NCT04224493

Brief Summary

The participants of this study would have relapsed/refractory follicular lymphoma. Follicular lymphoma is a type of blood cancer. It is referred to as 'relapsed' when the disease has come back after a period of improvement after that follows a treatment regimen and 'refractory' when treatment no longer works. Stage 1 of this trial will study the safety and the level that adverse effects of each of the study drug combinations can be tolerated (known as tolerability). It is also designed to establish a recommended study drug dosage for stage 2 and 3. Stage 1 of the study is completed. Stages 2 and 3 will evaluate and compare how long participants live without their disease getting worse when receiving the study drug in combination with other drug treatment versus the placebo (dummy drug) in combination with other drug treatment.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
555

participants targeted

Target at P75+ for phase_3

Timeline
34mo left

Started Jun 2020

Longer than P75 for phase_3

Geographic Reach
17 countries

204 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress68%
Jun 2020Mar 2029

First Submitted

Initial submission to the registry

December 12, 2019

Completed
1 month until next milestone

First Posted

Study publicly available on registry

January 13, 2020

Completed
5 months until next milestone

Study Start

First participant enrolled

June 11, 2020

Completed
6.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 13, 2027

Expected
2 years until next milestone

Study Completion

Last participant's last visit for all outcomes

March 1, 2029

Last Updated

April 20, 2026

Status Verified

April 1, 2026

Enrollment Period

6.7 years

First QC Date

December 12, 2019

Last Update Submit

April 17, 2026

Conditions

Keywords

EpizymeTazverikTazemetostat (EPZ-6438)LenalidomideRevlimidRituximabRituxanFollicular lymphomaEZH2

Outcome Measures

Primary Outcomes (3)

  • Recommended Phase 3 Dose (RP3D) of tazemetostat in combination with rituximab and lenalidomide (R2)

    The safety and tolerability of tazemetostat in combination with R2 in subjects with R/R FL will be evaluated. RP3D of tazemetostat for further evaluation in phase 3 will be selected as assessed by the occurrence of treatment-emergent dose-limiting toxicities (DLTs) and adverse events (AEs).

    Subjects are evaluated for DLTs during the first 28-day cycle. The RP3D for Phase 3 was selected at the end of Stage 1

  • Progression-Free Survival (PFS) in the Intent-to-treat wild-type (ITT-WT) population

    PFS is defined as the time from the date of randomization to the time of confirmed disease progression per the 2014 Lugano Classification or death, whichever occurs first, as assessed by Investigators.

    Stage 2: Up to 72 months

  • PFS in the Intent-to-treat mutant-type (ITT-MT) population

    PFS is defined as the time from the date of randomization to the time of confirmed disease progression per the 2014 Lugano Classification or death, whichever occurs first, as assessed by Investigators.

    Stage 2: Up to 72 months

Secondary Outcomes (38)

  • Pharmacokinetics (PK) of tazemetostat: Maximum (peak) Observed Plasma Drug Concentration (Cmax).

    Stage 1: In cycles 1 and 2 on days 1 and 15 (28 days cycle)

  • PK of tazemetostat, EPZ 6930 (desethyl metabolite), and lenalidomide as data permit: Time to Maximum Observed Drug Concentration (Tmax)

    Stage 1: In cycles 1 and 2 on days 1 and 15 (28 days cycle)

  • PK of tazemetostat: area under the plasma concentration-time curve (AUC) from time 0 to the time of the last quantifiable concentration [AUC(0-t)],

    Stage 1: In cycles 1 and 2 on days 1 and 15 (28 days cycle)

  • PK of tazemetostat: area under the plasma concentration-time curve (AUC) from time 0 to infinity [AUC(0-∞)]

    Stage 1: In cycles 1 and 2 on days 1 and 15 (28 days cycle)

  • The apparent terminal elimination half-life (t1/2) of tazemetostat, EPZ 6930 (desethyl metabolite), and lenalidomide as data permit

    Stage 1: In cycles 1 and 2 on days 1 and 15 (28 days cycle)

  • +33 more secondary outcomes

Study Arms (2)

