NCT06234605

Brief Summary

This is a Phase 1b, open-label, multicenter, safety, tolerability and efficacy study of HC-7366 in combination with belzutifan (WELIREG™). This is a multipart study that consists of a HC-7366 monotherapy cohort, a combination dose escalation, and a combination dose expansion. Approximately 80 patients will be enrolled in this study (up to 20 patients will be enrolled into the HC-7366 monotherapy cohort, up to 30 patients into the combination dose escalation, and up to 30 patients into the combination dose expansion). The primary purpose of this study is to determine the maximum tolerated dose of HC-7366 in combination with belzutifan in patients with locally advanced (inoperable) or metastatic RCC with predominantly clear cell histology, irrespective of VHL gene mutation status.

Trial Health

77
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
80

participants targeted

Target at P75+ for phase_1

Timeline
18mo left

Started Apr 2024

Typical duration for phase_1

Geographic Reach
1 country

20 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress58%
Apr 2024Nov 2027

First Submitted

Initial submission to the registry

January 9, 2024

Completed
22 days until next milestone

First Posted

Study publicly available on registry

January 31, 2024

Completed
3 months until next milestone

Study Start

First participant enrolled

April 29, 2024

Completed
2.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

November 1, 2026

Expected
1 year until next milestone

Study Completion

Last participant's last visit for all outcomes

November 1, 2027

Last Updated

January 15, 2026

Status Verified

January 1, 2026

Enrollment Period

2.5 years

First QC Date

January 9, 2024

Last Update Submit

January 13, 2026

Conditions

Keywords

ccRCCbelzutifankidney cancermetastaticlocally advancedHC-7366WELIREG™

Outcome Measures

Primary Outcomes (1)

  • Determination of MTD and RP2D (combination cohorts only)

    To identify the maximum tolerated dose (MTD) and/ or recommended Phase 2 dose (RP2D), and evaluate the safety, tolerability and dose-limiting toxicities (DLTs) of HC-7366 in combination with belzutifan in patients with locally advanced (inoperable) or metastatic RCC with predominantly clear cell histology irrespective of VHL gene mutation status

    30 months

Study Arms (2)

Monotherapy

EXPERIMENTAL

Participants will receive HC-7366 monotherapy \[dose to be determined\] daily

Drug: HC-7366

Combination

EXPERIMENTAL

Participants will receive HC-7366 monotherapy \[dose to be determined\] in combination with belzutifan \[120 mg\] daily

Drug: HC-7366Drug: Belzutifan

Interventions

HC-7366 is a novel, orally administered, highly selective and potent general control nonderepressible 2 (GCN2) kinase activator.

CombinationMonotherapy

Belzutifan is a potent and selective HIF-2α inhibitor

Also known as: WELIREG™, MK-6482
Combination

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Has diagnosis of locally advanced (inoperable) or metastatic RCC with a predominant clear cell component
  • Be age 18 years or older (male or female) at the time of consent

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (20)

University of Arizona Cancer Center

Tucson, Arizona, 85719, United States

RECRUITING

University of California San Diego Moores Cancer Center

La Jolla, California, 92093, United States

RECRUITING

Cedars-Sinai Medical Center

Los Angeles, California, 90048, United States

RECRUITING

University of Colorado Anschutz Medical Campus

Aurora, Colorado, 80045, United States

RECRUITING

Rocky Mountain Cancer Centers, LLP

Lone Tree, Colorado, 80124, United States

RECRUITING

Yale - New Haven Hospital

New Haven, Connecticut, 06520, United States

RECRUITING

HealthPartners Cancer Research Center

Saint Paul, Minnesota, 55101, United States

RECRUITING

Washington University School of Medicine

St Louis, Missouri, 63110, United States

RECRUITING

Memorial Sloan Kettering Cancer Center

New York, New York, 10065, United States

RECRUITING

University Hospitals Cleveland Medical Center

Cleveland, Ohio, 44106, United States

RECRUITING

Cleveland Clinic

Cleveland, Ohio, 44195, United States

RECRUITING

Providence Cancer Institute

Portland, Oregon, 97213, United States

RECRUITING

SCRI Oncology Partners

Nashville, Tennessee, 37203, United States

RECRUITING

Texas Oncology

Dallas, Texas, 75246, United States

RECRUITING

University of Texas Southwestern Medical Center

Dallas, Texas, 75390, United States

RECRUITING

University Medical Center & Texas Tech Health Science Center

Lubbock, Texas, 79430, United States

RECRUITING

Virginia Cancer Specialists

Fairfax, Virginia, 22031, United States

RECRUITING

Swedish Medical Center

Seattle, Washington, 98104, United States

RECRUITING

Fred Hutchinson Cancer Center

Seattle, Washington, 98109, United States

RECRUITING

University of Wisconsin - Carbone Cancer Center

Madison, Wisconsin, 53705, United States

RECRUITING

MeSH Terms

Conditions

Carcinoma, Renal CellKidney NeoplasmsNeoplasm Metastasis

Interventions

belzutifan

Condition Hierarchy (Ancestors)

AdenocarcinomaCarcinomaNeoplasms, Glandular and EpithelialNeoplasms by Histologic TypeNeoplasmsUrologic NeoplasmsUrogenital NeoplasmsNeoplasms by SiteFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesKidney DiseasesUrologic DiseasesMale Urogenital DiseasesNeoplastic ProcessesPathologic ProcessesPathological Conditions, Signs and Symptoms

Central Study Contacts

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 9, 2024

First Posted

January 31, 2024

Study Start

April 29, 2024

Primary Completion (Estimated)

November 1, 2026

Study Completion (Estimated)

November 1, 2027

Last Updated

January 15, 2026

Record last verified: 2026-01

Locations