NCT01818596

Brief Summary

The primary objective of this study is to evaluate the effect of elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide (E/C/F/TAF) fixed-dose combination (FDC) tablet on renal parameters at Week 24 in treatment-naive and treatment-experienced HIV-positive, adults with mild to moderate renal impairment.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
252

participants targeted

Target at P25-P50 for phase_3 hiv

Timeline
Completed

Started Mar 2013

Longer than P75 for phase_3 hiv

Geographic Reach
9 countries

70 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

March 22, 2013

Completed
4 days until next milestone

First Posted

Study publicly available on registry

March 26, 2013

Completed
1 day until next milestone

Study Start

First participant enrolled

March 27, 2013

Completed
1.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 31, 2014

Completed
1.6 years until next milestone

Results Posted

Study results publicly available

February 18, 2016

Completed
2.4 years until next milestone

Study Completion

Last participant's last visit for all outcomes

July 18, 2018

Completed
Last Updated

March 2, 2020

Status Verified

June 1, 2019

Enrollment Period

1.3 years

First QC Date

March 22, 2013

Results QC Date

December 4, 2015

Last Update Submit

February 18, 2020

Conditions

Keywords

HIVHIV-1 InfectedTreatment ExperiencedTreatment Naive

Outcome Measures

Primary Outcomes (3)

  • Change From Baseline in the Estimated Glomerular Filtration Rate Calculated by the Cockcroft-Gault Formula (eGFR_CG) at Week 24

    eGFR is a measurement of the kidney's ability to filter blood.

    Baseline; Week 24

  • Change From Baseline in eGFR Calculated by the Chronic Kidney Disease Epidemiology Collaboration Method Based on Cystatin C (eGFR_CKD-EPI,cysC) at Week 24

    eGFR is a measurement of the kidney's ability to filter blood. The eGFR\_CKD-EPI,cysC method is adjusted for age and sex.

    Baseline; Week 24

  • Change From Baseline in eGFR Calculated by the CKD-EPI Method Based on Serum Creatinine (eGFR_CKD-EPI,Creatinine) at Week 24

    eGFR is a measurement of the kidney's ability to filter blood. The eGFR\_CKD-EPI,creatinine method is adjusted for age, race, and sex.

    Baseline; Week 24

Secondary Outcomes (18)

  • Change From Baseline in Actual GFR (aGFR) of E/C/F/TAF for Participants Enrolled in the PK/PD Substudy

    Baseline; Week 2, 4, or 8; Week 24

  • Percent Change From Baseline in C-type Collagen Sequence (CTX) at Weeks 24 and 48

    Baseline; Weeks 24 and 48

  • Percent Change From Baseline in Procollagen Type 1 N-terminal Propeptide (P1NP) at Weeks 24 and 48

    Baseline; Weeks 24 and 48

  • Percent Change From Baseline in Retinol Binding Protein (RBP) to Creatinine Ratio (μg/g) at Weeks 24, 48, 96, and 144

    Baseline; Weeks 24, 48, 96, and 144

  • Percent Change From Baseline in Urine Beta-2-microglobulin to Creatinine Ratio (μg/g) at Weeks 24, 48, 96, and 144

    Baseline; Weeks 24, 48, 96, and 144

  • +13 more secondary outcomes

Study Arms (1)

E/C/F/TAF

EXPERIMENTAL

Participants will receive E/C/F/TAF for 144 weeks. Following Week 144, in countries where E/C/F/TAF is not available (except for the United Kingdom), participants will be given the option to continue in the study and receive E/C/F/TAF for another 48 weeks, or until the product becomes available through an access program, or until Gilead Sciences elects to discontinue the study in that country, whichever comes first.

