NCT01756703

Brief Summary

The purpose of this study is to evaluate pharmacodynamics, safety, tolerability and pharmacokinetics of MT-3995 in Type II Diabetic Nephropathy Subjects with Albuminuria

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
67

participants targeted

Target at P50-P75 for phase_2

Timeline
Completed

Started Nov 2012

Geographic Reach
5 countries

43 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

November 1, 2012

Completed
2 months until next milestone

First Submitted

Initial submission to the registry

December 20, 2012

Completed
7 days until next milestone

First Posted

Study publicly available on registry

December 27, 2012

Completed
1.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2014

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2014

Completed
Last Updated

February 9, 2015

Status Verified

February 1, 2015

Enrollment Period

1.7 years

First QC Date

December 20, 2012

Last Update Submit

February 5, 2015

Conditions

Keywords

Diabetic Nephropathy

Outcome Measures

Primary Outcomes (2)

  • Percentage change from baseline in Urine albumin-to-creatinine ratio (UACR) within group.

    up to 8 weeks

  • Frequency and nature of treatment-emergent adverse events and serious adverse events.

    up to 16 weeks

Secondary Outcomes (3)

  • Percentage change from baseline in UACR compared to placebo

    up to 8 weeks

  • Change from baseline in Systolic Blood Pressure and Diastolic Blood Pressure within group.

    up to 8 weeks

  • Plasma concentrations of MT-3995 and its major metabolite

    up to 16 weeks

Study Arms (3)

MT-3995 Low group

EXPERIMENTAL
Drug: MT-3995 Low

MT-3995 High group

EXPERIMENTAL
Drug: MT-3995 High

Placebo group

PLACEBO COMPARATOR
Drug: Placebo

Interventions

MT-3995 Low dose for 8 weeks

MT-3995 Low group

MT-3995 High dose for 8 weeks

MT-3995 High group

Placebo for 8 weeks

Placebo group

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Subjects with Type II diabetic nephropathy, who have been treated with angiotensin converting enzyme-inhibitor (ACE-I) or angiotensin II receptor blocker (ARB)
  • Glycosylated haemoglobin (HbA1c) ≤10.5%
  • An estimated glomerular filtration rate (eGFR) ≥60 mL/min/1.73m\^2
  • Subject with albuminuria

You may not qualify if:

  • History of Type I diabetes, pancreas or β-cell transplantation, or diabetes secondary to pancreatitis or pancreatectomy
  • Serum potassium level \<3.5 or \>5.0 mmol/L
  • Subjects who had acute kidney injury (AKI) within 3 months prior to baseline or have undergone renal dialysis at any time prior to randomisation
  • Subjects with a history of renal transplant
  • Subjects with clinically significant hypotension

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (43)

Investigational site

Blagoevgrad, Bulgaria

Location

Investigational site

Burgas, Bulgaria

Location

Investigational site

Byala, Bulgaria

Location

Investigational site

Golenci, Bulgaria

Location

Investigational site

Pazardzhik, Bulgaria

Location

Investigational site

Plovdiv, Bulgaria

Location

Investigational site

Rousse, Bulgaria

Location

Investigational site

Sofia, Bulgaria

Location

Investigational site

Varna, Bulgaria

Location

Investigational site

Baja, Hungary

Location

Investigational site

Budapest, Hungary

Location

Investigational site

Debrecen, Hungary

Location

Investigational site

Eger, Hungary

Location

Investigational site

Kistelek, Hungary

Location

Investigational site

Komárom, Hungary

Location

Investigational site

Pécs, Hungary

Location

Investigational site

Szigetvár, Hungary

Location

Investigational site

Szikszó, Hungary

Location

Investigational site

Zalaegerszeg, Hungary

Location

Investigational site

Kaunas, Lithuania

Location

Investigational site

Klaipėda, Lithuania

Location

Investigational site

Vilnius, Lithuania

Location

Investigational site

Bacau, Romania

Location

Investigational site

Baia Mare, Romania

Location

Investigational site

Brasov, Romania

Location

Investigational site

Brăila, Romania

Location

Investigational site

Bucharest, Romania

Location

Investigational site

Cluj-Napoca, Romania

Location

Investigational site

Iași, Romania

Location

Investigational site

Oradea, Romania

Location

Investigational site

Ploieşti, Romania

Location

Investigational site

Satu Mare, Romania

Location

Investigational site

Târgu Mureş, Romania

Location

Investigational site

Timișoara, Romania

Location

Investigational site

Banská Bystrica, Slovakia

Location

Investigational site

Bardejov, Slovakia

Location

Investigational site

Bratislava, Slovakia

Location

Investigational site

Lučenec, Slovakia

Location

Investigational site

Martin, Slovakia

Location

Investigational site

Nitra, Slovakia

Location

Investigational site

Šahy, Slovakia

Location

Investigational site

Štúrovo, Slovakia

Location

Investigational site

Žilina, Slovakia

Location

MeSH Terms

Conditions

Diabetic Nephropathies

Condition Hierarchy (Ancestors)

Kidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesDiabetes ComplicationsDiabetes MellitusEndocrine System Diseases

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

December 20, 2012

First Posted

December 27, 2012

Study Start

November 1, 2012

Primary Completion

August 1, 2014

Study Completion

August 1, 2014

Last Updated

February 9, 2015

Record last verified: 2015-02

Locations