Tazemetostat + R2 arm

EXPERIMENTAL

Stage 1 (Phase 1b): This phase is now completed. * Tazemetostat was escalated from a starting dose of 400 mg PO twice daily to 600 mg PO twice daily to 800 mg PO twice daily in 28-day cycles. * Rituximab 375 mg/m2 IV on days 1, 8, 15, and 22 of cycle 1; then on day 1 of cycles 2 to 5. * Lenalidomide 20 mg or 10 mg (if creatinine clearance ≥60 mL/minute or \<60 mL/minute), administred PO QD on days 1 to 21 for 12 cycles. Stage 2: * Tazemetostat 800 mg administered PO twice daily in continuous 28-day cycles. * Rituximab 375 mg/m2 IV on days 1, 8, 15, and 22 of cycle 1; then on day 1 of cycles 2 to 5. * Lenalidomide 20 mg or 10 mg (if creatinine clearance ≥60 mL/minute or \<60 mL/minute), PO QD on days 1 to 21 for 12 cycles. Maintenance Therapy (Stages 1 and 2): Tazemetostat will be administered as monotherapy at an 800 mg twice daily dose for up to 2 years after the initial 12 months of combination therapy.

Drug: TazemetostatCombination Product: LenalidomideCombination Product: Rituximab

Placebo + R2 Arm

PLACEBO COMPARATOR

Stage 2: * Placebo administered PO twice daily in continuous 28-day cycles. * Rituximab 375 mg/m2 IV on days 1, 8, 15, and 22 of cycle 1; then on day 1 of cycles 2 to 5. * Lenalidomide 20 mg or 10 mg (if creatinine clearance ≥60 mL/minute or \<60 mL/minute), administered PO QD on days 1 to 21 for 12 cycles. Maintenance Therapy (Stage 2): Placebo will be administered as monotherapy twice daily dose for up to 2 years after the initial 12 months of combination therapy. During maintenance, placebo will be continued until disease progression or unacceptable toxicity, or participant withdraws consent.

Drug: Placebo oral tabletCombination Product: LenalidomideCombination Product: Rituximab

Interventions

Stage 2: Placebo administered orally twice daily in continuous 28-day cycles. Placebo will be administered as monotherapy twice daily dose for up to 2 years after the initial 12 months of combination therapy.

Placebo + R2 Arm
LenalidomideCOMBINATION_PRODUCT

Lenalidomide 20 mg capsules or 10 mg capsules (if creatinine clearance ≥60 mL/minute or \<60 mL/minute), administered PO QD on days 1 to 21 for 12 cycles.

Placebo + R2 ArmTazemetostat + R2 arm
RituximabCOMBINATION_PRODUCT

Rituximab 375 mg/m2 IV on days 1, 8, 15, and 22 of cycle 1; then on day 1 of cycles 2 to 5.

Placebo + R2 ArmTazemetostat + R2 arm

Stage 1 (Phase 1b): Tazemetostat was escalated from a starting dose of 400 mg orally twice daily to 600 mg orally twice daily to 800 mg PO twice daily in 28-day cycles as tolerated in a standard 3 + 3 design. Tazemetostat will be administered as monotherapy at an 800 mg twice daily dose for up to 2 years after the initial 12 months of combination therapy.

Also known as: EPZ-6438, IPN60200
Tazemetostat + R2 arm

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Have voluntarily agreed to provide written informed consent and demonstrated willingness and ability to comply with all aspects of the protocol.
  • Males or females are ≥18 years of age, or per country adult legal age regulations, at the time of providing voluntary written informed consent.
  • Life expectancy ≥3 months before enrollment.
  • Meet requirement for hepatitis and human immunodeficiency virus (HIV) infection as follows
  • Negative serologic or polymerase chain reaction (PCR) test results for acute or chronic hepatitis B virus (HBV) infection Note: Participants whose HBV infection status could not be determined by serologic test results have to be negative for HBV-DNA by PCR to be eligible for study participation. Participants seropositive for HBV with undetectable HBV DNA by PCR are permitted with appropriate antiviral prophylaxis.
  • Negative test results for hepatitis C virus (HCV) Note: Participants who are positive for HCV antibody must be negative for HCV RNA by PCR to be eligible for study participation

