NCT06247085

Brief Summary

The purpose of this study is to measure efficacy and safety of pegtibatinase treatment compared with placebo in participants with classical HCU receiving standard of care. Study details include:

  • Total Study duration: up to 38 weeks
  • Screening:
  • Initial Screening duration: up to 4 weeks
  • Pre-treatment Diet Standardization Period duration: up to 6 weeks
  • Blinded Treatment Duration: 24 weeks
  • 2-week blinded dose titration period
  • 22-week blinded assessment period
  • Safety Follow-Up: 4 weeks after last dose (as applicable for those not enrolling in the long term extension study, ENSEMBLE)

Trial Health

88
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
70

participants targeted

Target at below P25 for phase_3

Timeline
13mo left

Started Dec 2023

Typical duration for phase_3

Geographic Reach
14 countries

52 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress71%
Dec 2023Sep 2027

Study Start

First participant enrolled

December 28, 2023

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

January 30, 2024

Completed
8 days until next milestone

First Posted

Study publicly available on registry

February 7, 2024

Completed
3.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2027

Expected
1 month until next milestone

Study Completion

Last participant's last visit for all outcomes

September 1, 2027

Last Updated

May 8, 2026

Status Verified

May 1, 2026

Enrollment Period

3.6 years

First QC Date

January 30, 2024

Last Update Submit

May 5, 2026

Conditions

Keywords

HCUcystathionine beta synthase deficiencyClassical Homocystinuria

Outcome Measures

Primary Outcomes (1)

  • Change from baseline in plasma tHcy levels - Weeks 6 to 12

    Change between baseline and average of 6 to 12 week (6, 8, 10, and 12 week) plasma tHcy levels in participants receiving pegtibatinase vs. placebo. Baseline tHcy level defined as average of Week -3, Week -1, and Day 1 pre-dose plasma tHcy

    Weeks 6 - 12

Secondary Outcomes (1)

  • Change from baseline in plasma tHcy levels - Weeks 16 to 24

    Weeks 16 - 24

Study Arms (2)

pegtibatinase

EXPERIMENTAL
Drug: Pegtibatinase

placebo

PLACEBO COMPARATOR
Other: Placebo

Interventions

Pegtibatinase BIW

Also known as: OT-058, TVT-058
pegtibatinase
PlaceboOTHER

volume-matched saline SC BIW

placebo

Eligibility Criteria

Age12 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsChild (0-17), Adult (18-64), Older Adult (65+)

You may qualify if:

  • Must be ≥12 to ≤65 years of age, at the time of signing the informed consent
  • Must have a diagnosis of classical HCU based on clinical, biochemical, and/or molecular genetic testing
  • Plasma tHcy ≥80 µM at Screening visit, with allowance for up to 18 participants who may be enrolled with a Screening plasma tHcy ≥50 to \<80 µM
  • Participants who can become pregnant must have a negative pregnancy test before starting the study and must use a highly effective form of birth control (less than 1% risk of pregnancy per year) during the study and for at least 4 weeks after the last dose.
  • Willing to maintain a generally stable diet for the duration of the study (unless changes are required based on medical/safety reasons)
  • Willing to maintain generally stable intake and doses of betaine, pyridoxine, and medical food for the duration of the study (unless changes are required based on medical/safety reasons)

You may not qualify if:

  • Diagnosis of Marfan syndrome, methylenetetrahydrofolate reductase (MTHFR) deficiency, or disorder of cobalamin metabolism
  • Concurrent disease or condition (eg, history or presence of clinically significant cardiovascular, pulmonary, hepatic, renal, hematologic, gastrointestinal, endocrine, immunologic, dermatologic, neurological, oncologic, or psychiatric disease) that would interfere with study participation or safety (excluding complications of HCU).
  • History of major thrombotic event (eg, cerebrovascular accident, myocardial infarction, pulmonary embolism) in the previous 6 months.
  • Body weight ≥160 kg.
  • Use or planned use of any injectable drugs containing PEG (excluding PEG-containing vaccines)
  • Any previous exposure to pegtibatinase and/or previous participation in a clinical study that included administration of pegtibatinase or pegtarviliase
  • Prior severe immune reaction to a PEG-containing product

