NCT00688688

Brief Summary

The study is intended to test the safety, tolerability, efficacy of two doses of long term once daily (qd) treatment of Mirabegron in patients with symptoms of overactive bladder and secondly to compare these with active comparator.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
2,792

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Apr 2008

Geographic Reach
28 countries

303 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

April 25, 2008

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

May 29, 2008

Completed
5 days until next milestone

First Posted

Study publicly available on registry

June 3, 2008

Completed
1.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 6, 2010

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 6, 2010

Completed
2.5 years until next milestone

Results Posted

Study results publicly available

October 19, 2012

Completed
Last Updated

November 20, 2024

Status Verified

October 1, 2024

Enrollment Period

2 years

First QC Date

May 29, 2008

Results QC Date

July 23, 2012

Last Update Submit

October 29, 2024

Conditions

Keywords

FrequencyOveractive BladderUrgencyUrinary urge incontinenceUrinary incontinenceMicturition

Outcome Measures

Primary Outcomes (1)

  • Number of Participants With and Severity of Treatment-emergent Adverse Events (TEAEs)

    An adverse event (AE) was defined as any untoward medical occurrence in a patient administered a study drug and which did not necessarily have a causal relationship with the treatment. The investigator assessed the severity of each AE, including abnormal laboratory values, as follows: Mild: No disruption of normal daily activities; Moderate: Affected normal daily activities; Severe: Inability to perform daily activities.

    From the first dose of double-blind study drug up until 30 days after the last dose of study drug, up to 13 months.

Secondary Outcomes (27)

  • Change From Baseline to Months 1, 3, 6, 9, 12 and Final Visit in Mean Number of Micturitions Per 24 Hours

    Baseline and Months 1, 3, 6, 9 and 12

  • Change From Baseline to Months 1, 3, 6, 9, 12 and Final Visit in Mean Number of Incontinence Episodes Per 24 Hours

    Baseline and Months 1, 3, 6, 9 and 12

  • Change From Baseline to Months 1, 3, 6, 9, 12 and Final Visit in Mean Volume Voided Per Micturition

    Baseline and Months 1, 3, 6, 9 and 12

  • Change From Baseline to Months 1, 3, 6, 9, 12 and Final Visit in Mean Number of Urgency Incontinence Episodes Per 24 Hours

    Baseline and Months 1, 3, 6, 9 and 12

  • Change From Baseline to Months 1, 3, 6, 9, 12 and Final Visit in Mean Number of Urgency Episodes (Grade 3 and/or 4) Per 24 Hours

    Baseline and Months 1, 3, 6, 9 and 12

  • +22 more secondary outcomes

Study Arms (3)

Mirabegron 50 mg

EXPERIMENTAL

Participants received mirabegron 50 mg tablets and matching tolterodine extended release (ER) placebo capsules orally once a day for 12 months.

Drug: MirabegronDrug: Placebo to Tolterodine

Mirabegron 100 mg

EXPERIMENTAL

Participants received mirabegron 100 mg tablets and matching tolterodine ER placebo capsules orally once a day for 12 months.

Drug: MirabegronDrug: Placebo to Tolterodine

Tolterodine ER 4 mg

ACTIVE COMPARATOR

Participants received tolterodine ER 4 mg capsules and matching mirabegron placebo tablets orally once a day for 12 months.

Drug: TolterodineDrug: Placebo to Mirabegron

Interventions

Tablets

Also known as: Myrbetriq, YM178
Mirabegron 100 mgMirabegron 50 mg

Extended release capsules

Tolterodine ER 4 mg

Matching mirabegron placebo tablets.

Tolterodine ER 4 mg

Matching tolterodine placebo capsules.

Mirabegron 100 mgMirabegron 50 mg

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Patient is willing and able to complete the micturition diary and questionnaires correctly
  • Patient has symptoms of overactive bladder for ≥ 3 months
  • Patient experiences frequency of micturition on average ≥ 8 times per 24-hour period during the 3-day micturition diary period
  • Patient must experience at least 3 episodes of urgency (grade 3 or 4) with or without incontinence, during the 3-day micturition diary period

You may not qualify if:

