NCT06470282

Brief Summary

This phase Ib/II trial studies the side effects, best dose, and effectiveness of enfortumab vedotin (EV) in combination with pembrolizumab and radiation therapy for treating patients with muscle invasive bladder cancer. Standard of care treatment for muscle invasive bladder cancer is chemotherapy, to shrink the tumor before the main treatment is given (neoadjuvant), followed by surgery to remove all of the bladder as well as nearby tissues and organs (radical cystectomy). In cases where patients are not candidates for the standard of care approach or prefer a bladder sparing option, tri-modality therapy with transurethral resection of bladder tumor (TURBT) followed by combined chemotherapy and radiation therapy is used. Enfortumab vedotin is a monoclonal antibody, enfortumab, linked to an anticancer drug called vedotin. It works by helping the immune system to slow or stop the growth of tumor cells. Enfortumab attaches to a protein called nectin-4 on tumor cells in a targeted way and delivers vedotin to kill them. It is a type of antibody-drug conjugate. Immunotherapy with monoclonal antibodies, such as pembrolizumab, may help the body's immune system attack the cancer, and may interfere with the ability of tumor cells to grow and spread. Intensity-modulated radiation therapy is a type of 3-dimensional radiation therapy that uses computer-generated images to show the size and shape of the tumor. Thin beams of radiation of different intensities are aimed at the tumor from many angles. This type of radiation therapy reduces the damage to healthy tissue near the tumor. Giving enfortumab vedotin with pembrolizumab and radiation therapy may work better in treating patients with muscle invasive bladder cancer.

Trial Health

77
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
47

participants targeted

Target at P50-P75 for phase_1

Timeline
22mo left

Started Mar 2025

Typical duration for phase_1

Geographic Reach
1 country

1 active site

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress39%
Mar 2025Jan 2028

First Submitted

Initial submission to the registry

June 17, 2024

Completed
7 days until next milestone

First Posted

Study publicly available on registry

June 24, 2024

Completed
9 months until next milestone

Study Start

First participant enrolled

March 31, 2025

Completed
2.8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 31, 2028

Expected
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

January 31, 2028

Last Updated

February 18, 2026

Status Verified

February 1, 2026

Enrollment Period

2.8 years

First QC Date

June 17, 2024

Last Update Submit

February 13, 2026

Conditions

Outcome Measures

Primary Outcomes (4)

  • Recommended phase II dose (RP2D) (Phase Ib)

    The RP2D is the last dose cohort at which no more than one instance of a dose limiting toxicity (DLT) is observed among 6 participants treated. If the maximum tolerated dose (MTD) cannot be determined due to lack of DLT during the DLT window, the maximum dose level of enfortumab vedotin administered during the study will be declared the RP2D. For the purposes of this study, the RP2D is the MTD.

    Up to 72 days

  • Proportion of participants reporting dose limiting toxicities (DLTs) (Phase Ib)

    The DLT evaluation period will be within the first three cycles (e.g., 56 days or eight weeks, and not to exceed 72 days) of treatment start with enfortumab-vedotin, pembrolizumab, and standard of care fractionation radiation therapy. Participants who receive \> 75% of intended enfortumab vedotin, pembrolizumab, and standard of care radiation doses will be considered DLT evaluable (DE).

    Up to 72 days

  • Frequency of treatment-emergent adverse events

    The frequency of adverse events by highest grade and overall attribution to study drugs, according to the NCI Common Terminology Criteria for Adverse Events (CTCAE) version 5.0

    Up to 14 months

  • Percentage of participants with Clinical complete response (cCR) (Phase II)

    The rate of clinical complete response to treatment (cCR) will be measured as the percentage of participants with cCR based on cystoscopy and TURBT done at 6 months from treatment start. cCR is defined as no visual tumor AND no histological presence of tumor (i.e., ypT0).