Drug: E/C/F/TAF

Interventions

E/C/F/TAF (150/150/200/10 mg) FDC tablet administered orally once daily with food

Also known as: Genvoya®
E/C/F/TAF

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Cohort 1 (treatment-experienced switch)
  • Must not have a history of known resistance to elvitegravir (EVG), tenofovir disoproxil fumarate (TDF), or emtricitabine (FTC)
  • Plasma HIV-1 RNA concentrations (at least two measurements) at undetectable levels (according to the local assay being used) in the 6 months preceding the screening visit and have HIV-1 RNA \< 50 copies/mL at screening
  • Estimated glomerular filtration rate (GFR) 30-69 mL/min according to the Cockcroft-Gault formula for creatinine clearance, using actual weight
  • May be currently enrolled in Gilead studies GS-US-236-0102, GS-US-236-0103, and GS-US-216-0114, but will be eligible to enroll only after the Week 144 visit for that study is complete; or currently receiving Stribild® (STB) or atazanavir (ATV)/cobicistat (COBI) + Truvada (TVD) in Gilead studies GS-US-236-0104 or GS-US-216-0105, but will be eligible to enroll only after the Week 48 visit for that study is complete.
  • Cohort 2 (treatment-naive)
  • Plasma HIV-1 RNA levels ≥ 1,000 copies/mL at screening
  • Screening genotype report provided by Gilead Sciences must show sensitivity to EVG, FTC, and TDF
  • No prior use of any approved or investigational antiretroviral drug for any length of time, except the use for pre-exposure prophylaxis (PrEP), or post-exposure prophylaxis (PEP), up to 6 months prior to screening
  • Estimated GFR 30-69 mL/min according to the Cockcroft Gault formula for creatinine clearance, using actual weight
  • All Cohorts:
  • The ability to understand and sign a written informed consent form, which must be obtained prior to initiation of study procedures
  • CD4+ count of ≥ 50 cells/μL
  • Stable renal function: serum creatinine measurements to be taken at least once (within three months of screening)
  • Cause of underlying chronic kidney disease (eg hypertension, diabetes) stable, without change in medical management, for 3 months prior to baseline
  • +8 more criteria

You may not qualify if:

  • A new AIDS-defining condition (excluding CD4 cell count and percentage criteria) diagnosed within the 30 days prior to screening,with the exception of the first two bullet points
  • Hepatitis C virus (HCV) antibody positive. Individuals who are HCV positive, but have a documented negative HCV RNA, are eligible
  • Hepatitis B surface antigen (HBVsAg) positive
  • Individuals receiving drug treatment for Hepatitis C, or individuals who are anticipated to receive treatment for Hepatitis C during the course of the study
  • Individuals experiencing decompensated cirrhosis (eg, ascites, encephalopathy, etc.)
  • Females who are breastfeeding
  • Positive serum pregnancy test
  • Have an implanted defibrillator or pacemaker
  • Current alcohol or substance use judged by the Investigator to potentially interfere with study compliance
  • A history of malignancy within the past 5 years or ongoing malignancy other than cutaneous Kaposi's sarcoma, basal cell carcinoma, or resected, non-invasive cutaneous squamous carcinoma
  • Active, serious infections (other than HIV-1 infection) requiring parenteral antibiotic or antifungal therapy within 30 days prior to baseline
  • Individuals on hemodialysis, other forms of renal replacement therapy, or on treatment for underlying kidney diseases (including prednisolone and dexamethasone)
  • Individuals receiving ongoing therapy with any medications not to be used with EVG, COBI, FTC, or TAF or individuals with any known allergies to the excipients of E/C/F/TAF

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (70)