  • Patient is breastfeeding, pregnant, intends to become pregnant during the study, or of childbearing potential, sexually active and not practicing a highly reliable method of birth control
  • Patient has significant stress incontinence or mixed stress/urge incontinence where stress is the predominant factor
  • Patient has an indwelling catheter or practices intermittent self-catheterization
  • Patient has diabetic neuropathy
  • Patient has evidence of a symptomatic urinary tract infection, chronic inflammation such as interstitial cystitis, bladder stones, previous pelvic radiation therapy or previous or current malignant disease of the pelvic organs
  • Patient receives non-drug treatment including electro-stimulation therapy
  • Patient has severe hypertension
  • Patient has a known or suspected hypersensitivity to tolterodine, other anticholinergics, YM178, other beta-adrenoreceptor (ß-AR) agonists, or lactose or any of the other inactive ingredients
  • Patient has been treated with any investigational drug or device within 30 days (90 days in the UK for all clinical studies except 178-CL-046)
  • Patient had an average total daily urine volume \> 3000 mL as recorded in the 3-day micturition diary period
  • Patient has serum creatinine \>150 umol/L, aspartate aminotransferase (AST) and/or alanine aminotransferase (ALT) \> 2x upper limit of normal range (ULN), or gamma-glutamyl transpeptidase (γ-GT) \> 3x ULN
  • Patient has a clinically significant abnormal electrocardiogram (ECG)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (308)

Unknown Facility

Homewood, Alabama, 35209, United States

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Huntsville, Alabama, 35801, United States

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Mobile, Alabama, 36608, United States

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Montgomery, Alabama, 36117, United States

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Anchorage, Alaska, 99508, United States

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Phoenix, Arizona, 85051, United States

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Tucson, Arizona, 85712, United States

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Tucson, Arizona, 85741, United States

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Atherton, California, 94027, United States

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Beverly Hills, California, 90211, United States

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Buena Park, California, 90620, United States

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Fresno, California, 93720, United States

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La Mesa, California, 91942, United States

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Mission Hills, California, 91345, United States

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Newport Beach, California, 92660, United States

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Orange, California, 92869, United States

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Sacramento, California, 95831, United States

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San Bernardino, California, 92404, United States

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San Diego, California, 92108, United States

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San Diego, California, 92120, United States

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Tarzana, California, 91356, United States

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Torrance, California, 90505, United States

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Aurora, Colorado, 80012, United States

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Denver, Colorado, 80211, United States

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Denver, Colorado, 80218, United States

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Englewood, Colorado, 80112, United States

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New Britain, Connecticut, 06052, United States

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Waterbury, Connecticut, 06708, United States

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Aventura, Florida, 33180, United States

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Clearwater, Florida, 33756, United States

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Clearwater, Florida, 33761, United States

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Fort Myers, Florida, 33916, United States

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Miami, Florida, 33136, United States

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Ocala, Florida, 34471, United States

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Orlando, Florida, 32803, United States

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Pembroke Pines, Florida, 33024, United States

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Pembroke Pines, Florida, 33027, United States

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Sarasota, Florida, 34237, United States

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Tallahassee, Florida, 32308, United States

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Tampa, Florida, 33606, United States

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Wellington, Florida, 33414, United States

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West Palm Beach, Florida, 33407, United States

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Atlanta, Georgia, 30328, United States

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Decatur, Georgia, 30034, United States

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Marietta, Georgia, 30060, United States

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Roswell, Georgia, 30076, United States

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Coeur d'Alene, Idaho, 83814, United States

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Idaho Falls, Idaho, 83404, United States

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Melrose Park, Illinois, 60160, United States

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Fort Wayne, Indiana, 46825, United States

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Jeffersonville, Indiana, 47130, United States

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Newburgh, Indiana, 47630, United States

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Des Moines, Iowa, 50309, United States

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Wichita, Kansas, 57207, United States

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Greenbelt, Maryland, 20770, United States

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Watertown, Massachusetts, 02472, United States

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North Kansas City, Missouri, 64116, United States

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Billings, Montana, 59102, United States

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Lincoln, Nebraska, 68516, United States

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Omaha, Nebraska, 68114, United States

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Las Vegas, Nevada, 89148, United States

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New Brunswick, New Jersey, 08901, United States

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West Orange, New Jersey, 07052, United States

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Albuquerque, New Mexico, 87109, United States

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Albany, New York, 12205, United States

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Albany, New York, 12208, United States

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Endwell, New York, 13760, United States

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Garden City, New York, 11530, United States

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Kingston, New York, 12401, United States

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New York, New York, 10016, United States

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Poughkeepsie, New York, 12601, United States

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Cary, North Carolina, 27518, United States

