NCT03654274

Brief Summary

The purpose of this study is to evaluate the long-term efficacy and safety of relugolix 40 milligram (mg) once daily co-administered with low-dose estradiol (E2) and norethindrone acetate (NETA) for up to 104 weeks on endometriosis-associated pain in participants who previously completed a 24-week treatment period in one of the parent studies (MVT-601-3101 or MVT-601-3102).

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
802

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started May 2018

Longer than P75 for phase_3

Geographic Reach
20 countries

169 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

May 22, 2018

Completed
3 months until next milestone

First Submitted

Initial submission to the registry

August 29, 2018

Completed
2 days until next milestone

First Posted

Study publicly available on registry

August 31, 2018

Completed
3.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 16, 2021

Completed
1.1 years until next milestone

Study Completion

Last participant's last visit for all outcomes

January 31, 2023

Completed
6 months until next milestone

Results Posted

Study results publicly available

July 20, 2023

Completed
Last Updated

August 8, 2023

Status Verified

August 1, 2023

Enrollment Period

3.6 years

First QC Date

August 29, 2018

Results QC Date

March 3, 2023

Last Update Submit

August 4, 2023

Conditions

Keywords

EndometriosisDysmenorrheaPainDyspareuniaPelvic Pain

Outcome Measures

Primary Outcomes (4)

  • Percentage Of Participants Who Meet The Dysmenorrhea Responder Criteria At Week 52

    Assessed using an NRS score (11-point scale) for pain recorded daily in an electronic diary. A participant was defined as a responder if the NRS score for dysmenorrhea declined from baseline to Week 52 by at least 2.8 points without increased use of protocol-specified analgesics for pelvic pain at Week 52 relative to baseline. Participants rated their pelvic pain on a scale from 0 to 10, with 0 indicating no pain and 10 indicating pain as bad as you can imagine.

    Week 52

  • Percentage Of Participants Who Meet The NMPP Responder Criteria At Week 52

    Assessed using an NRS score (11-point scale) for pain recorded daily in an electronic diary. A participant was defined as a responder if the NRS score for NMPP declined from baseline to Week 52 by at least 2.1 points without increased use of protocol-specified analgesics for pelvic pain at Week 52 relative to baseline. Participants rated their pelvic pain on a scale from 0 to 10, with 0 indicating no pain and 10 indicating pain as bad as you can imagine.

    Week 52

  • Percentage Of Participants Who Meet The Dysmenorrhea Responder Criteria At Week 104

    Assessed using an NRS score (11-point scale) for pain recorded daily in an electronic diary. A participant was defined as a responder if the NRS score for dysmenorrhea declined from baseline to Week 104 by at least 2.8 points without increased use of protocol-specified analgesics for pelvic pain at Week 104 relative to baseline. Participants rated their pelvic pain on a scale from 0 to 10, with 0 indicating no pain and 10 indicating pain as bad as you can imagine.

    Week 104

  • Percentage Of Participants Who Meet The NMPP Responder Criteria At Week 104

    Assessed using an NRS score (11-point scale) for pain recorded daily in an electronic diary. A participant was defined as a responder if the NRS score for NMPP declined from baseline to Week 104 by at least 2.1 points without increased use of protocol-specified analgesics for pelvic pain at Week 104 relative to baseline. Participants rated their pelvic pain on a scale from 0 to 10, with 0 indicating no pain and 10 indicating pain as bad as you can imagine.

    Week 104

Secondary Outcomes (37)

  • Change From The Pivotal Phase 3 Study Baseline In The Endometriosis Health Profile (EHP)-30 Pain Domain Scores At Week 52

    Week 52

  • Change From The Pivotal Phase 3 Study Baseline In The Endometriosis Health Profile (EHP)-30 Pain Domain Scores At Week 104

    Week 104

  • Percentage Of Participants Who Have A Reduction Of At Least 20 Points In The EHP-30 Pain Domain Scores From The Pivotal Phase 3 Study Baseline At Week 52

    Week 52

  • Percentage Of Participants Who Have A Reduction Of At Least 20 Points In The EHP-30 Pain Domain Scores From The Pivotal Phase 3 Study Baseline At Week 104

    Week 104

  • Change From The Pivotal Phase 3 Study Baseline In The Mean Dysmenorrhea NRS Score At Week 52

    Week 52

  • +32 more secondary outcomes

Study Arms (1)

Relugolix plus E2/NETA

EXPERIMENTAL

Relugolix co-administered with E2/NETA for 80 weeks.

