NCT01447147

Brief Summary

The purpose of this study is to evaluate the safety and efficacy of treatment with CCX140-B in subjects with diabetic nephropathy.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
332

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Oct 2011

Typical duration for phase_2

Geographic Reach
6 countries

83 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

October 1, 2011

Completed
3 days until next milestone

First Submitted

Initial submission to the registry

October 4, 2011

Completed
2 days until next milestone

First Posted

Study publicly available on registry

October 6, 2011

Completed
2.8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2014

Completed
4 months until next milestone

Study Completion

Last participant's last visit for all outcomes

December 1, 2014

Completed
Last Updated

February 27, 2025

Status Verified

February 1, 2025

Enrollment Period

2.8 years

First QC Date

October 4, 2011

Last Update Submit

February 25, 2025

Conditions

Outcome Measures

Primary Outcomes (1)

  • Subject incidence of adverse events

    The primary objective of this study is to evaluate the safety and tolerability of CCX140-B in subjects with diabetic nephropathy.

    Up to 365 days

Secondary Outcomes (1)

  • Change from baseline in first morning urinary albumin:creatinine ratio (ACR)

    Up to 365 days

Study Arms (3)

Placebo (Group A)

PLACEBO COMPARATOR
Drug: Placebo

CCX140-B (Group B)

EXPERIMENTAL
Drug: CCX140-B

CCX140-B (Group C)

EXPERIMENTAL
Drug: CCX140-B

Interventions

Placebo capsules once daily

Placebo (Group A)

CCX140-B capsules once daily (Group B)

CCX140-B (Group B)

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Aged 18-75 years inclusive, with documented previously diagnosed type 2 diabetes mellitus (per American Diabetes Association \[ADA\] criteria)
  • Residual albuminuria despite stable treatment with an angiotensin-converting enzyme (ACE) inhibitor or an angiotensin receptor blocker (ARB) for at least 8 weeks prior to screening (Albumin:creatinine ratio \[ACR\] of 100 to 3000 mg/g creatinine, inclusive)
  • Estimated glomerular filtration rate based on serum creatinine (eGFR, determined by Modification of Diet in Renal Disease \[MDRD\] equation) of ≥ 25 mL/min/1.73 m(2)
  • Must be on a stable dose of an ACE inhibitor or ARB for at least 8 weeks prior to screening, but subjects must not be on both an ACE inhibitor and an ARB
  • Hemoglobin A1c (HbA1c) \> 6.0% but not \> 10.0% and fasting plasma glucose less than 270 mg/dL at screening

You may not qualify if:

  • Type 1 diabetes mellitus or history of diabetic ketoacidosis
  • Previous renal transplant or known non-diabetic renal disease, except related to hypertension
  • Undergone renal dialysis at any time in the past
  • Received chronic (more than 7 days continuously) systemic glucocorticoid or other immunosuppressive treatment within 8 weeks of screening
  • Use of bardoxolone, atrasentan or other endothelin antagonist within 8 weeks of screening
  • Received chronic (more than 7 days continuously) non-steroidal anti-inflammatory drug (NSAID) treatment within 2 weeks of screening
  • Cardiac failure (class III or IV), history of unstable angina, symptomatic coronary artery disease, myocardial infarction or stroke within 12 weeks of screening
  • Poorly-controlled blood pressure (systolic blood pressure \>155 or diastolic blood pressure \>95, with blood pressure measured in the seated position after at least 5 minutes of rest)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (83)