    Up to 6 months

Secondary Outcomes (9)

  • Proportion of participants with Clinical Complete Response (cCR) (Phase Ib)

    Up to 6 months

  • Median Recurrence Free Survival Rate (RFS) at 1 year

    Up to 1 year

  • Median Cystectomy Free Survival rate (CFS) at 2 years

    Up to 2 years

  • Median Overall Survival (OS) at 2 years

    Up to 2 years

  • Median Overall OS

    Up to 5 years

  • +4 more secondary outcomes

Study Arms (4)

Dose Level 1: 0.75 mg/kg Enfortumab Vedotin (Starting Dose)

EXPERIMENTAL

Participants receive 0.75 mg/kg enfortumab vedotin intravenously (IV) over 30 minutes on days 1 and 8 of cycles 1-5 and pembrolizumab IV on day 1 of each cycle. Cycles repeat every 21 days for up to 5 cycles of enfortumab vedotin and up to 17 cycles of pembrolizumab in the absence of disease progression or unacceptable toxicity. Beginning on cycle 1 day 1, participants also undergo standard of care intensity modulated radiation therapy (IMRT) once daily (QD) for 32 days over 6.5-8 weeks. Participants also undergo TURBT, cystoscopy, as well as imaging throughout the study.

Drug: Enfortumab VedotinBiological: PembrolizumabRadiation: Intensity Modulated Radiation Therapy (IMRT)Procedure: Transurethral Resection of Bladder TumorProcedure: Cystoscopy (CS)Procedure: Computed Tomography (CT)Procedure: Magnetic Resonance Imaging (MRI)Procedure: Positron Emission Tomography (PET)

Dose Level 2: 1.0 mg/kg Enfortumab Vedotin

EXPERIMENTAL

Participants receive 1.05 mg/kg enfortumab vedotin intravenously (IV) over 30 minutes on days 1 and 8 of cycles 1-5 and pembrolizumab IV on day 1 of each cycle. Cycles repeat every 21 days for up to 5 cycles of enfortumab vedotin and up to 17 cycles of pembrolizumab in the absence of disease progression or unacceptable toxicity. Beginning on cycle 1 day 1, participants also undergo standard of care intensity modulated radiation therapy (IMRT) once daily (QD) for 32 days over 6.5-8 weeks. Participants also undergo TURBT, cystoscopy, as well as imaging throughout the study.

Drug: Enfortumab VedotinBiological: PembrolizumabRadiation: Intensity Modulated Radiation Therapy (IMRT)Procedure: Transurethral Resection of Bladder TumorProcedure: Cystoscopy (CS)Procedure: Computed Tomography (CT)Procedure: Magnetic Resonance Imaging (MRI)Procedure: Positron Emission Tomography (PET)

Dose Level 3: 1.25 mg/kg Enfortumab Vedotin

EXPERIMENTAL

Participants receive 1.25 mg/kg enfortumab vedotin intravenously (IV) over 30 minutes on days 1 and 8 of cycles 1-5 and pembrolizumab IV on day 1 of each cycle. Cycles repeat every 21 days for up to 5 cycles of enfortumab vedotin and up to 17 cycles of pembrolizumab in the absence of disease progression or unacceptable toxicity. Beginning on cycle 1 day 1, participants also undergo standard of care intensity modulated radiation therapy (IMRT) once daily (QD) for 32 days over 6.5-8 weeks. Participants also undergo TURBT, cystoscopy, as well as imaging throughout the study.

Drug: Enfortumab VedotinBiological: PembrolizumabRadiation: Intensity Modulated Radiation Therapy (IMRT)Procedure: Transurethral Resection of Bladder TumorProcedure: Cystoscopy (CS)Procedure: Computed Tomography (CT)Procedure: Magnetic Resonance Imaging (MRI)Procedure: Positron Emission Tomography (PET)

Dose Expansion; Recommended Phase 2 Dose (RP2D)

EXPERIMENTAL

Participants receive RP2D of enfortumab vedotin intravenously (IV) over 30 minutes on days 1 and 8 of cycles 1-5 and pembrolizumab IV on day 1 of each cycle. Cycles repeat every 21 days for up to 5 cycles of enfortumab vedotin and up to 17 cycles of pembrolizumab in the absence of disease progression or unacceptable toxicity. Beginning on cycle 1 day 1, participants also undergo standard of care intensity modulated radiation therapy (IMRT) once daily (QD) for 32 days over 6.5-8 weeks. Participants also undergo TURBT, cystoscopy, as well as imaging throughout the study.

