NCT02920450

Brief Summary

The purpose of this research study is to determine if the study drug, Gedatolisib (PF-05212384), given in combination with paclitaxel and carboplatin will work against unresectable non-small cell lung cancer.

Trial Health

57
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
3

participants targeted

Target at below P25 for phase_1 nonsmall-cell-lung-cancer

Timeline
Completed

Started Sep 2017

Shorter than P25 for phase_1 nonsmall-cell-lung-cancer

Geographic Reach
1 country

1 active site

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 27, 2016

Completed
3 days until next milestone

First Posted

Study publicly available on registry

September 30, 2016

Completed
12 months until next milestone

Study Start

First participant enrolled

September 25, 2017

Completed
1.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 2, 2019

Completed
3 months until next milestone

Study Completion

Last participant's last visit for all outcomes

April 4, 2019

Completed
6 months until next milestone

Results Posted

Study results publicly available

October 3, 2019

Completed
Last Updated

October 4, 2019

Status Verified

October 1, 2019

Enrollment Period

1.3 years

First QC Date

September 27, 2016

Results QC Date

July 16, 2019

Last Update Submit

October 2, 2019

Conditions

Keywords

lungcarcinoma

Outcome Measures

Primary Outcomes (2)

  • Dose Tolerability

    To identify the maximum tolerated dose of PF-05212384 in combination with paclitaxel and carboplatin in subjects with NSCLC.

    1 year

  • Objective Response Rate (ORR)

    To estimate the objective rate of response of PF-05212384 in combination with paclitaxel and carboplatin administered to subjects with unresectable or metastatic NSCLC, according to current RECIST criteria. ORR is defined as the number of participants who achieved either a partial or complete response by RECIST 1.1 criteria. By these criteria, Complete Response (CR) is defined as the disappearance of all target lesions and Partial Response (PR) is defined as a decrease of at least 30% in the sum of the longest diameter of the target lesions.

    1 year

Study Arms (4)

Treatment Arm (Phase 1b; Gedatolisib Dose Level 1[110 mg])

EXPERIMENTAL
Drug: GedatolisibDrug: PaclitaxelDrug: Carboplatin

Treatment Arm (Phase 1b; Gedatolisib Dose Level 2[150 mg])

EXPERIMENTAL
Drug: GedatolisibDrug: PaclitaxelDrug: Carboplatin

Treatment Arm (Phase 1b; Gedatolisib Dose Level 3[180 mg])

EXPERIMENTAL
Drug: GedatolisibDrug: PaclitaxelDrug: Carboplatin

Treatment Arm (Phase 2; MTD of Gedatolisib from Phase Ib)

EXPERIMENTAL
Drug: GedatolisibDrug: PaclitaxelDrug: Carboplatin

Interventions

During the first phase, subjects will be sequentially enrolled to each increasing dose level, beginning with dose level 1 (110 mg) until the first dose limiting toxicity occurs, or safely accrued to dose level 3. PF-05212384 is intravenously infused over a thirty minute period. The dose given in the phase 2 portion will be the MTD determined in the phase Ib portion of the study. Dose Level 1: 110 mg Dose Level 2: 150 mg Dose Level 3: 180 mg

Also known as: PF-05212384
Treatment Arm (Phase 1b; Gedatolisib Dose Level 1[110 mg])Treatment Arm (Phase 1b; Gedatolisib Dose Level 2[150 mg])Treatment Arm (Phase 1b; Gedatolisib Dose Level 3[180 mg])Treatment Arm (Phase 2; MTD of Gedatolisib from Phase Ib)

Given as 200 mg/m2 infusion over a three hour period at every twenty-one days; the dose will not adjust as part of the study design.

Also known as: Taxol®, NSC-673089
Treatment Arm (Phase 1b; Gedatolisib Dose Level 1[110 mg])Treatment Arm (Phase 1b; Gedatolisib Dose Level 2[150 mg])Treatment Arm (Phase 1b; Gedatolisib Dose Level 3[180 mg])Treatment Arm (Phase 2; MTD of Gedatolisib from Phase Ib)

The carboplatin dose (mg) = AUC x (CrCl + 25) where AUC = 6 depending on the dose level. carboplatin is intravenously infused over a thirty minute period following paclitaxel administration; the dose will not adjust as part of the study design.

