NCT01780506

Brief Summary

The primary objective of this study is to evaluate the efficacy of elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide (E/C/F/TAF) fixed-dose combination (FDC) versus elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate (E/C/F/TDF) FDC in HIV-1 positive, antiretroviral treatment-naive adults.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
872

participants targeted

Target at P75+ for phase_3 hiv

Timeline
Completed

Started Dec 2012

Longer than P75 for phase_3 hiv

Geographic Reach
11 countries

112 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

December 26, 2012

Completed
21 days until next milestone

First Submitted

Initial submission to the registry

January 16, 2013

Completed
15 days until next milestone

First Posted

Study publicly available on registry

January 31, 2013

Completed
1.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 26, 2014

Completed
1.4 years until next milestone

Results Posted

Study results publicly available

January 8, 2016

Completed
1.7 years until next milestone

Study Completion

Last participant's last visit for all outcomes

September 6, 2017

Completed
Last Updated

November 19, 2018

Status Verified

August 1, 2018

Enrollment Period

1.7 years

First QC Date

January 16, 2013

Results QC Date

December 4, 2015

Last Update Submit

October 19, 2018

Conditions

Keywords

HIVTreatment NaiveHIV 1 InfectedFemaleWomen

Outcome Measures

Primary Outcomes (1)

  • Percentage of Participants With HIV-1 RNA < 50 Copies/mL at Week 48

    The percentage of participants achieving HIV-1 RNA \< 50 copies/mL at Week 48 was analyzed using the snapshot algorithm, which defines a patient's virologic response status using only the viral load at the predefined time point within an allowed window of time, along with study drug discontinuation status.

    Week 48

Secondary Outcomes (23)

  • Percentage of Participants With HIV-1 RNA < 50 Copies/mL at Weeks 96 and 144

    Weeks 96 and 144

  • Percentage of Participants With HIV-1 RNA < 20 Copies/mL at Weeks 48, 96, and 144

    Weeks 48, 96. and 144

  • Change From Baseline in CD4+ Cell Count at Week 48

    Baseline; Week 48

  • Change From Baseline in CD4+ Cell Count at Week 96

    Baseline; Week 96

  • Change From Baseline in CD4+ Cell Count at Week 144

    Baseline; Week 144

  • +18 more secondary outcomes

Study Arms (3)

E/C/F/TAF (Double-Blind Phase)

EXPERIMENTAL

E/C/F/TAF plus E/C/F/TDF placebo for 144 weeks

Drug: E/C/F/TAFDrug: E/C/F/TDF Placebo

E/C/F/TDF (Double-Blind Phase)

ACTIVE COMPARATOR

E/C/F/TDF plus E/C/F/TAF placebo for 144 weeks

Drug: E/C/F/TDFDrug: E/C/F/TAF Placebo

Open-Label Extension Phase

EXPERIMENTAL

After study unblinding, participants who complete 144 weeks of the study had the option to receive open-label E/C/F/TAF until commercially available, or until Gilead Sciences terminated the study in that country.

Drug: E/C/F/TAF

Interventions

150/150/200/10 mg FDC tablet administered orally once daily

Also known as: Genvoya®
E/C/F/TAF (Double-Blind Phase)Open-Label Extension Phase

150/150/200/300 mg FDC tablet administered orally once daily

Also known as: Stribild®
E/C/F/TDF (Double-Blind Phase)

Tablet administered orally once daily

E/C/F/TAF (Double-Blind Phase)

Tablet administered orally once daily

E/C/F/TDF (Double-Blind Phase)

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Ability to understand and sign a written informed consent form, which must be obtained prior to initiation of study procedures
  • Plasma HIV-1 RNA levels ≥ 1,000 copies/mL at screening
  • No prior use of any approved or investigational antiretroviral drug for any length of time, except the use for pre-exposure prophylaxis (PREP) or post-exposure prophylaxis (PEP), up to 6 months prior to screening
  • Screening genotype report must show sensitivity to elvitegravir, emtricitabine, tenofovir disoproxil fumarate (tenofovir DF)
  • Normal electrocardiogram (ECG)
  • Estimated glomerular filtration rate (eGFR) ≥ 50 mL/min according to the Cockcroft-Gault formula for creatinine clearance
  • Hepatic transaminases (AST and ALT) ≤ 5 × upper limit of normal (ULN)
  • Total bilirubin ≤ 1.5 mg/dL, or normal direct bilirubin
  • Adequate hematologic function
  • Serum amylase ≤ 5 × ULN
  • Males and females of childbearing potential must agree to utilize highly effective contraception methods or be non-heterosexually active or practice sexual abstinence from screening throughout the duration of study treatment and for 30 days following the last dose of study drug
  • Females who utilize hormonal contraceptive as one of their birth control methods must have used the same method for at least three months prior to study dosing
  • Females who have stopped menstruating for ≥ 12 months but do not have documentation of ovarian hormonal failure must have a serum follicle stimulating hormone (FSH) level at screening within the post-menopausal range based on the Central Laboratory reference range