Drug: RelugolixDrug: Estradiol/norethindrone acetate

Interventions

Relugolix 40-mg tablet administered orally once daily

Also known as: TAK-385, MVT-601
Relugolix plus E2/NETA

Capsule containing co-formulated tablet of E2 (1.0 mg) and NETA (0.5 mg) administered orally once daily

Also known as: E2/NETA, low-dose hormonal add-back
Relugolix plus E2/NETA

Eligibility Criteria

Age18 Years - 51 Years
Sexfemale
Healthy VolunteersNo
Age GroupsAdult (18-64)

You may qualify if:

  • Completed 24 weeks of study drug treatment and study participation in either parent study, MVT-601-3101 or MVT-601-3102.
  • Is not expected to undergo gynecological surgery or other surgical procedures for treatment of endometriosis (including ablation, shaving, or excision) during the study, including during the Follow-Up Period, and the participant does not desire such treatment during this time frame.
  • Has agreed to continue to use only study-specified analgesic medications during the study and is not known to be intolerant to these.

You may not qualify if:

  • Has had a surgical procedure for treatment for endometriosis at any time during the parent study (MVT-601-3101 or MVT-601-3102).
  • Has any chronic pain or frequently recurring pain condition, other than endometriosis, that is treated with opioids or requires analgesics for ≥ 7 days per month.
  • Has a Z-score \< -2.0 or has a ≥ 7% decrease in bone mineral density from the parent study Baseline at lumbar spine, total hip, or femoral neck based on the parent study Week 24 DXA assessment of bone mineral density.
  • Has any contraindication to treatment with low-dose E2 and NETA, including:
  • Known, suspected, or history of breast cancer;
  • Known or suspected estrogen-dependent neoplasia;
  • Active deep vein thrombosis or pulmonary embolism, or history of these conditions prior to the Week 24/Baseline visit;
  • History of or active arterial thromboembolic disease, including stroke and myocardial infarction;
  • Known anaphylactic reaction or angioedema or hypersensitivity to E2 or NETA;
  • Known protein C, protein S, or antithrombin deficiency, or other known thrombophilia disorders, including Factor V Leiden;
  • Migraine with aura;
  • History of porphyria.
  • Had any of the following clinical laboratory abnormalities at the parent study Week 20 visit or, if available, any subsequent visit in one of the parent studies (MVT-601-3101 or MVT-601-3102):
  • Alanine aminotransferase or aspartate aminotransferase \> 2.0 times the upper limit of normal (ULN); or
  • Bilirubin (total bilirubin) \> 1.5 x ULN (or \> 2.0 x ULN if secondary to Gilbert syndrome or pattern consistent with Gilbert syndrome).

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (169)