Also known as: CBDCA, NSC-241240
Treatment Arm (Phase 1b; Gedatolisib Dose Level 1[110 mg])Treatment Arm (Phase 1b; Gedatolisib Dose Level 2[150 mg])Treatment Arm (Phase 1b; Gedatolisib Dose Level 3[180 mg])Treatment Arm (Phase 2; MTD of Gedatolisib from Phase Ib)

Eligibility Criteria

Age18 Years - 90 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Signed Institutional Review Board (IRB)-approved informed consent prior to any study-related procedures
  • Age of 18 years or older
  • Advanced-stage unresectable NSCLC, as confirmed by pathological and/or radiological analysis (subjects will be classified as having advanced disease if they were not eligible for, or had disease progression after, surgical or locoregional therapies)
  • Prior chemotherapy will be allowed for other invasive malignancies, provided therapy was completed at least five years before the start of protocol therapy, and participants have recovered from all toxicities of that prior therapy
  • Participants may have received prior chemotherapy for NSCLC
  • In the Phase II portion, subjects must have disease which lacks PTEN expression by immunohistochemistry, or has known prior activating PI3K or inactivating PTEN gene mutations (mutations will not be assayed for specifically)
  • Eastern Cooperative Oncology Group (ECOG) performance status score \< 2
  • Life expectancy ≥ 12 week
  • Participants must have measureable disease by RECIST criteria
  • Absolute neutrophil count \> 1500 mm3 (individuals with benign ethnic neutropenia may be enrolled if they have no evidence of infectious diathesis, or febrile neutropenia at the time of enrollment)
  • Platelet count ≥ 100×109 L
  • Hgb ≥ 8.5 g/dL (subjects may receive transfusions to achieve this, in the absence of overt bleeding)
  • Total Bilirubin ≤ 2 mg/dL
  • aspartate aminotransferase/alanine aminotransferase (AST/ALT) ≤ 3 times the upper limit of normal range
  • Serum creatinine ≤1.5 times the upper limit of the normal range
  • +4 more criteria

You may not qualify if:

  • Uncontrolled cardiac disease, congestive heart failure, angina, arrhythmias or hypertension.
  • Myocardial infarction or unstable angina within 2 months of treatment.
  • Known human immunodeficiency virus (HIV) infection or chronic active Hepatitis B (subjects will not be screened for this).
  • Active clinically serious infection \> CTCAE Grade 2.
  • Thrombotic or embolic events such as a cerebrovascular accident including transient ischemic attacks within the past 6 months.
  • Pulmonary hemorrhage/bleeding event ≥ CTCAE Grade 2 within 4 weeks of first dose of study drug.
  • Any other hemorrhage/bleeding event ≥ CTCAE Grade 3 within 4 weeks of first dose of study drug.
  • Serious non-healing wound, ulcer, or bone fracture.
  • Evidence or history of bleeding diathesis or coagulopathy
  • Major surgery, open biopsy or significant traumatic injury within 4 weeks of first study drug
  • Women or men of childbearing potential who are unwilling or unable to use an acceptable method to avoid pregnancy for the entire study period and for at least 6 months after the last dose of study drug
  • Women who are pregnant or breastfeeding.
  • History of any other disease, metabolic dysfunction, physical examination finding, or clinical laboratory finding giving reasonable suspicion of a disease or condition that contraindicates the use of protocol therapy or that might affect the interpretation of the results of the study or that puts the subject at high risk for treatment complications, in the opinion of the treating physician.
  • Prisoners or subjects who are involuntarily incarcerated.
  • Subjects who are compulsorily detained for treatment of either a psychiatric or physical illness.
  • +1 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

UF Health Cancer Center

Gainesville, Florida, 32608, United States

Location

MeSH Terms

Conditions

Carcinoma, Non-Small-Cell LungCarcinoma

Interventions

gedatolisibPaclitaxelCarboplatin

Condition Hierarchy (Ancestors)

Carcinoma, BronchogenicBronchial NeoplasmsLung NeoplasmsRespiratory Tract NeoplasmsThoracic NeoplasmsNeoplasms by SiteNeoplasmsLung DiseasesRespiratory Tract DiseasesNeoplasms, Glandular and EpithelialNeoplasms by Histologic Type

Intervention Hierarchy (Ancestors)

TaxoidsCyclodecanesCycloparaffinsHydrocarbons, AlicyclicHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsDiterpenesTerpenesCoordination Complexes

Results Point of Contact

Title
Protocol Development Manager
Organization
University of Florida Heath Cancer Center

Study Officials

  • Dennie Jones, MD

    University of Florida

    PRINCIPAL INVESTIGATOR

Publication Agreements

PI is Sponsor Employee
No
Restrictive Agreement
No

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
OTHER
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 27, 2016

First Posted

September 30, 2016

Study Start

September 25, 2017

Primary Completion

January 2, 2019

Study Completion

April 4, 2019

Last Updated

October 4, 2019

Results First Posted

October 3, 2019

Record last verified: 2019-10

Data Sharing

IPD Sharing
Will not share

Locations