NCT07030257

Brief Summary

The goal of this clinical trial is to learn if an investigational drug CP-383 works to treat advanced cancer. It will also learn about the safety of CP-383. The main questions if aims to answer are:

  • Does CP-383 slow or stop the growth of cancer in patients with advanced cancer
  • What medical problems do participants have when taking CP-383 Researchers will test CP-383 in all kinds of cancers at various dose levels to determine what the best dose is to study further. Researchers will also see if certain cancers that have gene mutations respond better to CP-383 Participants will:
  • Take CP-383 every day by mouth until the researcher learns whether CP-383 is helping slow or reduce the cancer growth
  • Visit the clinic weekly for the first 6 weeks for checkups and tests
  • Visit the clinic every 3 weeks thereafter for checkups and tests

Trial Health

77
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
150

participants targeted

Target at P75+ for phase_1

Timeline
34mo left

Started Aug 2025

Typical duration for phase_1

Geographic Reach
1 country

13 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress20%
Aug 2025Feb 2029

First Submitted

Initial submission to the registry

May 20, 2025

Completed
1 month until next milestone

First Posted

Study publicly available on registry

June 22, 2025

Completed
2 months until next milestone

Study Start

First participant enrolled

August 27, 2025

Completed
3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 15, 2028

Expected
6 months until next milestone

Study Completion

Last participant's last visit for all outcomes

February 1, 2029

Last Updated

February 18, 2026

Status Verified

January 1, 2026

Enrollment Period

3 years

First QC Date

May 20, 2025

Last Update Submit

February 17, 2026

Conditions

Keywords

Phase 1Dose EscalationDose ExpansionLoss of FunctionFAT1P300

Outcome Measures

Primary Outcomes (2)

  • Part 1: Determine the maximum tolerated dose (MTD)

    Determine the MTD of CP-383 in subjects with advanced solid tumors

    21 days

  • Part 2: Evaluate the efficacy of CP-383 at the recommended phase 2 dose in selected tumor types

    Objective response rate assessed by the investigator according to RECIST

    From enrollment through study completion, an average of 1 year

Secondary Outcomes (9)

  • Part 1: Determine the pharmacokinetics parameters of CP-383

    From enrollment through study completion, an average of 1 year

  • Part 1: Determine the pharmacokinetics parameters of CP-383

    From enrollment through study completion, an average of 1 year

  • Part 1: Determine the pharmacokinetics parameters of CP-383

    From enrollment through study completion, an average of 1 year

  • Part 1: Assess safety and tolerability of CP-383 in participants with advanced solid tumors

    From enrollment through study completion, an average of 1 year

  • Part 2: Evaluate safety and tolerability of CP-383 at the recommended Phase 2 dose in selected tumor types

    From enrollment through study completion, an average of 1 year

  • +4 more secondary outcomes

Study Arms (10)

Dose Level 1

EXPERIMENTAL

CP-383, single daily oral capsule, 0.8 mg

Drug: CP-383

Dose Level 2

EXPERIMENTAL

CP-383, single daily oral capsule, 1.6 mg

Drug: CP-383

Dose Level 3

EXPERIMENTAL

CP-383, single daily oral capsule, 3.0 mg

Drug: CP-383

Dose Level 4

EXPERIMENTAL

CP-383, single daily oral capsule, 5.0 mg

Drug: CP-383

Dose Level 5

EXPERIMENTAL

CP-383, single daily oral capsule, 8.0 mg

Drug: CP-383

Dose Level 6

EXPERIMENTAL

CP-383, single daily oral capsule, 12 mg

Drug: CP-383

Expansion Arm 1

EXPERIMENTAL

Expansion in selected tumor type at recommended Phase 2 Dose of CP-383

Drug: CP-383

Expansion Arm 2

EXPERIMENTAL

Expansion in selected tumor type at recommended Phase 2 Dose of CP-383

Drug: CP-383

Expansion Arm 3

EXPERIMENTAL

Expansion in selected tumor type at recommended Phase 2 Dose of CP-383

Drug: CP-383

Expansion Arm 4

EXPERIMENTAL

Expansion in selected tumor type at recommended Phase 2 Dose of CP-383

Drug: CP-383

Interventions

CP-383DRUG

Novel anti-cancer agent inhibiting pyrimidine synthesis in cancer cells

Dose Level 1Dose Level 2Dose Level 3Dose Level 4Dose Level 5Dose Level 6Expansion Arm 1Expansion Arm 2Expansion Arm 3Expansion Arm 4