You may not qualify if:

  • A new acquired immunodeficiency syndrome (AIDS) defining condition diagnosed within the 30 days prior to screening
  • Hepatitis B surface antigen (HBsAg) positive
  • Hepatitis C antibody positive
  • Individuals experiencing decompensated cirrhosis
  • Females who are breastfeeding
  • Positive serum pregnancy test
  • Have an implanted defibrillator or pacemaker
  • Current alcohol or substance use judged by the Investigator to potentially interfere with study compliance
  • History of malignancy within the past 5 years or ongoing malignancy other than cutaneous Kaposi's sarcoma, basal cell carcinoma, or resected, noninvasive cutaneous squamous carcinoma
  • Active, serious infections (other than HIV-1 infection) requiring parenteral antibiotic or antifungal therapy within 30 days prior to baseline
  • Any other clinical condition or prior therapy that, in the opinion of the Investigator, would make the individual unsuitable for the study or unable to comply with dosing requirements
  • Participation in any other clinical trial (including observational trials) without prior approval
  • Individuals receiving ongoing therapy with drugs not to be used with elvitegravir, cobicistat, emtricitabine, tenofovir DF, and TAF or individuals with any known allergies to the excipients of E/C/F/TDF or E/C/F/TAF single-tablet regimen tablets

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (117)

The University of Alabama at Birmingham

Birmingham, Alabama, 35294, United States

Location

Spectrum Medical Group

Phoenix, Arizona, 85012, United States

Location

Kaiser Permanente Los Angeles

Los Angeles, California, 90027, United States

Location

University of California, Los Angeles

Los Angeles, California, 90035, United States

Location

Peter J. Ruane, MD, Inc.

Los Angeles, California, 90036, United States

Location

Anthony Mills MD Inc

Los Angeles, California, 90069, United States

Location

East Bay AIDS Center

Oakland, California, 94609, United States

Location

Kaiser Permanente - Sacramento

Sacramento, California, 95825, United States

Location

La Playa Medical Group and Clinical Research

San Diego, California, 92103, United States

Location

University of California, San Diego

San Diego, California, 92103, United States

Location

Los Angeles Biomedical Research Institute at Harbor-UCLA Medical Center

Torrance, California, 90502, United States

Location

Apex Research, LLC

Denver, Colorado, 80209, United States

Location

Yale University School of Medicine

New Haven, Connecticut, 06510, United States

Location

Dupont Circle Physicians Group, P.C.

Washington D.C., District of Columbia, 20009, United States

Location

Whitman Walker Clinic

Washington D.C., District of Columbia, 20009, United States

Location

Capital Medical Associates, P.C.

Washington D.C., District of Columbia, 20036, United States

Location

Gary Richmond, MD, PA, Inc.

Fort Lauderdale, Florida, 33316, United States

Location

Midway Immunology & Research Center, LLC

Ft. Pierce, Florida, 34982, United States

Location

The Kinder Medical Group

Miami, Florida, 33133, United States

Location

AIDS Healthcare Foundation

Miami Beach, Florida, 33139, United States

Location

Orlando Immunology Center

Orlando, Florida, 32803, United States

Location

IDOCF/ValuHealthMD, LLC

Orlando, Florida, 32806, United States

Location

Infectious Diseases Associates

Pensacola, Florida, 32504, United States

Location

The University of South Florida

Tampa, Florida, 33602, United States

Location

Infectious Disease Research Institute Inc.

