NCT01497899

Brief Summary

The primary objective of this study is to evaluate the efficacy of elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide (Genvoya®; E/C/F/TAF) fixed-dose combination (FDC) versus elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate (Stribild®; E/C/F/TDF) FDC in HIV-1 infected, antiretroviral treatment-naive adults.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
279

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Dec 2011

Longer than P75 for phase_2

Geographic Reach
2 countries

41 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

December 14, 2011

Completed
9 days until next milestone

First Posted

Study publicly available on registry

December 23, 2011

Completed
5 days until next milestone

Study Start

First participant enrolled

December 28, 2011

Completed
10 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 17, 2012

Completed
3.2 years until next milestone

Results Posted

Study results publicly available

January 8, 2016

Completed
8 months until next milestone

Study Completion

Last participant's last visit for all outcomes

August 22, 2016

Completed
Last Updated

November 19, 2018

Status Verified

August 1, 2017

Enrollment Period

10 months

First QC Date

December 14, 2011

Results QC Date

December 4, 2015

Last Update Submit

October 19, 2018

Conditions

Keywords

HIV-1HIVTreatment-Naive

Outcome Measures

Primary Outcomes (1)

  • Percentage of Participants With HIV-1 RNA < 50 Copies/mL at Week 24

    The percentage of participants achieving HIV-1 RNA \< 50 copies/mL at Week 24 was analyzed using the snapshot algorithm, which defines a patient's virologic response status using only the viral load at the predefined time point within an allowed window of time, along with study drug discontinuation status.

    Week 24

Secondary Outcomes (3)

  • Percentage of Participants With HIV-1 RNA < 50 Copies/mL at Week 48

    Week 48

  • Change From Baseline in log10 HIV-1 RNA at Weeks 24 and 48

    Baseline; Weeks 24 and 48

  • Change From Baseline in CD4+ Cell Count at Weeks 24 and 48

    Baseline; Weeks 24 and 48

Study Arms (3)

E/C/F/TAF

EXPERIMENTAL

E/C/F/TAF plus E/C/F/TDF placebo for at least 48 weeks

Drug: E/C/F/TAFDrug: E/C/F/TDF Placebo

E/C/F/TDF

ACTIVE COMPARATOR

E/C/F/TDF plus E/C/F/TAF placebo for at least 48 weeks

Drug: E/C/F/TDFDrug: E/C/F/TAF Placebo

E/C/F/TAF Open-Label

EXPERIMENTAL

Following study unblinding, participants from the E/C/F/TAF and E/C/F/TDF arms may have the option to receive E/C/F/TAF during an open-label extension phase. Also, participants who are actively participating in a Gilead-sponsored study of cobicistat-boosted darunavir plus nucleoside/nucleotide reverse transcriptase inhibitors (NRTI) who have reached the protocol-defined secondary endpoint (Week 48) and remain virologically suppressed are eligible to participate and receive E/C/F/TAF in this open-label extension phase.