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (52)

Phoenix Children's Hospital

Phoenix, Arizona, 85006, United States

NOT YET RECRUITING

Yale University School of Medicine

New Haven, Connecticut, 06519, United States

RECRUITING

Emory University

Atlanta, Georgia, 30322, United States

RECRUITING

Ann & Robert H. Lurie Children's Hospital of Chicago

Chicago, Illinois, 60611, United States

NOT YET RECRUITING

Maine Health - Maine Medical Center

Portland, Maine, 04102, United States

RECRUITING

Uncommon Cures

Chevy Chase, Maryland, 20815, United States

RECRUITING

The Mount Sinai Hospital

New York, New York, 10029, United States

RECRUITING

Science 37 - Virtual Site

Morrisville, North Carolina, 27560, United States

RECRUITING

Oregon Health and Science University

Portland, Oregon, 97239, United States

NOT YET RECRUITING

Children's Hospital of Philadelphia

Philadelphia, Pennsylvania, 19104, United States

RECRUITING

University of Pittsburgh Medical Center - Children's Hospital of Pittsburgh

Pittsburgh, Pennsylvania, 15224, United States

RECRUITING

University of Texas Southwestern Medical Center

Dallas, Texas, 75390, United States

RECRUITING

Utah Health - The University of Utah Primary Children's Hospital

Salt Lake City, Utah, 84113, United States

NOT YET RECRUITING

Royal Adelaide Hospital

Adelaide, Australia

NOT YET RECRUITING

Royal Children's Hospital Melbourne

Parkville, Australia

NOT YET RECRUITING

Westmead Hospital

Westmead, Australia

NOT YET RECRUITING

Cliniques Universitaires Saint-Luc

Brussels, Belgium

NOT YET RECRUITING

Universitair Ziekenhuis Antwerpen (UZA)

Edegem, Belgium

NOT YET RECRUITING

Assistance Publique - Hôpitaux de Paris (AP-HP) - Hôpital Necker-Enfants Malades

Paris, France

NOT YET RECRUITING

CHRU Hôpitaux de Tours - Hôpital Bretonneau

Tours, France

NOT YET RECRUITING

Centre Hospitalier Régional Universitaire de Nancy (CHRU) - Hopitaux de Brabois - Hôpital d'enfants

Vandœuvre-lès-Nancy, France

NOT YET RECRUITING

Universitätsklinikum Hamburg-Eppendorf

Hamburg, Germany

NOT YET RECRUITING

Universitätsklinikum Leipzig

Leipzig, Germany

NOT YET RECRUITING

Universitätsklinikum Münster

Münster, Germany

NOT YET RECRUITING

Children's Health Ireland (CHI) at Temple Street

Dublin, Ireland

NOT YET RECRUITING

Ospedale Pediatrico Giovanni XXIII

Bari, Italy

NOT YET RECRUITING

IRCCS Istituto Giannina Gaslini

Genova, Italy

NOT YET RECRUITING

Fondazione IRCCS Ca' Granda Ospedale Maggiore Policlinico (Policlinico di Milano)