Tampa, Florida, 33614, United States

Location

St. Joseph's Comprenhensive Research Inisitute

Tampa, Florida, 33614, United States

Location

AIDS Research and Treatment Center of the Treasure Coast

Vero Beach, Florida, 32960, United States

Location

AIDS Research Consortium of Atlanta

Atlanta, Georgia, 30308, United States

Location

Emory University

Atlanta, Georgia, 30308, United States

Location

Atlanta ID Group, PC

Atlanta, Georgia, 30309, United States

Location

Infectious Disease Specialist of Atlanta

Decatur, Georgia, 30033, United States

Location

Mercer University School of Medicine

Macon, Georgia, 31201, United States

Location

University of Hawaii - Hawaii Center for AIDS

Honolulu, Hawaii, 96816, United States

Location

Northwestern University

Chicago, Illinois, 60611, United States

Location

Ruth M. Rothstein CORE Center

Chicago, Illinois, 60612, United States

Location

Howard Brown Health Center

Chicago, Illinois, 60613, United States

Location

Institute of Human Virology, University of Maryland

Baltimore, Maryland, 21201, United States

Location

Community Research Initative

Boston, Massachusetts, 02111, United States

Location

Brigham & Women's Hospital

Boston, Massachusetts, 02115, United States

Location

Metrowest Medical Center

Framingham, Massachusetts, 01702, United States

Location

Baystate Infectious Diseases Clinical Research

Springfield, Massachusetts, 01199, United States

Location

Be Well Medical Center

Berkley, Michigan, 48072, United States

Location

Henry Ford Hospital

Detroit, Michigan, 48202, United States

Location

Hennepin County Medical Center

Minneapolis, Minnesota, 55415, United States

Location

Central West Clinical Research, Inc.

St Louis, Missouri, 63108, United States

Location

Southampton Healthcare, Inc.

St Louis, Missouri, 63139, United States

Location

ID Care

Hillsborough, New Jersey, 08844, United States

Location

Saint Michael's Medical Center

Newark, New Jersey, 07102, United States

Location

Southwest C.A.R.E. Center

Santa Fe, New Mexico, 87505, United States

Location

Albany Medical College

Albany, New York, 12208, United States

Location

Upstate Infectious Diseases Associates

Albany, New York, 12208, United States

Location

New York Hospital Queens

Flushing, New York, 11355, United States

Location

North Shore University Hospital - Division of Infectious Diseases

Manhasset, New York, 11030, United States

Location

Mount Sinai School of Medicine

New York, New York, 10029, United States

Location

Jacobi Medical Center

The Bronx, New York, 10461, United States

Location

Montefiore Medical Center

The Bronx, New York, 10467, United States

Location

University of North Carolina

Chapel Hill, North Carolina, 27514, United States

Location

Infectious Disease Consultants, PA

Charlotte, North Carolina, 28209, United States

Location

Duke University

Durham, North Carolina, 22710, United States

Location

Rosedale Infectious Diseases

Huntersville, North Carolina, 28078, United States

Location

Summa Health Care Center

Akron, Ohio, 44304, United States

Location

University of Pennsylvania

Philadelphia, Pennsylvania, 19104, United States

Location

Thomas Jefferson University

Philadelphia, Pennsylvania, 19107, United States

Location

The Miriam Hospital

Providence, Rhode Island, 02906, United States

Location

Medical University of South Carolina

Charleston, South Carolina, 29425, United States

Location

University of South Carolina School of Medicine

Columbia, South Carolina, 29203, United States

Location

Central Texas Clinical Research

Austin, Texas, 78705, United States

Location

St. Hope Foundation, Inc.

Bellaire, Texas, 77401, United States

Location

Trinity Health and Wellness Center/AIDS Arms, Inc.

Dallas, Texas, 75208, United States

Location

North Texas Infectious Diseases Consultants

Dallas, Texas, 75246, United States

Location

Tarrant County Infectious Disease Associates

Fort Worth, Texas, 76104, United States

Location

Garcias' Family Health Group

Harlingen, Texas, 78550, United States

Location

Therapeutic Concepts, PA

Houston, Texas, 77004, United States

Location

Gordon E. Crofoot, MD, PA

Houston, Texas, 77098, United States

Location

DCOL Center for Clinical Research

Longview, Texas, 75605, United States

Location

Clinical Alliance for Research & Education - Infectious Diseases, LLC (CARE-ID)