Drug: Enfortumab VedotinBiological: PembrolizumabRadiation: Intensity Modulated Radiation Therapy (IMRT)Procedure: Transurethral Resection of Bladder TumorProcedure: Cystoscopy (CS)Procedure: Computed Tomography (CT)Procedure: Magnetic Resonance Imaging (MRI)Procedure: Positron Emission Tomography (PET)

Interventions

Undergo CT imaging

Also known as: CT Scan
Dose Expansion; Recommended Phase 2 Dose (RP2D)Dose Level 1: 0.75 mg/kg Enfortumab Vedotin (Starting Dose)Dose Level 2: 1.0 mg/kg Enfortumab VedotinDose Level 3: 1.25 mg/kg Enfortumab Vedotin

Undergo MRI imaging

Also known as: MRI Scan
Dose Expansion; Recommended Phase 2 Dose (RP2D)Dose Level 1: 0.75 mg/kg Enfortumab Vedotin (Starting Dose)Dose Level 2: 1.0 mg/kg Enfortumab VedotinDose Level 3: 1.25 mg/kg Enfortumab Vedotin

Undergo TURBT

Also known as: Transurethral resection (TURBT)
Dose Expansion; Recommended Phase 2 Dose (RP2D)Dose Level 1: 0.75 mg/kg Enfortumab Vedotin (Starting Dose)Dose Level 2: 1.0 mg/kg Enfortumab VedotinDose Level 3: 1.25 mg/kg Enfortumab Vedotin

Undergo cystoscopy

Also known as: CS
Dose Expansion; Recommended Phase 2 Dose (RP2D)Dose Level 1: 0.75 mg/kg Enfortumab Vedotin (Starting Dose)Dose Level 2: 1.0 mg/kg Enfortumab VedotinDose Level 3: 1.25 mg/kg Enfortumab Vedotin

Undergo PET Scan, may be combined with CT (PET/CT)

Also known as: PET Scan
Dose Expansion; Recommended Phase 2 Dose (RP2D)Dose Level 1: 0.75 mg/kg Enfortumab Vedotin (Starting Dose)Dose Level 2: 1.0 mg/kg Enfortumab VedotinDose Level 3: 1.25 mg/kg Enfortumab Vedotin

Given intravenously (IV)

Also known as: Padcev
Dose Expansion; Recommended Phase 2 Dose (RP2D)Dose Level 1: 0.75 mg/kg Enfortumab Vedotin (Starting Dose)Dose Level 2: 1.0 mg/kg Enfortumab VedotinDose Level 3: 1.25 mg/kg Enfortumab Vedotin
PembrolizumabBIOLOGICAL

Given IV

Also known as: Keytruda
Dose Expansion; Recommended Phase 2 Dose (RP2D)Dose Level 1: 0.75 mg/kg Enfortumab Vedotin (Starting Dose)Dose Level 2: 1.0 mg/kg Enfortumab VedotinDose Level 3: 1.25 mg/kg Enfortumab Vedotin

Undergo standard of care, IMRT

Also known as: Standard of care IMRT
Dose Expansion; Recommended Phase 2 Dose (RP2D)Dose Level 1: 0.75 mg/kg Enfortumab Vedotin (Starting Dose)Dose Level 2: 1.0 mg/kg Enfortumab VedotinDose Level 3: 1.25 mg/kg Enfortumab Vedotin

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Biopsy-confirmed muscle-invasive bladder cancer (cT2,T3,T4a). (Note: Tissue samples are required.) (Participants with cT3/T4a staged disease will be capped at 25% of patients treated at RP2D).
  • Urothelial histology present. Mixed histologies other than small cell/neuroendocrine are allowed as long as some urothelial histology is present. Neuroendocrine histology of any component and pure variant (non-urothelial) histology tumors will be excluded. (Patients with \< 50% urothelial histology will be capped at 25% of patients treated at RP2D).
  • Must be judged by the investigator to be ineligible for radical cystectomy or electing not to undergo radical cystectomy.
  • Must be eligible for and agree to receive bladder irradiation as determined by the treating investigator.
  • Must have a TURBT within 8 weeks of combination treatment start with viable tumor content. If no viable tumor content is present on TURBT, the patient will be replaced in the study.
  • Patients who have autoimmune disease will be evaluated on a case-by-case basis and can only enroll so long as participants are not on active immunosuppression with a corticoid steroid allowance exceeding 10mg of prednisone or equivalent per day.
  • Age \>= 18 years.
  • Eastern Cooperative Oncology Group (ECOG) performance status \<= 1.
  • Absolute neutrophil count ≥ 1,500/microliter (mcL).
  • Platelets \>= 100,000/mcL.
  • Hemoglobin \>= 9.0 g/dL or ≥ 5.6 mmol/L.
  • \* Criteria must be met without erythropoietin dependency and without packed red blood cell (pRBC) transfusion within last 2 weeks
  • Total bilirubin \<= 1.5 × upper limit of normal, unless elevated due to Gilbert's syndrome and direct bilirubin is within normal limits.
  • Aspartate aminotransferase (AST) (serum glutamic oxaloacetic transaminase (SGOT)) \<= 2.5 X institutional upper limit of normal.
  • Alanine aminotransferase (ALT) (serum glutamic pyruvic transaminase (SGPT)) \<= 2.5 X institutional upper limit of normal.
  • +13 more criteria