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Charlotte, North Carolina, 28209, United States

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Concord, North Carolina, 28025, United States

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Wilmington, North Carolina, 28401, United States

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Winston-Salem, North Carolina, 27103, United States

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Fargo, North Dakota, 58104, United States

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Cincinnati, Ohio, 45212, United States

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Cleveland, Ohio, 44122, United States

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Columbus, Ohio, 43214, United States

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Lyndhurst, Ohio, 44124, United States

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Wadsworth, Ohio, 44281, United States

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Bethany, Oklahoma, 73008, United States

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Edmond, Oklahoma, 73008, United States

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Edmond, Oklahoma, 73034, United States

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Bala-Cynwyd, Pennsylvania, 19004, United States

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Jenkintown, Pennsylvania, 19046, United States

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Lancaster, Pennsylvania, 17604, United States

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Reading, Pennsylvania, 19611, United States

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Uniontown, Pennsylvania, 15401, United States

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Warwick, Rhode Island, 02886, United States

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Greer, South Carolina, 29650, United States

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Mt. Pleasant, South Carolina, 29464, United States

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Simpsonville, South Carolina, 29681, United States

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Bristol, Tennessee, 37620, United States

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Arlington, Texas, 76017, United States

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Austin, Texas, 78759, United States

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Corpus Christi, Texas, 78414, United States

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Dallas, Texas, 75231, United States

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Houston, Texas, 77024, United States

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Salt Lake City, Utah, 84107, United States

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Virginia Beach, Virginia, 23454, United States

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Mountlake Terrace, Washington, 98043, United States

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Seattle, Washington, 98166, United States

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Spokane, Washington, 99204, United States

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Tacoma, Washington, 98405, United States

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Woolloongabba, Australia

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Graz, 8036, Austria

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Innsbruck, 6020, Austria

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Linz, 4020, Austria

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Minsk, 220036, Belarus

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Minsk, 223041, Belarus

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Antwerp, 2020, Belgium

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Antwerp, 2030, Belgium

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Edegem, 2650, Belgium

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Ghent, 9000, Belgium

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Kortrijk, 8500, Belgium

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Leper, 8900, Belgium

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Leuven, 3000, Belgium

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Liège, 4000, Belgium

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Sint-Truiden, 3800, Belgium

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Calgary, Alberta, T2V 4R6, Canada

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Edmonton, Alberta, T5H 3V9, Canada

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Surrey, British Columbia, V3V 1N1, Canada

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Victoria, British Columbia, V8T 5G1, Canada

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Victoria, British Columbia, V8V 3N1, Canada

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Saint John, New Brunswick, E2L 3J8, Canada

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Dartmouth, Nova Scotia, B2W 2S7, Canada

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Kentville, Nova Scotia, B4N 4K9, Canada

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Barrie, Ontario, L4M 7G1, Canada

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Brampton, Ontario, L6T 4S5, Canada

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Kitchener, Ontario, N2N 2B9, Canada

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Markham, Ontario, L6B 1A1, Canada

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Newmarket, Ontario, L3X 1W1, Canada

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North Bay, Ontario, P1B 7K8, Canada

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Oshawa, Ontario, L1H 1B9, Canada

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Saint Denis, Ontario, H2X 3J4, Canada

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Thunder Bay, Ontario, P7E 6E7, Canada

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Toronto, Ontario, M4N 3M5, Canada

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Toronto, Ontario, M5T 2S8, Canada

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Granby, Quebec, J2G 8Z9, Canada

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Montreal, Quebec, H3A 1A1, Canada

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Point Claire, Quebec, H9R 4S3, Canada

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Montreal, Canada

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Brno, 60200, Czechia

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Mělník, 27601, Czechia

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Olomouc, 77200, Czechia

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Ostrava-Poruba, 70853, Czechia

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Pilsen, 30599, Czechia

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Prague, 12851, Czechia

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Prague, 14056, Czechia

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Prague, 18081, Czechia

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Štětí, 41108, Czechia

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Ústí nad Labem, 40001, Czechia

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Aalborg, 9100, Denmark

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Aarhus, 8200, Denmark

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Glostrup Municipality, 2600, Denmark

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Roskilde, Denmark

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Helsinki, 00029, Finland

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Oulu, 90220, Finland

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Tampere, 33521, Finland

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Turku, 20100, Finland

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Paris, Cedex 10, 75020, France