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Antwerp, Belgium

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Brussels, Belgium

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Edegem, Belgium

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Ghent, Belgium

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Leuven, Belgium

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Liège, Belgium

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Roeselare, Belgium

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Beroun, Czechia

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Brno, Czechia

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Hlučín, Czechia

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Neratovice, Czechia

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Nový Jičín, Czechia

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NZdar Nad Sazavou, Czechia

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Pardubice, Czechia

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Prague, Czechia

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Přelouč, Czechia

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Rakovník, Czechia

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Slaný, Czechia

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Třebíč, Czechia

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Uherský Brod, Czechia

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Uničov, Czechia

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Berlin, Germany

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Bosenheim, Germany

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Cologne, Germany

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Deggingen, Germany

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Dresden, Germany

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Erlangen, Germany

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Hanover, Germany

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Heidelberg, Germany

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Heilbronn, Germany

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Hoyerswerda, Germany

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Munich, Germany

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Neuwied, Germany

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Nuremberg, Germany

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Pirna, Germany

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Potsdam, Germany

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Saarlouis, Germany

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Speyer, Germany

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Wiesbaden, Germany

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Baja, Hungary

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Balatonfüred, Hungary

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Békéscsaba, Hungary

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Budapest, Hungary

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Debrecen, Hungary

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Eger, Hungary

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Gyula, Hungary

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Hatvan, Hungary

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Kaposvár, Hungary

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Kisvárda, Hungary

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Sátoraljaújhely, Hungary

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Szekszard, Tolna, Hungary

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Szikszó, Hungary

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Bialystok, Poland

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Ciechanów, Poland

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Gdansk, Poland

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Grodzisk Mazowiecki, Poland

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Krakow, Poland

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Poznan, Poland

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Radom, Poland

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Rzeszów, Poland

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Szczecin, Poland

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Warsaw, Poland

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Wroclaw, Poland

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Bath, United Kingdom

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Belfast, United Kingdom

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Birmingham, United Kingdom

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Bristol, United Kingdom

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Chester, United Kingdom

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Coventry, United Kingdom

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Doncaster, United Kingdom

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Edmonton, United Kingdom

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Liverpool, United Kingdom

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Livingston, United Kingdom

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London, United Kingdom

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Londonderry, United Kingdom

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Manchester, United Kingdom

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Middlesbrough, United Kingdom

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Norfolk, United Kingdom

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Preston, United Kingdom

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Salford, United Kingdom

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Sheffield, United Kingdom

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Swansea, United Kingdom

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Welwyn Garden City, United Kingdom

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Related Publications (2)

  • de Zeeuw D, Bekker P, Henkel E, Hasslacher C, Gouni-Berthold I, Mehling H, Potarca A, Tesar V, Heerspink HJ, Schall TJ; CCX140-B Diabetic Nephropathy Study Group. The effect of CCR2 inhibitor CCX140-B on residual albuminuria in patients with type 2 diabetes and nephropathy: a randomised trial. Lancet Diabetes Endocrinol. 2015 Sep;3(9):687-96. doi: 10.1016/S2213-8587(15)00261-2. Epub 2015 Aug 9.

  • Sullivan T, Miao Z, Dairaghi DJ, Krasinski A, Wang Y, Zhao BN, Baumgart T, Ertl LS, Pennell A, Seitz L, Powers J, Zhao R, Ungashe S, Wei Z, Boring L, Tsou CL, Charo I, Berahovich RD, Schall TJ, Jaen JC. CCR2 antagonist CCX140-B provides renal and glycemic benefits in diabetic transgenic human CCR2 knockin mice. Am J Physiol Renal Physiol. 2013 Nov 1;305(9):F1288-97. doi: 10.1152/ajprenal.00316.2013. Epub 2013 Aug 28.

MeSH Terms

Conditions

Diabetic NephropathiesDiabetes Mellitus, Type 2

Interventions

CCX140-B

Condition Hierarchy (Ancestors)

Kidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesDiabetes ComplicationsDiabetes MellitusEndocrine System DiseasesGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic Diseases

Study Officials

  • MD

    Amgen

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 4, 2011

First Posted

October 6, 2011

Study Start

October 1, 2011

Primary Completion

August 1, 2014

Study Completion

December 1, 2014

Last Updated

February 27, 2025

Record last verified: 2025-02

Locations