Andalusia

Andalusia, Alabama, 36420, United States

Location

Scottsdale

Scottsdale, Arizona, 85251, United States

Location

Tucson

Tucson, Arizona, 85704, United States

Location

Tuscon

Tucson, Arizona, 85712, United States

Location

Canoga Park

Canoga Park, California, 91303, United States

Location

Los Angeles

Los Angeles, California, 70433, United States

Location

San Diego

San Diego, California, 92111, United States

Location

Greenwood Village

Greenwood Village, Colorado, 80111, United States

Location

Washington

Washington D.C., District of Columbia, 20036, United States

Location

Aventura

Aventura, Florida, 33180, United States

Location

Fort Myers

Fort Myers, Florida, 33912, United States

Location

Hialeah

Hialeah, Florida, 33012, United States

Location

Hialeah

Hialeah, Florida, 33016, United States

Location

Margate

Margate, Florida, 33063, United States

Location

Miami

Miami, Florida, 33126, United States

Location

Miami

Miami, Florida, 33155, United States

Location

Sarasota

Sarasota, Florida, 34239, United States

Location

Tampa

Tampa, Florida, 33606, United States

Location

Atlanta

Atlanta, Georgia, 30312, United States

Location

Atlanta

Atlanta, Georgia, 30363, United States

Location

Augusta

Augusta, Georgia, 30909, United States

Location

Norcross

Norcross, Georgia, 30093, United States

Location

Idaho Falls

Idaho Falls, Idaho, 83404, United States

Location

Oakbrook

Oakbrook Terrace, Illinois, 60523, United States

Location

Park Ridge

Park Ridge, Illinois, 60068, United States

Location

Shawnee

Shawnee Mission, Kansas, 66218, United States

Location

Marrero

Marrero, Louisiana, 70072, United States

Location

Towson

Towson, Maryland, 21204, United States

Location

Saginaw

Saginaw, Michigan, 48602, United States

Location

Jefferson City

Jefferson City, Missouri, 65109, United States

Location

St. Louis

St Louis, Missouri, 63141, United States

Location

Omaha

Omaha, Nebraska, 68130, United States

Location

Las Vegas

Las Vegas, Nevada, 89113, United States

Location

Durham

Durham, North Carolina, 27713, United States

Location

New Bern

New Bern, North Carolina, 28562, United States

Location

Winston Salem

Winston-Salem, North Carolina, 27103, United States

Location

Akron

Akron, Ohio, 44313, United States

Location

Columbus

Columbus, Ohio, 43235, United States

Location

Englewood

Englewood, Ohio, 45322, United States

Location

Hershey

Hershey, Pennsylvania, 17033-0850, United States

Location

Columbia

Columbia, South Carolina, 29201, United States

Location

Chattanooga

Chattanooga, Tennessee, 37404, United States

Location

Memphis

Memphis, Tennessee, 38120, United States

Location

Beaumont

Beaumont, Texas, 77702, United States

Location

Corpus Christi

Corpus Christi, Texas, 78412, United States

Location

Dallas

Dallas, Texas, 75231, United States

Location

Fort Worth

Fort Worth, Texas, 76104, United States

Location

Houston

Houston, Texas, 77030, United States

Location

Houston

Houston, Texas, 77054, United States

Location

Irving

Irving, Texas, 75062, United States

Location

San Antonio

San Antonio, Texas, 78258, United States

Location

Sugar Land

Sugar Land, Texas, 77479, United States

Location

Webster

Webster, Texas, 77598, United States

Location

Salt Lake City

Salt Lake City, Utah, 84102, United States

Location

Salt Lake City

Salt Lake City, Utah, 84107, United States

Location

Salt Lake City

Salt Lake City, Utah, 84124, United States

Location

Norfolk

Norfolk, Virginia, 23507, United States

Location

Richmond

Richmond, Virginia, 23235, United States

Location

Virginia Beach

Virginia Beach, Virginia, 23502, United States

Location

Seattle

Seattle, Washington, 98105, United States

Location

Ciudad de Buenos Aires

Ciudad de Buenos Aires, Buenos Aires, C1128AAF, Argentina

Location

San Isidro

San Isidro, Buenos Aires, B1642CKL, Argentina

