NCT01278134

Brief Summary

This multicenter, randomized, double-blind, parallel group study will evaluate the safety and efficacy of the combination RO5024048 and ritonavir-boosted danoprevir with and without Copegus (ribavirin) in patients with chronic hepatitis C genotype 1. In arm A and B, interferon treatment-naïve patients will receive 1000 mg RO5024048 orally twice daily and 100 mg danoprevir with 100 mg ritonavir orally twice daily plus either Copegus (1000 mg or 1200 mg orally daily) or placebo for 12 weeks. Depending on viral response and treatment arm patients will be re-randomized to continue assigned treatment for additional 12 weeks or stop all treatment. The anticipated time on study treatment is up to 24 weeks plus a 24-week follow-up. As of 29. September 2011, Arm B patients (placebo-containing arm) will be offered, in conjunction with the current treatment, Pegasys (peginterferon alfa-2a) 180 mcg subcutaneously weekly plus Copegus 1000mg or 1200 mg orally daily for 24 weeks, with a 24-week follow-up.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
170

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Feb 2011

Geographic Reach
4 countries

32 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

January 14, 2011

Completed
3 days until next milestone

First Posted

Study publicly available on registry

January 17, 2011

Completed
15 days until next milestone

Study Start

First participant enrolled

February 1, 2011

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 1, 2012

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

October 1, 2012

Completed
Last Updated

November 2, 2016

Status Verified

November 1, 2016

Enrollment Period

1.7 years

First QC Date

January 14, 2011

Last Update Submit

November 1, 2016

Conditions

Outcome Measures

Primary Outcomes (2)

  • Sustained virological response, defined as undetectable HVC RNA measured by Roche COBAS TaqMan HCV test

    24 weeks after end of treatment

  • Safety: Incidence of adverse events

    1.5 years

Secondary Outcomes (7)

  • Virological response (HCV RNA measured by Roche COBAS Taqman HCV test)

    up to 48 weeks

  • Impact of Copegus (ribavirin) on efficacy of the direct-acting antiviral combination regimen: viral response (HCV RNA measured by Roche COBAS TaqMan HCV test)

    1.5 years

  • Comparison of 12 and 24 weeks of treatment duration: viral response (HCV RNA measured by Roche COBAS TaqMan HCV test)

    1.5 years

  • Pharmacokinetics: Plasma concentrations of danoprevir, ritonavir, RO4995855 (parent drug of RO5024048) and ribavirin

    up to 24 weeks

  • Viral resistance: HCV RNA sequencing and phenotypic analyses

    up to 48 weeks

  • +2 more secondary outcomes

Study Arms (3)

Arm B Extension

EXPERIMENTAL

All patients in treatment arm B were offered to receive Pegasys/Cogepus therapy for an additional 24 weeks.

Drug: peginterferon alfa-2a [Pegasys]Drug: ribavirin [Copegus]

RO5024048 & ritonavir-boosted danoprevir without Ribavirin (B)

EXPERIMENTAL
Drug: Copegus placeboDrug: RO5024048Drug: danoprevirDrug: ritonavir

RO5024048 and ritonavir-boosted danoprevir with Ribavirin (A)

EXPERIMENTAL
Drug: RO5024048Drug: danoprevirDrug: ribavirin [Copegus]Drug: ritonavir

Interventions

1000 mg or 1200 mg daily orally in split doses (morning/evening), up to 24 weeks

RO5024048 & ritonavir-boosted danoprevir without Ribavirin (B)

1000 mg bid orally, up to 24 weeks

RO5024048 & ritonavir-boosted danoprevir without Ribavirin (B)RO5024048 and ritonavir-boosted danoprevir with Ribavirin (A)

100 mg bid orally, up to 24 weeks

RO5024048 & ritonavir-boosted danoprevir without Ribavirin (B)RO5024048 and ritonavir-boosted danoprevir with Ribavirin (A)

180 mcg sc weekly, 24 weeks

Arm B Extension

1000 mg or 1200 mg daily orally in split doses (morning/evening), up to 24 weeks

Arm B ExtensionRO5024048 and ritonavir-boosted danoprevir with Ribavirin (A)

100 mg bid orally, up to 24 weeks

RO5024048 & ritonavir-boosted danoprevir without Ribavirin (B)RO5024048 and ritonavir-boosted danoprevir with Ribavirin (A)

