NCT00869661

Brief Summary

This 6-arm study will assess the efficacy and safety of RO5024048 (R7128) in combination with the approved doses of Pegasys (180micrograms sc weekly) + Copegus (1000/1200mg po daily) (SOC), versus SOC in treatment-naive patients with chronic hepatitis C, genotype 1 and 4. The first 3 groups will receive 1) RO5024048 500mg bid + Pegasys + Copegus for 12 weeks, followed by SOC for 12 weeks; 2)RO5024048 1000mg bid + Pegasys + Copegus for 8 weeks, followed by SOC for 16 weeks; 3) RO5024048 1000mg bid + Pegasys + Copegus for 12 weeks, followed by SOC for 12 weeks. After 24 weeks, patients in these 3 groups who have achieved rapid viral response will stop treatment, and those who have not will receive SOC for a further 24 weeks. Group 4 will receive RO5024048 1000mg bid + Pegasys + Copegus for 12 weeks, followed by SOC for 36 weeks, and group 5 will receive SOC for 48 weeks. Group 6 provides retreatment on an open-label basis for patients of Group 5 who failed treatment. Patients will receive RO5024048 1000mg bid + Pegasys + Copegus for 24 weeks, followed by SOC for 24 weeks. The anticipated time on study treatment is 6-12 months.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
413

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Feb 2001

Longer than P75 for phase_2

Geographic Reach
9 countries

65 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

February 1, 2001

Completed
8.1 years until next milestone

First Submitted

Initial submission to the registry

March 25, 2009

Completed
1 day until next milestone

First Posted

Study publicly available on registry

March 26, 2009

Completed
2.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 1, 2012

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

February 1, 2012

Completed
Last Updated

November 2, 2016

Status Verified

November 1, 2016

Enrollment Period

11 years

First QC Date

March 25, 2009

Last Update Submit

November 1, 2016

Conditions

Outcome Measures

Primary Outcomes (1)

  • Sustained virologic response: Percentage of patients with undetectable Hepatitis C RNA level

    24 weeks after end of treatment

Secondary Outcomes (4)

  • Virologic response: Percentage of patients with undetectable Hepatitis C RNA level

    60 Weeks

  • Virologic response: Percentage of patients with undetectable Hepatitis C RNA level

    12 weeks post-treatment

  • Relapse rate: Percentage of patients who achieved a virologic response at the end of treatment but had detectable Hepatitis C RNA level at the last assessment post treatment

    72 weeks

  • Safety: Incidence of adverse events

    72 weeks

Study Arms (6)

Group 1

EXPERIMENTAL

RO5024048 500 mg bid + Pegasys + Copegus for 12 weeks, followed by SOC for 12 weeks. After 24 weeks, patients who have achieved rapid viral response will stop treatment, and those who have not will receive SOC for a further 24 weeks.

Drug: CopegusDrug: PegasysDrug: RO5024048

Group 2

EXPERIMENTAL

RO5024048 1000mg bid + Pegasys + Copegus for 8 weeks, followed by SOC for 16 weeks. After 24 weeks, patients who have achieved rapid viral response will stop treatment, and those who have not will receive SOC for a further 24 weeks.

Drug: CopegusDrug: PegasysDrug: RO5024048

Group 3

EXPERIMENTAL

RO5024048 1000mg bid + Pegasys + Copegus for 12 weeks, followed by SOC for 12 weeks. After 24 weeks, patients who have achieved rapid viral response will stop treatment, and those who have not will receive SOC for a further 24 weeks.

Drug: CopegusDrug: PegasysDrug: RO5024048

Group 4

EXPERIMENTAL

Group 4 will receive RO5024048 1000mg bid + Pegasys + Copegus for 12 weeks, followed by SOC for 36 weeks

Drug: CopegusDrug: PegasysDrug: RO5024048

Group 5

ACTIVE COMPARATOR

Group 5 will receive SOC for 48 weeks

Drug: CopegusDrug: Pegasys

Group 6

EXPERIMENTAL

Group 6 provides retreatment on an open-label basis for patients of Group 5 who failed treatment. Patients will receive RO5024048 1000mg bid + Pegasys + Copegus for 24 weeks, followed by SOC for 24 weeks.