You may not qualify if:

  • Have histologically confirmed FL, Grades 1 to 3A.
  • Must have been previously treated with at least 1 prior systemic chemotherapy, immunotherapy, or chemoimmunotherapy:
  • a. Systemic therapy includes treatments such as:
  • i. Rituximab monotherapy
  • ii. Chemotherapy given with or without rituximab
  • iii. Radioimmunoconjugates such as 90Y-ibritumomab tiuxetan and 131I-tositumomab.
  • b. Systemic therapy does not include, for example:
  • i. Local involved field radiotherapy for limited-stage disease
  • ii. Helicobacter pylori eradication
  • d. Prior autologous/allogeneic hematopoietic stem cell transplant (HSCT) will be allowed.
  • e. Prior chimeric antigen receptor T-cell therapy (CAR T) will be allowed.
  • Must have documented relapsed, refractory, or PD after treatment with systemic therapy (refractory defined as less than PR or disease progression \<6 months after last dose).
  • Have measurable disease as defined by the Lugano Classification (Cheson, 2014; Appendix 5).
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0, 1, or 2.
  • Within 7 days prior to randomization, all clinically significant toxicity related to a prior anticancer treatment (ie, chemotherapy, immunotherapy, and/or radiotherapy must have either resolved to Grade 1 per NCI CTCAE Version 5.0 OR are clinically stable and no longer clinically significant.
  • +63 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (204)

Southern Cancer Center

Mobile, Alabama, 36608, United States

Location

Arizona Oncology Associates - Tuscon-Rusadill Road

Tucson, Arizona, 85704, United States

Location

TOI - Clinical Research

Cerritos, California, 90703, United States

Location

UCSF Fresno

Clovis, California, 93611, United States

Location

UC San Diego Health Sciences

La Jolla, California, 92093, United States

Location

UCLA Clinical Research Unit Hematology/Oncology

Santa Monica, California, 90404, United States

Location

Rocky Mountain Cancer Centers (RMCC) - Boulder

Boulder, Colorado, 80303, United States

Location

St. Mary's Hospital and Regional Medical Center - St. Mary's

Grand Junction, Colorado, 81501, United States

Location

Cancer Specialists of North Florida

Fleming Island, Florida, 32003, United States

Location

Florida Cancer Specialists & Research Institute (FCS) - Fort Myers Cancer Center

Fort Myers, Florida, 33908, United States

Location

Mayo Clinic

Jacksonville, Florida, 32224, United States

Location

Florida Cancer Affiliates/Ocala Oncology - Clinic

Ocala, Florida, 34474, United States

Location

BRCR Medical Center, INC

Plantation, Florida, 33322, United States

Location

Florida Cancer Specialists

St. Petersburg, Florida, 33705, United States

Location

Florida Cancer Specialists - Panhandle

Tallahassee, Florida, 32308, United States

Location

H Lee Moffitt Cancer Center and Research Institute I

Tampa, Florida, 33612, United States

Location

Florida Cancer Specialists & Research Institute (FCS) - Atlantis

West Palm Beach, Florida, 33401, United States

Location

University of Chicago

Chicago, Illinois, 60637, United States

Location

Illinois Cancer Specialists

Niles, Illinois, 60714, United States

Location

University of Michigan Comprehensive Cancer Center

Ann Arbor, Michigan, 48109, United States

Location

St. Joseph Mercy Hospital

Ypsilanti, Michigan, 48197, United States

Location

Mayo Clinic - Rochester

Rochester, Minnesota, 55901, United States

Location

University Of Nebraska Medical Center

Omaha, Nebraska, 68198, United States

Location

Astera Cancer Care

East Brunswick, New Jersey, 08816, United States

Location

Astera Cancer Center

East Brunswick, New Jersey, 08816, United States

Location

Regional Cancer Care Associates-Freehold

Freehold, New Jersey, 07728, United States

Location

Regional Cancer Care Associates LLC - Little Silver

Little Silver, New Jersey, 07739, United States

Location

New Mexico Cancer Care Alliance

Albuquerque, New Mexico, 87131-0001, United States

Location

Weill Cornell Medicine-New York Presbyterian Hospital

New York, New York, 10021, United States

Location

Columbia U - Herbert Irving Comprehensive Cancer Center

New York, New York, 10032, United States

Location

Memorial Sloan-Kettering Cancer Center

New York, New York, 10065, United States

Location

Hematology Oncology Associates of Rockland, P.C.