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Adult patient, \>/= 18 years of age
  • Chronic Hepatitis C of \>/= 6 months duration at screening
  • HCV genotype 1 and quantifiable HCV RNA at screening (Roche COBAS TaqMan HCV test)
  • Naïve for treatment with interferon (pegylated or non-pegylated)
  • Body Mass Index (BMI) 18-35 inclusive, minimum weight 45 kg
  • Females of child-bearing potential and males with female partners of childbearing potential must use 2 forms of effective non-hormonal contraception

You may not qualify if:

  • Pregnant or lactating women and males with female partners who are pregnant or lactating
  • Decompensated liver disease or impaired liver function
  • Cirrhosis or incomplete/transition to cirrhosis
  • Non-hepatitis C chronic liver disease
  • Hepatitis B or HIV infection
  • History of neoplastic disease within the last 5 years, except for localized or in situ carcinoma of the skin
  • History of pre-existing renal disease (except for nephrolithiasis) or severe cardiac disease
  • History of drug or alcohol abuse within the last year or alcohol consumption of \> 2 units per day; cannabinoid use is excepted

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (32)

Unknown Facility

La Jolla, California, 92037-1030, United States

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Unknown Facility

Sacramento, California, 95817, United States

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Unknown Facility

Orlando, Florida, 32809, United States

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Marietta, Georgia, 30060, United States

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Unknown Facility

Honolulu, Hawaii, 96814, United States

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Unknown Facility

Honolulu, Hawaii, 96817, United States

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Unknown Facility

Chicago, Illinois, 60637, United States

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Unknown Facility

Indianapolis, Indiana, 46202, United States

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Unknown Facility

Lutherville, Maryland, 21093, United States

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Unknown Facility

Detroit, Michigan, 48202, United States

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Newark, New Jersey, 07102, United States

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Unknown Facility

Albuquerque, New Mexico, 87131, United States

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Unknown Facility

New York, New York, 10021, United States

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Unknown Facility

Providence, Rhode Island, 02905, United States

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Unknown Facility

Nashville, Tennessee, 37211, United States

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Unknown Facility

Houston, Texas, 77030, United States

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Unknown Facility

Newport News, Virginia, 23602, United States

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Vancouver, Washington, 98664, United States

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Clichy, 92118, France

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Unknown Facility

Créteil, 94010, France

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Lille, 59037, France

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Unknown Facility

Marseille, 13285, France

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Unknown Facility

Montpellier, 34295, France

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Paris, 75651, France

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Berlin, 10969, Germany

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Unknown Facility

Berlin, 13353, Germany

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Unknown Facility

Frankfurt am Main, 60590, Germany

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Unknown Facility

Hamburg, 20099, Germany

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Unknown Facility

Hanover, 30625, Germany

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Unknown Facility

Kiel, 24146, Germany

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Unknown Facility

Leipzig, 04103, Germany

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Unknown Facility

Grafton, 1010, New Zealand

Location

Related Publications (1)

  • Tong X, Li L, Haines K, Najera I. Identification of the NS5B S282T resistant variant and two novel amino acid substitutions that affect replication capacity in hepatitis C virus-infected patients treated with mericitabine and danoprevir. Antimicrob Agents Chemother. 2014 Jun;58(6):3105-14. doi: 10.1128/AAC.02672-13. Epub 2014 Mar 17.

MeSH Terms

Conditions

Hepatitis C, Chronic

Interventions

danoprevirpeginterferon alfa-2aRibavirinRitonavir

Condition Hierarchy (Ancestors)

Hepatitis CBlood-Borne InfectionsCommunicable DiseasesInfectionsHepatitis, Viral, HumanVirus DiseasesFlaviviridae InfectionsRNA Virus InfectionsHepatitis, ChronicHepatitisLiver DiseasesDigestive System DiseasesChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

RibonucleosidesNucleosidesNucleic Acids, Nucleotides, and NucleosidesThiazolesSulfur CompoundsOrganic ChemicalsAzolesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Officials

  • Clinical Trials

    Hoffmann-La Roche

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 14, 2011

First Posted

January 17, 2011

Study Start

February 1, 2011

Primary Completion

October 1, 2012

Study Completion

October 1, 2012

Last Updated

November 2, 2016

Record last verified: 2016-11

Locations