Drug: E/C/F/TAF

Interventions

150/150/200/300 mg FDC tablet administered orally once daily

Also known as: Stribild®
E/C/F/TDF

Tablet administered orally once daily

E/C/F/TDF

150/150/200/10 mg FDC tablet administered orally once daily

Also known as: Genvoya®
E/C/F/TAFE/C/F/TAF Open-Label

Tablet administered orally once daily

E/C/F/TAF

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Ability to understand and sign a written informed consent form
  • Plasma HIV 1 RNA levels ≥ 5,000 copies/mL
  • No prior use of any approved or experimental anti-HIV drug for any length of time
  • Screening genotype report must show sensitivity to TDF and emtricitabine (FTC)
  • Normal ECG
  • Adequate renal function: Estimated glomerular filtration rate ≥ 70 mL/min according to the Cockcroft Gault formula
  • Hepatic transaminases ≤ 2.5 x upper limit of the normal range (ULN)
  • Total bilirubin ≤ 1.5 mg/dL, or normal direct bilirubin
  • Adequate hematologic function
  • CD4+ cell count \> 50 cells/µL
  • Serum amylase ≤ 5 x ULN
  • Normal thyroid-stimulating hormone (TSH)
  • Females of childbearing potential must have a negative serum pregnancy test
  • Females of childbearing potential must agree to utilize highly effective contraception methods from screening throughout the duration of study treatment and for 30 days following the last dose of study drugs
  • Female subjects who utilize hormonal contraceptive as one of their birth control methods must have used the same method for at least three months prior to study dosing
  • +5 more criteria

You may not qualify if:

  • New AIDS-defining condition diagnosed within the 30 days prior to screening
  • Hepatitis B surface Antigen positive
  • Hepatitis C Antibody positive
  • Proven acute hepatitis in the 30 days prior to study entry
  • Subjects experiencing decompensated cirrhosis
  • Females who are breastfeeding
  • Positive serum pregnancy test (female of childbearing potential)
  • Have an implanted defibrillator or pacemaker
  • Receiving ongoing therapy with any of the disallowed medications, including drugs not to be used with elvitegravir and cobicistat
  • Have been treated with immunosuppressant therapies or chemotherapeutic agents within 3 months of study screening, or expected to receive these agents or systemic steroids during the study
  • Current alcohol or substance
  • History of or ongoing malignancy (including untreated carcinoma in-situ) other than cutaneous Kaposi's sarcoma (KS), basal cell carcinoma or resected, non-invasive cutaneous squamous carcinoma
  • Active, serious infections (other than HIV 1 infection) requiring parenteral antibiotic or antifungal therapy within 30 days prior to Baseline
  • Participation in any other clinical trial without prior approval is prohibited while participating in this trial
  • Medications contraindicated for use with emtricitabine or tenofovir disoproxil fumarate
  • +2 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (41)

University of Alabama at Birmingham (UAB)

Birmingham, Alabama, 35233, United States

Location

Spectrum Medical Group

Phoenix, Arizona, 85012, United States

Location

AHF Research Center

Beverly Hills, California, 90211, United States

Location

Kaiser Permanente

Los Angeles, California, 90027, United States

Location

Peter J. Ruane, MD, Inc.

Los Angeles, California, 90036, United States

Location

Anthony Mills MD, Inc

Los Angeles, California, 90069, United States

Location

East Bay AIDS Center

Oakland, California, 94609, United States

Location

St. Joseph Heritage Healthcare

Orange, California, 92869, United States

Location

Stanford University

Palo Alto, California, 94304, United States

Location

Kaiser Permanente Medical Group

Sacramento, California, 95825, United States

Location

La Playa Medical Group and Clinical Research

San Diego, California, 92103, United States

Location

Metropolis Medical

San Francisco, California, 94107, United States

Location

Kaiser Permanente Medical Group-Clinical Trials Unit

San Francisco, California, 94118, United States

Location

Apex Research, LLC

Denver, Colorado, 80220, United States

Location

Dupont Circle Physician's Group

Washington D.C., District of Columbia, 20009, United States

Location

Whitman-Walker Health

Washington D.C., District of Columbia, 20009, United States

Location

Capital Medical Associates, PC

Washington D.C., District of Columbia, 20036, United States

Location

Gary J. Richmond,M.D.,P.A.