Maricopa Integrated Health System - McDowell Clinic

Phoenix, Arizona, 85006, United States

Location

Pueblo Family Physicians

Phoenix, Arizona, 85015, United States

Location

Health for Life Clinic PLLC

Little Rock, Arkansas, 72207, United States

Location

Pacific Oaks Medical Group

Beverly Hills, California, 90211, United States

Location

Kaiser Permanente

Hayward, California, 94545, United States

Location

Long Beach Education and Research Consultants

Long Beach, California, 90813, United States

Location

LA Gay & Lesbian Center - Jeffrey Goodman Special Care Clinic

Los Angeles, California, 90028, United States

Location

Peter J Ruane, MD, Inc

Los Angeles, California, 90036, United States

Location

Anthony Mills MD, Inc

Los Angeles, California, 90069, United States

Location

Desert Medical Group Inc. dba Desert Oasis Healthcare Medical Group

Palm Springs, California, 92262, United States

Location

Kaiser Permanente Medical Group

Sacramento, California, 95825, United States

Location

Metropolis Medical

San Francisco, California, 94109, United States

Location

Kaiser Permanente CTU San Francisco

San Francisco, California, 94118, United States

Location

University of Colorado

Aurora, Colorado, 80045, United States

Location

National Jewish Health

Denver, Colorado, 80206, United States

Location

Dupont Circle Physician's Group

Washington D.C., District of Columbia, 20009, United States

Location

Gary J. Richmond, MD PA

Fort Lauderdale, Florida, 33316, United States

Location

Midway Immunology and Research Center

Ft. Pierce, Florida, 34982, United States

Location

Idocf/Valuhealthmd

Orlando, Florida, 32806, United States

Location

University of South Florida

Tampa, Florida, 33602, United States

Location

Triple O Research Institute, P.A.

West Palm Beach, Florida, 33401, United States

Location

Rowan Tree Medical, P.A.

Wilton Manors, Florida, 33305, United States

Location

Infectious Disease Specialists of Atlanta

Decatur, Georgia, 30033, United States

Location

Mercer University

Macon, Georgia, 31210, United States

Location

Indiana University School of Medicine

Indianapolis, Indiana, 46202, United States

Location

Community Research Initiative of New England

Boston, Massachusetts, 02111, United States

Location

The Research Institute

Springfield, Massachusetts, 01105, United States

Location

Be Well Medical Center, P.C.

Berkley, Michigan, 48210, United States

Location

Henry Ford Health System

Detroit, Michigan, 48202, United States

Location

Hennepin County Medical Center

Minneapolis, Minnesota, 55415, United States

Location

The Kansas City Care Clinic (KC Free Health Clinic)

Kansas City, Missouri, 64111, United States

Location

Southampton Healthcare, Inc.

St Louis, Missouri, 63139, United States

Location

Jersey Shore University Medical Center

Neptune City, New Jersey, 07754, United States

Location

Saint Michael's Medical Center

Newark, New Jersey, 07102, United States

Location

Southwest CARE Center

Santa Fe, New Mexico, 87505, United States

Location

Albany Medical College

Albany, New York, 12208, United States

Location

Upstate Infectious Diseases Associates

Albany, New York, 12208, United States

Location

North Shore University Hospital/Division of Infectious Diseases

Manhasset, New York, 11030, United States

Location

Aids Care

Rochester, New York, 14607, United States

Location

Jacobi Medical Center

The Bronx, New York, 10461, United States

Location

Montefiore Medical Center

The Bronx, New York, 10467, United States

Location

University of Cincinnati

Cincinnati, Ohio, 45267-0405, United States

Location

MetroHealth Medical Center

Cleveland, Ohio, 44109, United States

Location

University of PA HIV Clinical Trials Unit

Philadelphia, Pennsylvania, 19104, United States

Location

Thomas Jefferson University

Philadelphia, Pennsylvania, 19107, United States

Location

St. Hope Foundation

Bellaire, Texas, 77401, United States

Location

North Texas Infectious Diseases Consultants, PA

Dallas, Texas, 75246, United States

Location

Garcias' Family Health Group

Harlingen, Texas, 78550, United States

Location

Therapeutic Concepts, PA

Houston, Texas, 77004, United States

Location

Gordon E. Crofoot MD, PA

Houston, Texas, 77098, United States

Location

Peter Shalit, MD

Seattle, Washington, 98104, United States

Location

Holdsworth House Medical Practice

Darlinghurst, New South Wales, 2010, Australia

Location

Clinical Research Infectious Diseases Department- Alfred Hospital

Melbourne, Victoria, 3004, Australia

Location

Prahran Market Clinic

Prahran, Victoria, 3181, Australia

Location

Instituto Dominicano de Estudios Virologicos (IDEV)

Santo Domingo, 99999, Dominican Republic

Location

Hopital de la Croix Rousse

Lyon, 69004, France

Location

GHPS Service des maladies infectieuses et tropicales pavillon Laveran unité de recherche clinique