Nyack, New York, 10960, United States

Location

Messino Cancer Center

Asheville, North Carolina, 28806, United States

Location

Levine Cancer Institute - Concord

Concord, North Carolina, 28205, United States

Location

FirstHealth of the Carolinas

Pinehurst, North Carolina, 28374, United States

Location

Regional Medical Oncology Center

Wilson, North Carolina, 27895, United States

Location

Gabrail Cancer Center Research

Canton, Ohio, 44718, United States

Location

Oncology Hematology Care (OHC), Inc. - Kenwood Office

Cincinnati, Ohio, 45236, United States

Location

Willamette Valley Cancer Institute and Research Center - Oncology

Eugene, Oregon, 97401, United States

Location

Western Pennsylvania Hospital Hematology & Cellular Therapy

Pittsburgh, Pennsylvania, 15524, United States

Location

Sarah Cannon Research Institute

Nashville, Tennessee, 37203, United States

Location

Texas Oncology - Amarillo

Amarillo, Texas, 79124, United States

Location

Texas Oncology-Austin Midtown

Austin, Texas, 78705, United States

Location

Texas Oncology - Medical City Dallas Pediatric Hematology

Dallas, Texas, 75230, United States

Location

Texas Oncology-Baylor Charles A. Sammons Cancer Center

Dallas, Texas, 75246, United States

Location

The University of Texas MD Anderson Cancer Center

Houston, Texas, 77030, United States

Location

Millennium Physicians - Oncology

Houston, Texas, 77090, United States

Location

Texas Oncology

Plano, Texas, 75075, United States

Location

Mays Cancer Center

San Antonio, Texas, 78229, United States

Location

UT Health East Texas HOPE Cancer Center - Tyler

Tyler, Texas, 75701, United States

Location

USO Texas Oncology - Tyler

Tyler, Texas, 75702, United States

Location

Texas Oncology- Weslaco

Weslaco, Texas, 78596, United States

Location

Utah Cancer Specialists/ IHO Corp

Salt Lake City, Utah, 84106, United States

Location

Huntsman Cancer Institute; The University of Utah

Salt Lake City, Utah, 84112, United States

Location

Virginia Cancer Specialists

Gainesville, Virginia, 22155, United States

Location

Oncology and Hematology Associates of Southwest Virginia Inc.

