NCT00864175

Brief Summary

This is a single arm, modified dose escalation, open label trial with the objectives of: (1) Determining a safe optimal dose of INCB007839 in combination with trastuzumab and docetaxel (2) Determining clinical efficacy and safety of INCB007839 in combination with trastuzumab and docetaxel.

Trial Health

57
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
68

participants targeted

Target at P50-P75 for phase_1 breast-cancer

Timeline
Completed

Started Jul 2007

Typical duration for phase_1 breast-cancer

Geographic Reach
1 country

12 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

July 1, 2007

Completed
1.6 years until next milestone

First Submitted

Initial submission to the registry

January 26, 2009

Completed
2 months until next milestone

First Posted

Study publicly available on registry

March 18, 2009

Completed
2.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 1, 2011

Completed
4 months until next milestone

Study Completion

Last participant's last visit for all outcomes

October 1, 2011

Completed
Last Updated

January 18, 2018

Status Verified

January 1, 2018

Enrollment Period

3.9 years

First QC Date

January 26, 2009

Last Update Submit

January 16, 2018

Conditions

Outcome Measures

Primary Outcomes (1)

  • Overall response rate (complete + partial response) using RECIST (Response Evaluation Criteria in Solid Tumor) criteria

    Day 1 of each completed subsequent 21-day treatment cycle and the End of Study Visit.

Secondary Outcomes (1)

  • To determine the plasma pharmacokinetic (PK) profile of INCB007839 and trastuzumab when given in combination

    Monthly

Study Arms (4)

Treatment A - INCB007839 and Trastuzumab

EXPERIMENTAL

INCB007839 100 mg BID and trastuzumab In Cycle 1, trastuzumab will be administered at a loading dose of 8 mg/kg as a 90 minute intravenous infusion on Day 8. In all subsequent 21-day cycles, trastuzumab will be administered at 6 mg/kg as a 90 minute intravenous infusion on Day 1.

Drug: INCB007839Drug: trastuzumab

Treatment B - INCB007839 and Trastuzumab

EXPERIMENTAL

INCB007839 200 mg BID and trastuzumab In Cycle 1, trastuzumab will be administered at a loading dose of 8 mg/kg as a 90 minute intravenous infusion on Day 8. In all subsequent 21-day cycles, trastuzumab will be administered at 6 mg/kg as a 90 minute intravenous infusion on Day 1.

Drug: INCB007839Drug: trastuzumab

Treatment C - INCB007839 and Trastuzumab

EXPERIMENTAL

INCB007839 300 mg BID and trastuzumab In Cycle 1, trastuzumab will be administered at a loading dose of 8 mg/kg as a 90 minute intravenous infusion on Day 8. In all subsequent 21-day cycles, trastuzumab will be administered at 6 mg/kg as a 90 minute intravenous infusion on Day 1.

Drug: INCB007839Drug: trastuzumab

Treatment D - INCB007839 and Docetaxel

EXPERIMENTAL

INCB007839 300mg BID with docetaxel

Drug: INCB007839Drug: Docetaxel

Interventions

100 mg BID

Treatment A - INCB007839 and Trastuzumab

trastuzumab will be administered at a loading dose of 8 mg/kg as a 90 minute intravenous infusion on Day 8. In all subsequent 21-day cycles, trastuzumab will be administered at 6 mg/kg as a 90 minute intravenous infusion on Day 1.

Treatment A - INCB007839 and TrastuzumabTreatment B - INCB007839 and TrastuzumabTreatment C - INCB007839 and Trastuzumab
Treatment D - INCB007839 and Docetaxel

Eligibility Criteria

Age18 Years+
Sexfemale
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Histologically or cytologically confirmed metastatic breast carcinoma that is HER2 positive
  • Measurable disease as defined by the RECIST criteria
  • Life expectancy greater than or equal to 6 months
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1

You may not qualify if:

  • Received any anticancer medications in the 28 days prior to enrollment into this study
  • Received any anticancer medications for cancers other than breast cancer within 6 months prior to enrollment in this study.
  • History of deep venous thrombosis within the last year
  • Contraindication to low dose warfarin therapy
  • Clinically significant cardiomyopathy
  • Prior treatment with INCB007839 or trastuzumab or lapatinib

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (12)

Unknown Facility

Visakhapatnam, Andhra Pradesh, India

Location

Unknown Facility

New Delhi, Ansari Nagar, India

Location

Unknown Facility

Mangalore, Attavar, India

Location

Unknown Facility

Bangalore, Karnataka, India

Location

Unknown Facility

Hyderabaad, Punjagutta, India

Location

Unknown Facility

Bangalore, Ram Nagar, India

Location

Unknown Facility

Delhi, Rohini, India

Location

Unknown Facility

Delhi, Vasundhara Enclave, India

Location

Unknown Facility

Bhopal, India

Location

Unknown Facility

Kolkata, India

Location

Unknown Facility

Nashik, India

Location

Unknown Facility

Pune, India

Location

MeSH Terms

Conditions

Breast Neoplasms

Interventions

TrastuzumabDocetaxel

Condition Hierarchy (Ancestors)

Neoplasms by SiteNeoplasmsBreast DiseasesSkin DiseasesSkin and Connective Tissue Diseases

Intervention Hierarchy (Ancestors)

Antibodies, Monoclonal, HumanizedAntibodies, MonoclonalAntibodiesImmunoglobulinsImmunoproteinsBlood ProteinsProteinsAmino Acids, Peptides, and ProteinsSerum GlobulinsGlobulinsTaxoidsCyclodecanesCycloparaffinsHydrocarbons, AlicyclicHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsDiterpenesTerpenes

Study Officials

  • Bijyoyesh Mookerjee, MD

    Incyte Corporation

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 26, 2009

First Posted

March 18, 2009

Study Start

July 1, 2007

Primary Completion

June 1, 2011

Study Completion

October 1, 2011

Last Updated

January 18, 2018

Record last verified: 2018-01

Locations