You may not qualify if:

  • Presence of distant metastases on imaging (M1 disease).
  • Presence of ≥ N2 disease on imaging (N1 disease allowed, but participants with N1 disease will be capped at 25% of patients treated at RP2D).
  • Presence of small cell / neuroendocrine histology in tumor sample (any content).
  • Absence of urothelial histology in TURBT tumor sample (pure variant histology).
  • Presence of untreated upper tract urothelial cancer.
  • Presence of severe hydronephrosis precluding therapy in the judgement of the treating physician.
  • Baseline neuropathy grade 2 (G2) or greater.
  • Baseline uncontrolled diabetes mellitus.Uncontrolled diabetes is defined as hemoglobin A1c (HbA1c) ≥ 8% or HbA1c 7 to \< 8% with associated diabetes symptoms (polyuria or polydipsia) that are not otherwise explained.
  • \* Note: Patients with prior diagnosis but with disease under control are eligible
  • Prior treatment with systemic immunotherapy or chemotherapy for urothelial cancer. (with the exception of prior systematic therapy treatment \>12 months prior). Note: Prior bacillus calmette-guerin (BCG) and intravesical treatments are allowed
  • Has received prior systemic anti-cancer therapy including investigational agents within 4 weeks prior to cycle 1 day 1.
  • Has received prior radiotherapy within 2 weeks of cycle 1 day 1 or had radiation-related toxicities requiring corticosteroids.
  • Has received a live vaccine or live-attenuated vaccine within 30 days before the first dose of study intervention.
  • \* Note: Administration of killed vaccines is allowed. Any licensed coronavirus 2019 (COVID-19) vaccine (including for emergency use) is allowed in the study as long as they are messenger ribonucleic acid (mRNA) vaccines, replication-incompetent adenoviral vaccines, or inactivated vaccines.
  • Major surgery within 2 weeks prior to first dose of EV.
  • +15 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

University of California, San Francisco

San Francisco, California, 94143, United States

RECRUITING

MeSH Terms

Conditions

Urinary Bladder Neoplasms

Interventions

enfortumab vedotinpembrolizumabRadiotherapy, Intensity-ModulatedTransurethral Resection of BladderCystoscopyMagnetic Resonance Spectroscopy

Condition Hierarchy (Ancestors)

Urologic NeoplasmsUrogenital NeoplasmsNeoplasms by SiteNeoplasmsFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesUrinary Bladder DiseasesUrologic DiseasesMale Urogenital Diseases

Intervention Hierarchy (Ancestors)

Radiotherapy, ConformalRadiotherapy, Computer-AssistedRadiotherapyTherapeuticsUrologic Surgical ProceduresUrogenital Surgical ProceduresSurgical Procedures, OperativeEndoscopyDiagnostic Techniques, SurgicalDiagnostic Techniques and ProceduresDiagnosisDiagnostic Techniques, UrologicalMinimally Invasive Surgical ProceduresSpectrum AnalysisChemistry Techniques, AnalyticalInvestigative Techniques

Study Officials

  • Vadim Koshkin, MD

    University of California, San Francisco

    PRINCIPAL INVESTIGATOR

Central Study Contacts

UCSF Genitourinary Medical Oncology Recruitment

CONTACT

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
OTHER
Responsible Party
PRINCIPAL INVESTIGATOR
PI Title
Principal Investigator, IND Holder

Study Record Dates

First Submitted

June 17, 2024

First Posted

June 24, 2024

Study Start

March 31, 2025

Primary Completion (Estimated)

January 31, 2028

Study Completion (Estimated)

January 31, 2028

Last Updated

February 18, 2026

Record last verified: 2026-02

Data Sharing

IPD Sharing
Will not share

Locations