Roanoke, Virginia, 24014, United States

Location

Wheeling Hospital

Wheeling, West Virginia, 26003, United States

Location

Royal Adelaide Hospital

Adelaide, South Australia, 5000, Australia

Location

Flinders Medical Centre

Bedford Park, South Australia, 5042, Australia

Location

Monash Health

Clayton, Victoria, 3168, Australia

Location

Barwon Health, University Hospital Geelong

Geelong, Victoria, 3220, Australia

Location

Hollywood Private Hospital

Nedlands, Western Australia, 6009, Australia

Location

GenesisCare - St Andrew's

Adelaide, Australia

Location

Peninsula Health - Frankston

Frankston, Australia

Location

Royal Hobart Hospital

Hobart, Australia

Location

Gold Coast University Hosptial

Southport, Australia

Location

Universitair Ziekenhuis Gent

Ghent, Oost-Vlaanderen, 9000, Belgium

Location

UZ Leuven - Campus Gasthuisberg

Leuven, Vlaams Brabant, 3000, Belgium

Location

Hospital Haroldo Juacaba - Instituto do Cancer do Ceara

Ceará, Brazil

Location

Hospital Santa Cruz

Curitiba, Brazil

Location

HC-UFG - Hospital das CLINICAS da Universidade Federal de Go

Goiânia, Brazil

Location

Association Hospital de Caridade de Iju

Ijuí, Brazil

Location

Liga Norte Riograndense Contra o Cancer

Natal, Brazil

Location

Hospital de Clinicas de Porto Alegre - Centro de Pesquisa Clinica

Porto Alegre, Brazil

Location

Instituto D'Or de Pesquisa e Ensino- Recife

Recife, Brazil

Location

Instituto de Psiquiatria - UFRJ

Rio de Janeiro, Brazil

Location

Instituto Nacional de Câncer - INCA

Rio de Janeiro, Brazil

Location

Fundacao Antonio Prudente - Hospital A.C.Camargo Cancer Center

São Paulo, Brazil

Location

Hospital Alemao Oswaldo Cruz (HAOC)

São Paulo, Brazil

Location

Instituto D'or de Pesquisa e Ensino

São Paulo, Brazil

Location

Instituto de Oncologia e Hematologia - HEMOMED

São Paulo, Brazil

Location

Irmandade Santa Casa de Misericordia de Sao Paulo

São Paulo, Brazil

Location

University Health Network Princess Margaret Hospital

Toronto, Ontario, M5G 2M9, Canada

Location

Centre Hospitalier de l'Universite de Montreal (CHUM)