Location

Rosario

Rosario, Santa Fe Province, S2000PRB, Argentina

Location

Cordoba

Córdoba, X5000JHQ, Argentina

Location

Sydney

Sydney, New South Wales, 2000, Australia

Location

Wollongong

Wollongong, NS, 2522, Australia

Location

Taringa

Taringa, Queensland, 4068, Australia

Location

Adelaide

Adelaide, South Australia, 5000, Australia

Location

Nedlands

Nedlands, Western Australia, 6009, Australia

Location

Leuven

Leuven, Flemish Brabant, 3000, Belgium

Location

La Louvière

La Louvière, Hainaut, 7100, Belgium

Location

Gent

Ghent, Oost-vlaanderen, 9000, Belgium

Location

Brussels

Brussels, 1070, Belgium

Location

Passo Fundo

Passo Fundo, Rio Grande do Sul, 99010-080, Brazil

Location

Porto Alegre

Porto Alegre, Rio Grande do Sul, 90430-001, Brazil

Location

Porto Alegre

Porto Alegre, Rio Grande do Sul, 90510-040, Brazil

Location

Porto Alegre

Porto Alegre, Rio Grande do Sul, 90610-000, Brazil

Location

Porto Alegre

Porto Alegre, São Paulo, 90035-903, Brazil

Location

São Bernardo do Campo

São Bernardo do Campo, São Paulo, 09715-090, Brazil

Location

São Paulo

São Paulo, São Paulo, 04023-062, Brazil

Location

Sao Paulo

São Paulo, São Paulo, 04266-010, Brazil

Location

São Paulo

São Paulo, São Paulo, 04708-001, Brazil

Location

Sao Paulo

São Paulo, 01317-000, Brazil

Location

Sofia

Sofia, Sofia, 1233, Bulgaria

Location

Sofia

Sofia, Sofia, 1336, Bulgaria

Location

Sofia

Sofia, Sofia, 1431, Bulgaria

Location

Sofia

Sofia, Sofia, 1504, Bulgaria

Location

Blagoevgrad

Blagoevgrad, 2700, Bulgaria

Location

Pleven

Pleven, 5809, Bulgaria

Location

Stara Zagora

Stara Zagora, 6003, Bulgaria

Location

Varna

Varna, 9002, Bulgaria

Location

Red Deer

Red Deer, Alberta, T4N 6V7, Canada

Location

Waterloo

Waterloo, Ontario, N2J1C4, Canada

Location

Victoriaville

Victoriaville, Quebec, G6P 6P6, Canada

Location

Santiago

Santiago, 7510186, Chile

Location

Santiago

Santiago, 8320143, Chile

Location

Santiago

Santiago, 8880465, Chile

Location

Tábor

Tábor, Jihormoravsky Kraj, 390 03, Czechia

Location

Písek

Písek, Jihočeský kraj, 397 01, Czechia

Location

Vodňany

Vodňany, Jihočeský kraj, 389 01, Czechia

Location

Náchod

Náchod, Královéhradecký kraj, 547 01, Czechia

Location

Praha 10

Prague, Prague, 100 34, Czechia

Location

Praha 2

Prague, Prague, 128 08, Czechia

Location

České Budějovice

České Budějovice, 370 01, Czechia

Location

Olomouc

Olomouc, 772 00, Czechia

Location

Praha 8 - Libeň

Praha 8 - Libeň, 180 81, Czechia

Location

Kuopio

Kuopio, Eastern Finland, 70100, Finland

Location

Helsinki

Helsinki, Southern Finland, 00260, Finland

Location

Oulu

Oulu, 90100, Finland

Location

Tbilisi

Tbilisi, 0159, Georgia

Location

Pécs

Pécs, Baranya, 7624, Hungary

Location

Békéscsaba

Békéscsaba, Bekes County, 5600, Hungary

Location

Gyula

Gyula, Bekes County, 5700, Hungary

Location

Kecskemét

Kecskemét, Bács-Kiskun county, 6000, Hungary

Location

Szeged

Szeged, Csongrád megye, 6725, Hungary

Location

Debrecen

Debrecen, Hajdú-Bihar, 4024, Hungary

Location

Debrecen

Debrecen, Hajdú-Bihar, 4025, Hungary

Location

Debrecen

Debrecen, Hajdú-Bihar, 4032, Hungary

Location

Nyíregyháza

Nyíregyháza, Szabolcs-Szatmár-Bereg, 4400, Hungary

Location

Monserrato

Monserrato, Cagliari, 9042, Italy

Location

Catanzaro

Catanzaro, 88100, Italy

Location

Napoli

Napoli, 80131, Italy

Location

Pavia

Pavia, 27100, Italy

Location

Roma

Roma, 00168, Italy

Location

Remuera

Remuera, Auckland, 1050, New Zealand

Location

Palmerston North

Palmerston North, Manawatu-Wanganui, 4442, New Zealand

Location

Christchurch

Christchurch, 8013, New Zealand

Location

Skórzewo

Skórzewo, Greater Poland Voivodeship, 60-185, Poland

Location

Lublin

Lublin, Lublin Voivodeship, 20-064, Poland

Location

Lublin

Lublin, Lublin Voivodeship, 20-093, Poland

Location

Lublin

