022

Enrollment Period

1.1 years

First QC Date

May 18, 2020

Last Update Submit

January 31, 2022

Conditions

Keywords

AnalgesiaBunionectomy

Outcome Measures

Primary Outcomes (2)

  • Incidence of Treatment-emergent adverse events (TEAE's) (Phase 1B)

    42 days

  • Mean area under the curve (AUC) of the NRS scores through 72 hours (AUC0-72) for the pooled Phase 1b and Phase 2

    7 days

Secondary Outcomes (9)

  • Maximum plasma concentration (Cmax) of HTX-034

    29 days

  • Time of maximum plasma concentration (Tmax) of HTX-034

    29 days

  • Area under the concentration-time curve from Time 0 to the time of the last quantitative concentration (AUClast) of HTX-034

    29 days

  • Area under the concentration-time curve from Time 0 extrapolated to infinity (AUCinf) of HTX-034 (Phase 1B)

    22 days

  • Apparent terminal half-life (t½) of HTX-034 (Phase 1B)

    22 days

  • +4 more secondary outcomes

Study Arms (5)

Phase 1b (Cohort 1)

EXPERIMENTAL

Fixed dose of HTX-034.

Drug: HTX-034Device: Luer lock applicator

Phase 1b (Cohort 2)

EXPERIMENTAL

Individualized dose of HTX-034.

Drug: HTX-034Device: Luer lock applicator

Phase 2 (Expansion): Low Dose

EXPERIMENTAL

Fixed dose of HTX-034.

Drug: HTX-034Device: Luer lock applicator

Phase 2 (Expansion): High Dose

EXPERIMENTAL

Individualized dose of HTX-034.

Drug: HTX-034Device: Luer lock applicator

Phase 1b and Phase 2

ACTIVE COMPARATOR

Bupivacaine HCl.

Drug: Bupivacaine HCl

Interventions

HTX-034, low dose

Phase 1b (Cohort 1)Phase 2 (Expansion): Low Dose

Applicator for instillation

Phase 1b (Cohort 1)Phase 1b (Cohort 2)Phase 2 (Expansion): High DosePhase 2 (Expansion): Low Dose

Bupivacaine HCl, 50 mg

Phase 1b and Phase 2

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Is medically fit to undergo an elective unilateral, first metatarsal bunionectomy with osteotomy and internal fixation under regional anesthesia; no neuraxial technique (eg, no spinal, epidural, or general anesthesia).
  • Has an American Society of Anesthesiologists (ASA) Physical Status of I, II, or III.
  • Female subjects are eligible only if not pregnant, not lactating, not planning to become pregnant during the study; sterile, or using acceptable contraceptives.

You may not qualify if:

  • Had contralateral foot bunionectomy in the past 3 months.
  • Has a planned concurrent surgical procedure.
  • Has a contraindication or a known or suspected history of hypersensitivity or clinically significant idiosyncratic reaction to required study medications.
  • Has a pre-existing concurrent acute or chronic painful physical/restrictive condition expected to require analgesic treatment in the postoperative period for pain.
  • Has received or is taking a contraindicated or prohibited medications.
  • Received an investigational product or device in a clinical trial within 30 days or within 5 elimination half lives.
  • Has a known or suspected history of drug abuse, a positive drug screen on the day of surgery, or a recent history of alcohol abuse.
  • Has a history of clinically significant cardiac abnormality such as myocardial infarction within 6 months.
  • Has a history of coronary artery bypass graft surgery within 12 months.
  • Has a history of known or suspected coagulopathy.
  • As per subject history and/or medical records, has active infection or is currently undergoing treatment for Hepatitis B, Hepatitis C, or human immunodeficiency virus (HIV).
  • Has uncontrolled anxiety, psychiatric, or neurological disorder.
  • Had a malignancy in the last year, with the exception of nonmetastatic basal cell or squamous cell carcinoma of the skin or localized carcinoma in situ of the cervix.
  • Has undergone 3 or more surgeries within 12 months.
  • Has a known history of glucose-6-phosphate dehydrogenase deficiency.
  • +5 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (4)

Arizona Research Center

Phoenix, Arizona, 85053, United States

Location

First Surgical Hospital

Bellaire, Texas, 77401, United States

Location

Endeavor Clinical Trials, LLC

San Antonio, Texas, 78229, United States

Location

JBR Clinical Research

Salt Lake City, Utah, 84017, United States

Location

MeSH Terms

Conditions

BunionAgnosia

Interventions

Bupivacaine

Condition Hierarchy (Ancestors)

Foot Deformities, AcquiredFoot DeformitiesMusculoskeletal DiseasesPerceptual DisordersNeurobehavioral ManifestationsNeurologic ManifestationsNervous System DiseasesSigns and SymptomsPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

AnilidesAmidesOrganic ChemicalsAniline CompoundsAmines

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 18, 2020

First Posted

May 21, 2020

Study Start

May 18, 2020

Primary Completion

July 1, 2021

Study Completion

August 3, 2021

Last Updated

February 15, 2022

Record last verified: 2022-01

Locations