Montreal, Quebec, H2X 3E4, Canada

Location

Sir Mortimer B Davis/Jewish General Hospital

Montreal, Quebec, H3T 1E2, Canada

Location

Nova Scotia Health Centre for Clinical Research

Nova Scotia, Canada

Location

Sunnybrook Health Sciences Centre Odette Cancer Centre

Ottawa, Canada

Location

Fujian Medical University Union Hospital

Fuzhou, Fujian, 350001, China

Location

The First Affiliated Hospital of Xiamen University

Xiamen, Fujian, 361003, China

Location

The Affiliated Hospital of Guizhou Medical University

Guiyang, Guizhou, 550004, China

Location

The Second Affiliated Hospital Zhejiang University School of Medicine

Zhejiang, Hangzhou, 310000, China

Location

The Fourth Hospital of Hebei Medical University

Shijiazhuang, Hebei, 050011, China

Location

Henan Provincial People's Hospital

Zhengzhou, Henan, 450008, China

Location

Henan Cancer Hospital

Zhengzhou, Henan, 45008, China

Location

Hunan Cancer Hospital

Changsha, Hunan, 410013, China

Location

The First Bethune Hospital of Jilin University

Changchun, Jinlin, 130021, China

Location

The Affiliated Hospital of Qingdao University

Qingdao, Shandong, 266071, China

Location

Ruijin Hospital, Shanghai Jiaotong University School of Medicine

Shanghai, Shanghai Municipality, 20025, China

Location

Shanxi Bethune Hospital

Taiyuan, Shanxi, 30032, China

Location

Peking University Third Hospital

Beijing, 100191, China

Location

The First Affiliated Hospital Zhejiang University School of Medicine

Hangzhou, China

Location

Tongji Hospital of Tongji Medical College of HUST

Hangzhou, China

Location

Jiangxi Cancer Hospital

Nanchang, China

Location

Shandong Cancer Hospital

Shandong, China

Location

Tongji Hospital of Tongji University

Shanghai, China

Location

Sichuan Provincial People's Hospital

Sichuan, China

Location

Tianjin Medical University Cancer Institute & Hospital

Tianjin, 300060, China

Location

Centre Hospitalier Universitaire de Bordeaux-Hopital du Haut Leveque

Pessac, Aquitaine, 33600, France

Location

CHRU Brest Hôp Morvan

Brest, Brittany Region, 29609, France

Location

Institut Bergonie

Bordeaux, Gironde, 33000, France

Location

Centre Hosp Mulh Hop Emile Muller

Mulhouse, Haut-Rhin, 68100, France

Location

Centre Henri Becquerel

Rouen, Haute-Normandie, 76038, France

Location

CHU de Limoges Dupuytren

Limoges, Haute-Vienne, 87042, France

Location

CHU de Grenoble - Hopital Albe

La Tronche, Isere, 38700, France

Location

CHU de Nantes - Hematologie

Nantes, Loire-Atlantique, 44000, France

Location

CHRU de Lille Hop Claude Huriez

Lille, Nord, 59037, France

Location

Centre Hospitalier Le Mans

Le Mans, Sarthe, 72000, France

Location

Centre Hospitalier Universitaire D'Angers - Hématologie Clinique

Angers, France

Location

CHRU de Besançon- Hopital Jean Minjoz

Besançon, 25000, France

Location

CHU de Clermont-Ferrand, site Estaing

Clermont-Ferrand, 63000, France

Location

Centre Hospitalier Docteur Schaffner

Lens, France

Location

L'Hôpital Privé Confluent

Nantes, 44202, France

Location

L'hôpital Privé du Concluent

Nantes, France

Location

Hopital Saint Louis

Paris, 75010, France

Location

Centre Hospitalier - Hôpital de jour d'Hématologie

Périgueux, France

Location

Centre Hospitalier Universitaire de Poitiers

Poitiers, France

Location

CHU de Nancy Brabois

Vandœuvre-lès-Nancy, 54511, France

Location

Centre Hospitalier Bretagne Atlantique

Vannes, 56017, France

Location

Institut Gustave Roussy

Villejuif, France

Location

Hopital Henri Mondor - Hemopathies Lymphoides

Créteil, Île-de-France Region, 94010, France

Location

Diakoneo Diak Schwaebisch Hall gGmbH

Schwäbisch Hall, Baden-Wurttemberg, 74523, Germany

Location

Klinikum Der Universität München AöR

München, Bavaria, 81377, Germany

Location

Universitätsmedizin Mainz

Mainz, Hesse, 55131, Germany

Location

Universitaetsklinikum Bonn AöR

Bonn, North Rhine-Westphalia, 53127, Germany

Location

Kliniken Maria Hilf GmbH

Mönchengladbach, North Rhine-Westphalia, 41063, Germany

Location

Städt. Krankenhaus Kiel

Kiel, Schleswig-Holstein, 24116, Germany

Location

Vivantes Klinikum am Urban Hämatologie und Onkologie

Berlin, Germany

Location

University Medical Center Schleswig Holstein

Kiel, Germany

Location

Debreceni Egyetem Klinikai Központ

Debrecen, Hajdú-Bihar, 4032, Hungary

Location

Semmelweis Egyetem Általános Orvostudományi Kar

Budapest, 1088, Hungary

Location

Országos Onkológiai Intézet

Budapest, 1122, Hungary

Location

AOU Federico II

Naples, Campania, 80122, Italy

Location

Istituto Romagnolo per lo Studio dei Tumori (IRST) Dino Amadori IRCCS

Meldola, Forli-Cesena, 47014, Italy

Location

ASST Spedali Civili di Brescia

Brescia, 25123, Italy

Location

PO Garibaldi-Nesima, ARNAS Garibaldi

Catania, 95122, Italy

Location

AOU Careggi

Florence, 50134, Italy

Location

Ospedale Vito Fazzi, ASL Lecce

Lecce, Italy

Location

IEO - Istituto Europeo di Oncologia, IRCCS

Milan, Italy

Location

Ospedale Maggiore Policlinico, Fondazione IRCCS Ca' Granda

Milan, Italy

Location

Ospedale Niguarda, ASST Grande Ospedale Metropolitano Niguarda

Milan, Italy

Location

Ospedale San Gerardo, ASST di Monza

Monza, Italy

Location

Ospedale Civile S.Spirito, PO di Pescara, AUSL Pescara

Pescara, Italy

Location

Ospedale Infermi di Rimini, AUSL Rimini, Distretto di Rimini, Presidio di Rimini, Santarcangelo di Romagna e Novafeltria

