NCT03954327

Brief Summary

Placebo Controlled, double-blind randomized controlled trial (RCT) with 12 months Tenofovir Disoproxil and Raltegravir for primary biliary cholangitis (PBC) patients unresponsive to Ursodeoxycholic Acid (UDCA). Placebo patients will be offered 12 months open label therapy at unblinding. All patients will be offered an additional 12 months open label therapy. Observational, open label study will be performed in parallel using Emtricitabine (FTC)/Tenofovir Disoproxil (TDF) \& Raltegravir in liver transplant recipients meeting all entry criteria except for use of immunosuppression.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
37

participants targeted

Target at P25-P50 for phase_2

Timeline
Completed

Started Mar 2021

Typical duration for phase_2

Geographic Reach
1 country

6 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

May 7, 2019

Completed
10 days until next milestone

First Posted

Study publicly available on registry

May 17, 2019

Completed
1.8 years until next milestone

Study Start

First participant enrolled

March 1, 2021

Completed
1.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 1, 2022

Completed
1.3 years until next milestone

Study Completion

Last participant's last visit for all outcomes

January 1, 2024

Completed
Last Updated

February 16, 2024

Status Verified

February 1, 2024

Enrollment Period

1.6 years

First QC Date

May 7, 2019

Last Update Submit

February 15, 2024

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change in alkaline phosphatase levels

    Mean changes in alkaline phosphatase levels after 12 months treatment with combination antiretroviral therapy or placebo.

    12 months

Secondary Outcomes (7)

  • Serial changes in alkaline phosphatase

    Evaluation baseline, 3 months, 6 months and end of RCT; then 3 months, 6 monthly to end of open label therapy]

  • Serial changes in ALT

    Evaluation baseline, 3 months, 6 months and end of RCT; then 3 months, 6 monthly to end of open label therapy]

  • Serial changes in bilirubin

    Evaluation baseline, 3 months, 6 months and end of RCT; then 3 months, 6 monthly to end of open label therapy]

  • Achievement of the composite biochemistry endpoint

    6 and 12 months

  • Human Betaretrovirus load in peripheral blood

    Evaluation baseline, 3 months, 6 months and end of RCT; then 3 months, 6 monthly to end of open label therapy

  • +2 more secondary outcomes

Study Arms (2)

Emtricitabine (FTC)/Tenofovir Disoproxil (TDF) & Raltegravir

EXPERIMENTAL

one Emtricitabine 200mg and Tenofovir Disoproxil 300mg tablet two Raltegravir 600mg tablets

Drug: Emtricitabine (FTC)/Tenofovir Disoproxil (TDF)Drug: Raltegravir

Placebo

PLACEBO COMPARATOR

Identical tablets resembling one Emtricitabine 200mg and Tenofovir Disoproxil 300mg tablet two Raltegravir 600mg tablets

Drug: Placebo Oral Capsule [CEBOCAP]

Interventions

Emtricitabine (FTC) 200 mg/Tenofovir Disoproxil (TDF) 300 mg by mouth once per day

Also known as: Truvada
Emtricitabine (FTC)/Tenofovir Disoproxil (TDF) & Raltegravir

Raltegravir (RTF) 600 mg two tablets by mouth once per day

Also known as: Isentress
Emtricitabine (FTC)/Tenofovir Disoproxil (TDF) & Raltegravir

Two capsules identical to Raltegravir and one capsule identical to Truvada with no active ingredients by mouth once per day

Also known as: placebo
Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • over 18 years old of either sex,
  • Anti-mitochondrial antibody +ve or liver histology compatible with PBC,
  • stable UDCA dose of 13-15 mg/kg for \> 12 months or intolerant to UDCA,
  • ALP at least 1.67 x ULN or abnormal bilirubin less than 2x ULN
  • able to read and sign informed consent form.

You may not qualify if:

  • use of non-standard or experimental therapy within the last 6 months,
  • advanced liver disease: INR \> 1.2 ULN, Albumin \< 35 g/L lower limit of normal, platelets \< 120,000/microL unless varices with risk of bleeding excluded by endoscopy within the last 6 months, Childs Pugh class B or C cirrhosis, presence of grade 2 varices or previous variceal hemorrhage, encephalopathy, ascites or need for liver transplantation within the next two years;
  • secondary diagnosis such as HIV, viral hepatitis, drug induced liver injury, extrahepatic biliary obstruction, primary sclerosing cholangitis, metabolic liver - regular use of \> 30g alcohol/day in the last year;
  • a predicted survival of less than 3 years from malignant or other life threatening disease;
  • hepatic mass consistent with hepatocellular carcinoma ;
  • previous allergic reaction to study medications;
  • Glomerular Filtration Rate less than \< 30 mL/min as measured Cockcroft-Gault formula;
  • pregnancy, breast-feeding or pre-menopausal patients not using contraception.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (6)

University of Alberta

Edmonton, Alberta, T6G 2R3, Canada

Location

St Paul's Hospital, University of British Columbia

Vancouver, British Columbia, V6Z 1Y6, Canada

Location

Vancouver General Hospital, University of Brittish Columbia

Vancouver, British Columbia, V6Z 1Z4, Canada

Location

University of Toronto

Toronto, Ontario, M5S 1A1, Canada

Location

University of Montreal

Montreal, Quebec, Canada

Location

Royal University Hospital

Saskatoon, Saskatchewan, S7N 0W8, Canada

Location

MeSH Terms

Conditions

Liver Cirrhosis, Biliary

Interventions

EmtricitabineEmtricitabine, Tenofovir Disoproxil Fumarate Drug CombinationRaltegravir Potassium

Condition Hierarchy (Ancestors)

Cholestasis, IntrahepaticCholestasisBile Duct DiseasesBiliary Tract DiseasesDigestive System DiseasesLiver DiseasesLiver CirrhosisFibrosisPathologic ProcessesPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

DeoxycytidineCytidinePyrimidine NucleosidesPyrimidinesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsDeoxyribonucleosidesNucleosidesNucleic Acids, Nucleotides, and NucleosidesTenofovirOrganophosphonatesOrganophosphorus CompoundsOrganic ChemicalsAdeninePurinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingDrug CombinationsPharmaceutical PreparationsPyrrolidinonesPyrrolidines

Study Officials

  • Andrew Mason, MD

    University of Alberta

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Masking Details
Double-blind
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
OTHER
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 7, 2019

First Posted

May 17, 2019

Study Start

March 1, 2021

Primary Completion

October 1, 2022

Study Completion

January 1, 2024

Last Updated

February 16, 2024

Record last verified: 2024-02

Data Sharing

IPD Sharing
Will not share

Locations