Fort Lauderdale, Florida, 33316, United States

Location

Wohlfeiler, Piperato and Associates, LLC

Miami Beach, Florida, 33139, United States

Location

Orlando Immunology Center

Orlando, Florida, 32803, United States

Location

IDOCF/ValuhealthMD, LLC

Orlando, Florida, 32806, United States

Location

St. Joseph's Comprehensive Research Institute

Tampa, Florida, 33614, United States

Location

Infectious Disease Specialists of Atlanta

Decatur, Georgia, 30033, United States

Location

Mercer University Mercer Medicine

Macon, Georgia, 31201, United States

Location

Howard Brown Health Center

Chicago, Illinois, 60613, United States

Location

Brigham and Women's Hospital

Boston, Massachusetts, 02115, United States

Location

Be Well Medical Center

Berkley, Michigan, 48072, United States

Location

Henry Ford Health System

Detroit, Michigan, 48202, United States

Location

Hennepin County Medical Center

Minneapolis, Minnesota, 55415, United States

Location

Central West Clinical Research Inc

St Louis, Missouri, 63108, United States

Location

North Shore University Hospital / Division of Infectious Diseases

Manhasset, New York, 11030, United States

Location

ID Consultants, P.A.

Charlotte, North Carolina, 28209, United States

Location

Duke University Medical Center

Durham, North Carolina, 27710, United States

Location

University of South Carolina School of Medicine Division of Infectious Disease

Columbia, South Carolina, 29203, United States

Location

Southwest Infectious Disease Clinical Research Inc

Dallas, Texas, 75219, United States

Location

Tarrant County Infectious Disease Associates

Fort Worth, Texas, 76104, United States

Location

Therapeutic Concepts, PA

Houston, Texas, 77004, United States

Location

Gordon E. Crofoot, MD., PA

Houston, Texas, 77098, United States

Location

DCOL Center for Clinical Research

Longview, Texas, 75605, United States

Location

Peter Shalit, M.D.

Seattle, Washington, 98104, United States

Location

Clinical Research Puerto Rico

San Juan, 00909, Puerto Rico

Location

Related Publications (1)

  • Sax PE, Zolopa A, Brar I, Elion R, Ortiz R, Post F, Wang H, Callebaut C, Martin H, Fordyce MW, McCallister S. Tenofovir alafenamide vs. tenofovir disoproxil fumarate in single tablet regimens for initial HIV-1 therapy: a randomized phase 2 study. J Acquir Immune Defic Syndr. 2014 Sep 1;67(1):52-8. doi: 10.1097/QAI.0000000000000225.

MeSH Terms

Conditions

Acquired Immunodeficiency SyndromeHIV Infections

Interventions

Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination

Condition Hierarchy (Ancestors)

Blood-Borne InfectionsCommunicable DiseasesInfectionsSexually Transmitted Diseases, ViralSexually Transmitted DiseasesLentivirus InfectionsRetroviridae InfectionsRNA Virus InfectionsVirus DiseasesSlow Virus DiseasesGenital DiseasesUrogenital DiseasesImmunologic Deficiency SyndromesImmune System Diseases

Intervention Hierarchy (Ancestors)

CobicistatCarbamatesAcids, AcyclicCarboxylic AcidsOrganic ChemicalsTenofovirOrganophosphonatesOrganophosphorus CompoundsThiazolesSulfur CompoundsAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsEmtricitabineDeoxycytidineCytidinePyrimidine NucleosidesPyrimidinesAdeninePurinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingDeoxyribonucleosidesNucleosidesNucleic Acids, Nucleotides, and NucleosidesDrug CombinationsPharmaceutical Preparations

Limitations and Caveats

There were no limitations affecting the analysis or results.

Results Point of Contact

Title
Clinical Trial Disclosures
Organization
Gilead Sciences

Study Officials

  • Gilead Study Director

    Gilead Sciences

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

December 14, 2011

First Posted

December 23, 2011

Study Start

December 28, 2011

Primary Completion

October 17, 2012

Study Completion

August 22, 2016

Last Updated

November 19, 2018

Results First Posted

January 8, 2016

Record last verified: 2017-08

Data Sharing

IPD Sharing
Will share

Qualified external researchers may request IPD for this study after study completion. For more information, please visit our website at http://www.gilead.com/research/disclosure-and-transparency.

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
18 months after study completion
Access Criteria
A secured external environment with username, password, and RSA code.
More information

Locations