Milan, Italy

NOT YET RECRUITING

Fondazione IRCCS San Gerardo Dei Tintori - Ospedale San Gerardo

Monza, Italy

NOT YET RECRUITING

Azienda Ospedaliera di Padova

Padova, Italy

NOT YET RECRUITING

SP ZOZ Szpital Uniwersytecki w Krakowie

Krakow, Poland

NOT YET RECRUITING

Instytut Matki i Dziecka

Warsaw, Poland

NOT YET RECRUITING

Instytut Pomnik-Centrum Zdrowia Dziecka

Warsaw, Poland

NOT YET RECRUITING

Unidade Local de Saúde de Coimbra, EPE - Hospitais da Universidade de Coimbra

Coimbra, Portugal

NOT YET RECRUITING

Unidade Local de Saúde de Santa Maria, EPE - Hospital de Santa Maria

Lisbon, Portugal

NOT YET RECRUITING

Unidade Local de Saúde de São João, EPE - Hospital São João

Porto, Portugal

NOT YET RECRUITING

Hamad General Hospital

Doha, Qatar

NOT YET RECRUITING

Sidra Hospital

Doha, Qatar

NOT YET RECRUITING

King Abdullah International Medical Research Center

Riyadh, Saudi Arabia

NOT YET RECRUITING

King Faisal Specialist Hospital and Research Centre (KFSHRC) - Riyadh

Riyadh, Saudi Arabia

NOT YET RECRUITING

Hospital Sant Joan de Déu

Barcelona, Spain

NOT YET RECRUITING

Hospital Universitario 12 de Octubre

Madrid, Spain

NOT YET RECRUITING

Hospital Universitario Ramón y Cajal

Madrid, Spain

NOT YET RECRUITING

Complejo Hospitalario Universitario de Santiago (CHUS) - Hospital Clínico Universitario

Santiago de Compostela, Spain

NOT YET RECRUITING

Hospital Universitario Virgen del Rocío

Seville, Spain

NOT YET RECRUITING

Gazi University Hospital

Ankara, Turkey (Türkiye)

NOT YET RECRUITING

Ege Üniversitesi Hastanesi Bornova

Bornova, Turkey (Türkiye)

NOT YET RECRUITING

Istanbul University Cerrahpasa Hospital

Istanbul, Turkey (Türkiye)

NOT YET RECRUITING

Birmingham Women's and Children's NHS Foundation Trust

Birmingham, United Kingdom

NOT YET RECRUITING

University Hospitals Birmingham NHS Foundation Trust - Queen Elizabeth Hospital Birmingham

Birmingham, United Kingdom

NOT YET RECRUITING

University College London Hospitals NHS Foundation Trust - National Hospital for Neurology and Neurosurgery

London, United Kingdom

NOT YET RECRUITING

Salford Royal NHS Foundation Trust - Salford Royal Hospital

Salford, United Kingdom

NOT YET RECRUITING

MeSH Terms

Conditions

Homocystinuria

Condition Hierarchy (Ancestors)

Brain Diseases, Metabolic, InbornBrain Diseases, MetabolicBrain DiseasesCentral Nervous System DiseasesNervous System DiseasesHyperhomocysteinemiaAmino Acid Metabolism, Inborn ErrorsMetabolism, Inborn ErrorsGenetic Diseases, InbornCongenital, Hereditary, and Neonatal Diseases and AbnormalitiesConnective Tissue DiseasesSkin and Connective Tissue DiseasesMetabolic DiseasesNutritional and Metabolic Diseases

Study Officials

  • Michael Imperiale, MD

    Travere Therapeutics, Inc.

    STUDY DIRECTOR

Central Study Contacts

Travere Call Center

CONTACT

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 30, 2024

First Posted

February 7, 2024

Study Start

December 28, 2023

Primary Completion (Estimated)

August 1, 2027

Study Completion (Estimated)

September 1, 2027

Last Updated

May 8, 2026

Record last verified: 2026-05

Data Sharing

IPD Sharing
Will share

Requests for clinical trial data, including language stating its intended use, should be directed to datarequest@travere.com. If approved, the requested information will be provided to the requestor after signing a data access agreement. Requests can be made following completion of the study and full publication of the study data in a peer reviewed journal for up to 36 months following its publication. Travere reserves the right to decline or recommend modifications to a request if it does not comply with the data sharing policy or if it is determined that the request is made by a biased source.

Time Frame
Requests can be made following completion of the study and full publication of the study data in a peer reviewed journal for up to 36 months following its publication.
Access Criteria
Requires submission and approval of intended use and a data sharing agreement.

Locations