Rimini, Italy

Location

Catholic University Of Sacred Heart

Roma, 00168, Italy

Location

PU Campus Bio-Medico di Roma

Roma, Italy

Location

Regina Elena, Istituto Nazionale dei Tumori , IFO, IRCCS

Roma, Italy

Location

Azienda Ospedaliera Santa Maria di Terni

Terni, 05100, Italy

Location

Azienda Ospedaliera Ordine Mauriziano di Torino, Ospedale Umberto I di Torino

Torino, Italy

Location

Ospedale S.Giacomo Apostolo, PO Castelfranco Veneto, AULSS 2 Marca Trevigiana

Treviso, Italy

Location

Azienda Sanitaria Universitaria Giuliano Isontina (ASU GI), Ospedale Maggiore

Trieste, Italy

Location

Centrum Medyczne Pratia Poznan

Skórzewo, Greater Poland Voivodeship, 60-185, Poland

Location

Narodowy Instytut Onkologii im. Marii Skłodowskiej-Curie - Państwowy Instytut Badawczy

Warsaw, Masovian Voivodeship, 02-781, Poland

Location

Pratia Onkologia Katowice

Katowice, Poland

Location

Pratia MCM Krakow

Krakow, 30-727, Poland

Location

MICS Centrum Medyczne Torun

Torun, 87-100, Poland

Location

MTZ Clinical Research powered by Pratia

Warsaw, Poland

Location

Uniwersytecki Szpital Kliniczny im. J. Mikulicza-Radeckiego we Wroclawiu

Wroclaw, 50-367, Poland

Location

National Cancer Center Singapore

Singapore, Singapore

Location

Tan Tock Seng Hospital

Singapore, Singapore

Location

The Catholic University of Korea, Seoul St. Mary's Hospital

Seoul, Seoul Teugbyeolsi [Seoul-T'ukp], 06591, South Korea

Location

Severance Hospital, Yonsei University Health System

Seoul, Seoul Teugbyeolsi [Seoul-T'ukp, 03722, South Korea

Location

Samsung Medical Center

Seoul, Seoul Teugbyeolsi [Seoul-T'ukp, 06351, South Korea

Location

Seoul National University Hospital

Seoul, Seoul Teugbyeolsi, 03080, South Korea

Location

Pusan National University Hospital

Busan, South Korea

Location

Gachon University Gil Medical Center

Incheon, South Korea

Location

Ajou University Hospital

Suwon, South Korea

Location

Hospital Universitari Vall d'Hebrón

Barcelona, Cataluny, 08035, Spain

Location

Hospital Costa del Sol

Marbella, Málaga, 29603, Spain

Location

Hospital Del Mar

Barcelona, 08003, Spain

Location

Hospital Virgen de la Arrixaca

El Palmar, Spain

Location

Hospital Univ. Infanta Leonor

Madrid, 28031, Spain

Location

Hospital Universitario La Paz

Madrid, 28046, Spain

Location

Clínica Universidad de Navarra

Madrid, Spain

Location

C.H. de Navarra

Pamplona, Spain

Location

Hospital Universitario de Salamanca

Salamanca, 37007, Spain

Location

Hospital Universitario Nuestra Señora de Valme

Seville, 41014, Spain

Location

Hospital Universitario Virgen De La Macarena

Seville, Spain

Location

Buddihist Tzu Chi Medical Foundation- Hualien Tzu Chi Hospital

Hualien City, Taiwan

Location

Chang Gung Medical Foundation - Kaohsiung Chang Gung Memorial Hospital - Hemato-Oncology

Kaohsiung City, 833, Taiwan

Location

Taichung Veterans General Hospital

Taichung, 40705, Taiwan

Location

National Cheng Kung University Hospital

Tainan, 704, Taiwan

Location

National Taiwan University Hospital

Taipei, Taiwan

Location

Ankara University Medical Faculty - Hematology

Ankara, Turkey (Türkiye)

Location

Dr Abdurrahman Yurtaslan Ankara Oncology Training and Research

Ankara, Turkey (Türkiye)

Location

Gazi University Medical Faculty

Ankara, Turkey (Türkiye)

Location

Medipol Bagcilar Mega Hospital

Istanbul, Turkey (Türkiye)