Lublin, Lublin Voivodeship, 20-632, Poland

Location

Lublin

Lublin, Lublin Voivodeship, 20-880, Poland

Location

Warszawa

Warsaw, Masovian Voivodeship, 02-066, Poland

Location

Warszawa

Warsaw, Masovian Voivodeship, 02-201, Poland

Location

Warszawa

Warsaw, Masovian Voivodeship, 02-929, Poland

Location

Białystok

Bialystok, Podlaskie Voivodeship, 15-224, Poland

Location

Katowice

Katowice, Silesian Voivodeship, 40-081, Poland

Location

Katowice

Katowice, Silesian Voivodeship, 40-301, Poland

Location

Szczecin

Szczecin, West Pomeranian Voivodeship, 71-434, Poland

Location

Łódź

Lodz, Łódź Voivodeship, 90-602, Poland

Location

Almada

Almada, Lisbon District, 2805-267, Portugal

Location

Coimbra

Coimbra, 3000-075, Portugal

Location

Covilhã

Covilha, 6200-251, Portugal

Location

Porto

Porto, 4099-001, Portugal

Location

Brasov

Brasov, 500091, Romania

Location

Bucuresti

Bucharest, 012071, Romania

Location

Bucuresti

Bucharest, 022441, Romania

Location

Bucuresti

Bucharest, 024091, Romania

Location

București

Bucharest, 20475, Romania

Location

Port Elizabeth

Port Elizabeth, Eastern Cape, 6001, South Africa

Location

Centurion

Centurion, Gauteng, 0157, South Africa

Location

Roodepoort

Roodepoort, Gauteng, 1724, South Africa

Location

Durban

Durban, KwaZulu-Natal, 4126, South Africa

Location

Cape Town

Cape Town, Western Cape, 7405, South Africa

Location

Madrid

Madrid, 28041, Spain

Location

Valencia

Valencia, 46010, Spain

Location

Kyiv

Kyiv, Kiev City, 2232, Ukraine

Location

Kyiv

Kyiv, Kiev City, 4050, Ukraine

Location

Kyiv

Kyiv, Kyiv City, 1034, Ukraine

Location

Chernivtsi

Chernivtsi, 58001, Ukraine

Location

Ivano-Frankivsk

Ivano-Frankivsk, 76018, Ukraine

Location

Kharkiv

Kharkiv, 61052, Ukraine

Location

Kiev

Kiev, 3148, Ukraine

Location

Kiev

Kiev, 4112, Ukraine

Location

Kyiv

Kyiv, 04053, Ukraine

Location

Zaporizhzhya

Zaporizhzhya, 69063, Ukraine

Location

Zaporizhzhya

Zaporizhzhya, 69065, Ukraine

Location

Zaporizhzhya

Zaporizhzhya, 69068, Ukraine

Location

Zaporizhzhya

Zaporizhzhya, 69071, Ukraine

Location

Related Publications (2)

  • As-Sanie S, Abrao MS, Reznichenko G, Wilk K, Zhong Y, Perry J, Hunsche E, Soulban G, Becker CM. Impact of relugolix combination therapy on functioning and quality of life in women with endometriosis-associated pain. Fertil Steril. 2024 Oct;122(4):687-695. doi: 10.1016/j.fertnstert.2024.06.009. Epub 2024 Jun 19.

  • Becker CM, Johnson NP, As-Sanie S, Arjona Ferreira JC, Abrao MS, Wilk K, Imm SJ, Mathur V, Perry JS, Wagman RB, Giudice LC. Two-year efficacy and safety of relugolix combination therapy in women with endometriosis-associated pain: SPIRIT open-label extension study. Hum Reprod. 2024 Mar 1;39(3):526-537. doi: 10.1093/humrep/dead263.

MeSH Terms

Conditions

EndometriosisDysmenorrheaPainDyspareuniaPelvic Pain

Interventions

relugolixestradiol, norethindrone drug combination

Condition Hierarchy (Ancestors)

Genital Diseases, FemaleFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesGenital DiseasesMenstruation DisturbancesPathologic ProcessesPathological Conditions, Signs and SymptomsNeurologic ManifestationsSigns and SymptomsGenital Diseases, MaleSexual Dysfunction, PhysiologicalMale Urogenital DiseasesSexual Dysfunctions, PsychologicalMental Disorders

Results Point of Contact

Title
Clinical Trials at Myovant
Organization
Myovant Sciences GmbH

Study Officials

  • Myovant Medical Monitor

    Myovant Sciences

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Model Details: Open label extension
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

August 29, 2018

First Posted

August 31, 2018

Study Start

May 22, 2018

Primary Completion

December 16, 2021

Study Completion

January 31, 2023

Last Updated

August 8, 2023

Results First Posted

July 20, 2023

Record last verified: 2023-08

Data Sharing

IPD Sharing
Will not share

Locations