Annandale, Virginia, 22003, United States

Location

Peter Shalit, MD

Seattle, Washington, 98104, United States

Location

Medical College of Wisconsin

Milwaukee, Wisconsin, 53226, United States

Location

Holdsworth House Medical Practice

Darlinghurst, New South Wales, 2010, Australia

Location

Taylor Square Private Clinic

Darlington, New South Wales, 2010, Australia

Location

East Sydney Doctors

Sydney, New South Wales, 2010 NSW, Australia

Location

Albion Street Centre

Sydney, Southwest, 2010, Australia

Location

Melbourne Sexual Health Clinic

Carlton, Victoria, 3053, Australia

Location

DIAID, Department of Dermatology, Medical University Vienna

Vienna, 1090, Austria

Location

Otto-Wagner-Spital, Sozialmedizinisches Zentrum Baumgartner Hoehe

Vienna, 1140, Austria

Location

Hôpital Erasme-ULB

Anderlecht, Brussels Capital, 1070, Belgium

Location

CHU Saint-Pierre University Hospital

Brussels, 1000, Belgium

Location

Spectrum Health

Vancouver, British Columbia, V6Z 2T1, Canada

Location

Health Sciences Centre Winnipeg

Winnipeg, Manitoba, R3A 1R9, Canada

Location

The Ottawa Hospital

Ottawa, Ontario, K1H 8L6, Canada

Location

Maple Leaf Research

Toronto, Ontario, M5G 1K2, Canada

Location

Clinique Medicale Du Quartier Latin

Montreal, Quebec, H2L 5B1, Canada

Location

Clinique medicale l'Actuel

Montreal, Quebec, H2L 5B1, Canada

Location

Clinique OPUS

Montreal, Quebec, H3A 1T1, Canada

Location

Sunnybrook Health Science Center

Toronto, M4N 3M5, Canada

Location

Ospedale San Raffaele

Milan, 20127, Italy

Location

National Center for Global Health and Medicine AIDS Clinical Center

Shinjuku-ku, Tokyo, 162-8655, Japan

Location

HOPE Clinical Research

San Juan, 00909, Puerto Rico

Location

Hospital Germans Trias i Pujol

Badalona, 08916, Spain

Location

Hospital del Mar

Barcelona, 08003, Spain

Location

Hospital Universitari Vall D'Hebron

Barcelona, 08035, Spain

Location

Hospital Clinic i Provincial

Barcelona, 08036, Spain

Location

University Hospital Bellvitge

Barcelona, 08907, Spain

Location

Hospital General Universitario Gregorio Maranon

Madrid, 28007, Spain

Location

Hospital Universitario 12 de Octubre

Madrid, 28041, Spain

Location

Hospital Universitario La Paz

Madrid, 28046, Spain

Location

Complejo Hospitalario Universitario de Santiago (CHUS)

Santiago de Compostela, 15706, Spain

Location

Universitätsspital Bern

Bern, 3010, Switzerland

Location

Centre Hospitalier Universitaire Vaudois

Lausanne, 1011, Switzerland

Location

University Hospital, Zurich

Zurich, CH-8091, Switzerland

Location

The HIV Netherland Australia Thailand, Thai Red Cross AIDS Research Center (The HIV-NAT)

Bangkok, 10330, Thailand

Location

Ramathibodi Hospital, Mahidol University

Bangkok, 10400, Thailand

Location

Siriraj Hospital

Bangkok, 10700, Thailand

Location

Chiang Mai University

Chiang Mai, 50200, Thailand

Location

Khon Kaen University

Khon Kaen, 40002, Thailand

Location

Bamrasnaradura Infectious Diseases Institute

Nonthaburi, 11000, Thailand

Location

Chelsea & Westminster Hospital

London, SW10 9TH, United Kingdom

Location

Related Publications (7)

  • Sax PE, Wohl D, Yin MT, Post F, DeJesus E, Saag M, Pozniak A, Thompson M, Podzamczer D, Molina JM, Oka S, Koenig E, Trottier B, Andrade-Villanueva J, Crofoot G, Custodio JM, Plummer A, Zhong L, Cao H, Martin H, Callebaut C, Cheng AK, Fordyce MW, McCallister S; GS-US-292-0104/0111 Study Team. Tenofovir alafenamide versus tenofovir disoproxil fumarate, coformulated with elvitegravir, cobicistat, and emtricitabine, for initial treatment of HIV-1 infection: two randomised, double-blind, phase 3, non-inferiority trials. Lancet. 2015 Jun 27;385(9987):2606-15. doi: 10.1016/S0140-6736(15)60616-X. Epub 2015 Apr 15.

  • Arribas JR, Thompson M, Sax PE, Haas B, McDonald C, Wohl DA, DeJesus E, Clarke AE, Guo S, Wang H, Callebaut C, Plummer A, Cheng A, Das M, McCallister S. Brief Report: Randomized, Double-Blind Comparison of Tenofovir Alafenamide (TAF) vs Tenofovir Disoproxil Fumarate (TDF), Each Coformulated With Elvitegravir, Cobicistat, and Emtricitabine (E/C/F) for Initial HIV-1 Treatment: Week 144 Results. J Acquir Immune Defic Syndr. 2017 Jun 1;75(2):211-218. doi: 10.1097/QAI.0000000000001350.