Location

Ondokuz Mayis University Medical Faculty - Hematology

Samsun, Turkey (Türkiye)

Location

Western General Hospital - Haematology

Edinburgh, Edinburgh, City of, EH4 2XU, United Kingdom

Location

Imperial College Healthcare NHS Trust - Hammersmith Hospital

London, London City, W12 0HS, United Kingdom

Location

St Bartholomew's Hospital Barts Health NHS Trust

London, London, City of, EC1A 7BE, United Kingdom

Location

The Clatterbridge Cancer Centre NHS Foundation Trust - Clatterbridge Cancer Centre

Bebington, United Kingdom

Location

Royal Cornwall Hospitals NHS Trust - Royal Cornwall Hospital

Cornwell, United Kingdom

Location

Beatson West of Scotland Cancer Centre

Glasgow, G12 0YN, United Kingdom

Location

Northwick Park Hospital Middlesex, United Kindgom, HA1 3UJ

Middlesex, United Kingdom

Location

Related Publications (1)

  • Cao J, Chen G, Qiu L, Zhang L, Jiang M, Cheng Y, Zhang Q, Liu L, Li P, Shuang Y, Wang H, Xue H, Wu H, Zheng M, Zhou K, Li Z, Jing H, Yang W, Zhu Z, Li W, Wangwu J, Huang H, Jia Q, Chen D, Fan S, Shi MM, Su W. Efficacy and safety of tazemetostat, an EZH2 inhibitor, in Chinese patients with relapsed/refractory follicular lymphoma: a multicentre, single-arm, phase 2 study. EClinicalMedicine. 2025 Aug 18;87:103399. doi: 10.1016/j.eclinm.2025.103399. eCollection 2025 Sep.

MeSH Terms

Conditions

Lymphoma, Follicular

Interventions

tazemetostatLenalidomideRituximab

Condition Hierarchy (Ancestors)

Lymphoma, Non-HodgkinLymphomaNeoplasms by Histologic TypeNeoplasmsLymphoproliferative DisordersLymphatic DiseasesHemic and Lymphatic DiseasesImmunoproliferative DisordersImmune System Diseases

Intervention Hierarchy (Ancestors)

PhthalimidesPhthalic AcidsAcids, CarbocyclicCarboxylic AcidsOrganic ChemicalsPiperidonesPiperidinesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsIsoindolesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingAntibodies, Monoclonal, Murine-DerivedAntibodies, MonoclonalAntibodiesImmunoglobulinsImmunoproteinsBlood ProteinsProteinsAmino Acids, Peptides, and ProteinsSerum GlobulinsGlobulins

Study Officials

  • Ipsen Medical Director

    Ipsen

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Model Details: 3 stages study: Stage 1: Open-Label (Phase 1b: Safety run-in): All participants will receive Tazemetostat in combination with Lenalidomide and Rituximab Stage 2: Double-blinded (Phase 3): * Study drug arm: Tazemetostat in combination with Lenalidomide and Rituximab * Placebo arm: Placebo in combination with Lenalidomide and Rituximab Stage 3: Long-term Follow-up of participants in Stage 2 after treatment for response, when applicable, and overall survival for up to 5 years after the enrollment of the last patient in the study.
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

December 12, 2019

First Posted

January 13, 2020

Study Start

June 11, 2020

Primary Completion (Estimated)

February 13, 2027

Study Completion (Estimated)

March 1, 2029

Last Updated

April 20, 2026

Record last verified: 2026-04

Data Sharing

IPD Sharing
Will share

Qualified researchers may request access to patient level data and related study documents including the clinical study report, study protocol with any amendments, annotated case report form, statistical analysis plan, and dataset specifications. Patient level data will be anonymized and study documents will be redacted to protect the privacy of study participants.

Time Frame
Where applicable, data from eligible studies are available 6 months after the studied medicine and indication have been approved in the US and/or EU.
Access Criteria
Further details on Ipsen's sharing criteria and process for sharing are available here (https://www.ipsen.com/science/clinical-trials/clinical-data-transparency/).
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