Paris, 75651, France

Location

Hospital Civil de Guadalajara Dr. Juan I. Menchaca

Guadalajara, Jalisco, 44340, Mexico

Location

University Medical Center Utrecht

Utrecht, 3584 CX, Netherlands

Location

Hospital Universitari de Bellvitge

Barcelona, 8907, Spain

Location

Germans Trias i Pujol University Hospital

Barcelona, 8916, Spain

Location

Hospital La Paz

Madrid, 28046, Spain

Location

HIV-NAT, Thai Red Cross AIDS Research Centre

Bangkok, 10330, Thailand

Location

Faculty of Medicine Ramathibodi Hospital, Mahidol University

Bangkok, 10400, Thailand

Location

Department of Preventive and Social Medicine, Faculty of Medicine, Siriraj Hospital

Bangkok, 10700, Thailand

Location

Srinagarind Hospital, Khon Kaen University

Khon Kaen, 40002, Thailand

Location

Brighton & Sussex University Hospitals NHS Trust

Brighton, BN2 1ES, United Kingdom

Location

Kings College London

London, SE5 9RJ, United Kingdom

Location

Chelsea and Westminster NHS Foundation Trust Hospital

London, Sw10 9NH, United Kingdom

Location

Central Manchester University Hospitals NHS foundation Trust

Manchester, M13 0FH, United Kingdom

Location

Related Publications (2)

  • Pozniak A, Arribas JR, Gathe J, Gupta SK, Post FA, Bloch M, Avihingsanon A, Crofoot G, Benson P, Lichtenstein K, Ramgopal M, Chetchotisakd P, Custodio JM, Abram ME, Wei X, Cheng A, McCallister S, SenGupta D, Fordyce MW; GS-US-292-0112 Study Team. Switching to Tenofovir Alafenamide, Coformulated With Elvitegravir, Cobicistat, and Emtricitabine, in HIV-Infected Patients With Renal Impairment: 48-Week Results From a Single-Arm, Multicenter, Open-Label Phase 3 Study. J Acquir Immune Defic Syndr. 2016 Apr 15;71(5):530-7. doi: 10.1097/QAI.0000000000000908.

  • Post FA, Tebas P, Clarke A, Cotte L, Short WR, Abram ME, Jiang S, Cheng A, Das M, Fordyce MW. Brief Report: Switching to Tenofovir Alafenamide, Coformulated With Elvitegravir, Cobicistat, and Emtricitabine, in HIV-Infected Adults With Renal Impairment: 96-Week Results From a Single-Arm, Multicenter, Open-Label Phase 3 Study. J Acquir Immune Defic Syndr. 2017 Feb 1;74(2):180-184. doi: 10.1097/QAI.0000000000001186.

MeSH Terms

Conditions

HIV Infections

Interventions

Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination

Condition Hierarchy (Ancestors)

Blood-Borne InfectionsCommunicable DiseasesInfectionsSexually Transmitted Diseases, ViralSexually Transmitted DiseasesLentivirus InfectionsRetroviridae InfectionsRNA Virus InfectionsVirus DiseasesGenital DiseasesUrogenital DiseasesImmunologic Deficiency SyndromesImmune System Diseases

Intervention Hierarchy (Ancestors)

CobicistatCarbamatesAcids, AcyclicCarboxylic AcidsOrganic ChemicalsTenofovirOrganophosphonatesOrganophosphorus CompoundsThiazolesSulfur CompoundsAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsEmtricitabineDeoxycytidineCytidinePyrimidine NucleosidesPyrimidinesAdeninePurinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingDeoxyribonucleosidesNucleosidesNucleic Acids, Nucleotides, and NucleosidesDrug CombinationsPharmaceutical Preparations

Limitations and Caveats

Enrollment in Cohort 2 (treatment-naive) was low, which affects the interpretation of the data.

Results Point of Contact

Title
Gilead Clinical Study Information Center
Organization
Gilead Sciences

Study Officials

  • Gilead Study Director

    Gilead Sciences

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 22, 2013

First Posted

March 26, 2013

Study Start

March 27, 2013

Primary Completion

July 31, 2014

Study Completion

July 18, 2018

Last Updated

March 2, 2020

Results First Posted

February 18, 2016

Record last verified: 2019-06

Data Sharing

IPD Sharing
Will share

Qualified external researchers may request IPD for this study after study completion. For more information, please visit our website at https://www.gilead.com/science-and-medicine/research/clinical-trials-transparency-and-data-sharing-policy.

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
18 months after study completion
Access Criteria
A secured external environment with username, password, and RSA code.
More information

Locations