  • Margot N, Cox S, Das M, McCallister S, Miller MD, Callebaut C. Infrequent development of drug resistance in HIV-1-infected treatment-naive subjects after 96 weeks of treatment with elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide or elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate. Antivir Ther. 2017;22(5):443-446. doi: 10.3851/IMP3125. Epub 2017 Jan 11.

  • Margot NA, Kitrinos KM, Fordyce M, McCallister S, Miller MD, Callebaut C. Rare emergence of drug resistance in HIV-1 treatment-naive patients after 48 weeks of treatment with elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide. HIV Clin Trials. 2016 Mar;17(2):78-87. doi: 10.1080/15284336.2016.1142731.

  • Funderburg NT, McComsey GA, Kulkarni M, Bannerman T, Mantini J, Thornton B, Liu HC, Zhang Y, Song Q, Fang L, Dinoso J, Cheng A, McCallister S, Fordyce MW, Das M. Equivalent Decline in Inflammation Markers with Tenofovir Disoproxil Fumarate vs. Tenofovir Alafenamide. EBioMedicine. 2016 Nov;13:321-327. doi: 10.1016/j.ebiom.2016.10.009. Epub 2016 Oct 11.

  • Wohl D, Oka S, Clumeck N, Clarke A, Brinson C, Stephens J, Tashima K, Arribas JR, Rashbaum B, Cheret A, Brunetta J, Mussini C, Tebas P, Sax PE, Cheng A, Zhong L, Callebaut C, Das M, Fordyce M; GS-US-2,92-01040111 and Study Team. Brief Report: A Randomized, Double-Blind Comparison of Tenofovir Alafenamide Versus Tenofovir Disoproxil Fumarate, Each Coformulated With Elvitegravir, Cobicistat, and Emtricitabine for Initial HIV-1 Treatment: Week 96 Results. J Acquir Immune Defic Syndr. 2016 May 1;72(1):58-64. doi: 10.1097/QAI.0000000000000940.

  • Custodio JM, Garner W, Callebaut C, Fordyce M, Plummer A, Zhong L, et al. The Pharmacokinetics of Tenofovir and Tenofovir Diphosphate Following Administration of Tenofovir Alafenamide vs Tenofovir Disoproxil Fumarate [Oral Abstract #6]. The 16th International Workshop on Clinical Pharmacology of HIV & Hepatitis Therapy. Washington DC, USA, May 26-28, 2015.

    RESULT

MeSH Terms

Conditions

HIV Infections

Interventions

Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination

Condition Hierarchy (Ancestors)

Blood-Borne InfectionsCommunicable DiseasesInfectionsSexually Transmitted Diseases, ViralSexually Transmitted DiseasesLentivirus InfectionsRetroviridae InfectionsRNA Virus InfectionsVirus DiseasesGenital DiseasesUrogenital DiseasesImmunologic Deficiency SyndromesImmune System Diseases

Intervention Hierarchy (Ancestors)

CobicistatCarbamatesAcids, AcyclicCarboxylic AcidsOrganic ChemicalsTenofovirOrganophosphonatesOrganophosphorus CompoundsThiazolesSulfur CompoundsAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsEmtricitabineDeoxycytidineCytidinePyrimidine NucleosidesPyrimidinesAdeninePurinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingDeoxyribonucleosidesNucleosidesNucleic Acids, Nucleotides, and NucleosidesDrug CombinationsPharmaceutical Preparations

Results Point of Contact

Title
Gilead Clinical Study Information Center
Organization
Gilead Sciences

Study Officials

  • Gilead Study Director

    Gilead Sciences

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 16, 2013

First Posted

January 31, 2013

Study Start

December 26, 2012

Primary Completion

August 26, 2014

Study Completion

September 6, 2017

Last Updated

November 19, 2018

Results First Posted

January 8, 2016

Record last verified: 2018-08

Data Sharing

IPD Sharing
Will share

Qualified external researchers may request IPD for this study after study completion. For more information, please visit our website at http://www.gilead.com/research/disclosure-and-transparency.

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
18 months after study completion
Access Criteria
A secured external environment with username, password, and RSA code.
More information

Locations