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Measurable or non measurable cancer that the research can assess for changes
  • Not eligible or able to take existing standard therapies for cancer
  • Availability of a part of a tumor for laboratory testing or willing to have a safe biopsy taken from a tumor
  • Diagnosed with locally advanced, recurrent or metastatic incurable disease
  • Part 1: any solid tumor (with the exception of brain cancer) that has progressed, standard therapy is no longer or has not helped the cancer, or is too toxic and for whom a clinical trial is an option for continued treatment
  • Part 1: specific advanced, metastatic tumor types will also be enrolled: colorectal cancer, small cell lung cancer, head and neck cancer, non-small cell lung cancer, pancreatic cancer, bladder cancer - some of these will have a specific gene mutation in the cancer
  • Part 1: selected solid tumor cancer types (with the exception of brain cancers) that have a specific gene mutation in the cancer
  • Part 2: specific advanced, metastatic tumor types will also be enrolled: colorectal cancer, small cell lung cancer, head and neck cancer - some of these will have a specific gene mutation in the cancer
  • \_ Part 2: selected solid tumor cancer types (with the exception of brain cancers) that have a specific gene mutation in the cancer
  • Adequate blood and urine lab tests
  • Women and men of childbearing potential with adequate contraception
  • Provides written informed consent
  • Willing to comply with the requirements of the protocol

You may not qualify if:

  • Inability to swallow pills
  • Known history of HIV, HCV, HBV unless cured, controlled with undetectable viral load
  • Active tumor in the brain
  • Clinically significant liver disease
  • Significant gastrointestinal diseases
  • History of other cancer within past 5 years with certain exceptions for cancers that are likely cured
  • Significant cardiac disease
  • Other diseases that are not well controlled that could make taking the drug unsafe
  • pregnant or lactating females
  • Exposure to certain anti-cancer or other drugs within a certain period before the start of study drug

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (13)

Sarah Cannon Research Institute at HealthONE

Denver, Colorado, 80218, United States

RECRUITING

Florida Cancer Specialists-Lake Nona

Orlando, Florida, 32827, United States

RECRUITING

START Midwest

Grand Rapids, Michigan, 49546, United States

RECRUITING

Washington University

St Louis, Missouri, 63110, United States

RECRUITING

Nebraska Cancer Specialists

Omaha, Nebraska, 68130, United States

RECRUITING

Carolina BioOncology Institute

Huntersville, North Carolina, 28078, United States

RECRUITING

Cleveland Clinic

Cleveland, Ohio, 44195, United States

RECRUITING

Taylor Cancer Research Center

Maumee, Ohio, 43537, United States

RECRUITING

University of Pennsylvania

Philadelphia, Pennsylvania, 19104, United States

RECRUITING

NEXT Oncology - Dallas

Dallas, Texas, 75039, United States

RECRUITING

START San Antonio

San Antonio, Texas, 78229, United States

RECRUITING

START Mountain Region

West Valley City, Utah, 84119, United States

RECRUITING

NEXT Virginia

Fairfax, Virginia, 22031, United States

RECRUITING

MeSH Terms

Conditions

Colorectal NeoplasmsSmall Cell Lung CarcinomaSquamous Cell Carcinoma of Head and NeckUrinary Bladder NeoplasmsCarcinoma, Non-Small-Cell LungPancreatic NeoplasmsNeoplasm Metastasis

Condition Hierarchy (Ancestors)

Intestinal NeoplasmsGastrointestinal NeoplasmsDigestive System NeoplasmsNeoplasms by SiteNeoplasmsDigestive System DiseasesGastrointestinal DiseasesColonic DiseasesIntestinal DiseasesRectal DiseasesCarcinoma, BronchogenicBronchial NeoplasmsLung NeoplasmsRespiratory Tract NeoplasmsThoracic NeoplasmsLung DiseasesRespiratory Tract DiseasesCarcinoma, Squamous CellCarcinomaNeoplasms, Glandular and EpithelialNeoplasms by Histologic TypeHead and Neck NeoplasmsUrologic NeoplasmsUrogenital NeoplasmsFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesUrinary Bladder DiseasesUrologic DiseasesMale Urogenital DiseasesEndocrine Gland NeoplasmsPancreatic DiseasesEndocrine System DiseasesNeoplastic ProcessesPathologic ProcessesPathological Conditions, Signs and Symptoms

Central Study Contacts

Tasca Therapeutics

CONTACT

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 20, 2025

First Posted

June 22, 2025

Study Start

August 27, 2025

Primary Completion (Estimated)

August 15, 2028

Study Completion (Estimated)

February 1, 2029

Last Updated

February 18, 2026

Record last verified: 2026-01

Locations