Drug: CopegusDrug: PegasysDrug: RO5024048

Interventions

1000/1200mg po daily for 24 or 48 weeks

Group 1Group 2Group 3

180 micrograms sc weekly for 24 or 48 weeks

Group 1Group 2Group 3

1000mg bid for 24 weeks

Group 6

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Adult patients, 18-65 years of age
  • Chronic hepatitis C, genotype 1 or 4
  • Treatment-naive

You may not qualify if:

  • No previous treatment with any interferon- or ribavirin-based therapy
  • Other forms of liver disease
  • HIV infection

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (66)

Unknown Facility

Birmingham, Alabama, 35294, United States

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La Jolla, California, 92037-1030, United States

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Sacramento, California, 95817, United States

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San Diego, California, 92103-8465, United States

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San Francisco, California, 94115, United States

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Washington D.C., District of Columbia, 20037, United States

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Bradenton, Florida, 34209, United States

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Gainesville, Florida, 32610-0214, United States

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Marietta, Georgia, 30060, United States

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Chicago, Illinois, 60637, United States

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Lutherville, Maryland, 21093, United States

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Kansas City, Missouri, 64131, United States

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Newark, New Jersey, 07102, United States

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New York, New York, 10021, United States

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Hershey, Pennsylvania, 17033, United States

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Providence, Rhode Island, 02905, United States

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Columbia, South Carolina, 29204, United States

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Nashville, Tennessee, 37211, United States

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Houston, Texas, 77030, United States

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San Antonio, Texas, 78234, United States

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Richmond, Virginia, 23249, United States

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Sydney, New South Wales, 2050, Australia

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Greenslopes, Queensland, 4120, Australia

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Herston, Queensland, 4006, Australia

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Woolloongabba, Queensland, 4102, Australia

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Fitzroy, Victoria, 3065, Australia

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Melbourne, Victoria, 3004, Australia

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Nedlands, Western Australia, 6009, Australia

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Perth, Western Australia, 6001, Australia

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Vienna, 1090, Austria

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Calgary, Alberta, T2N 4Z6, Canada

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Edmonton, Alberta, T6G 2B7, Canada

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Vancouver, British Columbia, V5Z 1M9, Canada

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Vancouver, British Columbia, V6Z 2K5, Canada

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London, Ontario, N6A 5A5, Canada

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Toronto, Ontario, M5G 1L7, Canada

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Montreal, Quebec, H2X 3J4, Canada

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Créteil, 94010, France

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La Tronche, 38700, France

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Lille, 59037, France

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Nice, 06202, France

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Paris, 75651, France

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Paris, 75679, France

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Pessac, 33604, France

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Vandœuvre-lès-Nancy, 54511, France

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Berlin, 13353, Germany

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Frankfurt am Main, 60590, Germany

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Freiburg im Breisgau, 79106, Germany

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Hanover, 30625, Germany

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München, 81377, Germany

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Ulm, 89081, Germany

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Bologna, Emilia-Romagna, 40138, Italy

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Milan, Lombardy, 20121, Italy

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Turin, Piedmont, 10126, Italy

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Pisa, Tuscany, 56124, Italy

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Santurce, 00909, Puerto Rico

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Badalona, Barcelona, 08915, Spain

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Barcelona, Barcelona, 08003, Spain

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Barcelona, Barcelona, 08036, Spain

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Granada, Granada, 18003, Spain

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A Coruña, La Coruña, 15006, Spain

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Madrid, Madrid, 28222, Spain

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Seville, Sevilla, 41014, Spain

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Valencia, Valencia, 46014, Spain

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London, SE5 9RS, United Kingdom

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London, W1 1TF, United Kingdom

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Related Publications (1)

  • Tong X, Le Pogam S, Li L, Haines K, Piso K, Baronas V, Yan JM, So SS, Klumpp K, Najera I. In vivo emergence of a novel mutant L159F/L320F in the NS5B polymerase confers low-level resistance to the HCV polymerase inhibitors mericitabine and sofosbuvir. J Infect Dis. 2014 Mar 1;209(5):668-75. doi: 10.1093/infdis/jit562. Epub 2013 Oct 23.

MeSH Terms

Conditions

Hepatitis C, Chronic

Interventions

Ribavirinpeginterferon alfa-2a

Condition Hierarchy (Ancestors)

Hepatitis CBlood-Borne InfectionsCommunicable DiseasesInfectionsHepatitis, Viral, HumanVirus DiseasesFlaviviridae InfectionsRNA Virus InfectionsHepatitis, ChronicHepatitisLiver DiseasesDigestive System DiseasesChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

RibonucleosidesNucleosidesNucleic Acids, Nucleotides, and Nucleosides

Study Officials

  • Clinical Trials

    Hoffmann-La Roche

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 25, 2009

First Posted

March 26, 2009

Study Start

February 1, 2001

Primary Completion

February 1, 2012

Study Completion

February 1, 2012

Last Updated

November 2, 2016

Record last verified: 2016-11

Locations