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Colmar, 68024, France

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Marseille, 13274, France

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Mulhouse, 68070, France

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Nîmes, 30029, France

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Orléans, 45067, France

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Paris-Cedex12, 75571, France

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Saint-Priest-en-Jarez, 42055, France

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Strasbourg, 67000, France

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Toulouse, 31059, France

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Aichach, 86551, Germany

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Bad Ems, 56130, Germany

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Bautzen, 02625, Germany

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Berlin, 13347, Germany

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Duisburg, 47051, Germany

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Eisleben Lutherstadt, 06295, Germany

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Frankfurt, 65933, Germany

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Ganderkesee, 27777, Germany

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Hagenow, 19230, Germany

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Halle, 06132, Germany

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Hamburg, 20253, Germany

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Henningsdorf, 16761, Germany

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Hettstedt, 06333, Germany

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Kiel, Germany

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Koblenz, 56068, Germany

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Leipzig, 04105, Germany

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Muenchen-Bogenhausen, 81925, Germany

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Munich, Germany

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Neustadt in Sachsen, 01844, Germany

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Oranienburg, 16151, Germany

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Radebeul, 01445, Germany

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Sangerhausen, 06526, Germany

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Trier, 54290, Germany

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Uetersen, 25436, Germany

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Budapest, 1047, Hungary

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Budapest, 1076, Hungary

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Nyíregyháza, 4400, Hungary

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Sopron, Hungary

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Szeged, 6725, Hungary

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Szekszárd, 7100, Hungary

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Székesfehérvár, 8000, Hungary

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Tatabánya, 2800, Hungary

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Reykjavik, 101, Iceland

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Dublin, Ireland

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Mullingar, Ireland

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Bari, 70124, Italy

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Catanzaro, 88100, Italy

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Genoa, 16128, Italy

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Latina, 04100, Italy

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Milan, 20142, Italy

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Modena, 41100, Italy

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Naples, 80131, Italy

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Perugia, 06122, Italy

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Treviglio, 24047, Italy

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Varese, 21100, Italy

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Liepāja, Latvia

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Riga, Latvia

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Kaunas, Lithuania

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Amsterdam, 1105 AZ, Netherlands

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Apeldoorn, 7334 DZ, Netherlands

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Eindhoven, 5623 EJ, Netherlands

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Enschede, 7511 JX, Netherlands

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Leiden, 2334 CK, Netherlands

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Nijmegen, 6532 SZ, Netherlands

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Sneek, 8600 BA, Netherlands

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Tilburg, 5022 GC, Netherlands

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Winterswijk, 7101 BN, Netherlands

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Bergen, 5021, Norway

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Drammen, 3016, Norway

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Hamar, 2317, Norway

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Oslo, 0257, Norway

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Tønsberg, 3103, Norway

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Bialystok, 15-278, Poland

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Lodz, 93-338, Poland

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Lodz, 93-513, Poland

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Lublin, 20-954, Poland

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Warsaw, 00-846, Poland

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Warsaw, 02-005, Poland

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Warsaw, 02-507, Poland

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Warsaw, Poland

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Wroclaw, 50-556, Poland

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Amadora, 2700, Portugal

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Porto, 4099-005, Portugal

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Tomar, 2304-909, Portugal

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Bucharest, 22328, Romania

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Bucharest, Romania

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Lasi, Romania

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Oradea, Romania

Location

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Moscow, 101000, Russia

Location

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Moscow, 105425, Russia

Location

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Moscow, 111020, Russia

Location

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Moscow, 111123, Russia

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Moscow, 117049, Russia

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Moscow, 117815, Russia

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Moscow, 119435, Russia

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Moscow, 123836, Russia

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Moscow, 125206, Russia

Location

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Saint Petersburg, 115516, Russia

Location

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Saint Petersburg, 197089, Russia

Location

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Saint Petersburg, 198013, Russia

Location

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Martin, 03659, Slovakia

Location

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Poprad, 05801, Slovakia

Location

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Skalica, 90982, Slovakia

Location

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Trenčín, 91101, Slovakia

Location

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Žilina, 01207, Slovakia

Location

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Hatfield, South Africa

Location

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Lyttelton, South Africa

Location

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Paarl, South Africa

Location

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Pietermaritzburg, South Africa

Location

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Roodepoort, South Africa

Location

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Barcelona, 08020, Spain

Location

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Barcelona, 08036, Spain

Location

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Bilbao, 48013, Spain

Location

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Getafe, 28905, Spain

Location

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Madrid, 28016, Spain

Location

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Madrid, 28046, Spain

Location

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Mataró, 8304, Spain

Location

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Miranda de Ebro, 09200, Spain

Location

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Seville, 41013, Spain

Location

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Toledo, 45071, Spain

Location

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Valencia, 46010, Spain

Location

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Huddinge, 75185, Sweden

Location

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Örebro, 70185, Sweden

Location

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Skövde, 54130, Sweden

Location

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Sonkoping, 11883, Sweden

Location

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Stockholm, 14186, Sweden

Location

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Stockholm, 17176, Sweden

Location

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Stockholm, 18288, Sweden

Location

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Umeå, 90185, Sweden

Location

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Frauenfeld, 8501, Switzerland

Location

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Lucerne, 6000, Switzerland

Location

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Kiev, 01023, Ukraine

Location

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Kiev, 04053, Ukraine

Location

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Bristol, B15 2TG, United Kingdom

Location

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Chorley, PR7 7NA, United Kingdom

Location

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Croydon, CR7 7YE, United Kingdom

Location

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Liverpool, L22 OLG, United Kingdom

Location

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London, SE5 9RS, United Kingdom

Location

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London, W2 2YP, United Kingdom

Location

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Manchester, M15 6SX, United Kingdom

Location

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Newcastle upon Tyne, NE7 7DN, United Kingdom

Location

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Northwood, HA6 2RN, United Kingdom

Location

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Reading, RG1 5AN, United Kingdom

Location

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Reading, RG2 7AG, United Kingdom

Location

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Sheffield, S10 2JF, United Kingdom

Location

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Swansea, SA6 6NL, United Kingdom

Location

Related Publications (1)

  • Chapple CR, Kaplan SA, Mitcheson D, Klecka J, Cummings J, Drogendijk T, Dorrepaal C, Martin N. Randomized double-blind, active-controlled phase 3 study to assess 12-month safety and efficacy of mirabegron, a beta(3)-adrenoceptor agonist, in overactive bladder. Eur Urol. 2013 Feb;63(2):296-305. doi: 10.1016/j.eururo.2012.10.048. Epub 2012 Nov 6.

    PMID: 23195283BACKGROUND

Related Links

MeSH Terms

Conditions

Urinary Bladder, OveractiveUrinary Incontinence, UrgeUrinary Incontinence

Interventions

mirabegronTolterodine Tartrate

Condition Hierarchy (Ancestors)

Urinary Bladder DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesLower Urinary Tract SymptomsUrological ManifestationsSigns and SymptomsPathological Conditions, Signs and SymptomsUrination Disorders

Intervention Hierarchy (Ancestors)

PhenylpropanolaminePropanolaminesAmino AlcoholsAlcoholsOrganic ChemicalsPropanolsAminesBenzhydryl CompoundsBenzene DerivativesHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsCresolsPhenols

Limitations and Caveats

Company makes no warranties or representations of any kind as to the posting, expressed or implied, including warranties of merchantability and fitness for a particular purpose, and shall not be liable for any damages.

Results Point of Contact

Title
Medical Director, Global Medical Sciences
Organization
Astellas Pharma Global Development, Inc.

Study Officials

  • Central Contact

    Astellas Pharma Europe B.V.

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 29, 2008

First Posted

June 3, 2008

Study Start

April 25, 2008

Primary Completion

May 6, 2010

Study Completion

May 6, 2010

Last Updated

November 20, 2024

Results First Posted

October 19, 2012

Record last verified: 2024-10

Data Sharing

IPD Sharing
Will share

Access to anonymized individual participant level data collected during the study, in addition to study-related supporting documentation, is planned for studies conducted with approved product indications and formulations, as well as products terminated during development. Studies conducted with product indications or formulations that remain active in development are assessed after study completion to determine if Individual Participant Data can be shared. Further details on Astellas' data sharing policy can be found at https://www.clinicaltrials.astellas.com/transparency/.

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
Access to participant level data is offered to researchers after publication of the primary manuscript (if applicable) and is available as long as Astellas has legal authority to provide the data.
Access Criteria
Researchers must submit a proposal to conduct a scientifically relevant analysis of the study data. The research proposal is reviewed by an Independent Research Panel. If the proposal is approved, access to the study data is provided in a secure data sharing environment after receipt of a signed Data Sharing Agreement.
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